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320 KiB
320 KiB
| 1 | Peptide | Cell line | Cargo | PubmedID | Uptake | Units | Conc. | Time | Temp. | Method | Type | Sequence |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 2 | Tat (49-57) | Jurkat cells | Fluorescein | 11087855 | 650 | Mean Fluorescence intensity | 12.5 uM | 15 min | 23ºC | Flow cytometry | Cellular uptake | RKKRRQRRR |
| 3 | Tat (49-56) | Jurkat cells | Fluorescein | 11087855 | 31.25 | Mean Fluorescence intensity | 12.5 uM | 10 min | 23ºC | Flow cytometry | Cellular uptake | RKKRRQRR |
| 4 | Tat (49-55) | Jurkat cells | Fluorescein | 11087855 | 10 | Mean Fluorescence intensity | 12.5 uM | 10 min | 23ºC | Flow cytometry | Cellular uptake | RKKRRQR |
| 5 | Tat (50-57) | Jurkat cells | Fluorescein | 11087855 | 22.5 | Mean Fluorescence intensity | 12.5 uM | 10 min | 23ºC | Flow cytometry | Cellular uptake | KKRRQRRR |
| 6 | Tat (51-57) | Jurkat cells | Fluorescein | 11087855 | 20 | Mean Fluorescence intensity | 12.5 uM | 10 min | 23ºC | Flow cytometry | Cellular uptake | KRRQRRR |
| 7 | D-Tat (49-57) | Jurkat cells | Fluorescein | 11087855 | 1800 | Mean Fluorescence intensity | 12.5 uM | 15 min | 23ºC | Flow cytometry | Cellular uptake | rkkrrqrrr |
| 8 | Retro - Tat (57-49) | Jurkat cells | Fluorescein | 11087855 | 2450 | Mean Fluorescence intensity | 12.5 uM | 15 min | 23ºC | Flow cytometry | Cellular uptake | RRRQRRKKR |
| 9 | D-Tat (57-49) | Jurkat cells | Fluorescein | 11087855 | 3600 | Mean Fluorescence intensity | 12.5 uM | 15 min | 23ºC | Flow cytometry | Cellular uptake | rrrqrrkkr |
| 10 | Ala49 substitution mutant of Tat (49-57) | Jurkat cells | Fluorescein | 11087855 | 16.25 | Mean Fluorescence intensity | 12.5 uM | 10 min | 23ºC | Flow cytometry | Cellular uptake | AKKRRQRRR |
| 11 | Ala50 substitution mutant of Tat (49-57) | Jurkat cells | Fluorescein | 11087855 | 32.5 | Mean Fluorescence intensity | 12.5 uM | 10 min | 23ºC | Flow cytometry | Cellular uptake | RAKRRQRRR |
| 12 | Ala51 substitution mutant of Tat (49-57) | Jurkat cells | Fluorescein | 11087855 | 37.5 | Mean Fluorescence intensity | 12.5 uM | 10 min | 23ºC | Flow cytometry | Cellular uptake | RKARRQRRR |
| 13 | Ala52 substitution mutant of Tat (49-57) | Jurkat cells | Fluorescein | 11087855 | 20 | Mean Fluorescence intensity | 12.5 uM | 10 min | 23ºC | Flow cytometry | Cellular uptake | RKKARQRRR |
| 14 | Ala53 substitution mutant of Tat (49-57) | Jurkat cells | Fluorescein | 11087855 | 30 | Mean Fluorescence intensity | 12.5 uM | 10 min | 23ºC | Flow cytometry | Cellular uptake | RKKRAQRRR |
| 15 | Ala54 substitution mutant of Tat (49-57) | Jurkat cells | Fluorescein | 11087855 | 132.5 | Mean Fluorescence intensity | 12.5 uM | 10 min | 23ºC | Flow cytometry | Cellular uptake | RKKRRARRR |
| 16 | Ala55 substitution mutant of Tat (49-57) | Jurkat cells | Fluorescein | 11087855 | 32.5 | Mean Fluorescence intensity | 12.5 uM | 10 min | 23ºC | Flow cytometry | Cellular uptake | RKKRRQARR |
| 17 | Ala56 substitution mutant of Tat (49-57) | Jurkat cells | Fluorescein | 11087855 | 35 | Mean Fluorescence intensity | 12.5 uM | 10 min | 23ºC | Flow cytometry | Cellular uptake | RKKRRQRAR |
| 18 | Ala57 substitution mutant of Tat (49-57) | Jurkat cells | Fluorescein | 11087855 | 12.5 | Mean Fluorescence intensity | 12.5 uM | 10 min | 23ºC | Flow cytometry | Cellular uptake | RKKRRQRRA |
| 19 | R5 | Jurkat cells | Fluorescein | 11087855 | 100 | Mean Fluorescence intensity | 12.5 uM | 15 min | 23ºC | Flow cytometry | Cellular uptake | RRRRR |
| 20 | R6 | Jurkat cells | Fluorescein | 11087855 | 500 | Mean Fluorescence intensity | 12.5 uM | 15 min | 23ºC | Flow cytometry | Cellular uptake | RRRRRR |
| 21 | R7 | Jurkat cells | Fluorescein | 11087855 | 1225 | Mean Fluorescence intensity | 12.5 uM | 15 min | 23ºC | Flow cytometry | Cellular uptake | RRRRRRR |
| 22 | R8 | Jurkat cells | Fluorescein | 11087855 | 1700 | Mean Fluorescence intensity | 12.5 uM | 15 min | 23ºC | Flow cytometry | Cellular uptake | RRRRRRRR |
| 23 | R9 | Jurkat cells | Fluorescein | 11087855 | 2650 | Mean Fluorescence intensity | 12.5 uM | 15 min | 23ºC | Flow cytometry | Cellular uptake | RRRRRRRRR |
| 24 | D-R5 | Jurkat cells | Fluorescein | 11087855 | 150 | Mean Fluorescence intensity | 12.5 uM | 15 min | 23ºC | Flow cytometry | Cellular uptake | rrrrr |
| 25 | D-R6 | Jurkat cells | Fluorescein | 11087855 | 950 | Mean Fluorescence intensity | 12.5 uM | 15 min | 23ºC | Flow cytometry | Cellular uptake | rrrrrr |
| 26 | D-R7 | Jurkat cells | Fluorescein | 11087855 | 3100 | Mean Fluorescence intensity | 12.5 uM | 15 min | 23ºC | Flow cytometry | Cellular uptake | rrrrrrr |
| 27 | D-R8 | Jurkat cells | Fluorescein | 11087855 | 4400 | Mean Fluorescence intensity | 12.5 uM | 15 min | 23ºC | Flow cytometry | Cellular uptake | rrrrrrrr |
| 28 | D-R9 | Jurkat cells | Fluorescein | 11087855 | 5125 | Mean Fluorescence intensity | 12.5 uM | 15 min | 23ºC | Flow cytometry | Cellular uptake | rrrrrrrrr |
| 29 | I | Aortic endothelial cells | Fluorescein | 10323198 | 228 ± 54 | pmol internalized peptide / mg protein | 1.8 uM | 30 min | 37ºC | HPCL-analysis | Internalization | KLALKLALKALKAALKLA |
| 30 | KLA1 | Aortic endothelial cells | NA | 10323198 | 161 ± 21 | pmol internalized peptide / mg protein | 1.8 uM | 30 min | 37ºC | HPCL-analysis | Internalization | KLALKLALKAWKAALKLA |
| 31 | KLA2 | Aortic endothelial cells | NA | 10323198 | 15 ± 6 | pmol internalized peptide / mg protein | 1.8 uM | 30 min | 37ºC | HPCL-analysis | Internalization | KLALKAALKAWKAAAKLA |
| 32 | KLA3 | Aortic endothelial cells | NA | 10323198 | <10 | pmol internalized peptide / mg protein | 1.8 uM | 30 min | 37ºC | HPCL-analysis | Internalization | KLALKAAAKAWKAAAKAA |
| 33 | KLA11 | Aortic endothelial cells | NA | 10323198 | 47 ± 7 | pmol internalized peptide / mg protein | 1.8 uM | 30 min | 37ºC | HPCL-analysis | Internalization | KITLKLAIKAWKLALKAA |
| 34 | KLA5 | Aortic endothelial cells | NA | 10323198 | 68 ± 2 | pmol internalized peptide / mg protein | 1.8 uM | 30 min | 37ºC | HPCL-analysis | Internalization | KIAAKSIAKIWKSILKIA |
| 35 | KLA12 | Aortic endothelial cells | NA | 10323198 | 149 ± 20 | pmol internalized peptide / mg protein | 1.8 uM | 30 min | 37ºC | HPCL-analysis | Internalization | KALAKALAKLWKALAKAA |
| 36 | KLA13 | Aortic endothelial cells | NA | 10323198 | 15 ± 4 | pmol internalized peptide / mg protein | 1.8 uM | 30 min | 37ºC | HPCL-analysis | Internalization | KLALKLALKWAKLALKAA |
| 37 | KLA14 | Aortic endothelial cells | NA | 10323198 | 29 ± 14 | pmol internalized peptide / mg protein | 1.8 uM | 30 min | 37ºC | HPCL-analysis | Internalization | KLLAKAAKKWLLLALKAA |
| 38 | KLA9 | Aortic endothelial cells | NA | 10323198 | 44 ± 10 | pmol internalized peptide / mg protein | 1.8 uM | 30 min | 37ºC | HPCL-analysis | Internalization | KLLAKAALKWLLKALKAA |
| 39 | KLA10 | Aortic endothelial cells | NA | 10323198 | 218 ± 31 | pmol internalized peptide / mg protein | 1.8 uM | 30 min | 37ºC | HPCL-analysis | Internalization | KALKKLLAKWLAAAKALL |
| 40 | KLA15 | Aortic endothelial cells | NA | 10323198 | 226 ± 19 | pmol internalized peptide / mg protein | 1.8 uM | 30 min | 37ºC | HPCL-analysis | Internalization | KLAAALLKKWKKLAAALL |
| 41 | KLA8 | Aortic endothelial cells | Fluorescein | 10323198 | 341 ± 58 | pmol internalized peptide / mg protein | 1.8 uM | 30 min | 37ºC | HPCL-analysis | Internalization | KALAALLKKWAKLLAALK |
| 42 | CPP-II | Aortic endothelial cells | Fluorescein | 10323198 | 371 ± 56 | pmol internalized peptide / mg protein | 1.8 uM | 30 min | 37ºC | HPCL-analysis | Internalization | KALAALLKKLAKLLAALK |
| 43 | CPP-III | Aortic endothelial cells | Fluorescein | 10323198 | 218 ± 23 | pmol internalized peptide / mg protein | 1.8 uM | 30 min | 37ºC | HPCL-analysis | Internalization | KLALKLALKALKAALK |
| 44 | CPP-IV | Aortic endothelial cells | Fluorescein | 10323198 | <30 | pmol internalized peptide / mg protein | 1.8 uM | 30 min | 37ºC | HPCL-analysis | Internalization | KLALKALKAALKLA |
| 45 | CPP-V | Aortic endothelial cells | Fluorescein | 10323198 | <30 | pmol internalized peptide / mg protein | 1.8 uM | 30 min | 37ºC | HPCL-analysis | Internalization | KLALKLALKALKAA |
| 46 | CPP-VI | Aortic endothelial cells | Fluorescein | 10323198 | <30 | pmol internalized peptide / mg protein | 1.8 uM | 30 min | 37ºC | HPCL-analysis | Internalization | KLGLKLGLKGLKGGLKLG |
| 47 | CPP-VII | Aortic endothelial cells | Fluorescein | 10323198 | 42 ± 12.4 | pmol internalized peptide / mg protein | 1.8 uM | 30 min | 37ºC | HPCL-analysis | Internalization | KLALKLALKALQAALQLA |
| 48 | CPP-VIII | Aortic endothelial cells | Fluorescein | 10323198 | 461 ± 44 | pmol internalized peptide / mg protein | 1.8 uM | 30 min | 37ºC | HPCL-analysis | Internalization | KLALQLALQALQAALQLA |
| 49 | CPP-IX | Aortic endothelial cells | Fluorescein | 10323198 | 5670 ± 3971 | pmol internalized peptide / mg protein | 1.8 uM | 30 min | 37ºC | HPCL-analysis | Internalization | QLALQLALQALQAALQLA |
| 50 | CPP-X | Aortic endothelial cells | Fluorescein | 10323198 | 135 ± 14.6 | pmol internalized peptide / mg protein | 1.8 uM | 30 min | 37ºC | HPCL-analysis | Internalization | ELALELALEALEAALELA |
| 51 | CPP-XI | Aortic endothelial cells | Fluorescein | 10323198 | 539 ± 80 | pmol internalized peptide / mg protein | 1.8 uM | 30 min | 37ºC | HPCL-analysis | Internalization | LKTLATALTKLAKTLTTL |
| 52 | CPP-XIII | Aortic endothelial cells | Fluorescein | 10323198 | 141 ± 54 | pmol internalized peptide / mg protein | 1.8 uM | 30 min | 37ºC | HPCL-analysis | Internalization | LKTLTETLKELTKTLTEL |
| 53 | pAntpHD (43-58) | Cortical striatal cells | Biotin | 8663410 | 0.24 | OD (optical density values) | 44 uM | 2h | 4ºC | ELISA | Internalization | RQIKIWFQNRRMKWKK |
| 54 | pAntpHD (58-43) | Cortical striatal cells | Biotin | 8663410 | 0.26 | OD (optical density values) | 44 uM | 2h | 4ºC | ELISA | Internalization | KKWKMRRNQFWIKIQR |
| 55 | D form of pAntpHD (43-58) | Cortical striatal cells | Biotin | 8663410 | 0.45 | OD (optical density values) | 44 uM | 2h | 4ºC | ELISA | Internalization | rqikiwfqnrrmkwkk |
| 56 | pAntpHD (Pro50) | Cortical striatal cells | Biotin | 8663410 | 0.88 | OD (optical density values) | 44 uM | 2h | 4ºC | ELISA | Internalization | RQIKIWFPNRRMKWKK |
| 57 | pAntpHD (3Pro) | Cortical striatal cells | Biotin | 8663410 | 0.18 | OD (optical density values) | 44 uM | 2h | 4ºC | ELISA | Internalization | RQPKIWFPNRRKPWKK |
| 58 | pAntp (43-58) | HaCaT cells | Biotin | 10784032 | 100.0 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | NA | Fluorescent Microscopy | Cellular uptake | RQIKIWFQNRRMKWKK |
| 59 | pAntp (43-57) | HaCaT cells | Biotin | 10784032 | 57 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | NA | Fluorescent Microscopy | Cellular uptake | RQIKIWFQNRRMKWK |
| 60 | pAntp (43-56) | HaCaT cells | Biotin | 10784032 | 47.5 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | NA | Fluorescent Microscopy | Cellular uptake | RQIKIWFQNRRMKW |
| 61 | pAntp (43-55) | HaCaT cells | Biotin | 10784032 | 28 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | NA | Fluorescent Microscopy | Cellular uptake | RQIKIWFQNRRMK |
| 62 | pAntp (43-54) | HaCaT cells | Biotin | 10784032 | 19.5 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | NA | Fluorescent Microscopy | Cellular uptake | RQIKIWFQNRRM |
| 63 | pAntp (43-53) | HaCaT cells | Biotin | 10784032 | 25 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | NA | Fluorescent Microscopy | Cellular uptake | RQIKIWFQNRR |
| 64 | pAntp (43-52) | HaCaT cells | Biotin | 10784032 | 15 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | NA | Fluorescent Microscopy | Cellular uptake | RQIKIWFQNR |
| 65 | pAntp (43-51) | HaCaT cells | Biotin | 10784032 | 18 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | NA | Fluorescent Microscopy | Cellular uptake | RQIKIWFQN |
| 66 | pAntp (43-50) | HaCaT cells | Biotin | 10784032 | 13 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | NA | Fluorescent Microscopy | Cellular uptake | RQIKIWFQ |
| 67 | pAntp (43-48) | HaCaT cells | Biotin | 10784032 | 20 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | NA | Fluorescent Microscopy | Cellular uptake | RQIKIW |
| 68 | pAntp (44-58) | HaCaT cells | Biotin | 10784032 | 87 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | NA | Fluorescent Microscopy | Cellular uptake | QIKIWFQNRRMKWKK |
| 69 | pAntp (45-58) | HaCaT cells | Biotin | 10784032 | 94 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | NA | Fluorescent Microscopy | Cellular uptake | IKIWFQNRRMKWKK |
| 70 | pAntp (46-58) | HaCaT cells | Biotin | 10784032 | 67 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | NA | Fluorescent Microscopy | Cellular uptake | KIWFQNRRMKWKK |
| 71 | pAntp (47-58) | HaCaT cells | Biotin | 10784032 | 48 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | NA | Fluorescent Microscopy | Cellular uptake | IWFQNRRMKWKK |
| 72 | pAntp (48-58) | HaCaT cells | Biotin | 10784032 | 52 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | NA | Fluorescent Microscopy | Cellular uptake | WFQNRRMKWKK |
| 73 | pAntp (49-58) | HaCaT cells | Biotin | 10784032 | 64 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | NA | Fluorescent Microscopy | Cellular uptake | FQNRRMKWKK |
| 74 | pAntp (50-58) | HaCaT cells | Biotin | 10784032 | 60 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | NA | Fluorescent Microscopy | Cellular uptake | QNRRMKWKK |
| 75 | pAntp (51-58) | HaCaT cells | Biotin | 10784032 | 60 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | NA | Fluorescent Microscopy | Cellular uptake | NRRMKWKK |
| 76 | pAntp (52-58) | HaCaT cells | Biotin | 10784032 | 50 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | NA | Fluorescent Microscopy | Cellular uptake | RRMKWKK |
| 77 | pAntp (53-58) | HaCaT cells | Biotin | 10784032 | 22 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | NA | Fluorescent Microscopy | Cellular uptake | RMKWKK |
| 78 | Ala43 substitution mutant of pAntp (43-58) | HaCaT cells | Biotin | 10784032 | 89 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | NA | Fluorescent Microscopy | Cellular uptake | AQIKIWFQNRRMKWKK |
| 79 | Ala44 substitution mutant of pAntp (43-58) | HaCaT cells | Biotin | 10784032 | 67 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | NA | Fluorescent Microscopy | Cellular uptake | RAIKIWFQNRRMKWKK |
| 80 | Ala45 substitution mutant of pAntp (43-58) | HaCaT cells | Biotin | 10784032 | 82 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | NA | Fluorescent Microscopy | Cellular uptake | RQAKIWFQNRRMKWKK |
| 81 | Ala46 substitution mutant of pAntp (43-58) | HaCaT cells | Biotin | 10784032 | 52 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | NA | Fluorescent Microscopy | Cellular uptake | RQIAIWFQNRRMKWKK |
| 82 | Ala47 substitution mutant of pAntp (43-58) | HaCaT cells | Biotin | 10784032 | 56 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | NA | Fluorescent Microscopy | Cellular uptake | RQIKAWFQNRRMKWKK |
| 83 | Ala48 substitution mutant of pAntp (43-58) | HaCaT cells | Biotin | 10784032 | 68 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | NA | Fluorescent Microscopy | Cellular uptake | RQIKIAFQNRRMKWKK |
| 84 | Ala49 substitution mutant of pAntp (43-58) | HaCaT cells | Biotin | 10784032 | 89.5 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | NA | Fluorescent Microscopy | Cellular uptake | RQIKIWAQNRRMKWKK |
| 85 | Ala50 substitution mutant of pAntp (43-58) | HaCaT cells | Biotin | 10784032 | 90 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | NA | Fluorescent Microscopy | Cellular uptake | RQIKIWFANRRMKWKK |
| 86 | Ala51 substitution mutant of pAntp (43-58) | HaCaT cells | Biotin | 10784032 | 61 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | NA | Fluorescent Microscopy | Cellular uptake | RQIKIWFQARRMKWKK |
| 87 | Ala52 substitution mutant of pAntp (43-58) | HaCaT cells | Biotin | 10784032 | 42 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | NA | Fluorescent Microscopy | Cellular uptake | RQIKIWFQNARMKWKK |
| 88 | Ala53 substitution mutant of pAntp (43-58) | HaCaT cells | Biotin | 10784032 | 31 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | NA | Fluorescent Microscopy | Cellular uptake | RQIKIWFQNRAMKWKK |
| 89 | Ala54 substitution mutant of pAntp (43-58) | HaCaT cells | Biotin | 10784032 | 87.5 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | NA | Fluorescent Microscopy | Cellular uptake | RQIKIWFQNRRAKWKK |
| 90 | Ala55 substitution mutant of pAntp (43-58) | HaCaT cells | Biotin | 10784032 | 26 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | NA | Fluorescent Microscopy | Cellular uptake | RQIKIWFQNRRMAWKK |
| 91 | Ala56 substitution mutant of pAntp (43-58) | HaCaT cells | Biotin | 10784032 | 41 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | NA | Fluorescent Microscopy | Cellular uptake | RQIKIWFQNRRMKAKK |
| 92 | Ala57 substitution mutant of pAntp (43-58) | HaCaT cells | Biotin | 10784032 | 21 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | NA | Fluorescent Microscopy | Cellular uptake | RQIKIWFQNRRMKWAK |
| 93 | Ala58 substitution mutant of pAntp (43-58) | HaCaT cells | Biotin | 10784032 | 23 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | NA | Fluorescent Microscopy | Cellular uptake | RQIKIWFQNRRMKWKA |
| 94 | Crot (27-39) | NIH-3T3 cells | FITC | 21319732 | 3176 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KMDCRWRWKCCKK |
| 95 | Crot (27-39) derevative 1 | NIH-3T3 cells | FITC | 21319732 | 3344 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | MDCRWRWKCCKK |
| 96 | Crot (27-39) derevative 2 | NIH-3T3 cells | FITC | 21319732 | 1909 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | DCRWRWKCCKK |
| 97 | CyLoP-1 | NIH-3T3 cells | FITC | 21319732 | 4050 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | CRWRWKCCKK |
| 98 | Crot (27-39) derevative 3 | NIH-3T3 cells | FITC | 21319732 | 1511 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | RWRWKCCKK |
| 99 | Crot (27-39) derevative 4 | NIH-3T3 cells | FITC | 21319732 | 1516 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KMDCRWRWKCKK |
| 100 | Crot (27-39) derevative 5 | NIH-3T3 cells | FITC | 21319732 | 1202 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KMDCRWRWKKK |
| 101 | Crot (27-39) derevative 6 | NIH-3T3 cells | FITC | 21319732 | 100 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KMDRWRWKKK |
| 102 | Crot (27-39) derevative 7 | NIH-3T3 cells | FITC | 21319732 | 1043 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KDCRWRWKCCKK |
| 103 | Crot (27-39) derevative 8 | NIH-3T3 cells | FITC | 21319732 | 1583 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KCRWRWKCCKK |
| 104 | Crot (27-39) derevative 9 | NIH-3T3 cells | FITC | 21319732 | 1226 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KRWRWKCCKK |
| 105 | Crot (27-39) derevative 10 | NIH-3T3 cells | FITC | 21319732 | 1937 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | MDCRWRWKXCKK |
| 106 | Crot (27-39) derevative 11 | NIH-3T3 cells | FITC | 21319732 | 1741 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | DCRWRWKXCKK |
| 107 | Crot (27-39) derevative 12 | NIH-3T3 cells | FITC | 21319732 | 943 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | DCRWRWKCXKK |
| 108 | Crot (27-39) derevative 13 | NIH-3T3 cells | FITC | 21319732 | 2044 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | CRWRWKXCKK |
| 109 | Crot (27-39) derevative 14 | NIH-3T3 cells | FITC | 21319732 | 1347 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | CRWRWKCXKK |
| 110 | Crot (27-39) derevative 15 | NIH-3T3 cells | FITC | 21319732 | 1211 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | RWRWKXCKK |
| 111 | Crot (27-39) derevative 16 | NIH-3T3 cells | FITC | 21319732 | 1256 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | MDCRWRWKXXKK |
| 112 | Crot (27-39) derevative 17 | NIH-3T3 cells | FITC | 21319732 | 872 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | DCRWRWKXXKK |
| 113 | Crot (27-39) derevative 18 | NIH-3T3 cells | FITC | 21319732 | 1390 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | CRWRWKXXKK |
| 114 | Crot (27-39) derevative 19 | NIH-3T3 cells | FITC | 21319732 | 405 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | RWRWKXXKK |
| 115 | Crot (27-39) derevative 20 | NIH-3T3 cells | FITC | 21319732 | 2172 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | CRWRWKCSKK |
| 116 | Crot (27-39) derevative 21 | NIH-3T3 cells | FITC | 21319732 | 1867 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | SRWRWKCCKK |
| 117 | Crot (27-39) derevative 22 | NIH-3T3 cells | FITC | 21319732 | 572 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | SRWRWKCSKK |
| 118 | Crot (27-39) derevative 23 | NIH-3T3 cells | FITC | 21319732 | 475 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | SRWRWKSCKK |
| 119 | Crot (27-39) derevative 24 | NIH-3T3 cells | FITC | 21319732 | 415 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | CRWRWKSSKK |
| 120 | Crot (27-39) derevative 25 | NIH-3T3 cells | FITC | 21319732 | 193 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | SRWRWKSSKK |
| 121 | Crot (27-39) derevative 26 | NIH-3T3 cells | FITC | 21319732 | 2656 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | CRFRWKCCKK |
| 122 | Crot (27-39) derevative 27 | NIH-3T3 cells | FITC | 21319732 | 2476 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | CRWRFKCCKK |
| 123 | Crot (27-39) derevative 28 | NIH-3T3 cells | FITC | 21319732 | 2569 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | CRFRFKCCKK |
| 124 | Crot (27-39) derevative 29 | NIH-3T3 cells | FITC | 21319732 | 2109 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | crwrwkcckk |
| 125 | Crot (27-39) derevative 30 | NIH-3T3 cells | FITC | 21319732 | 1713 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KCCKWRWRCK |
| 126 | Crot (27-39) derevative 31 | NIH-3T3 cells | FITC | 21319732 | 1449 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | kcckwrwrck |
| 127 | Crot (27-39) derevative 32 | NIH-3T3 cells | FITC | 21319732 | 1529 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | CrWRWKCCKK |
| 128 | Crot (27-39) derevative 33 | NIH-3T3 cells | FITC | 21319732 | 1229 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | CRwRWKCCKK |
| 129 | Crot (27-39) derevative 34 | NIH-3T3 cells | FITC | 21319732 | 1304 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | CRWrWKCCKK |
| 130 | Crot (27-39) derevative 35 | NIH-3T3 cells | FITC | 21319732 | 1412 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | CRWRwKCCKK |
| 131 | Crot (27-39) derevative 36 | NIH-3T3 cells | FITC | 21319732 | 1488 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | CrwrwKCCKK |
| 132 | Crot (27-39) derevative 37 | NIH-3T3 cells | FITC | 21319732 | 2376 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | CRWRWKCGCKK |
| 133 | Crot (27-39) derevative 38 | NIH-3T3 cells | FITC | 21319732 | 3056 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KCGCRWRWKCGCKK |
| 134 | Crot (27-39) derevative 39 | NIH-3T3 cells | FITC | 21319732 | 1922 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | CRWRWKCG |
| 135 | Crot (27-39) derevative 40 | NIH-3T3 cells | FITC | 21319732 | 1943 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KMDXRWRWKCCKK |
| 136 | Crot (27-39) derevative 41 | NIH-3T3 cells | FITC | 21319732 | 734 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KMDXRWRWKXCKK |
| 137 | Crot (27-39) derevative 42 | NIH-3T3 cells | FITC | 21319732 | 162 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KMDXRWRWKXXKK |
| 138 | Crot (27-39) derevative 43 | NIH-3T3 cells | FITC | 21319732 | 2816 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KMDXRWRWKCXKK |
| 139 | Crot (27-39) derevative 44 | NIH-3T3 cells | FITC | 21319732 | 1542 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | MDCRWRWKCXKK |
| 140 | Crot (27-39) derevative 45 | NIH-3T3 cells | FITC | 21319732 | 2335 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KMDCRWRWKCSKK |
| 141 | Crot (27-39) derevative 46 | NIH-3T3 cells | FITC | 21319732 | 1188 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KMDCRWRWKSCKK |
| 142 | Crot (27-39) derevative 47 | NIH-3T3 cells | FITC | 21319732 | 987 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KMDSRWRWKCCKK |
| 143 | Crot (27-39) derevative 48 | NIH-3T3 cells | FITC | 21319732 | 615 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KMDCRWRWKSSKK |
| 144 | Crot (27-39) derevative 49 | NIH-3T3 cells | FITC | 21319732 | 496 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KMDSRWRWKSSKK |
| 145 | Crot (27-39) derevative 50 | NIH-3T3 cells | FITC | 21319732 | 856 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KMDSRWRWKSCKK |
| 146 | Crot (27-39) derevative 51 | NIH-3T3 cells | FITC | 21319732 | 1244 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KMDSRWRWKCSKK |
| 147 | Crot (27-39) derevative 52 | NIH-3T3 cells | FITC | 21319732 | 1272 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KMDCRWRPKCCKK |
| 148 | Crot (27-39) derevative 53 | NIH-3T3 cells | FITC | 21319732 | 347 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KMDCRPRPKCCKK |
| 149 | Crot (27-39) derevative 54 | NIH-3T3 cells | FITC | 21319732 | 251 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KMDXRPRPKCCKK |
| 150 | Crot (27-39) derevative 55 | NIH-3T3 cells | FITC | 21319732 | 222 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KMDXRPRPKXCKK |
| 151 | Crot (27-39) derevative 56 | NIH-3T3 cells | FITC | 21319732 | 257 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KMDXRPRPKCXKK |
| 152 | Crot (27-39) derevative 57 | NIH-3T3 cells | FITC | 21319732 | 294 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KMDCRPRPKXCKK |
| 153 | Crot (27-39) derevative 58 | NIH-3T3 cells | FITC | 21319732 | 353 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KMDCRPRPKCXKK |
| 154 | Penetratin (pAntp) | NIH-3T3 cells | FITC | 21319732 | 27.5 | % Intracellular fluorescence of CyLoP-1 | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | RQIKIWFQNRRMKWKK |
| 155 | Tat (49-57) | NIH-3T3 cells | FITC | 21319732 | 55.0 | % Intracellular fluorescence of CyLoP-1 | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | rkkrrqrrr |
| 156 | Tat (57-49) | NIH-3T3 cells | FITC | 21319732 | 46.25 | % Intracellular fluorescence of CyLoP-1 | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | rrrqrrkkr |
| 157 | R8 | NIH-3T3 cells | FITC | 21319732 | 47.5 | % Intracellular fluorescence of CyLoP-1 | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | rrrrrrrr |
| 158 | Bip1 | DAMI cells | Fluorescein | 21359136 | 97± 4.3 | Cellular uptake (%) | 200 uM | 3h | 37ºC | Flow cytometry | Cell-Penetration | VPMLK |
| 159 | Bip2 | DAMI cells | Fluorescein | 21359136 | 61±1.7 | Cellular uptake (%) | 200 uM | 3h | 37ºC | Flow cytometry | Cell-Penetration | VPTLK |
| 160 | Bip2 | HeLa cells | Fluorescein | 21359136 | 1280 | Mean Fluorescence intensity | 1600 uM | 3h | NA | Flow cytometry | Cell-Penetration | VPTLK |
| 161 | Bip3 | DAMI cells | Fluorescein | 21359136 | 79 ± 1.5 | Cellular uptake (%) | 200 uM | 3h | 37ºC | Flow cytometry | Cell-Penetration | VPALR |
| 162 | Bip4 | DAMI cells | Fluorescein | 21359136 | 90 ± 3 | Cellular uptake (%) | 200 uM | 3h | 37ºC | Flow cytometry | Cell-Penetration | VSALK |
| 163 | Bip5 | DAMI cells | Fluorescein | 21359136 | 65 ± 3.7 | Cellular uptake (%) | 200 uM | 3h | 37ºC | Flow cytometry | Cell-Penetration | PMLKE |
| 164 | Bip6 | DAMI cells | Fluorescein | 21359136 | 71 ± 2.2 | Cellular uptake (%) | 200 uM | 3h | 37ºC | Flow cytometry | Cell-Penetration | VPALK |
| 165 | Bip9 | DAMI cells | Fluorescein | 21359136 | 100 ± 2.3 | Cellular uptake (%) | 200 uM | 3h | 37ºC | Flow cytometry | Cell-Penetration | KLPVM |
| 166 | Bip10 | DAMI cells | Fluorescein | 21359136 | 47 ± 1.4 | Cellular uptake (%) | 200 uM | 3h | 37ºC | Flow cytometry | Cell-Penetration | IPMIK |
| 167 | Bip16 | DAMI cells | Fluorescein | 21359136 | 70 ± 4 | Cellular uptake (%) | 200 uM | 3h | 37ºC | Flow cytometry | Cell-Penetration | VPTLQ |
| 168 | Bip19 | DAMI cells | Fluorescein | 21359136 | 80±1.9 | Cellular uptake (%) | 200 uM | 3h | 37ºC | Flow cytometry | Cell-Penetration | VPTLE |
| 169 | Inv1 | HeLa cells | (FITC)-labeled latex microspheres | 16620748 | 47.5 | Fluorescence intensity | 0.05 umol | NA | 37ºC | Flow cytometry | Uptake | VNADIKATTVFGGKYVSLTTP |
| 170 | Inv2 | HeLa cells | (FITC)-labeled latex microspheres | 16620748 | 104.5 | Fluorescence intensity | 0.05 umol | NA | 37ºC | Flow cytometry | Uptake | GKYVSLTTPKNPTKRRITPKDV |
| 171 | Inv3 | HeLa cells | (FITC)-labeled latex microspheres | 16620748 | 607.5 / 2400 | Fluorescence intensity | 0.05 umol | NA | 37ºC | Flow cytometry | Uptake | TKRRITPKDVIDVRSVTTEINT |
| 172 | Inv4 | HeLa cells | (FITC)-labeled latex microspheres | 16620748 | 104.5 | Fluorescence intensity | 0.05 umol | NA | 37ºC | Flow cytometry | Uptake | RSVTTEINTLFQTLTSIAEKVDP |
| 173 | Inv5 | HeLa cells | (FITC)-labeled latex microspheres | 16620748 | 626.5 | Fluorescence intensity | 0.05 umol | NA | 37ºC | Flow cytometry | Uptake | AEKVDPVKLNLTLSAAAEALTGLGDK |
| 174 | Inv6 | HeLa cells | (FITC)-labeled latex microspheres | 16620748 | 155 | Fluorescence intensity | 0.05 umol | NA | 37ºC | Flow cytometry | Uptake | GLGDKFGESIVNANTVLDDLNSRMPQSRHDIQQL |
| 175 | Inv7 | HeLa cells | (FITC)-labeled latex microspheres | 16620748 | 57 / 75 | Fluorescence intensity | 0.05 umol | NA | 37ºC | Flow cytometry | Uptake | GDVYADAAPDLFDFLDSSVTTARTINA |
| 176 | Inv8 | HeLa cells | (FITC)-labeled latex microspheres | 16620748 | 47.5 | Fluorescence intensity | 0.05 umol | NA | 37ºC | Flow cytometry | Uptake | ARTINAQQAELDSALLAAAGFGNTTADVFDRG |
| 177 | Inv9 | HeLa cells | (FITC)-labeled latex microspheres | 16620748 | 76 | Fluorescence intensity | 0.05 umol | NA | 37ºC | Flow cytometry | Uptake | ADVFDRGGPYLQRGVADLVPTATLLDTYSP |
| 178 | Inv10 | HeLa cells | (FITC)-labeled latex microspheres | 16620748 | 33.25 | Fluorescence intensity | 0.05 umol | NA | 37ºC | Flow cytometry | Uptake | LDTYSPELFCTIRNFYDADRPDRGAAA |
| 179 | Inv11 | HeLa cells | (FITC)-labeled latex microspheres | 16620748 | 123.5 | Fluorescence intensity | 0.05 umol | NA | 37ºC | Flow cytometry | Uptake | TKRRITPKDVIDVRSVTTEINT |
| 180 | Inv3.3 | HeLa cells | (FITC)-labeled latex microspheres | 16620748 | 50 | Fluorescence intensity | 0.05 umol | NA | 37ºC | Flow cytometry | Uptake | TKRRITPDDVIDVRSVTTEINT |
| 181 | Inv3.4 | HeLa cells | (FITC)-labeled latex microspheres | 16620748 | 1200 | Fluorescence intensity | 0.05 umol | NA | 37ºC | Flow cytometry | Uptake | TKRRITPKKVIDVRSVTTEINT |
| 182 | Inv3.5 | HeLa cells | (FITC)-labeled latex microspheres | 16620748 | 2650 | Fluorescence intensity | 0.05 umol | NA | 37ºC | Flow cytometry | Uptake | TKRRITPKDVIDVRSVTTKINT |
| 183 | Inv3.6 | HeLa cells | (FITC)-labeled latex microspheres | 16620748 | 50 | Fluorescence intensity | 0.05 umol | NA | 37ºC | Flow cytometry | Uptake | TKRRITPKDVIDV |
| 184 | Inv3.7 | HeLa cells | (FITC)-labeled latex microspheres | 16620748 | 75 | Fluorescence intensity | 0.05 umol | NA | 37ºC | Flow cytometry | Uptake | TKRRITPKDVIDVESVTTEINT |
| 185 | Inv3.8 | HeLa cells | (FITC)-labeled latex microspheres | 16620748 | 150 | Fluorescence intensity | 0.05 umol | NA | 37ºC | Flow cytometry | Uptake | TARRITPKDVIDVRSVTTEINT |
| 186 | Inv3.9 | HeLa cells | (FITC)-labeled latex microspheres | 16620748 | 100 | Fluorescence intensity | 0.05 umol | NA | 37ºC | Flow cytometry | Uptake | TKAARITPKDVIDVRSVTTEINT |
| 187 | Inv3.10 | HeLa cells | (FITC)-labeled latex microspheres | 16620748 | 1925 | Fluorescence intensity | 0.05 umol | NA | 37ºC | Flow cytometry | Uptake | HHHHHHTKRRITPKDVIDVRSVTTEINT |
| 188 | No.14 | CHO cells | Fluorescein | 19956900 | 790 | Fluorescence intensity | 50 uM | 1h | 37ºC | Flow cytometry | Translocation | KLWMRWYSPTTRRYG |
| 189 | No.14-1 | CHO cells | Fluorescein | 19956900 | 650 | Fluorescence intensity | 50 uM | 1h | 37ºC | Flow cytometry | Translocation | RLWMRWYSPTTRRYG |
| 190 | No.14-2 | CHO cells | Fluorescein | 19956900 | 790 | Fluorescence intensity | 50 uM | 1h | 37ºC | Flow cytometry | Translocation | KLWMRWYSATTRRYG |
| 191 | No.14-7 | CHO cells | Fluorescein | 19956900 | 850 | Fluorescence intensity | 50 uM | 1h | 37ºC | Flow cytometry | Translocation | KLWMRWYSPWTRRYG |
| 192 | No.14-8 | CHO cells | Fluorescein | 19956900 | 650 | Fluorescence intensity | 50 uM | 1h | 37ºC | Flow cytometry | Translocation | RLWMRWYSPWTRRYG |
| 193 | No.14-9 | CHO cells | Fluorescein | 19956900 | 530 | Fluorescence intensity | 50 uM | 1h | 37ºC | Flow cytometry | Translocation | RLWMRWYSPWTRRWG |
| 194 | No.14-11 | CHO cells | Fluorescein | 19956900 | 220 | Fluorescence intensity | 50 uM | 1h | 37ºC | Flow cytometry | Translocation | ALWMRWYSPTTRRYG |
| 195 | No.14-12 | CHO cells | Fluorescein | 19956900 | 800 | Fluorescence intensity | 50 uM | 1h | 37ºC | Flow cytometry | Translocation | RAWMRWYSPTTRRYG |
| 196 | No.14-13 | CHO cells | Fluorescein | 19956900 | 750 | Fluorescence intensity | 50 uM | 1h | 37ºC | Flow cytometry | Translocation | RLAMRWYSPTTRRYG |
| 197 | No.14-14 | CHO cells | Fluorescein | 19956900 | 750 | Fluorescence intensity | 50 uM | 1h | 37ºC | Flow cytometry | Translocation | RLWARWYSPTTRRYG |
| 198 | No.14-15 | CHO cells | Fluorescein | 19956900 | 90 | Fluorescence intensity | 50 uM | 1h | 37ºC | Flow cytometry | Translocation | RLWMAWYSPTTRRYG |
| 199 | No.14-16 | CHO cells | Fluorescein | 19956900 | 50 | Fluorescence intensity | 50 uM | 1h | 37ºC | Flow cytometry | Translocation | RLWMRAYSPTTRRYG |
| 200 | No.14-17 | CHO cells | Fluorescein | 19956900 | 790 | Fluorescence intensity | 50 uM | 1h | 37ºC | Flow cytometry | Translocation | RLWMRWASPTTRRYG |
| 201 | No.14-18 | CHO cells | Fluorescein | 19956900 | 800 | Fluorescence intensity | 50 uM | 1h | 37ºC | Flow cytometry | Translocation | RLWMRWYAPTTRRYG |
| 202 | No.14-20 | CHO cells | Fluorescein | 19956900 | 880 | Fluorescence intensity | 50 uM | 1h | 37ºC | Flow cytometry | Translocation | RLWMRWYSPATRRYG |
| 203 | No.14-21 | CHO cells | Fluorescein | 19956900 | 810 | Fluorescence intensity | 50 uM | 1h | 37ºC | Flow cytometry | Translocation | RLWMRWYSPTARRYG |
| 204 | No.14-22 | CHO cells | Fluorescein | 19956900 | 370 | Fluorescence intensity | 50 uM | 1h | 37ºC | Flow cytometry | Translocation | RLWMRWYSPTTARYG |
| 205 | No.14-3R | CHO cells | Fluorescein | 19956900 | 150 | Fluorescence intensity | 50 uM | 1h | 37ºC | Flow cytometry | Translocation | RLWMRWYSPTTRAYG |
| 206 | No.14-23 | CHO cells | Fluorescein | 19956900 | 840 | Fluorescence intensity | 50 uM | 1h | 37ºC | Flow cytometry | Translocation | RLWMRWYSPTTRRAG |
| 207 | No.14-35 | CHO cells | Fluorescein | 19956900 | 860 | Fluorescence intensity | 50 uM | 1h | 37ºC | Flow cytometry | Translocation | RLWMRWYSPTTRRYA |
| 208 | No.14-24 | CHO cells | Fluorescein | 19956900 | 440 | Fluorescence intensity | 50 uM | 1h | 37ºC | Flow cytometry | Translocation | RLLMRLYSPTTRRYG |
| 209 | No.14-25 | CHO cells | Fluorescein | 19956900 | 830 | Fluorescence intensity | 50 uM | 1h | 37ºC | Flow cytometry | Translocation | RLFMRFYSPTTRRYG |
| 210 | No.14-26 | CHO cells | Fluorescein | 19956900 | 860 | Fluorescence intensity | 50 uM | 1h | 37ºC | Flow cytometry | Translocation | RLIMRIYSPTTRRYG |
| 211 | No.14-29 | CHO cells | Fluorescein | 19956900 | 590 | Fluorescence intensity | 50 uM | 1h | 37ºC | Flow cytometry | Translocation | RLVMRVYSPTTRRYG |
| 212 | No.14-30 | CHO cells | Fluorescein | 19956900 | 890 | Fluorescence intensity | 50 uM | 1h | 37ºC | Flow cytometry | Translocation | RLYMRYYSPTTRRYG |
| 213 | pVEC | Human bowes melanoma cells | Fluorescein | 16808894 | 1350 | pmol/mg protein Cellular uptake | 10 uM | 1h | 37ºC | Fluorescence spectroscopy | Uptake | LLIILRRRIRKQAHAHSK |
| 214 | pVEC mutant 1 | Human bowes melanoma cells | Fluorescein | 16808894 | 300 | pmol/mg protein Cellular uptake | 10 uM | 1h | 37ºC | Fluorescence spectroscopy | Uptake | ALIILRRRIRKQAHAHSK |
| 215 | pVEC mutant 2 | Human bowes melanoma cells | Fluorescein | 16808894 | 500 | pmol/mg protein Cellular uptake | 10 uM | 1h | 37ºC | Fluorescence spectroscopy | Uptake | LAIILRRRIRKQAHAHSK |
| 216 | pVEC mutant 3 | Human bowes melanoma cells | Fluorescein | 16808894 | 375 | pmol/mg protein Cellular uptake | 10 uM | 1h | 37ºC | Fluorescence spectroscopy | Uptake | LLAILRRRIRKQAHAHSK |
| 217 | pVEC mutant 4 | Human bowes melanoma cells | Fluorescein | 16808894 | 700 | pmol/mg protein Cellular uptake | 10 uM | 1h | 37ºC | Fluorescence spectroscopy | Uptake | LLIALRRRIRKQAHAHSK |
| 218 | pVEC mutant 5 | Human bowes melanoma cells | Fluorescein | 16808894 | 450 | pmol/mg protein Cellular uptake | 10 uM | 1h | 37ºC | Fluorescence spectroscopy | Uptake | LLIIARRRIRKQAHAHSK |
| 219 | pVEC mutant 6 | Human bowes melanoma cells | Fluorescein | 16808894 | 2500 | pmol/mg protein Cellular uptake | 10 uM | 1h | 37ºC | Fluorescence spectroscopy | Uptake | LLIILARRIRKQAHAHSK |
| 220 | pVEC mutant 7 | Human bowes melanoma cells | Fluorescein | 16808894 | 1125 | pmol/mg protein Cellular uptake | 10 uM | 1h | 37ºC | Fluorescence spectroscopy | Uptake | LLIILRARIRKQAHAHSK |
| 221 | pVEC mutant 8 | Human bowes melanoma cells | Fluorescein | 16808894 | 2175 | pmol/mg protein Cellular uptake | 10 uM | 1h | 37ºC | Fluorescence spectroscopy | Uptake | LLIILRRAIRKQAHAHSK |
| 222 | pVEC mutant 9 | Human bowes melanoma cells | Fluorescein | 16808894 | 800 | pmol/mg protein Cellular uptake | 10 uM | 1h | 37ºC | Fluorescence spectroscopy | Uptake | LLIILRRRARKQAHAHSK |
| 223 | pVEC mutant 10 | Human bowes melanoma cells | Fluorescein | 16808894 | 1500 | pmol/mg protein Cellular uptake | 10 uM | 1h | 37ºC | Fluorescence spectroscopy | Uptake | LLIILRRRIARKQAHAHSK |
| 224 | pVEC mutant 11 | Human bowes melanoma cells | Fluorescein | 16808894 | 1800 | pmol/mg protein Cellular uptake | 10 uM | 1h | 37ºC | Fluorescence spectroscopy | Uptake | LLIILRRRIRAQAHAHSK |
| 225 | pVEC mutant 12 | Human bowes melanoma cells | Fluorescein | 16808894 | 1500 | pmol/mg protein Cellular uptake | 10 uM | 1h | 37ºC | Fluorescence spectroscopy | Uptake | LLIILRRRIRKAAHAHSK |
| 226 | pVEC mutant 13 | Human bowes melanoma cells | Fluorescein | 16808894 | 1850 | pmol/mg protein Cellular uptake | 10 uM | 1h | 37ºC | Fluorescence spectroscopy | Uptake | LLIILRRRIRKQaHAHSK |
| 227 | pVEC mutant 14 | Human bowes melanoma cells | Fluorescein | 16808894 | 550 | pmol/mg protein Cellular uptake | 10 uM | 1h | 37ºC | Fluorescence spectroscopy | Uptake | LLIILRRRIRKQAAAHSK |
| 228 | pVEC mutant 15 | Human bowes melanoma cells | Fluorescein | 16808894 | 1125 | pmol/mg protein Cellular uptake | 10 uM | 1h | 37ºC | Fluorescence spectroscopy | Uptake | LLIILRRRIRKQAHaHSK |
| 229 | pVEC mutant 16 | Human bowes melanoma cells | Fluorescein | 16808894 | 1550 | pmol/mg protein Cellular uptake | 10 uM | 1h | 37ºC | Fluorescence spectroscopy | Uptake | LLIILRRRIRKQAHAASK |
| 230 | pVEC mutant 17 | Human bowes melanoma cells | Fluorescein | 16808894 | 2150 | pmol/mg protein Cellular uptake | 10 uM | 1h | 37ºC | Fluorescence spectroscopy | Uptake | LLIILRRRIRKQAHAHAK |
| 231 | pVEC mutant 18 | Human bowes melanoma cells | Fluorescein | 16808894 | 2100 | pmol/mg protein Cellular uptake | 10 uM | 1h | 37ºC | Fluorescence spectroscopy | Uptake | LLIILRRRIRKQAHAHSA |
| 232 | Retro-pVEC | Human bowes melanoma cells | Fluorescein | 16808894 | 400 | pmol/mg protein Cellular uptake | 10 uM | 1h | 37ºC | Fluorescence spectroscopy | Uptake | KSHAHAQKRIRRRLIILL |
| 233 | D form of pVEC | Human bowes melanoma cells | Fluorescein | 16808894 | 1150 | pmol/mg protein Cellular uptake | 10 uM | 1h | 37ºC | Fluorescence spectroscopy | Uptake | lliilrrrirkqahahsk |
| 234 | Bac1-7 | RAW264.7 cells | Fluorescein | 12450378 | 90 | Intracellular Fluorescence | 5 uM | 30 min | 37ºC | Fluorescence spectroscopy | Uptake | RRIRPRP |
| 235 | Bac-1-15 | RAW264.7 cells | Fluorescein | 12450378 | 200 | Intracellular Fluorescence | 5 uM | 30 min | 37ºC | Fluorescence spectroscopy | Uptake | RRIRPRPPRLPRPRP |
| 236 | Bac1-24 | RAW264.7 cells | Fluorescein | 12450378 | 35 | Intracellular Fluorescence | 5 uM | 30 min | 37ºC | Fluorescence spectroscopy | Uptake | RRIRPRPPRLPRPRPRPLPFPRPG |
| 237 | Bac1-17 | RAW264.7 cells | Fluorescein | 12450378 | 130 | Intracellular Fluorescence | 5 uM | 30 min | 37ºC | Fluorescence spectroscopy | Uptake | RRIRPRPPRLPRPRPRP |
| 238 | Bac5-24 | RAW264.7 cells | Fluorescein | 12450378 | 60 | Intracellular Fluorescence | 5 uM | 30 min | 37ºC | Fluorescence spectroscopy | Uptake | PRPPRLPRPRPRPLPFPRPG |
| 239 | Bac7-24 | RAW264.7 cells | Fluorescein | 12450378 | 90 | Intracellular Fluorescence | 5 uM | 30 min | 37ºC | Fluorescence spectroscopy | Uptake | PPRLPRPRPRPLPFPRPG |
| 240 | Bac9-24 | RAW264.7 cells | Fluorescein | 12450378 | 100 | Intracellular Fluorescence | 5 uM | 30 min | 37ºC | Fluorescence spectroscopy | Uptake | RLPRPRPRPLPFPRPG |
| 241 | Bac13-24 | RAW264.7 cells | Fluorescein | 12450378 | 80 | Intracellular Fluorescence | 5 uM | 30 min | 37ºC | Fluorescence spectroscopy | Uptake | PRPRPLPFPRPG |
| 242 | Bac15-24 | RAW264.7 cells | Fluorescein | 12450378 | 555 | Intracellular Fluorescence | 5 uM | 30 min | 37ºC | Fluorescence spectroscopy | Uptake | PRPLPFPRPG |
| 243 | ARF(1-22) | MCF7 cells | Fluorescein | 17984975 | 1300 | pmol/mg protein Cellular uptake | 5 umol/L | 1h | NA | Fluorescence spectroscopy | Uptake | MVRRFLVTLRIRRACGPPRVRV |
| 244 | ARF(1-22) scr | MCF7 cells | Fluorescein | 17984975 | 1000 | pmol/mg protein Cellular uptake | 5 umol/L | 1h | NA | Fluorescence spectroscopy | Uptake | FVTRGCPRRLVARLIRVMVPRR |
| 245 | ARF(2-14) | MCF7 cells | Fluorescein | 17984975 | 750 | pmol/mg protein Cellular uptake | 5 umol/L | 1h | NA | Fluorescence spectroscopy | Uptake | VRRFLVTLRIRRA |
| 246 | ARF(2-14) scr | MCF7 cells | Fluorescein | 17984975 | 150 | pmol/mg protein Cellular uptake | 5 umol/L | 1h | NA | Fluorescence spectroscopy | Uptake | RVRILARFLRTRV |
| 247 | ARF(19-31) | MCF7 cells | Fluorescein | 17984975 | 1050 | pmol/mg protein Cellular uptake | 5 umol/L | 1h | NA | Fluorescence spectroscopy | Uptake | RVRVFVVHIPRLT |
| 248 | ARF(19-31) scr | MCF7 cells | Fluorescein | 17984975 | 250 | pmol/mg protein Cellular uptake | 5 umol/L | 1h | NA | Fluorescence spectroscopy | Uptake | VIRVHFRLPVRTV |
| 249 | Cyt C 71-101 | U373 MG cells | NA | 20659686 | 100 | Fluorescence intensity | 5 uM | 1h | 37ºC | Fluorescence spectroscopy | Translocation | GTKMIFVGIKKKEERADLIAYLKKA |
| 250 | Cyt C 86-101 | U373 MG cells | NA | 20659686 | 4 | Fluorescence intensity | 5 uM | 1h | 37ºC | Fluorescence spectroscopy | Translocation | KKKEERADLIAYLKKA |
| 251 | Cyt 79-92 | U373 MG cells | NA | 20659686 | 8 | Fluorescence (fold/basal) | 5 uM | 1h | 37ºC | Fluorescence spectroscopy | Translocation | KMIFVGIKKKEERA |
| 252 | Cyt 79-88 | U373 MG cells | NA | 20659686 | 4.5 | Fluorescence intensity | 5 uM | 1h | 37ºC | Fluorescence spectroscopy | Translocation | KMIFVGIKKK |
| 253 | Cyt 4-13 | U373 MG cells | NA | 20659686 | 7 | Fluorescence intensity | 5 uM | 1h | 37ºC | Fluorescence spectroscopy | Translocation | EKGKKIFIMK |
| 254 | Cyt 5-13 | U373 MG cells | NA | 20659686 | 41 | Fluorescence intensity | 5 uM | 1h | 37ºC | Fluorescence spectroscopy | Translocation | KGKKIFIMK |
| 255 | hLF peptide | HeLa cells | Fluorescein | 19858187 | 40 | Fluorescence intensity | 10 uM | 30 min | NA | Flow cytometry | Uptake | KCFQWQRNMRKVRGPPVSCIKR |
| 256 | M1 | HeLa cells | Fluorescein | 19858187 | 33.75 | Fluorescence intensity | 10 uM | 30 min | NA | Flow cytometry | Uptake | KCFQWQRNMRKVRGPPVSC |
| 257 | M2 | HeLa cells | Fluorescein | 19858187 | 7.5 | Fluorescence intensity | 10 uM | 30 min | NA | Flow cytometry | Uptake | KCFQWQRNMRKVRGPPVSSIKR |
| 258 | M3 | HeLa cells | Fluorescein | 19858187 | 6.25 | Fluorescence intensity | 10 uM | 30 min | NA | Flow cytometry | Uptake | KCFQWQRNMRKVR |
| 259 | M4 | HeLa cells | Fluorescein | 19858187 | 4.375 | Fluorescence intensity | 10 uM | 30 min | NA | Flow cytometry | Uptake | FQWQRNMRKVRGPPVS |
| 260 | M5 | HeLa cells | Fluorescein | 19858187 | 7.5 | Fluorescence intensity | 10 uM | 30 min | NA | Flow cytometry | Uptake | QWQRNMRKVRGPPVSCIKR |
| 261 | M6 | HeLa cells | Fluorescein | 19858187 | 3.75 | Fluorescence intensity | 10 uM | 30 min | NA | Flow cytometry | Uptake | QWQRNMRKVR |
| 262 | MPG Mutant | HS-68 | Fluorescein | 12771197 | 70 | Fluorescence intensity (%) | Charge ratio = 5:1 (MPG/DNA) | 30 min | 37ºC | Fluorescent Microscopy | Transfection | GALFLGFLGAAGSTMGAWSQPKSKRKV |
| 263 | MPG Mutant | Cos-7 cells | Fluorescein | 12771197 | 5 | Fluorescence intensity (%) | Charge ratio = 10:1 | 30 min | 37ºC | Fluorescent Microscopy | Transfection | GALFLGFLGAAGSTMGAWSQPKSKRKV |
| 264 | MPG Mutant | HeLa cells | Fluorescein | 12771197 | 10 | Fluorescence intensity (%) | Charge ratio = 10:1 | 30 min | 37ºC | Fluorescent Microscopy | Transfection | GALFLGFLGAAGSTMGAWSQPKSKRKV |
| 265 | Sweet Arrow Protein (SAP) (E) | HeLa cells | Fluorescein | 21365733 | 11.15 | Fluorescence intensity | 50 uM | 3h | 37ºC | Flow cytometry | Cellular internalization | VELPPPVELPPPVELPPP |
| 266 | Sweet Arrow Protein (SAP) (E) | A549 cells | Fluorescein | 21365733 | 5 | Fluorescence intensity | 50 uM | 3h | 37ºC | Flow cytometry | Cellular internalization | VELPPPVELPPPVELPPP |
| 267 | Glu-Oct-6 | DU-145 | FITC | 21029412 | 600 | Geo Mean Fluorescence intensity | 300 uM | 4h | 37ºC | Flow cytometry | Uptake | EEEAAGRKRKKRT |
| 268 | Glu | DU-145 | FITC | 21029412 | 140 | Geo Mean Fluorescence intensity | 300 uM | 4h | 37ºC | Flow cytometry | Uptake | EEE |
| 269 | Glu-Ala | DU-145 | FITC | 21029412 | 120 | Geo Mean Fluorescence intensity | 300 uM | 4h | 37ºC | Flow cytometry | Uptake | EEEAA |
| 270 | Glu-Lys | DU-145 | FITC | 21029412 | 280 | Geo Mean Fluorescence intensity | 300 uM | 4h | 37ºC | Flow cytometry | Uptake | EEEAAKKK |
| 271 | 6-Oct | DU-145 | FITC | 21029412 | 580 | Geo Mean Fluorescence intensity | 300 uM | 4h | 37ºC | Flow cytometry | Uptake | GRKRKKRT |
| 272 | Phe-Oct-6 | DU-145 | FITC | 21029412 | 100 | Geo Mean Fluorescence intensity | 300 uM | 1h | 37ºC | Flow cytometry | Uptake | FFFAAGRKRKKRT |
| 273 | Asn-Oct-6 | DU-145 | FITC | 21029412 | 55 | Geo Mean Fluorescence intensity | 300 uM | 1h | 37ºC | Flow cytometry | Uptake | NNNAAGRKRKKRT |
| 274 | Tyr-Oct-6 | DU-145 | FITC | 21029412 | 115 | Geo Mean Fluorescence intensity | 300 uM | 1h | 37ºC | Flow cytometry | Uptake | YYYAAGRKRKKRT |
| 275 | M918 | HeLa cells | Fluorescein | 17622242 | 3400 | pmol/mg protein Cellular uptake | 5 umol/l | 1h | NA | Fluorescence spectroscopy | Internalization | MVTVLFRRLRIRRACGPPRVRV |
| 276 | M918 | MCF7 cells | Fluorescein | 17622242 | 1700 | pmol/mg protein Cellular uptake | 5 umol/l | 1h | NA | Fluorescence spectroscopy | Internalization | MVTVLFRRLRIRRACGPPRVRV |
| 277 | M918 | Hifko cells | Fluorescein | 17622242 | 2700 | pmol/mg protein Cellular uptake | 5 umol/l | 1h | NA | Fluorescence spectroscopy | Internalization | MVTVLFRRLRIRRACGPPRVRV |
| 278 | TP10 | HeLa cells | Fluorescein | 17622242 | 1000 | pmol/mg protein Cellular uptake | 5 umol/l | 1h | NA | Fluorescence spectroscopy | Internalization | AGYLLGKINLKALAALAKKIL |
| 279 | NF-kB | MCF7 cells | Fluorescein | 12204694 | 4 | Mnlog FITC | 50 uM | 4h | NA | Flow cytometry | Cellular uptake | VQRKRQKLMP |
| 280 | TFIIE BETA | MCF7 cells | Fluorescein | 12204694 | 5 | Mnlog FITC | 50 uM | 4h | NA | Flow cytometry | Cellular uptake | SKKKKTKV |
| 281 | 6-Oct | MCF7 cells | Fluorescein | 12204694 | 14 | Mnlog FITC | 50 uM | 4h | NA | Flow cytometry | Cellular uptake | GRKRKKRT |
| 282 | TCF1-ALPHA | MCF7 cells | Fluorescein | 12204694 | 7 | Mnlog FITC | 50 uM | 4h | NA | Flow cytometry | Cellular uptake | GKKKKRKREKL |
| 283 | SV40 | MCF7 cells | Fluorescein | 12204694 | 3 | Mnlog FITC | 50 uM | 4h | NA | Flow cytometry | Cellular uptake | PKKKRKV |
| 284 | HATF3 | MCF7 cells | Fluorescein | 12204694 | 4 | Mnlog FITC | 50 uM | 4h | NA | Flow cytometry | Cellular uptake | ERKKRRRE |
| 285 | C.e SDC3 | MCF7 cells | Fluorescein | 12204694 | 2.8 | Mnlog FITC | 50 uM | 4h | NA | Flow cytometry | Cellular uptake | FKKFRKF |
| 286 | D-SynB1 | K562 cells | NBD | 12783857 | 7.5 | Fluorescence intensity | 6 uM | 65 min | 37ºC | Flow cytometry | Internalization | rggrlsysrrrfststgr |
| 287 | D-SynB3 | K562 cells | NBD | 12783857 | 17.5 | Fluorescence intensity | 6 uM | 65 min | 37ºC | Flow cytometry | Internalization | rrlsysrrrf |
| 288 | MG2d | HeLa cells | Texas Red | 12417587 | 16 | nmol/mg protein | 15 uM | 30 min | 37ºC | Fluorescence spectroscopy | Uptake | GIGKFLHSAKKWGKAFVGQIMNC |
| 289 | BF2d | HeLa cells | Texas Red | 12417587 | 1.5 | nmol/mg protein | 15 uM | 30 min | 37ºC | Fluorescence spectroscopy | Uptake | TRSSRAGLQWPVGRVHRLLRKGGC |
| 290 | PolyP 1 | HeLa cells | Fluorescein | 15054781 | 0 | Fluorescence intensity | 50 uM | 3h | 37ºC | Fluorescent Microscopy | Cellular uptake | VRLPPP |
| 291 | PolyP 2 | HeLa cells | Fluorescein | 15054781 | 100 | Fluorescence intensity | 50 uM | 3h | 37ºC | Fluorescent Microscopy | Cellular uptake | VRLPPPVRLPPP |
| 292 | PolyP 3 (SAP) | HeLa cells | Fluorescein | 15054781 | 575 | Fluorescence intensity | 50 uM | 3h | 37ºC | Fluorescent Microscopy | Cellular uptake | VRLPPPVRLPPPVRLPPP |
| 293 | PolyP 4 | HeLa cells | Fluorescein | 15054781 | 0 | Fluorescence intensity | 50 uM | 3h | 37ºC | Fluorescent Microscopy | Cellular uptake | VHLPPP |
| 294 | PolyP 5 | HeLa cells | Fluorescein | 15054781 | 10 | Fluorescence intensity | 50 uM | 3h | 37ºC | Fluorescent Microscopy | Cellular uptake | VHLPPPVHLPPP |
| 295 | PolyP 6 | HeLa cells | Fluorescein | 15054781 | 160 | Fluorescence intensity | 50 uM | 3h | 37ºC | Fluorescent Microscopy | Cellular uptake | VHLPPPVHLPPPVHLPPP |
| 296 | PolyP 7 | HeLa cells | Fluorescein | 15054781 | 0 | Fluorescence intensity | 50 uM | 3h | 37ºC | Fluorescent Microscopy | Cellular uptake | VKLPPP |
| 297 | PolyP 8 | HeLa cells | Fluorescein | 15054781 | 200 | Fluorescence intensity | 50 uM | 3h | 37ºC | Fluorescent Microscopy | Cellular uptake | VKLPPPVKLPPP |
| 298 | PolyP 9 | HeLa cells | Fluorescein | 15054781 | 230 | Fluorescence intensity | 50 uM | 3h | 37ºC | Fluorescent Microscopy | Cellular uptake | VKLPPPVKLPPPVKLPPP |
| 299 | hClock-(35-47) | ECV304 cells | FITC | 15346201 | 74 | Mean Fluorescence intensity | 4 uM | 1h | 37ºC | Fluorescent Microscopy | Internalization | KRVSRNKSEKKRR |
| 300 | Penetratin {pAntp-(43-58)} | CHO-K1 cells | Rho | 15937518 | 21.25 | Fold Change in GeoMean Fluorescence of control sample | 5 uM | 30 min | NA | Flow cytometry | Uptake | RQIKIWFQNRRMKWKK |
| 301 | Penetratin {pAntp-(43-58)} | HeLa cells | Rho | 15937518 | 3.13 | Fold Change in GeoMean Fluorescence of control sample | 5 uM | 30 min | NA | Flow cytometry | Uptake | RQIKIWFQNRRMKWKK |
| 302 | Penetratin {pAntp-(43-58)} | A549 cells | Rho | 15937518 | 2.29 | Fold Change in GeoMean Fluorescence of control sample | 5 uM | 30 min | NA | Flow cytometry | Uptake | RQIKIWFQNRRMKWKK |
| 303 | pAntpƒ-PKI | CHO-K1 cells | Rho | 15937518 | 21.5 | Fold Change in GeoMean Fluorescence of control sample | 5 uM | 30 min | NA | Flow cytometry | Uptake | RQIKIWFQNRRMKWKKTYADFIASGRTGRRNAI |
| 304 | pAntpƒ-PKI | HeLa cells | Rho | 15937518 | 8.13 | Fold Change in GeoMean Fluorescence of control sample | 5 uM | 30 min | NA | Flow cytometry | Uptake | RQIKIWFQNRRMKWKKTYADFIASGRTGRRNAI |
| 305 | pAntpƒ-PKI | A549 cells | Rho | 15937518 | 4.16 | Fold Change in GeoMean Fluorescence of control sample | 5 uM | 30 min | NA | Flow cytometry | Uptake | RQIKIWFQNRRMKWKKTYADFIASGRTGRRNAI |
| 306 | Tat | CHO-K1 cells | Rho | 15937518 | 3.54 | Fold Change in GeoMean Fluorescence of control sample | 5 uM | 30 min | NA | Flow cytometry | Uptake | GRKKRRQRRRPPQ |
| 307 | Tat | HeLa cells | Rho | 15937518 | 1.83 | Fold Change in GeoMean Fluorescence of control sample | 5 uM | 30 min | NA | Flow cytometry | Uptake | GRKKRRQRRRPPQ |
| 308 | Tat | A549 cells | Rho | 15937518 | 1.68 | Fold Change in GeoMean Fluorescence of control sample | 5 uM | 30 min | NA | Flow cytometry | Uptake | GRKKRRQRRRPPQ |
| 309 | Tat-PKI | CHO-K1 cells | Rho | 15937518 | 5.41 | Fold Change in GeoMean Fluorescence of control sample | 5 uM | 30 min | NA | Flow cytometry | Uptake | GRKKRRQRRRPPQTYADFIASGRTGRRNAI |
| 310 | Tat-PKI | HeLa cells | Rho | 15937518 | 2.5 | Fold Change in GeoMean Fluorescence of control sample | 5 uM | 30 min | NA | Flow cytometry | Uptake | GRKKRRQRRRPPQTYADFIASGRTGRRNAI |
| 311 | Tat-PKI | A549 cells | Rho | 15937518 | 1.84 | Fold Change in GeoMean Fluorescence of control sample | 5 uM | 30 min | NA | Flow cytometry | Uptake | GRKKRRQRRRPPQTYADFIASGRTGRRNAI |
| 312 | Transportan | CHO-K1 cells | Rho | 15937518 | 2 | Fold Change in GeoMean Fluorescence of control sample | 5 uM | 30 min | NA | Flow cytometry | Uptake | AGYLLGKINLKALAALAKKIL |
| 313 | Transportan | HeLa cells | Rho | 15937518 | 1.6 | Fold Change in GeoMean Fluorescence of control sample | 5 uM | 30 min | NA | Flow cytometry | Uptake | AGYLLGKINLKALAALAKKIL |
| 314 | Transportan | A549 cells | Rho | 15937518 | 1 | Fold Change in GeoMean Fluorescence of control sample | 5 uM | 30 min | NA | Flow cytometry | Uptake | AGYLLGKINLKALAALAKKIL |
| 315 | Transportan-PKI | CHO-K1 cells | Rho | 15937518 | 18 | Fold Change in GeoMean Fluorescence of control sample | 5 uM | 30 min | NA | Flow cytometry | Uptake | AGYLLGKINLKALAALAKKILTYADFIASGRTGRRNAI |
| 316 | Transportan-PKI | HeLa cells | Rho | 15937518 | 15.6 | Fold Change in GeoMean Fluorescence of control sample | 5 uM | 30 min | NA | Flow cytometry | Uptake | AGYLLGKINLKALAALAKKILTYADFIASGRTGRRNAI |
| 317 | Transportan-PKI | A549 cells | Rho | 15937518 | 9 | Fold Change in GeoMean Fluorescence of control sample | 5 uM | 30 min | NA | Flow cytometry | Uptake | AGYLLGKINLKALAALAKKILTYADFIASGRTGRRNAI |
| 318 | R11 | CHO-K1 cells | Rho | 15937518 | 31.16 | Fold Change in GeoMean Fluorescence of control sample | 5 uM | 30 min | NA | Flow cytometry | Uptake | RRRRRRRRRRR |
| 319 | R11 | HeLa cells | Rho | 15937518 | 43.93 | Fold Change in GeoMean Fluorescence of control sample | 5 uM | 30 min | NA | Flow cytometry | Uptake | RRRRRRRRRRR |
| 320 | R11 | A549 cells | Rho | 15937518 | 12.12 | Fold Change in GeoMean Fluorescence of control sample | 5 uM | 30 min | NA | Flow cytometry | Uptake | RRRRRRRRRRR |
| 321 | R11-PKI | CHO-K1 cells | Rho | 15937518 | 7.5 | Fold Change in GeoMean Fluorescence of control sample | 5 uM | 30 min | NA | Flow cytometry | Uptake | RRRRRRRRRRRTYADFIASGRTGRRNAI |
| 322 | R11-PKI | HeLa cells | Rho | 15937518 | 6.06 | Fold Change in GeoMean Fluorescence of control sample | 5 uM | 30 min | NA | Flow cytometry | Uptake | RRRRRRRRRRRTYADFIASGRTGRRNAI |
| 323 | R11-PKI | A549 cells | Rho | 15937518 | 3.63 | Fold Change in GeoMean Fluorescence of control sample | 5 uM | 30 min | NA | Flow cytometry | Uptake | RRRRRRRRRRRTYADFIASGRTGRRNAI |
| 324 | R9 | HeLa cells | Fluorescein | 21867915 | 100.0 | Cellular uptake (%) | 5 uM | 45 min | 37ºC | FCS | Uptake | RRRRRRRRR |
| 325 | R9 | MC57 | Fluorescein | 21867915 | 100.0 | Cellular uptake (%) | 5 uM | 45 min | 37ºC | FCS | Uptake | RRRRRRRRR |
| 326 | R9 | Jurkat cells | Fluorescein | 21867915 | 100.0 | Cellular uptake (%) | 5 uM | 45 min | 37ºC | FCS | Uptake | RRRRRRRRR |
| 327 | r9 | HeLa cells | Fluorescein | 21867915 | 53.13 | Cellular uptake (%) | 5 uM | 45 min | 37ºC | FCS | Uptake | rrrrrrrrr |
| 328 | r9 | MC57 | Fluorescein | 21867915 | 46.87 | Cellular uptake (%) | 5 uM | 45 min | 37ºC | FCS | Uptake | rrrrrrrrr |
| 329 | r9 | Jurkat cells | Fluorescein | 21867915 | 90.62 | Cellular uptake (%) | 5 uM | 45 min | 37ºC | FCS | Uptake | rrrrrrrrr |
| 330 | MAP | A549 cells | Fluorescein | 21875799 | 15 | Mean Fluorescence intensity/mg protein | 2 uM | 6h | 37ºC | Fluorescence spectroscopy | Internalization | KLALKLALKALKAALKLAGC |
| 331 | MAP (Aib) | A549 cells | Fluorescein | 21875799 | 160 | Mean Fluorescence intensity/mg protein | 2 uM | 6h | 37ºC | Fluorescence spectroscopy | Internalization | KLULKLULKULKAULKLUGC |
| 332 | HIV-1 Rev (34-50) | CHO-K1 cells | Alexa488 | 19707187 | 6.6 | Relative Cellular uptake | 5 umol/L | 30 min. | 37ºC | Flow cytometry | Uptake | TRQARRNRRRRWRERQRGC |
| 333 | HIV-1 Rev (34-50) | HeLa cells | Alexa488 | 19707187 | 6.0 | Relative Cellular uptake | 5 umol/L | 30 min. | 37ºC | Flow cytometry | Uptake | TRQARRNRRRRWRERQRGC |
| 334 | HIV-1 Rev (34-50) | Jurkat cells | Alexa488 | 19707187 | 2.5 | Relative Cellular uptake | 5 umol/L | 30 min. | 37ºC | Flow cytometry | Uptake | TRQARRNRRRRWRERQRGC |
| 335 | FHV coat (35-49) | CHO-K1 cells | Alexa488 | 19707187 | 21.1 | Relative Cellular uptake | 5 umol/L | 30 min. | 37ºC | Flow cytometry | Uptake | RRRRNRTRRNRRRVRGC |
| 336 | FHV coat (35-49) | HeLa cells | Alexa488 | 19707187 | 16.2 | Relative Cellular uptake | 5 umol/L | 30 min. | 37ºC | Flow cytometry | Uptake | RRRRNRTRRNRRRVRGC |
| 337 | FHV coat (35-49) | Jurkat cells | Alexa488 | 19707187 | 15.9 | Relative Cellular uptake | 5 umol/L | 30 min. | 37ºC | Flow cytometry | Uptake | RRRRNRTRRNRRRVRGC |
| 338 | BMV Gag (7-25) | CHO-K1 cells | Alexa488 | 19707187 | 1.2 | Relative Cellular uptake | 5 umol/L | 30 min. | 37ºC | Flow cytometry | Uptake | KMTRAQRRAAARRNRWTARGC |
| 339 | BMV Gag (7-25) | HeLa cells | Alexa488 | 19707187 | 1.3 | Relative Cellular uptake | 5 umol/L | 30 min. | 37ºC | Flow cytometry | Uptake | KMTRAQRRAAARRNRWTARGC |
| 340 | BMV Gag (7-25) | Jurkat cells | Alexa488 | 19707187 | 1.6 | Relative Cellular uptake | 5 umol/L | 30 min. | 37ºC | Flow cytometry | Uptake | KMTRAQRRAAARRNRWTARGC |
| 341 | HTLV-II Rex (4-16) | CHO-K1 cells | Alexa488 | 19707187 | 1.3 | Relative Cellular uptake | 5 umol/L | 30 min. | 37ºC | Flow cytometry | Uptake | TRRQRTRRARRNRGC |
| 342 | HTLV-II Rex (4-16) | HeLa cells | Alexa488 | 19707187 | 1.2 | Relative Cellular uptake | 5 umol/L | 30 min. | 37ºC | Flow cytometry | Uptake | TRRQRTRRARRNRGC |
| 343 | HTLV-II Rex (4-16) | Jurkat cells | Alexa488 | 19707187 | 1.8 | Relative Cellular uptake | 5 umol/L | 30 min. | 37ºC | Flow cytometry | Uptake | TRRQRTRRARRNRGC |
| 344 | Human cJun (252-279) | CHO-K1 cells | Alexa488 | 19707187 | 14.4 | Relative Cellular uptake | 5 umol/L | 30 min | 37ºC | Flow cytometry | Uptake | RIKAERKRMRNRIAASKSRKRKLERIARGC |
| 345 | Human cJun (252-279) | HeLa cells | Alexa488 | 19707187 | 12.4 | Relative Cellular uptake | 5 umol/L | 30 min | 37ºC | Flow cytometry | Uptake | RIKAERKRMRNRIAASKSRKRKLERIARGC |
| 346 | Human cJun (252-279) | Jurkat cells | Alexa488 | 19707187 | 10.5 | Relative Cellular uptake | 5 umol/L | 30 min | 37ºC | Flow cytometry | Uptake | RIKAERKRMRNRIAASKSRKRKLERIARGC |
| 347 | Human cFos (139-164) | CHO-K1 cells | Alexa488 | 19707187 | 0.9 | Relative Cellular uptake | 5 umol/L | 30 min. | 37ºC | Flow cytometry | Uptake | KRRIRRERNKMAAAKSRNRRRELTDTGC |
| 348 | Human cFos (139-164) | HeLa cells | Alexa488 | 19707187 | 0.8 | Relative Cellular uptake | 5 umol/L | 30 min. | 37ºC | Flow cytometry | Uptake | KRRIRRERNKMAAAKSRNRRRELTDTGC |
| 349 | Human cFos (139-164) | Jurkat cells | Alexa488 | 19707187 | 1.0 | Relative Cellular uptake | 5 umol/L | 30 min. | 37ºC | Flow cytometry | Uptake | KRRIRRERNKMAAAKSRNRRRELTDTGC |
| 350 | cTat | Rat alveolar epithelial cell monolayers (RAECM) | Insulin | 19228019 | 1.68 | % Amount transported into basolateral fluid | NA | 2h | 37ºC | Gamma-well counter | Absorption | crkkrrqrrr |
| 351 | cr9 | Rat alveolar epithelial cell monolayers (RAECM) | Insulin | 19228019 | 2.46 | % Amount transported into basolateral fluid | NA | 2h | 37ºC | Gamma-well counter | Absorption | crrrrrrrrr |
| 352 | ck9 | Rat alveolar epithelial cell monolayers (RAECM) | Insulin | 19228019 | 0.38 | % Amount transported into basolateral fluid | NA | 2h | 37ºC | Gamma-well counter | Absorption | ckkkkkkkkk |
| 353 | (RW)4 | SK-OV-3 cells | Doxorubicin | 23301519 | 31 | Mean Fluorescence intensity | 5 uM | 1h | 37ºC | Flow cytometry | Cellular uptake | RWRWRWRW |
| 354 | cyclic [W(RW)4] | SK-OV-3 cells | Doxorubicin | 23301519 | 81 | Mean Fluorescence intensity | 5 uM | 1h | 37ºC | Flow cytometry | Cellular uptake | WRWRWRWRW |
| 355 | PA 2 | PPC-1 | Rho | 23349939 | 6 | pmol/ug total protein | NA | NA | 37ºC | Fluorescence spectroscopy | Association | RPARPAR |
| 356 | PA 2 | M21 | Rho | 23349939 | 7.1 | pmol/ug total protein | NA | NA | 37ºC | Fluorescence spectroscopy | Association | RPARPAR |
| 357 | PA 3 | PPC-1 | Rho | 23349939 | 5 | pmol/ug total protein | NA | NA | 37ºC | Fluorescence spectroscopy | Association | RPARPAR |
| 358 | Peptide 599 | Human tongue squamous cell carcinoma (SCC) CAL 27 | siRNA | 24019920 | 45 | pmol siRNA / mg protein | 100:1 molar excess of siRNAs | 2.5 h | NA | Fluorescent Microscopy | Transfection | GLFEAIEGFIENGWEGMIDGWYGGGGrrrrrrrrrK |
| 359 | CH2 R4 H2 C | S-180 sarcoma cells | siRNA | 23911914 | 700 | Mean Fluorescence intensity/cell | N/P ratio 20 | 4h | NA | Flow cytometry | Transfection | CHHRRRRHHC |
| 360 | STR-R8 | CHO-K1 cells | GAPDH siRNA | 25193363 | 260 | Mean Fluorescence intensity | 100 nM siRNA | 3h | NA | Flow cytometry | Transfection | RRRRRRRR |
| 361 | STR-H8R8 | CHO-K1 cells | GAPDH siRNA | 25193363 | 160 | Mean Fluorescence intensity | 100 nM siRNA | 3h | NA | Flow cytometry | Transfection | HHHHHHHHRRRRRRRR |
| 362 | STR-H8R15 | CHO-K1 cells | GAPDH siRNA | 25193363 | 195 | Mean Fluorescence intensity | 100 nM siRNA | 3h | NA | Flow cytometry | Transfection | HHHHHHHHRRRRRRRRRRRRRRR |
| 363 | STR-H12R8 | CHO-K1 cells | GAPDH siRNA | 25193363 | 187 | Mean Fluorescence intensity | 100 nM siRNA | 3h | NA | Flow cytometry | Transfection | HHHHHHHHHHHHRRRRRRRRRRRRRRR |
| 364 | STR-H16R8 | CHO-K1 cells | GAPDH siRNA | 25193363 | 220 | Mean Fluorescence intensity | 100 nM siRNA | 3h | NA | Flow cytometry | Transfection | HHHHHHHHHHHHHHHHRRRRRRRRRRRRRRR |
| 365 | STR-H20R8 | CHO-K1 cells | GAPDH siRNA | 25193363 | 211 | Mean Fluorescence intensity | 100 nM | 3h | NA | Flow cytometry | Transfection | HHHHHHHHHHHHHHHHHHHHRRRRRRRRRRRRRRR |
| 366 | 1b | HeLa cells | Carboxyfluorescein | 25188671 | 0.18 | Cellular uptake | 100 nM | 2h | 37ºC | Fluorescence spectroscopy | Uptake | RLLRLLRLL |
| 367 | 2b | HeLa cells | Carboxyfluorescein | 25188671 | 0.23 | Cellular uptake | 100 nM | 2h | 37ºC | Fluorescence spectroscopy | Uptake | RLLRLLRLX |
| 368 | 3b | HeLa cells | Carboxyfluorescein | 25188671 | 0.23 | Cellular uptake | 100 nM | 2h | 37ºC | Fluorescence spectroscopy | Uptake | RLLRLXRLX |
| 369 | 4b | HeLa cells | Carboxyfluorescein | 25188671 | 0.85 | Cellular uptake | 100 nM | 2h | 37ºC | Fluorescence spectroscopy | Uptake | RLXRLXRLX |
| 370 | Penetratin | NA | Insulin | 24973720 | 13 | Plasma insulin concentration (uU/mL) | 5 mM | 30 min | NA | NA | Absorption | RQIKIWFQNRRMKWKK |
| 371 | Penetratin | NA | Insulin | 24973720 | 55 | Plasma insulin concentration (uU/mL) | 5 mM | 30 min | NA | NA | Absorption | RQIKIWFQNRRMKWKK |
| 372 | RALA peptide | ZR-75-1 human breast cancer | pDNA | 24995949 | 57.0 | % Transfection | N/P ratio 10 | 48h | NA | Flow cytometry | Transfection | WEARLARALARALARHLARALARA |
| 373 | RALA peptide | PC3 cells | pDNA | 24995949 | 27.0 | % Transfection | N/P ratio 10 | 48h | NA | Flow cytometry | Transfection | WEARLARALARALARHLARALARA |
| 374 | C24-LMWP | A549 cells | PLGA-NPs | 25003794 | 492 | Median Fluorescence intensity | Equal to a DOX dose of 10 ug/mL | 4h | NA | Flow cytometry | Uptake | VSRRRRRRGGRRRR |
| 375 | C24-LMWP | MCF7 cells | PLGA-NPs | 25003794 | 93.2 | Median Fluorescence intensity | Equal to a DOX dose of 10 ug/mL | 4h | NA | Flow cytometry | Uptake | VSRRRRRRGGRRRR |
| 376 | hLF WT | HeLa cells | Fluorescein | 24270856 | 100 | Median Normalized Fluorescence | 5 uM | 30 min | 37ºC | Flow cytometry | Uptake | KCFQWQRNMRKVRGPPVSCIKR |
| 377 | hLF WT | Jurkat cells | Fluorescein | 24270856 | 100 | Median Normalized Fluorescence | 5 uM | 30 min | 37ºC | Flow cytometry | Uptake | KCFQWQRNMRKVRGPPVSCIKR |
| 378 | hLF WT | Ovcar-3 cells | Fluorescein | 24270856 | 100 | Median Normalized Fluorescence | 5 uM | 30 min | 37ºC | Flow cytometry | Uptake | KCFQWQRNMRKVRGPPVSCIKR |
| 379 | hLF WT | Caco-2 cells | Fluorescein | 24270856 | 100 | Median Normalized Fluorescence | 5 uM | 30 min | 37ºC | Flow cytometry | Uptake | KCFQWQRNMRKVRGPPVSCIKR |
| 380 | hLF W5A | HeLa cells | Fluorescein | 24270856 | 52.5 | Median Normalized Fluorescence | 5 uM | 30 min | 37ºC | Flow cytometry | Uptake | KCFQWQRNMRKVRGPPVSCIKR |
| 381 | hLF Q6A | HeLa cells | Fluorescein | 24270856 | 72.5 | Median Normalized Fluorescence | 5 uM | 30 min | 37ºC | Flow cytometry | Uptake | KCFQWQRNMRKVRGPPVSCIKR |
| 382 | hLF M9A | HeLa cells | Fluorescein | 24270856 | 55 | Median Normalized Fluorescence | 5 uM | 30 min | 37ºC | Flow cytometry | Uptake | KCFQWQRNMRKVRGPPVSCIKR |
| 383 | hLF P15A | HeLa cells | Fluorescein | 24270856 | 72.5 | Median Normalized Fluorescence | 5 uM | 30 min | 37ºC | Flow cytometry | Uptake | KCFQWQRNMRKVRGPPVSCIKR |
| 384 | hLF V12R | HeLa cells | Fluorescein | 24270856 | 75 | Median Normalized Fluorescence | 5 uM | 30 min | 37ºC | Flow cytometry | Uptake | KCFQWQRNMRKVRGPPVSCIKR |
| 385 | hLF R7A | HeLa cells | Fluorescein | 24270856 | 70 | Median Normalized Fluorescence | 5 uM | 30 min | 37ºC | Flow cytometry | Uptake | KCFQWQRNMRKVRGPPVSCIKR |
| 386 | hLF R13A | HeLa cells | Fluorescein | 24270856 | 72.5 | Median Normalized Fluorescence | 5 uM | 30 min | 37ºC | Flow cytometry | Uptake | KCFQWQRNMRKVRGPPVSCIKR |
| 387 | hLF R7A/V12R | HeLa cells | Fluorescein | 24270856 | 70 | Median Normalized Fluorescence | 5 uM | 30 min | 37ºC | Flow cytometry | Uptake | KCFQWQRNMRKVRGPPVSCIKR |
| 388 | hLF R13A/P15R | HeLa cells | Fluorescein | 24270856 | 57.5 | Median Normalized Fluorescence | 5 uM | 30 min | 37ºC | Flow cytometry | Uptake | KCFQWQRNMRKVRGPPVSCIKR |
| 389 | hLF +4R | HeLa cells | Fluorescein | 24270856 | 240 | Median Normalized Fluorescence | 5 uM | 30 min | 37ºC | Flow cytometry | Uptake | KCFQWQRNMRKVRGPPVSCIKR |
| 390 | hLF +4R | Jurkat cells | Fluorescein | 24270856 | 95 | Median Normalized Fluorescence | 5 uM | 30 min | 37ºC | Flow cytometry | Uptake | KCFQWQRNMRKVRGPPVSCIKR |
| 391 | hLF +4R | Ovcar-3 cells | Fluorescein | 24270856 | 90 | Median Normalized Fluorescence | 5 uM | 30 min | 37ºC | Flow cytometry | Uptake | KCFQWQRNMRKVRGPPVSCIKR |
| 392 | hLF +4R | Caco-2 cells | Fluorescein | 24270856 | 132.5 | Median Normalized Fluorescence | 5 uM | 30 min | 37ºC | Flow cytometry | Uptake | KCFQWQRNMRKVRGPPVSCIKR |
| 393 | hLF lin+4R | HeLa cells | Fluorescein | 24270856 | 137.5 | Median Normalized Fluorescence | 5 uM | 30 min | 37ºC | Flow cytometry | Uptake | KCFQWQRNMRKVRGPPVSCIKR |
| 394 | hLF lin+4R | Jurkat cells | Fluorescein | 24270856 | 200 | Median Normalized Fluorescence | 5 uM | 30 min | 37ºC | Flow cytometry | Uptake | KCFQWQRNMRKVRGPPVSCIKR |
| 395 | hLF lin+4R | Ovcar-3 cells | Fluorescein | 24270856 | 165 | Median Normalized Fluorescence | 5 uM | 30 min | 37ºC | Flow cytometry | Uptake | KCFQWQRNMRKVRGPPVSCIKR |
| 396 | hLF lin+4R | Caco-2 cells | Fluorescein | 24270856 | 460 | Median Normalized Fluorescence | 5 uM | 30 min | 37ºC | Flow cytometry | Uptake | KCFQWQRNMRKVRGPPVSCIKR |
| 397 | hLF R7 | HeLa cells | Fluorescein | 24270856 | 57.5 | Median Normalized Fluorescence | 5 uM | 30 min | 37ºC | Flow cytometry | Uptake | KCFQWQRNMRKVRGPPVSCIKR |
| 398 | hLF R7 | Jurkat cells | Fluorescein | 24270856 | 87.5 | Median Normalized Fluorescence | 5 uM | 30 min | 37ºC | Flow cytometry | Uptake | KCFQWQRNMRKVRGPPVSCIKR |
| 399 | hLF R7 | Ovcar-3 cells | Fluorescein | 24270856 | 55 | Median Normalized Fluorescence | 5 uM | 30 min | 37ºC | Flow cytometry | Uptake | KCFQWQRNMRKVRGPPVSCIKR |
| 400 | hLF R7 | Caco-2 cells | Fluorescein | 24270856 | 85 | Median Normalized Fluorescence | 5 uM | 30 min | 37ºC | Flow cytometry | Uptake | KCFQWQRNMRKVRGPPVSCIKR |
| 401 | hLF K7 | HeLa cells | Fluorescein | 24270856 | 50 | Median Normalized Fluorescence | 5 uM | 30 min | 37ºC | Flow cytometry | Uptake | KCFQWQRNMRKVRGPPVSCIKR |
| 402 | hLF K7 | Jurkat cells | Fluorescein | 24270856 | 75 | Median Normalized Fluorescence | 5 uM | 30 min | 37ºC | Flow cytometry | Uptake | KCFQWQRNMRKVRGPPVSCIKR |
| 403 | hLF K7 | Ovcar-3 cells | Fluorescein | 24270856 | 60 | Median Normalized Fluorescence | 5 uM | 30 min | 37ºC | Flow cytometry | Uptake | KCFQWQRNMRKVRGPPVSCIKR |
| 404 | hLF K7 | Caco-2 cells | Fluorescein | 24270856 | 87.5 | Median Normalized Fluorescence | 5 uM | 30 min | 37ºC | Flow cytometry | Uptake | KCFQWQRNMRKVRGPPVSCIKR |
| 405 | hLF Hcy | HeLa cells | Fluorescein | 24270856 | 85 | Median Normalized Fluorescence | 5 uM | 30 min | 37ºC | Flow cytometry | Uptake | K-Hey-FQWQRNMRKVRGPPVS-Hey-IKR |
| 406 | Pep1 | HeLa cells | Plasmid DNA | 24462902 | 150 | Mean Fluorescence intensity/cell | N/P ratio 20 | NA | NA | Flow cytometry | Transfection | GRGDSPRR |
| 407 | Pep1 | A549 cells | Plasmid DNA | 24462902 | 20 | Mean Fluorescence intensity/cell | N/P ratio 20 | NA | NA | Flow cytometry | Transfection | GRGDSPRR |
| 408 | Pep2 | HeLa cells | Plasmid DNA | 24462902 | 200 | Mean Fluorescence intensity/cell | N/P ratio 20 | NA | NA | Flow cytometry | Transfection | GRGDSPRRSPRR |
| 409 | Pep2 | A549 cells | Plasmid DNA | 24462902 | 30 | Mean Fluorescence intensity/cell | N/P ratio 20 | NA | NA | Flow cytometry | Transfection | GRGDSPRRSPRR |
| 410 | Pep3 | HeLa cells | Plasmid DNA | 24462902 | 700 | Mean Fluorescence intensity/cell | N/P ratio 20 | NA | NA | Flow cytometry | Transfection | GRGDSPRRKKKKSPRRKKKKSPRR |
| 411 | Pep3 | A549 cells | Plasmid DNA | 24462902 | 38 | Mean Fluorescence intensity/cell | N/P ratio 20 | NA | NA | Flow cytometry | Transfection | GRGDSPRRKKKKSPRRKKKKSPRR |
| 412 | Pep3(Mutant) | HeLa cells | Plasmid DNA | 24462902 | 750 | Mean Fluorescence intensity/cell | N/P ratio 20 | NA | NA | Flow cytometry | Transfection | GRGDGPRRKKKKGPRRKKKKGPRR |
| 413 | Pep3(Mutant) | A549 cells | Plasmid DNA | 24462902 | 37.5 | Mean Fluorescence intensity/cell | N/P ratio 20 | NA | NA | Flow cytometry | Transfection | GRGDGPRRKKKKGPRRKKKKGPRR |
| 414 | FAM-1 | HeLa cells | Carboxyfluorescein | 24661993 | 1500 | pmol/mg protein Cellular uptake | 3 uM | 2 h | 37°C | Fluorescence spectroscopy | Uptake | BRRXRRXRRX |
| 415 | ent FAM-1 | HeLa cells | Carboxyfluorescein | 24661993 | 1940 | pmol/mg protein Cellular uptake | 3 uM | 2 h | 37°C | Fluorescence spectroscopy | Uptake | BrrXrrXrrX |
| 416 | FAM-2 | HeLa cells | Carboxyfluorescein | 24661993 | 845 | pmol/mg protein Cellular uptake | 3 uM | 2 h | 37°C | Fluorescence spectroscopy | Uptake | BRrXRrXRrX |
| 417 | FAM-3 | HeLa cells | Carboxyfluorescein | 24661993 | 625 | pmol/mg protein Cellular uptake | 3 uM | 2 h | 37°C | Fluorescence spectroscopy | Uptake | BXRXRXXRXRXXRXRX |
| 418 | RIPL | LNCaP | FITC | 24704199 | 78.3 | Mean Fluorescence intensity | 1 uM | 2h | 37ºC | Flow cytometry | Uptake | IPLVVPLRRRRRRRRC |
| 419 | RIPL | SK-OV-3 cells | FITC | 24704199 | 16.6 | Mean Fluorescence intensity | 1 uM | 2h | 37ºC | Flow cytometry | Uptake | IPLVVPLRRRRRRRRC |
| 420 | RIPL | MCF7 cells | FITC | 24704199 | 31.6 | Mean Fluorescence intensity | 1 uM | 2h | 37ºC | Flow cytometry | Uptake | IPLVVPLRRRRRRRRC |
| 421 | RIPL | DU-145 | FITC | 24704199 | 10 | Mean Fluorescence intensity | 1 uM | 2h | 37ºC | Flow cytometry | Uptake | IPLVVPLRRRRRRRRC |
| 422 | RIPL | PC3 cells | FITC | 24704199 | 23.3 | Mean Fluorescence intensity | 1 uM | 2h | 37ºC | Flow cytometry | Uptake | IPLVVPLRRRRRRRRC |
| 423 | RIPL | HaCaT cells | FITC | 24704199 | 4.16 | Mean Fluorescence intensity | 1 uM | 2h | 37ºC | Flow cytometry | Uptake | IPLVVPLRRRRRRRRC |
| 424 | R8 | LNCaP | FITC | 24704199 | 12.4 | Mean Fluorescence intensity | 3 uM | 2h | 37ºC | Flow cytometry | Uptake | RRRRRRRRC |
| 425 | IPL | LNCaP | FITC | 24704199 | 9 | Mean Fluorescence intensity | 3 uM | 2h | 37ºC | Flow cytometry | Uptake | IPLVVPLC |
| 426 | EGFP-TAT | Mouse macrophage-like cell line J774 A.1 | eGFP | 24746937 | 79.2 | % Positive cells | 10 umol/L | 1h | 37ºC | Flow cytometry | Internalization | YGRKKRRQRRR |
| 427 | EGFP-VP_22 | Mouse macrophage-like cell line J774 A.3 | eGFP | 24746937 | 58.1 | % Positive cells | 10 umol/L | 1h | 37ºC | Flow cytometry | Internalization | DAATARGRGRSAASRPTERPRAPARSASRPRRPVD |
| 428 | EGFP-LMWP | Mouse macrophage-like cell line J774 A.5 | eGFP | 24746937 | 98.8 | % Positive cells | 10 umol/L | 1h | 37ºC | Flow cytometry | Internalization | GSVSRRRRRRGGRRRR |
| 429 | EGFP-hcT(9-32) | Mouse macrophage-like cell line J774 A.6 | eGFP | 24746937 | 35.6 | % Positive cells | 10 umol/L | 1h | 37ºC | Flow cytometry | Internalization | LGTYTQDFNKFHTFPQTAIGVGAP |
| 430 | EGFP-R12 | Mouse macrophage-like cell line J774 A.10 | eGFP | 24746937 | 75.2 | % Positive cells | 10 umol/L | 1h | 37ºC | Flow cytometry | Internalization | RRRRRRRRRRRR |
| 431 | Hph-1 | HeLa cells | Hph1Hph1dsRBD/FAM-labeled siRNA complex | 24768403 | 99.0 | % Positive cells | 100 uM siRNA | 1h | NA | Flow cytometry | Uptake | YARVRRRGPRR |
| 432 | Mgpe-9 | CHO-K1 cells | Plasmid DNA | 24816284 | 5900 | Mean Fluorescence intensity | Charge ratio = 0.5 / Charge ratio 5 | 4h | 37ºC | Flow cytometry | Cellular uptake | CRRLRHLRHHYRRRWHRFRC |
| 433 | Mgpe-10 | CHO-K1 cells | Plasmid DNA | 24816284 | 400 | Mean Fluorescence intensity | Charge ratio = 0.5 / Charge ratio 5 | 4h | 37ºC | Flow cytometry | Cellular uptake | CLLYWFRRRHRHHRRRHRRC |
| 434 | ACPP | A549 cells | ACPP-HPMA Copolymer-Coated Adenovirus Conjugates | 25000246 | 85 | Relative fluorescence | 10^4 particles | 1h | 37ºC | Fluoroskan plate reader | Uptake | EEEEEEEEPLGLAGRRRRRRRRN |
| 435 | ACPP | MDA-MB-231 cells | ACPP-HPMA Copolymer-Coated Adenovirus Conjugates | 25000246 | 86 | Relative fluorescence | 10^4 particles | 1h | 37ºC | Fluoroskan plate reader | Uptake | EEEEEEEEPLGLAGRRRRRRRRN |
| 436 | ACPP | Human bronchial epithelial (HBE) cells | ACPP-HPMA Copolymer-Coated Adenovirus Conjugates | 25000246 | 9.6 | Relative fluorescence | 10^4 particles | 1h | 37ºC | Fluoroskan plate reader | Uptake | EEEEEEEEPLGLAGRRRRRRRRN |
| 437 | ACPP | HepG2 cells | ACPP-HPMA Copolymer-Coated Adenovirus Conjugates | 25000246 | 96 | Relative fluorescence | 10^4 particles | 1h | 37ºC | Fluoroskan plate reader | Uptake | EEEEEEEEPLGLAGRRRRRRRRN |
| 438 | LMWP | Pluripotent mouse mesenchymal progenitor cell line (C3H10T1/2) | TAZ | 24648725 | 98.9 | % Positive cells | 100 nM | 20 min | 37ºC | Flow cytometry | Internalization | VSRRRRRRGGRRRR |
| 439 | R7 | NA | ESRRB recombinant protein | 24693491 | 53.3 | Relative fluorescence | 2 ug/ml | 24h | NA | Immunocytochemistry | Transduction | RRRRRRR |
| 440 | Pip6a | Murine H2k mdx myoblasts | phosphorodiamidate morpholino oligomers (PMO) | 24366877 | 12812 | RFU/mg | 1 uM | 4h | NA | Fluorescence spectroscopy | Internalization | RXRRBRRXRYQFLIRXRBRXRB |
| 441 | Pip6a | C2C12 cells | phosphorodiamidate morpholino oligomers (PMO) | 24366877 | 7916 | RFU/mg | 1 uM | 4h | NA | Fluorescence spectroscopy | Internalization | RXRRBRRXRYQFLIRXRBRXRB |
| 442 | R9 | CHO-K1 cells | Biotin-gly4 | 25112713 | 8.0 | Internalized peptide (uM) | 10 uM | 70 min | 37ºC | MALDI-TOF | Internalization | RRRRRRRRR |
| 443 | R9 | xylose transferase- or GAG-deficient CHO-pgsA745 cells (GAGneg) | Biotin-gly4 | 25112713 | 2.5 | Internalized peptide (uM) | 10 uM | 70 min | 37ºC | MALDI-TOF | Internalization | RRRRRRRRR |
| 444 | TAT(47-57) | CHO-K1 cells | Biotin-gly4 | 25112713 | 0.2 | Internalized peptide (uM) | 10 uM | 70 min | 37ºC | MALDI-TOF | Internalization | YGRKKRRQRRR |
| 445 | TAT(47-57) | xylose transferase- or GAG-deficient CHO-pgsA745 cells (GAGneg) | Biotin-gly4 | 25112713 | 0.725 | Internalized peptide (uM) | 10 uM | 70 min | 37ºC | MALDI-TOF | Internalization | YGRKKRRQRRR |
| 446 | R6L3 | CHO-K1 cells | Biotin-gly4 | 25112713 | 0.3 | Internalized peptide (uM) | 10 uM | 70 min | 37ºC | MALDI-TOF | Internalization | RRLLRRLRR |
| 447 | R6L3 | xylose transferase- or GAG-deficient CHO-pgsA745 cells (GAGneg) | Biotin-gly4 | 25112713 | 0.2 | Internalized peptide (uM) | 10 uM | 70 min | 37ºC | MALDI-TOF | Internalization | RRLLRRLRR |
| 448 | Penetratin | CHO-K1 cells | Biotin-gly4 | 25112713 | 0.3 | Internalized peptide (uM) | 10 uM | 70 min | 37ºC | MALDI-TOF | Internalization | RQIKIWFQNRRMKWKK |
| 449 | Penetratin | xylose transferase- or GAG-deficient CHO-pgsA745 cells (GAGneg) | Biotin-gly4 | 25112713 | 0.2 | Internalized peptide (uM) | 10 uM | 70 min | 37ºC | MALDI-TOF | Internalization | RQIKIWFQNRRMKWKK |
| 450 | R6W3 | CHO-K1 cells | Biotin-gly4 | 25112713 | 9 | Internalized peptide (uM) | 10 uM | 70 min | 37ºC | MALDI-TOF | Internalization | RRWWRRWRR |
| 451 | R6W3 | xylose transferase- or GAG-deficient CHO-pgsA745 cells (GAGneg) | Biotin-gly4 | 25112713 | 5.0 | Internalized peptide (uM) | 10 uM | 70 min | 37ºC | MALDI-TOF | Internalization | RRWWRRWRR |
| 452 | MCa UF1-9-C-Cy5 | Undifferentiated malignant glioma rat (F98) cell line | Cy5 | 24276021 | 4.7e+5 | Fluorescence intensity | 10 uM | 2h | 37ºC | Flow cytometry | Penetration | GD(Abu)LPHLKLC |
| 453 | Tat-C-Cy5 | Undifferentiated malignant glioma rat (F98) cell line | Cy5 | 24276021 | 9.0e+4 | Fluorescence intensity | 10 uM | 2h | 37ºC | Flow cytometry | Penetration | YGRKKRRQRRRC |
| 454 | Pen-C-Cy5 | Undifferentiated malignant glioma rat (F98) cell line | Cy5 | 24276021 | 1.3e+5 | Fluorescence intensity | 10 uM | 2h | 37ºC | Flow cytometry | Penetration | RQIKIWFQNRRMKWKKC |
| 455 | PolyR-C-Cy5 | Undifferentiated malignant glioma rat (F98) cell line | Cy5 | 24276021 | 1.4e+5 | Fluorescence intensity | 10 uM | 2h | 37ºC | Flow cytometry | Penetration | RRRRRRRRRC |
| 456 | CF-BP16 | MCF7 cells | Carboxyfluorescein | 24480922 | 1431 ± 307 | Mean Fluorescence intensity | 50 uM | 1h | 37ºC | Flow cytometry | Uptake | KKLFKKILKKL |
| 457 | CF-BP16 | mouse embryonic fibroblast 3T3 | Carboxyfluorescein | 24480922 | 1829 ± 335 | Mean Fluorescence intensity | 50 uM | 1h | 37ºC | Flow cytometry | Uptake | KKLFKKILKKL |
| 458 | BP328 | MCF7 cells | Carboxyfluorescein | 24480922 | 1789 ± 221 | Mean Fluorescence intensity | 25 uM | 3h | 37ºC | Flow cytometry | Uptake | CREKA-KKLFKKILKKL |
| 459 | BP328 | mouse embryonic fibroblast 3T3 | Carboxyfluorescein | 24480922 | 1300 ± 221 | Mean Fluorescence intensity | 25 uM | 3h | 37ºC | Flow cytometry | Uptake | CREKA-KKLFKKILKKL |
| 460 | Penetratin | Wong-Kilbourne-derived human conjunctival epithelial cells (NHC) | Carboxyfluorescein | 24521351 | 13000 | Mean Fluorescence intensity | 57 umol/L | 1h | 37ºC | Flow cytometry | Uptake | RQIKIWFQNRRMKWKKK |
| 461 | Arg5-ELPBC | HeLa cells | BH3 peptide drug and ELPBC | 24611762 | 2.0 | Cell Fluorescence | 10 uM | 1h | 37ºC | Flow cytometry | Uptake | RRRRR |
| 462 | Arg8-ELPBC | HeLa cells | BH3 peptide drug and ELPBC | 24611762 | 10 | Cell Fluorescence | 10 uM | 1h | 37ºC | Flow cytometry | Uptake | RRRRRRRR |
| 463 | TAT-ELPBC | HeLa cells | BH3 peptide drug and ELPBC | 24611762 | 10 | Cell Fluorescence | 10 uM | 1h | 37ºC | Flow cytometry | Uptake | YGRKKRRQRRR |
| 464 | RTAT-ELPBC | HeLa cells | BH3 peptide drug and ELPBC | 24611762 | 4.0 | Cell Fluorescence | 10 uM | 1h | 37ºC | Flow cytometry | Uptake | YGRGGRRGRRR |
| 465 | IA0 (Bicyclic) (integral arginine peptides) | HeLa cells | FITC | 24697151 | 0 | Normalized Median Fluorescence | 5 uM | 1h | 37ºC | Flow cytometry | Uptake | ACSGSGSGCGSGSGSCG |
| 466 | IA2 | HeLa cells | FITC | 24697151 | 1.25 | Normalized Median Fluorescence | 5 uM | 1h | 37ºC | Flow cytometry | Uptake | ACSGRGSGCGSGRGSCG |
| 467 | IA4a | HeLa cells | FITC | 24697151 | 3.75 | Normalized Median Fluorescence | 5 uM | 1h | 37ºC | Flow cytometry | Uptake | ACRGSGRGCGRGSGRCG |
| 468 | IA4b | HeLa cells | FITC | 24697151 | 10 | Normalized Median Fluorescence | 5 uM | 1h | 37ºC | Flow cytometry | Uptake | ACSGRGRGCGRGRGSCG |
| 469 | IA6b | HeLa cells | FITC | 24697151 | 20 | Normalized Median Fluorescence | 5 uM | 1h | 37ºC | Flow cytometry | Uptake | ACGRGRGRCRGRGRGCG |
| 470 | IA8b | HeLa cells | FITC | 24697151 | 45 | Normalized Median Fluorescence | 5 uM | 1h | 37ºC | Flow cytometry | Uptake | ACRRSRRGCGRRSRRCG |
| 471 | GST-(HE)8EFG5YG(RG)6 | HeLa cells | GST | 24697211 | 240 | ng molecule / mg cell protein | 5 ug/ml | 1h | 37ºC | Gamma-well counter | Uptake | HEHEHEHEHEHEHEHEEFGGGGGYGRGRGRGRGRGRG |
| 472 | GST-(HE)10EFG5YG(RG)6 | HeLa cells | GST | 24697211 | 190 | ng molecule / mg cell protein | 5 ug/ml | 1h | 37ºC | Gamma-well counter | Uptake | HEHEHEHEHEHEHEHEHEHEEFGGGGGYGRGRGRGRGRGRG |
| 473 | GST-(HE)12EFG5YG(RG)6 | HeLa cells | GST | 24697211 | 80 | ng molecule / mg cell protein | 5 ug/ml | 1h | 37ºC | Gamma-well counter | Uptake | HEHEHEHEHEHEHEHEHEHEHEHEEFGGGGGYGRGRGRGRGRGRG |
| 474 | GST-(HE)8EFG5YGR6G6 | HeLa cells | GST | 24697211 | 370 | ng molecule / mg cell protein | 5 ug/ml | 1h | 37ºC | Gamma-well counter | Uptake | HEHEHEHEHEHEHEHEEFGGGGGYGRRRRRRGGGGGG |
| 475 | GST-(HE)10EFG5YGR6G6 | HeLa cells | GST | 24697211 | 335 | ng molecule / mg cell protein | 5 ug/ml | 1h | 37ºC | Gamma-well counter | Uptake | HEHEHEHEHEHEHEHEHEHEEFGGGGGYGRRRRRRGGGGGG |
| 476 | GST-(HE)12EFG5YGR6G6 | HeLa cells | GST | 24697211 | 100 | ng molecule / mg cell protein | 5 ug/ml | 1h | 37ºC | Gamma-well counter | Uptake | HEHEHEHEHEHEHEHEHEHEHEHEEFGGGGGYGRRRRRRGGGGGG |
| 477 | GST-(HE)12EFG5-TAT | HeLa cells | GST | 24697211 | 327 | ng molecule / mg cell protein | 5 ug/ml | 1h | 37ºC | Gamma-well counter | Uptake | HEHEHEHEHEHEHEHEHEHEHEHEEFGGGGGYGRKKRRQRRR |
| 478 | LK-1 | HeLa cells | FITC | 25056130 | 67 | % Positive cells | 100 nM | 12h | NA | Flow cytometry | Uptake | LKKLLKLLKKLLKLAG |
| 479 | LK-2 | HeLa cells | FITC | 25056130 | 70 | % Positive cells | 100 nM | 12h | NA | Flow cytometry | Uptake | LKKLCKLLKKLCKLAG |
| 480 | VG-21 | HEp-2 | FITC | 25154664 | 35.3 | % Positive cells | 1 nM | 48h | NA | Flow cytometry | Uptake | VTPHHVLVDEYTGEWVDSQFK |
| 481 | VG-21 | HeLa cells | FITC | 25154664 | 43.8 | % Positive cells | 1 nM | 48h | NA | Flow cytometry | Uptake | VTPHHVLVDEYTGEWVDSQFK |
| 482 | VG-21 | Vero | FITC | 25154664 | 32.4 | % Positive cells | 1 nM | 48h | NA | Flow cytometry | Uptake | VTPHHVLVDEYTGEWVDSQFK |
| 483 | VG-21 | Cos-7 cells | FITC | 25154664 | 26.6 | % Positive cells | 1 nM | 48h | NA | Flow cytometry | Uptake | VTPHHVLVDEYTGEWVDSQFK |
| 484 | PNIPAM-FL-TAT Peptide | A549 cells | poly(N-isopropylacrylamide) (PNIPAM) microgel particles | 25170605 | 1500 | Relative fluorescence | 200 ug/ml | 24h | NA | Flow cytometry | Uptake | YGRKKRRQRRR |
| 485 | Trehalose-KRKRWHW-Heparin | Mammalian cells | Trehalose | 24583082 | 20 | mM Intracellular concentration | 8 mM Trehalose | 1h | 37ºC | Flow cytometry | Interalization | KRKRWHW |
| 486 | SP-TatCherry | A549 cells | mCherry | 24928321 | 2800 | Mean Fluorescence intensity | 13 uM | 24h | NA | Fluorescence spectroscopy | Transduction | YGRKKRRQRRR |
| 487 | SP-Tatm3xCherry | A549 cells | mCherry | 24928321 | 3900 | Mean Fluorescence intensity | 13 uM | 24h | NA | Fluorescence spectroscopy | Transduction | YGRKKRRQRRRYGRKKRRQRRRYGRKKRRQRRR |
| 488 | SP-Tatm3xCherry | CHO-K1 cells | mCherry | 24928321 | 15900 | Mean Fluorescence intensity | 13 uM | 24h | NA | Fluorescence spectroscopy | Transduction | YGRKKRRQRRRYGRKKRRQRRRYGRKKRRQRRR |
| 489 | Penetratin | None | Insulin | 24973720 | 15 | Plasma insulin concentration (uU/mL) | 5 mM | 30 min | NA | NA | Absorption | RQIKIWFQNRRMKWKK |
| 490 | Penetratin | None | Insulin | 24973720 | 55 | Plasma insulin concentration (uU/mL) | 5 mM | 30 min | NA | NA | Absorption | RQIKIWFQNRRMKWKK |
| 491 | MCoTI-II | HeLa cells | Alexa488 | 24985034 | 1.0 | Normalized Mean Fluorescence intensity | 8 uM | 1h | 37ºC | Flow cytometry | Uptake | GGVCPKILKKCRRDSDCPGACICRGNGYCGSGSD |
| 492 | MCoTI-M1 | HeLa cells | Alexa488 | 24985034 | 0.95 | Normalized Mean Fluorescence intensity | 8 uM | 1h | 37ºC | Flow cytometry | Uptake | GGVCPKILKKCRRDSDCPGACICRGNGWCGSGSD |
| 493 | MCoTI-M2 | HeLa cells | Alexa488 | 24985034 | 1.08 | Normalized Mean Fluorescence intensity | 8 uM | 1h | 37ºC | Flow cytometry | Uptake | GGVCPKILRRCRRDSDCPGACICRGNGYCGSGSD |
| 494 | MCoTI-M3 | HeLa cells | Alexa488 | 24985034 | 0.52 | Normalized Mean Fluorescence intensity | 8 uM | 1h | 37ºC | Flow cytometry | Uptake | GGVCPKILRRCRRDSDCPGACICRGNGWCGSGSD |
| 495 | MCoTI-M4 | HeLa cells | Alexa488 | 24985034 | 1.65 | Normalized Mean Fluorescence intensity | 8 uM | 1h | 37ºC | Flow cytometry | Uptake | GGVCPKILRRCRRDSDCPGACICRGNGYCGSGSR |
| 496 | MCoTI-M5 | HeLa cells | Alexa488 | 24985034 | 1.73 | Normalized Mean Fluorescence intensity | 8 uM | 1h | 37ºC | Flow cytometry | Uptake | GGVCPRILRRCRRDSDCPGACICRGNGYCGSGSK |
| 497 | MCoTI-M6 | HeLa cells | Alexa488 | 24985034 | 1.95 | Normalized Mean Fluorescence intensity | 8 uM | 1h | 37ºC | Flow cytometry | Uptake | GGVCPKILKKCRRDSDCPGACICRGNGYCGSGSD |
| 498 | SFTI-1 | HeLa cells | Alexa488 | 24985034 | 1.00 | Normalized Mean Fluorescence intensity | 16 uM | 1h | 37ºC | Flow cytometry | Uptake | GRCTKSIPPICFPD |
| 499 | D-SFTI-1 | HeLa cells | Alexa488 | 24985034 | 1.17 | Normalized Mean Fluorescence intensity | 16 uM | 1h | 37ºC | Flow cytometry | Uptake | grctksippicfpd |
| 500 | SFTI-M1 | HeLa cells | Alexa488 | 24985034 | 1.04 | Normalized Mean Fluorescence intensity | 16 uM | 1h | 37ºC | Flow cytometry | Uptake | GACTKSIPPICFPD |
| 501 | SFTI-M2 | HeLa cells | Alexa488 | 24985034 | 0.86 | Normalized Mean Fluorescence intensity | 16 uM | 1h | 37ºC | Flow cytometry | Uptake | GRCTKSIPPICFPA |
| 502 | SFTI-M3 | HeLa cells | Alexa488 | 24985034 | 1.13 | Normalized Mean Fluorescence intensity | 16 uM | 1h | 37ºC | Flow cytometry | Uptake | GRCTKSIPPICWPD |
| 503 | SFTI-M4 | HeLa cells | Alexa488 | 24985034 | 1.00 | Normalized Mean Fluorescence intensity | 16 uM | 1h | 37ºC | Flow cytometry | Uptake | GRCTKSIPPICWPK |
| 504 | SFTI-M5 | HeLa cells | Alexa488 | 24985034 | 1.26 | Normalized Mean Fluorescence intensity | 16 uM | 1h | 37ºC | Flow cytometry | Uptake | GRCTRSIPPKCWPD |
| 505 | SFTI-M6 | HeLa cells | Alexa488 | 24985034 | 1.13 | Normalized Mean Fluorescence intensity | 16 uM | 1h | 37ºC | Flow cytometry | Uptake | GRXTKSIPPIXFPD |
| 506 | SFTI-M7 | HeLa cells | Alexa488 | 24985034 | 0.82 | Normalized Mean Fluorescence intensity | 16 uM | 1h | 37ºC | Flow cytometry | Uptake | GRXTKSIPPIXFPD |
| 507 | TAT | HeLa cells | Alexa488 | 24985034 | 3.0 / 6.0 | Mean Fluorescence intensity | 8 uM MCoTI-II / 16 uM SFTI-1 | 1h | 37ºC | Flow cytometry | Uptake | YGRKKRRQRRRPPQG |
| 508 | VIP-TAT | Neuro2a cells | FITC | 25086267 | 1.81 ± 0.34 | % Brain uptake efficiency (% of total peptide i. p. injection of VIP-TAT) | 100 nmol/kg | NA | NA | Fluorescence spectroscopy | Uptake | HSDAVFTDNYTALRKQMAVKKYLNSILNYGRKKRRQRRR |
| 509 | Cys(BSH)-Arg11-NH2 | U87 cells | BSH | 24452095 | 391.4 | ng^10B/10^6 cells Boron concentration | 10 uM BSH-11R | 2h | NA | Immunocytochemistry | Uptake | RRRRRRRRRRR |
| 510 | Cys(BSH)-Lys[Cys(BSH)-]Arg11-NH2 | U87 cells | BSH | 24452095 | 391.4 | ng^10B/10^6 cells Boron concentration | 10 uM BSH-11R | 2h | NA | Immunocytochemistry | Uptake | RRRRRRRRRRR |
| 511 | [Cys(BSH)]4-(Lys)3-Arg11-NH2 | U87 cells | BSH | 24452095 | 588.8 | ng^10B/10^6 cells Boron concentration | 10 uM BSH-11R | 2h | NA | Immunocytochemistry | Uptake | RRRRRRRRRRR |
| 512 | Cys(BSH)-TAT | U87 cells | BSH | 24452095 | 150 | ng^10B/10^6 cells | 10 uM BSH-11R (Boron concentration) | 12h | NA | Immunocytochemistry | Uptake | GRKKRRQRRR |
| 513 | Cys(BSH)-R11 | U87 cells | BSH | 24452095 | 219.4 | ng^10B/10^6 cells Boron concentration | 10 uM BSH-11R | 2h | NA | Immunocytochemistry | Uptake | RRRRRRRRRRR |
| 514 | Peptide I | CHO-K1 cells | Carboxyfluorescein | 25096299 | 64 | Mean Fluorescence intensity | 10 uM | 4h | 37ºC | Flow cytometry | Uptake | RXRRXRRXRRXR |
| 515 | Peptide II | CHO-K1 cells | Carboxyfluorescein | 25096299 | 71 | Mean Fluorescence intensity | 10 uM | 4h | 37ºC | Flow cytometry | Uptake | RXRRXRRXRRXR |
| 516 | Peptide III | CHO-K1 cells | Carboxyfluorescein | 25096299 | 85 | Mean Fluorescence intensity | 10 uM | 4h | 37ºC | Flow cytometry | Uptake | RXRRXRRXRRXR |
| 517 | Peptide IV | CHO-K1 cells | Carboxyfluorescein | 25096299 | 75 | Mean Fluorescence intensity | 10 uM | 4h | 37ºC | Flow cytometry | Uptake | RXRRXRRXRRXR |
| 518 | Peptide V | CHO-K1 cells | Carboxyfluorescein | 25096299 | 31 | Mean Fluorescence intensity | 10 uM | 4h | 37ºC | Flow cytometry | Uptake | RXRRXRRXRRXR |
| 519 | MAP | Rat basophilic leukemia RBL-2H3 cells | Fluorescein | 25016968 | 6000 | Fluorescence intensity | 1 uM | 30 min | NA | Flow cytometry | Uptake | KLALKLALKALKAALKLA |
| 520 | pAntp | Rat basophilic leukemia RBL-2H3 cells | Fluorescein | 25016968 | 3300 | Fluorescence intensity | 1 uM | 30 min | NA | Flow cytometry | Uptake | RQIKIWFQNRRMKWKK |
| 521 | Arg9 | Rat basophilic leukemia RBL-2H3 cells | Fluorescein | 25016968 | 7500 | Fluorescence intensity | 1 uM | 30 min | NA | Flow cytometry | Uptake | RRRRRRRRR |
| 522 | R8-lipo | C6 cells | CFPE-labeled liposomes | 24651033 | 100 | Mean Fluorescence intensity | 1.5 ug/mL lipossomes | 4h | 37ºC | Flow cytometry | Uptake | RRRRRRRR |
| 523 | R8-lipo | bEnd.3 cells | CFPE-labeled liposomes | 24651033 | 120 | Mean Fluorescence intensity | 1.5 ug/mL lipossomes | 4h | 37ºC | Flow cytometry | Uptake | RRRRRRRR |
| 524 | R8-lipo | HeLa cells | CFPE-labeled liposomes | 24651033 | 11 | Mean Fluorescence intensity | 1.5 ug/mL lipossomes | 4h | 37ºC | Flow cytometry | Uptake | RRRRRRRR |
| 525 | TAT-BID | PC3 cells | BID | 25326334 | 70.0 | Cellular uptake (%) | 40 ug/ml | 120 min | NA | Western blot | NA | YGRKKRRQRRR |
| 526 | TAT-BID | LNCaP | BID | 25326334 | 100.0 | Cellular uptake (%) | 30 ug/ml | 120 min | NA | Western blot | NA | YGRKKRRQRRR |
| 527 | TAT-BID | A549 cells | BID | 25326334 | 60.0 | Cellular uptake (%) | 40 ug/ml | 120 min | NA | Western blot | NA | YGRKKRRQRRR |
| 528 | TAT-BID | HeLa cells | BID | 25326334 | 20.0 | Cellular uptake (%) | 40 ug/ml | 120 min | NA | Western blot | NA | YGRKKRRQRRR |
| 529 | TAT-lyophiliosomes | HeLa cells | Lyophiliosomes and FITC labelled | 25369131 | 86±3 | % Positive cells | 25 µg/ml | 1h | NA | Flow cytometry | Internalization | YGRKKRRQRRR |
| 530 | TAT-lyophiliosomes | Ovcar-3 cells | Lyophiliosomes and FITC labelled | 25369131 | 97±3 | % Positive cells | 25 µg/ml | 1h | NA | Flow cytometry | Internalization | YGRKKRRQRRR |
| 531 | TAT-lyophiliosomes | Caco-2 cells | Lyophiliosomes and FITC labelled | 25369131 | 87±3 | % Positive cells | 25 µg/ml | 1h | NA | Flow cytometry | Internalization | YGRKKRRQRRR |
| 532 | TAT-lyophiliosomes | SK-OV-3 cells | Lyophiliosomes and FITC labelled | 25369131 | 95±10 | % Positive cells | 25 µg/ml | 1h | NA | Flow cytometry | Internalization | YGRKKRRQRRR |
| 533 | KST | K562 cells | Avidin-FITC | 25387797 | 26 | Fluorescence intensity | 5 uM | 18h | 37ºC | Flow cytometry | Uptake | KSTGKANKITITNDKGRLSK |
| 534 | TP-biot1 | HT29 cells | Streptavidin conjugated with FITC | 25511292 | 400 | Fluorescence intensity | 4 uM CPP | 2h | 25ºC | Flow cytometry | Uptake | GWTLNSAGYLLGKINLKALAALAKKIL |
| 535 | TP-biot1 | HCT116 cells | Streptavidin conjugated with FITC | 25511292 | 220 | Fluorescence intensity | 4 uM CPP | 2h | 25ºC | Flow cytometry | Uptake | GWTLNSAGYLLGKINLKALAALAKKIL |
| 536 | TP-biot13 | HT29 cells | Streptavidin conjugated with FITC | 25511292 | 80 | Fluorescence intensity | 4 uM CPP | 2h | 25ºC | Flow cytometry | Uptake | GWTLNSAGYLLGKINLKALAALAKKIL |
| 537 | TP-biot13 | HCT116 cells | Streptavidin conjugated with FITC | 25511292 | 90 | Fluorescence intensity | 4 uM CPP | 2h | 25ºC | Flow cytometry | Uptake | GWTLNSAGYLLGKINLKALAALAKKIL |
| 538 | TP10-biot1 | HT29 cells | Streptavidin conjugated with FITC | 25511292 | 50 | Fluorescence intensity | 4 uM CPP | 2h | 25ºC | Flow cytometry | Uptake | AGYLLGKINLKALAALAKKIL |
| 539 | TP10-biot1 | HCT116 cells | Streptavidin conjugated with FITC | 25511292 | 150 | Fluorescence intensity | 4 uM CPP | 2h | 25ºC | Flow cytometry | Uptake | AGYLLGKINLKALAALAKKIL |
| 540 | cTAT-GFP | HeLa cells | eGFP | 25521313 | 80.0 | Cellular uptake (%) | 150 uM | 60 min | 37ºC | CLSM | Uptake | rRrGrKkRr |
| 541 | TAT-GFP | HeLa cells | eGFP | 25521313 | 1.0 | Cellular uptake (%) | 150 uM | 60 min | 37ºC | CLSM | Uptake | rRrGrKkRr |
| 542 | V1 | Jurkat cells | FITC labelled peptide | 25524829 | 931 | Mean Fluorescence intensity | 10 uM | 10 min | 37ºC | Flow cytometry | Uptake | RRGRRG |
| 543 | V2 | Jurkat cells | FITC labelled peptide | 25524829 | 2750 | Mean Fluorescence intensity | 10 uM | 10 min | 37ºC | Flow cytometry | Uptake | RRRRRR |
| 544 | V2R | Jurkat cells | FITC labelled peptide | 25524829 | 0 | Mean Fluorescence intensity | 10 uM | 10 min | 37ºC | Flow cytometry | Uptake | RRRRRR |
| 545 | RVG-9LR | Neuro2a cells | siRNA | 25544044 | 1527±121 | Mean Fluorescence intensity | Final Concentration between 1/5 uM | 24h | NA | Flow cytometry | Transfection | RRRRRRRRR |
| 546 | RVG-9LR | Jurkat cells | siRNA | 25544044 | 20.97±0.99 | Mean Fluorescence intensity | Final Concentration between 1/5 uM | NA | NA | Flow cytometry | Transfection | RRRRRRRRR |
| 547 | RVG-9DR | Neuro2a cells | siRNA | 25544044 | 627±124 | Mean Fluorescence intensity | Final Concentration between 1/5 uM | 24h | NA | Flow cytometry | Transfection | rrrrrrrrr |
| 548 | RVG-9DR | Jurkat cells | siRNA | 25544044 | 18.60±0.82 | Mean Fluorescence intensity | Final Concentration between 1/5 uM | NA | NA | Flow cytometry | Transfection | rrrrrrrrr |
| 549 | R8-GALA-liposome | HeLa cells | Liposome | 25546552 | 68 | Geo Mean Fluorescence intensity | NA | 1 h | NA | Flow cytometry | Uptake | RRRRRRRR |
| 550 | R8-liposome | HeLa cells | Liposome | 25546552 | 94 | Geo Mean Fluorescence intensity | NA | 1h | NA | Flow cytometry | Uptake | RRRRRRRR |
| 551 | 5-FAM-H3R8 | MCF7 cells | Carboxyfluorescein | 25547808 | 24.67 | Geo Mean Fluorescence intensity | 1 uM | 4h | NA | Flow cytometry | Uptake | HHHRRRRRRRR |
| 552 | CS-Lin-Pen | HEK293 cells | FITC labeled CS-Lin | 24083483 | 85 | % Transfection | NA | 4h | 37ºC | Flow cytometry | Transfection | RQIKIWFQNRRMKWKKGG |
| 553 | CS-Lin-Pen | CHO cells | FITC labeled CS-Lin | 24083483 | 60 | % Transfection | NA | 4h | 37ºC | Flow cytometry | Transfection | RQIKIWFQNRRMKWKKGG |
| 554 | CS-Lin-Pen | Human cervical adenocarcinoma | FITC labeled CS-Lin | 24083483 | 55 | % Transfection | NA | 4h | 37ºC | Flow cytometry | Transfection | RQIKIWFQNRRMKWKKGG |
| 555 | Bac-ELP-H1 | D54 cells | Rhodamine labeled ELP | 23372821 | 50 | ug CPP-ELP / g tissue (C6) | NA | 4h | NA | Fluorescent Microscopy | Uptake | MRRIRPRPPRLPRPRPRPLPFPRPGGCYPG |
| 556 | SynB1-ELP-H1 | D54 cells | Rhodamine labeled ELP | 23372821 | 92 | ug CPP-ELP / g tissue (C6) | NA | 4h | NA | Fluorescent Microscopy | Uptake | RGGRLSYSRRRFSTSTGRA |
| 557 | I-TYR-L-Mca | F98 glioma cell culture | Radiolabelled Iodine (125I) | 24667409 | 20 | Intracellular concenctration (uM) | 10000 nM | 2h | 37ºC | Gamma-well counter | Uptake | YGDCLPHLKLCKENKDCCSKKCKRRGTNIEKRCR |
| 558 | PC-CC9/miRNA | Panc-1 | miRNA | 23298779 | 78.08 | Cellular uptake (%) | 0.15 uM | 2h | NA | Flow cytometry | Uptake | CRGDKGPDC |
| 559 | PC-CC9/miRNA | 293T cells | miRNA | 23298779 | 51.07 | Cellular uptake (%) | 0.15 uM | 2h | NA | Flow cytometry | Uptake | CRGDKGPDC |
| 560 | Tm3+-DOTA-CAT | SN56 cells | MRI probe [DOTA-caged metal ion (Tmü?)] | 23281285 | 19.0 ± 2.0 | % Positive cells | 5 uM | 30 min | 37ºC | CLSM | Uptake | GRKKRRQRRR |
| 561 | TAT-EGFP | The mouse macrophage J774 A.1 cells | eGFP | 24746937 | 79.2 | % Positive cells | 10 umol/L | 1h | 37ºC | Flow cytometry | Uptake | YGRKKRRQRRR |
| 562 | LMWP-EGFP | The mouse macrophage J774 A.1 cells | eGFP | 24746937 | 98.8 | % Positive cells | 10 umol/L | 1h | 37ºC | Flow cytometry | Uptake | GSVSRRRRRRGGRRRR |
| 563 | R8-lip | Bone marrow dendritic cells | Liposome | 24901376 | 10.7 | Fluorescence intensity | 40 uM | 2h | 37ºC | Flow cytometry | Uptake | RRRRRRRR |
| 564 | fTAT | HeLa cells | TMR | 24930129 | 1300 | Normalized Mean Fluorescence intensity | 1 uM | 1h | NA | Flow cytometry | Uptake | CKYGRKKRRQRRR |
| 565 | KW | MEF cells | Trehalose | 24583082 | 86 | % Positive cells | 100 uM | 4h | 37ºC | Flow cytometry | Uptake | KRKRWHW |
| 566 | LMWP-TAZ | Cultured Human Dental Pulp Stem Cells (hDPSCs) | TAZ | 21990606 | 100.0 | % Positive cells | 500 nM | 30 min | NA | Flow cytometry | Transduction | VSRRRRRRGGRRRR |
| 567 | pVEC | CHO-K1 cells | Plasmid DNA | 21996011 | 14 | Mean Fluorescence intensity | Charge ratio = 10 | 4h | 37ºC | Flow cytometry | Uptake | LLIILRRRIRKQAHAHSK |
| 568 | S6KR | CHO-K1 cells | Plasmid DNA | 21996011 | 15 | Mean Fluorescence intensity / % FITC Positive cells | Charge ratio = 10 | 4h | 37ºC | Flow cytometry | Uptake | LLHILRRSIRKQAHAIRK |
| 569 | S9R | CHO-K1 cells | Plasmid DNA | 21996011 | 58 | Mean Fluorescence intensity | Charge ratio = 10 | 4h | 37ºC | Flow cytometry | Uptake | LLRILRRSIRRARRAIRR |
| 570 | S6R | CHO-K1 cells | Plasmid DNA | 21996011 | 18 | Mean Fluorescence intensity | Charge ratio = 10 | 4h | 37ºC | Flow cytometry | Uptake | LLHILRRSIRRQAHAIRR |
| 571 | CPPK | HEK | FITC | 22076844 | 900 | Fold change in average fluorescence | 10 nM | 3 h | 37°C | Confocal laser scanning system (clss) | Uptake | MAMPGEPRRANVMAHKLEPASLQLR NSCA |
| 572 | CPPK | HeLa cells | FITC | 22076844 | 930 | Fold change in average fluorescence | 10 nM | 3 h | 37°C | Confocal laser scanning system (clss) | Uptake | MAMPGEPRRANVMAHKLEPASLQLR NSCA |
| 573 | CPPL | HEK | FITC | 22076844 | 1500 | Fold change in average fluorescence | 10 nM | 3 h | 37°C | Confocal laser scanning system (clss) | Uptake | MAPQRDTVGGRTTPPSWGPAKAQLRNSCA |
| 574 | CPPL | HeLa cells | FITC | 22076844 | 2500 | Fold change in average fluorescence | 10 nM | 3 h | 37°C | Confocal laser scanning system (clss) | Uptake | MAPQRDTVGGRTTPPSWGPAKAQLRNSCA |
| 575 | Tat | ARPE-19 cells | Fluorescein | 22100438 | 1.00 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRRQRRRPPQ |
| 576 | Tat | CHO cells | Fluorescein | 22100438 | 1.00 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRRQRRRPPQ |
| 577 | Tat | CHO cells | Fluorescein | 22100438 | 1.00 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRRQRRRPPQ |
| 578 | II | ARPE-19 cells | Fluorescein | 22100438 | 0.84 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRWWRQRRRPPQ |
| 579 | II | CHO cells | Fluorescein | 22100438 | 0.92 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRWWRQRRRPPQ |
| 580 | II | CHO cells | Fluorescein | 22100438 | 1.14 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRWWRQRRRPPQ |
| 581 | III | ARPE-19 cells | Fluorescein | 22100438 | 0.9 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRRQRRWWRPPQ |
| 582 | III | CHO cells | Fluorescein | 22100438 | 1.00 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRRQRRWWRPPQ |
| 583 | III | CHO cells | Fluorescein | 22100438 | 1.04 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRRQRRWWRPPQ |
| 584 | IV | ARPE-19 cells | Fluorescein | 22100438 | 0.96 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRRQRWWRRPPQ |
| 585 | IV | CHO cells | Fluorescein | 22100438 | 1.14 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRRQRWWRRPPQ |
| 586 | IV | CHO cells | Fluorescein | 22100438 | 1.07 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRRQRWWRRPPQ |
| 587 | V | ARPE-19 cells | Fluorescein | 22100438 | 0.82 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRWWRQRWWRWWRPPQ |
| 588 | V | CHO cells | Fluorescein | 22100438 | 0.84 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRWWRQRWWRWWRPPQ |
| 589 | V | CHO cells | Fluorescein | 22100438 | 0.98 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRWWRQRWWRWWRPPQ |
| 590 | VI | ARPE-19 cells | Fluorescein | 22100438 | 1.02 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRAARQRRRPPQ |
| 591 | VI | CHO cells | Fluorescein | 22100438 | 0.92 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRAARQRRRPPQ |
| 592 | VI | CHO cells | Fluorescein | 22100438 | 0.92 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRAARQRRRPPQ |
| 593 | VII | ARPE-19 cells | Fluorescein | 22100438 | 0.92 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRRQRRAARPPQ |
| 594 | VII | CHO cells | Fluorescein | 22100438 | 0.90 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRRQRRAARPPQ |
| 595 | VII | CHO cells | Fluorescein | 22100438 | 0.88 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRRQRRAARPPQ |
| 596 | VIII | ARPE-19 cells | Fluorescein | 22100438 | 0.88 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRRQRAARRPPQ |
| 597 | VIII | CHO cells | Fluorescein | 22100438 | 0.84 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRRQRAARRPPQ |
| 598 | VIII | CHO cells | Fluorescein | 22100438 | 0.83 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRRQRAARRPPQ |
| 599 | IX | ARPE-19 cells | Fluorescein | 22100438 | 0.84 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRAARQRAARAARPPQ |
| 600 | IX | CHO cells | Fluorescein | 22100438 | 0.76 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRAARQRAARAARPPQ |
| 601 | IX | CHO cells | Fluorescein | 22100438 | 0.84 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRAARQRAARAARPPQ |
| 602 | X | ARPE-19 cells | Fluorescein | 22100438 | 0.95 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRLLRQRRRPPQ |
| 603 | X | CHO cells | Fluorescein | 22100438 | 0.84 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRLLRQRRRPPQ |
| 604 | X | CHO cells | Fluorescein | 22100438 | 0.77 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRLLRQRRRPPQ |
| 605 | XI | ARPE-19 cells | Fluorescein | 22100438 | 0.84 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRRQRRLLRPPQ |
| 606 | XI | CHO cells | Fluorescein | 22100438 | 0.84 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRRQRRLLRPPQ |
| 607 | XI | CHO cells | Fluorescein | 22100438 | 0.73 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRRQRRLLRPPQ |
| 608 | XII | ARPE-19 cells | Fluorescein | 22100438 | 0.89 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRRQRLLRRPPQ |
| 609 | XII | CHO cells | Fluorescein | 22100438 | 0.88 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRRQRLLRRPPQ |
| 610 | XII | CHO cells | Fluorescein | 22100438 | 0.76 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRRQRLLRRPPQ |
| 611 | XIII | ARPE-19 cells | Fluorescein | 22100438 | 1.18 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRLLRQRLLRLLRPPQ |
| 612 | XIII | CHO cells | Fluorescein | 22100438 | 1.34 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRLLRQRLLRLLRPPQ |
| 613 | XIII | CHO cells | Fluorescein | 22100438 | 0.95 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRLLRQRLLRLLRPPQ |
| 614 | XIV | ARPE-19 cells | Fluorescein | 22100438 | 0.88 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRRQRR-Ahx-RPPQ |
| 615 | XIV | CHO cells | Fluorescein | 22100438 | 0.84 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRRQRR-Ahx-RPPQ |
| 616 | XIV | CHO cells | Fluorescein | 22100438 | 0.76 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRRQRR-Ahx-RPPQ |
| 617 | XV | ARPE-19 cells | Fluorescein | 22100438 | 0.97 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKR-Ahx-RQRRRPPQ |
| 618 | XV | CHO cells | Fluorescein | 22100438 | 0.88 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKR-Ahx-RQRRRPPQ |
| 619 | XV | CHO cells | Fluorescein | 22100438 | 0.76 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKR-Ahx-RQRRRPPQ |
| 620 | XVI | ARPE-19 cells | Fluorescein | 22100438 | 1.06 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRRQR-Ahx-RRPPQ |
| 621 | XVI | CHO cells | Fluorescein | 22100438 | 0.90 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRRQR-Ahx-RRPPQ |
| 622 | XVI | CHO cells | Fluorescein | 22100438 | 0.85 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRRQR-Ahx-RRPPQ |
| 623 | XVII | ARPE-19 cells | Fluorescein | 22100438 | 0.90 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKR-Ahx-RQR-Ahx-R-ahx-RPPQ |
| 624 | XVII | CHO cells | Fluorescein | 22100438 | 0.74 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKR-Ahx-RQR-Ahx-R-ahx-RPPQ |
| 625 | XVII | CHO cells | Fluorescein | 22100438 | 0.78 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKR-Ahx-RQR-Ahx-R-ahx-RPPQ |
| 626 | TAM-MP | U373 MG cells | TAMRA | 22148546 | 15.82 | Mean Fluorescence intensity | 5 uM | 1h | 37ºC | Fluorescence spectroscopy | Translocation | INLKALAALAKKIL |
| 627 | TAM-iMP | U373 MG cells | TAMRA | 22148546 | 100.0 | Mean Fluorescence intensity | 5 uM | 1h | 37ºC | Fluorescence spectroscopy | Translocation | inlkalaalakkil |
| 628 | TAM-rMP | U373 MG cells | TAMRA | 22148546 | 9.762 | Mean Fluorescence intensity | 5 uM | 1h | 37ºC | Fluorescence spectroscopy | Translocation | LIKKALAALAKLNI |
| 629 | TAM-riMP | U373 MG cells | TAMRA | 22148546 | 7.990 | Mean Fluorescence intensity | 5 uM | 1h | 37ºC | Fluorescence spectroscopy | Translocation | likkalaalaklni |
| 630 | TAM-MitP | U373 MG cells | TAMRA | 22148546 | 82.21 | Mean Fluorescence intensity | 5 uM | 1h | 37ºC | Fluorescence spectroscopy | Translocation | INLKKLAKL(Aib)KKIL |
| 631 | TAM-iMitP | U373 MG cells | TAMRA | 22148546 | 63.06 | Mean Fluorescence intensity | 5 uM | 1h | 37ºC | Fluorescence spectroscopy | Translocation | inlkklakl(Aib)kkil |
| 632 | TAM-rMitP | U373 MG cells | TAMRA | 22148546 | 14.75 | Mean Fluorescence intensity | 5 uM | 1h | 37ºC | Fluorescence spectroscopy | Translocation | LIKK(Aib)LKALKKLNI |
| 633 | TAM-riMitP | U373 MG cells | TAMRA | 22148546 | 23.23 | Mean Fluorescence intensity | 5 uM | 1h | 37ºC | Fluorescence spectroscopy | Translocation | likk(Aib)lkalkklni |
| 634 | Cyt c-ss-MAP | HEK293 cells | Cyt C protein | 22225540 | 1105.2 | ng molecule / mg cell protein | 10 ug/ml | 1h | 37ºC | Fluorescence spectroscopy | Uptake | KLALKLALKALKAALKLA |
| 635 | Cyt c-ss-MAP | HeLa cells | Cyt C protein | 22225540 | 1575 | ng molecule / mg cell protein | 10 ug/ml | 1h | 37ºC | Fluorescence spectroscopy | Uptake | KLALKLALKALKAALKLA |
| 636 | Cyt c-ss-R8 | HEK293 cells | Cyt C protein | 22225540 | 100 | ng molecule / mg cell protein | 10 ug/ml | 1h | 37ºC | Fluorescence spectroscopy | Uptake | RRRRRRRR |
| 637 | Cyt c-ss-R8 | HeLa cells | Cyt C protein | 22225540 | 262.5 | ng molecule / mg cell protein | 10 ug/ml | 1h | 37ºC | Fluorescence spectroscopy | Uptake | RRRRRRRR |
| 638 | PenArg | HEK293T cells | Plasmid DNA | 22281502 | 5.0 | Cellular uptake (%) | charge ratio = 2 | 2h | NA | Flow cytometry | Transfection | RQIRIWFQNRRMRWRR |
| 639 | PenArg-Cys | HEK293T cells | Plasmid DNA | 22281502 | 38.0 | Cellular uptake (%) | charge ratio = 2 | 2h | NA | Flow cytometry | Transfection | RQIRIWFQNRRMRWRRC |
| 640 | EB1 | HEK293T cells | Plasmid DNA | 22281502 | 48.0 | Cellular uptake (%) | charge ratio = 2 | 2h | NA | Flow cytometry | Transfection | LIRLWSHLIHIWFQNRRLKWKKK |
| 641 | EB1-Cys | HEK293T cells | Plasmid DNA | 22281502 | 49.0 | Cellular uptake (%) | charge ratio = 2 | 2h | NA | Flow cytometry | Transfection | LIRLWSHLIHIWFQNRRLKWKKKC |
| 642 | R8 | NA | Alexa600 | 22285548 | 378.0 | Relative fluorescence (%) | 3 nmol | 24h | NA | CLSM | Tumor accumulation | RRRRRRRRGC |
| 643 | r12 | NA | Alexa600 | 22285548 | 424.0 | Relative fluorescence (%) | 3 nmol | 24h | NA | CLSM | Tumor accumulation | rrrrrrrrrrrrGC |
| 644 | RV24 | T98G cell | b-galactosidase and eGFP | 22326265 | 82.46 | % Positive cells | Molar ratio 50 (v/w) or (w/w) eGFP | 4h | NA | Flow cytometry | Transduction | RRRRRRRRRGPGVTWTPQAWFQWV |
| 645 | RV24 | HepG2 cells | b-galactosidase and eGFP | 22326265 | 78.85 | % Positive cells | Molar ratio 50 (v/w) or (w/w) eGFP | 4h | NA | Flow cytometry | Transduction | RRRRRRRRRGPGVTWTPQAWFQWV |
| 646 | RV24 | HeLa cells | b-galactosidase and eGFP | 22326265 | 74.79 | % Positive cells | Molar ratio 50 (v/w) or (w/w) eGFP | 4h | NA | Flow cytometry | Transduction | RRRRRRRRRGPGVTWTPQAWFQWV |
| 647 | GST-HE-MAP | HeLa cells | GST | 22326404 | 32 | ng/ Cell monolayer | 5 ug/ml | 1h | 37ºC | Gamma-well counter | Internalization | HEHEHEHEHEHEHEHEHEHEGGGGGKLALKLALKALKAALKLA |
| 648 | TMR-R3 | U251 cells | TMR | 22465335 | 54.54 | Relative fluorescence | 1 uM | 30 min | NA | Fluorescence spectroscopy | Transduction | RRR |
| 649 | PasR8 (Alexa) | HeLa cells | Alexa | 22486588 | 61 | Mean Fluorescence intensity | 1 uM | 15 min | 37ºC | Flow cytometry | Uptake | FFLIPKGRRRRRRRRGC |
| 650 | LILIR8 (Alexa) | HeLa cells | Alexa | 22486588 | 18.5 | Mean Fluorescence intensity | 1 uM | 15 min | 37ºC | Flow cytometry | Uptake | LILIGRRRRRRRRGC |
| 651 | F2R8 (Alexa) | HeLa cells | Alexa | 22486588 | 22 | Mean Fluorescence intensity | 1 uM | 15 min | 37ºC | Flow cytometry | Uptake | FFGRRRRRRRGC |
| 652 | F4R8 (Alexa) | HeLa cells | Alexa | 22486588 | 100 | Mean Fluorescence intensity | 1 uM | 15 min | 37ºC | Flow cytometry | Uptake | FFFFGRRRRRRRRGC |
| 653 | (r-ahx-r)4_carbamate_CF (II) | CHO-K1 cells | Plasmid DNA | 22509923 | 362.5 | Mean Fluorescence intensity | 5 uM | 1h | 37ºC | Flow cytometry | Uptake | rXrrXrrXrrXr |
| 654 | r8_carbamate_CF15 (VI) | CHO-K1 cells | Plasmid DNA | 22509923 | 300 | Mean Fluorescence intensity | 5 uM | 1h | 37ºC | Flow cytometry | Uptake | rrrrrrrr |
| 655 | Tat | Caco-2 cells | Nanoparticle | 22531849 | 3.5 | Relative Median Fluorescence | 1.0 mg/ml | 4h | NA | Flow cytometry | Uptake | GCGGGYGRKKRRQRRR |
| 656 | TAT-NBD | MDA-MB-231 cells | TMTP1 | 22580115 | 15 | Mean Fluorescence intensity | 1 umol | 30 min | 37ºC | Fluorescent Microscopy | Association | YGRKKRRQRRRGTALDWSWLQTE |
| 657 | TAT-NBD | MCF7 cells | TMTP1 | 22580115 | 13 | Mean Fluorescence intensity | 1 umol | 30 min | 37ºC | Fluorescent Microscopy | Association | YGRKKRRQRRRGTALDWSWLQTE |
| 658 | TMTP1-TAT-NBD | MDA-MB-231 cells | TMTP1 | 22580115 | 28.75 | Mean Fluorescence intensity | 1 umol | 30 min | 37ºC | Fluorescent Microscopy | Association | CGNVVRQGC-G-YGRK-KRRQRRR-G-TALDWSWLQTE |
| 659 | TMTP1-TAT-NBD | MCF7 cells | TMTP1 | 22580115 | 2.25 | Mean Fluorescence intensity | 1 umol | 30 min | 37ºC | Fluorescent Microscopy | Association | CGNVVRQGC-G-YGRK-KRRQRRR-G-TALDWSWLQTE |
| 660 | SR9 | A549 cells | Plasmid DNA | 22669044 | 3.9 | Fold of transfection efficiency | N/P ratio = 3 | 10 min | 37ºC | Flow cytometry | Transfection | SRRRRRRRRR |
| 661 | PR9 | A549 cells | Plasmid DNA | 22669044 | 5.6 | Fold of transfection efficiency | N/P ratio = 3 | 10 min | 37ºC | Flow cytometry | Transfection | FFLIPKGRRRRRRRRR |
| 662 | CADY-1 | HeLa cells | Doxorubicin | 22688249 | 63 | % Positive cells | 10 uM | 1h | NA | HPCL-analysis | Penetration efficiencies | GLWWKAWWKAWWKSLWWRKRKRKA |
| 663 | RWR | CHO-K1 cells | Carboxyfluorescein | 22712882 | 750 | Mean Fluorescence intensity | 10 uM | 1h | 37ºC | Flow cytometry | Uptake | RRRRWWWWRRRR |
| 664 | RW MIX | CHO-K1 cells | Carboxyfluorescein | 22712882 | 1400 | Mean Fluorescence intensity | 10 uM | 1h | 37ºC | Flow cytometry | Uptake | RWRRWRRWRRWR |
| 665 | 1 (TAT) | NHDF | FITC | 22805558 | 1.89 | Relative fluorescence | 10 uM | 3h | NA | Flow cytometry | Uptake | YGRKKRPQRRR |
| 666 | CPP2 | HeLa cells | FITC | 22805558 | 4 | Relative fluorescence | 10 uM | 3h | NA | Fluorescent Microscopy | Penetration efficiencies | DSLKSYWYLQKFSWR |
| 667 | CPP2 | Lovo | FITC | 22805558 | 39 | Relative fluorescence | 10 uM | 3h | NA | Fluorescent Microscopy | Penetration efficiencies | DSLKSYWYLQKFSWR |
| 668 | CPP2 | A549 cells | FITC | 22805558 | 3 | Relative fluorescence | 10 uM | 3h | NA | Fluorescent Microscopy | Penetration efficiencies | DSLKSYWYLQKFSWR |
| 669 | CPP2 | MCF7 cells | FITC | 22805558 | 1 | Relative fluorescence | 10 uM | 3h | NA | Fluorescent Microscopy | Penetration efficiencies | DSLKSYWYLQKFSWR |
| 670 | CPP2 | HepG2 cells | FITC | 22805558 | 5 | Relative fluorescence | 10 uM | 3h | NA | Fluorescent Microscopy | Penetration efficiencies | DSLKSYWYLQKFSWR |
| 671 | CPP2 | U2OS cells | FITC | 22805558 | 6 | Relative fluorescence | 10 uM | 3h | NA | Fluorescent Microscopy | Penetration efficiencies | DSLKSYWYLQKFSWR |
| 672 | CPP2 | K562 cells | FITC | 22805558 | 2 | Relative fluorescence | 10 uM | 3h | NA | Fluorescent Microscopy | Penetration efficiencies | DSLKSYWYLQKFSWR |
| 673 | CPP2 | NHDF | FITC | 22805558 | 0 | Relative fluorescence | 10 uM | 3h | NA | Fluorescent Microscopy | Penetration efficiencies | DSLKSYWYLQKFSWR |
| 674 | CPP44 | HeLa cells | FITC | 22805558 | 3 | Relative fluorescence | 10 uM | 3h | NA | Fluorescent Microscopy | Penetration efficiencies | KRPTMRFRYTWNPMK |
| 675 | CPP44 | Lovo | FITC | 22805558 | 2 | Relative fluorescence | 10 uM | 3h | NA | Fluorescent Microscopy | Penetration efficiencies | KRPTMRFRYTWNPMK |
| 676 | CPP44 | A549 cells | FITC | 22805558 | 1 | Relative fluorescence | 10 uM | 3h | NA | Fluorescent Microscopy | Penetration efficiencies | KRPTMRFRYTWNPMK |
| 677 | CPP44 | MCF7 cells | FITC | 22805558 | 0 | Relative fluorescence | 10 uM | 3h | NA | Fluorescent Microscopy | Penetration efficiencies | KRPTMRFRYTWNPMK |
| 678 | CPP44 | HepG2 cells | FITC | 22805558 | 40 | Relative fluorescence | 10 uM | 3h | NA | Fluorescent Microscopy | Penetration efficiencies | KRPTMRFRYTWNPMK |
| 679 | CPP44 | U2OS cells | FITC | 22805558 | 3 | Relative fluorescence | 10 uM | 3h | NA | Fluorescent Microscopy | Penetration efficiencies | KRPTMRFRYTWNPMK |
| 680 | CPP44 | K562 cells | FITC | 22805558 | 70 | Relative fluorescence | 10 uM | 3h | NA | Fluorescent Microscopy | Penetration efficiencies | KRPTMRFRYTWNPMK |
| 681 | CPP44 | NHDF | FITC | 22805558 | 0 | Relative fluorescence | 10 uM | 3h | NA | Fluorescent Microscopy | Penetration efficiencies | KRPTMRFRYTWNPMK |
| 682 | Polyguanidine comparators 1 | MCF7 cells | Carboxyfluorescein | 22828784 | 56.8 | Mean Fluorescence intensity | 8 uM | 1h | 37ºC | Flow cytometry | Uptake | RRRRRRRR |
| 683 | Polyguanidine comparators 2 | MCF7 cells | Carboxyfluorescein | 22828784 | 36 | Mean Fluorescence intensity | 8 uM | 1h | 37ºC | Flow cytometry | Uptake | Nbtg-Nbtg-Nbtg-Nbtg-Nbtg-Nbtg-Nbtg-Nbtg |
| 684 | NLys(1/3) variants 1 | MCF7 cells | Carboxyfluorescein | 22828784 | 11.2 | Mean Fluorescence intensity | 8 uM | 1h | 37ºC | Flow cytometry | Uptake | NLys-Nspe-Nspe-NLys-Nspe-Nspe-NLys-Nspe-Nspe |
| 685 | NLys(1/3) variants 2 | MCF7 cells | Carboxyfluorescein | 22828784 | 92.8 | Mean Fluorescence intensity | 8 uM | 1h | 37ºC | Flow cytometry | Uptake | NLys-Nspe-Nspe-NLys-Nspe-Nspe-NLys-Nspe-Nspe-NLys-Nspe-Nspe |
| 686 | NLys(1/3) variants 3 | MCF7 cells | Carboxyfluorescein | 22828784 | 23.2 | Mean Fluorescence intensity | 8 uM | 1h | 37ºC | Flow cytometry | Uptake | NLys-Npm-Npm-NLys-Npm-Npm-NLys-Npm-Npm-NLys-Npm-Npm |
| 687 | NLys(1/3) variants 4 | MCF7 cells | Carboxyfluorescein | 22828784 | 7.2 | Mean Fluorescence intensity | 8 uM | 1h | 37ºC | Flow cytometry | Uptake | NLys-Nssb-Nssb-NLys-Nssb-Nssb-NLys-Nssb-Nssb-NLys-Nssb-Nssb |
| 688 | NLys(2/3) variants 1 | MCF7 cells | Carboxyfluorescein | 22828784 | 12 | Mean Fluorescence intensity | 8 uM | 1h | 37ºC | Flow cytometry | Uptake | NLys-NLys-Nspe-NLys-NLys-Nspe-NLys-NLys-Nspe-NLys-NLys-Nspe |
| 689 | NLys(2/3) variants 2 | MCF7 cells | Carboxyfluorescein | 22828784 | 20 | Mean Fluorescence intensity | 8 uM | 1h | 37ºC | Flow cytometry | Uptake | NLys-NLys-NLys-NLys-NLys-NLys-NLys-NLys-Nspe-Nspe-Nspe-Nspe |
| 690 | NLys(2/3) variants 3 | MCF7 cells | Carboxyfluorescein | 22828784 | 3.2 | Mean Fluorescence intensity | 8 uM | 1h | 37ºC | Flow cytometry | Uptake | NLys-NLys-NLys-NLys-NLys-NLys-NLys-NLys-NLeu-NLeu-NLeu-NLeu-Nleu |
| 691 | Guanidylated variants | MCF7 cells | Carboxyfluorescein | 22828784 | 98.4 | Mean Fluorescence intensity | 8 uM | 1h | 37ºC | Flow cytometry | Uptake | Nbtg-Nspe-Nspe-Nbtg-Nspe-Nspe-Nbtg-Nspe-Nspe-Nbtg-Nspe-Nspe |
| 692 | Guanidylated variants | MCF7 cells | Carboxyfluorescein | 22828784 | 92.8 | Mean Fluorescence intensity | 8 uM | 1h | 37ºC | Flow cytometry | Uptake | Nbtg-Nspe-Nspe-Nbtg-Nspe-Nspe-Nbtg-Nspe-Nspe-Nbtg-Nspe-Nspe |
| 693 | penetratin | MDCK-MDR cells | PEG-PLA | 22841849 | 20 | Nanoparticle uptake/cell | 100 ug/ml | 60 min | 37ºC | HCS analysis | Uptake | RQIKIWFQNRRMKWKK |
| 694 | low molecular weight protamine (LMWP) | Caco-2 cells | Insulin-PEG-LMWP | 23863452 | 0.205 | Insulin concentration | 0.5 uM | 8 hour | NA | Fluorescence spectroscopy | Absorption | VSRRRRRRGGRRRR |
| 695 | Peptide 1 | U87 cells | FITC | 25562654 | 95 | Fluorescence intensity | 10 uM | 2h | 37ºC | CLSM | Uptake | NTCTWLKYHS |
| 696 | Peptide 2 | U87 cells | FITC | 25562654 | 10 | Fluorescence intensity | 10 uM | 2h | 37ºC | CLSM | Uptake | CASGQQGLLKLC |
| 697 | Peptide 3 | U87 cells | FITC | 25562654 | 25 | Fluorescence intensity | 10 uM | 2h | 37ºC | CLSM | Uptake | YNNFAYSVFL |
| 698 | Peptide 4 | U87 cells | FITC | 25562654 | 16 | Fluorescence intensity | 10 uM | 2h | 37ºC | CLSM | Uptake | ECYPKKGQDP |
| 699 | Peptide 5 | U87 cells | FITC | 25562654 | 15 | Fluorescence intensity | 10 uM | 2h | 37ºC | CLSM | Uptake | RHVYHVLLSQ |
| 700 | Peptide 6 | U87 cells | FITC | 25562654 | 15 | Fluorescence intensity | 10 uM | 2h | 37ºC | CLSM | Uptake | HATKSQNINF |
| 701 | Peptide 7 | U87 cells | FITC | 25562654 | 10 | Fluorescence intensity | 10 uM | 2h | 37ºC | CLSM | Uptake | YRDRFAFQPH |
| 702 | Peptide 8 | U87 cells | FITC | 25562654 | 19 | Fluorescence intensity | 10 uM | 2h | 37ºC | CLSM | Uptake | IWRYSLASQQ |
| 703 | Peptide 9 | U87 cells | FITC | 25562654 | 19 | Fluorescence intensity | 10 uM | 2h | 37ºC | CLSM | Uptake | YQKQAKIMCS |
| 704 | Peptide 10 | U87 cells | FITC | 25562654 | 20 | Fluorescence intensity | 10 uM | 2h | 37ºC | CLSM | Uptake | VQLRRRWC |
| 705 | Peptide 1-C3G | U87 cells | FITC | 25562654 | 0.75 | Relative penetration efficiency | 10 uM | 2h | 37ºC | CLSM | Uptake | NTGTWLKYHS |
| 706 | Peptide 1-N? | U87 cells | FITC | 25562654 | 1.2 | Relative penetration efficiency | 10 uM | 2h | 37ºC | CLSM | Uptake | TCTWLKYHS |
| 707 | Peptide 1-S? | U87 cells | FITC | 25562654 | 1.15 | Relative penetration efficiency | 10 uM | 2h | 37ºC | CLSM | Uptake | NTCTWLKYH |
| 708 | Peptide 1-NS? | U87 cells | FITC | 25562654 | 2 | Relative penetration efficiency | 10 uM | 2h | 37ºC | CLSM | Uptake | TCTWLKYH |
| 709 | Peptide 1-NTS? | U87 cells | FITC | 25562654 | 1.3 | Relative penetration efficiency | 10 uM | 2h | 37ºC | CLSM | Uptake | CTWLKYH |
| 710 | Peptide 1-NTCS? | U87 cells | FITC | 25562654 | 0.5 | Relative penetration efficiency | 10 uM | 2h | 37ºC | CLSM | Uptake | TWLKYH |
| 711 | Peptide 1-NTHS? | U87 cells | FITC | 25562654 | 0.8 | Relative penetration efficiency | 10 uM | 2h | 37ºC | CLSM | Uptake | CTWLKY |
| 712 | P1 | HeLa cells | FITC | 25459448 | 112.5 | Mean Fluorescence (% of positive control TAT as 100 %) | 10 uM | 1h | 37ºC | Flow cytometry | Uptake | KKKKKKNKKLQQRGD |
| 713 | P2 | HeLa cells | FITC | 25459448 | 20.8 | Mean Fluorescence (% of positive control TAT as 100 %) | 10 uM | 1h | 37ºC | Flow cytometry | Uptake | RGDGPRRRPRKRRGR |
| 714 | P3 | HeLa cells | FITC | 25459448 | 166 | Mean Fluorescence (% of positive control TAT as 100 %) | 10 uM | 1h | 37ºC | Flow cytometry | Uptake | RRRQKRIVVRRRLIR |
| 715 | P4 | HeLa cells | FITC | 25459448 | 100 | Mean Fluorescence (% of positive control TAT as 100 %) | 10 uM | 1h | 37ºC | Flow cytometry | Uptake | RRVWRRYRRQRWCRR |
| 716 | P5 | HeLa cells | FITC | 25459448 | 75 | Mean Fluorescence (% of positive control TAT as 100 %) | 10 uM | 1h | 37ºC | Flow cytometry | Uptake | RRARRPRRLRPAPGR |
| 717 | P6 | HeLa cells | FITC | 25459448 | 208.3 | Mean Fluorescence (% of positive control TAT as 100 %) | 10 uM | 1h | 37ºC | Flow cytometry | Uptake | LLRARWRRRRSRRFR |
| 718 | P7 | HeLa cells | FITC | 25459448 | 83.3 | Mean Fluorescence (% of positive control TAT as 100 %) | 10 uM | 1h | 37ºC | Flow cytometry | Uptake | RGPRRQPRRHRRPRR |
| 719 | P8 | HeLa cells | FITC | 25459448 | 950 | Mean Fluorescence (% of positive control TAT as 100 %) | 10 uM | 1h | 37ºC | Flow cytometry | Uptake | RRWRRWNRFNRRRCR |
| 720 | Tat | HeLa cells | FITC | 25459448 | 100 | Mean Fluorescence (% of positive control TAT as 100 %) | 10 uM | 1h | 37ºC | Flow cytometry | Uptake | GRKKRRQRRRPPQ |
| 721 | PolyR | NA | Carboxyfluorescein | 25894337 | 70 ± 5 | % Average area uptake | 100 uM | NA | NA | Immunohistochemistry | Penetration | RRRRRRRRR |
| 722 | Antp | NA | Carboxyfluorescein | 25894337 | 0.0 | % Average area uptake | 100 uM | NA | NA | Immunohistochemistry | Penetration | RQIKIWFQNRRMKWKK |
| 723 | Tat(49-57) | NA | Carboxyfluorescein | 25894337 | 27 ±13 | % Average area uptake | 100 uM | NA | NA | Immunohistochemistry | Penetration | RKKRRQRRR |
| 724 | Trans | NA | Carboxyfluorescein | 25894337 | 70 ± 4 | % Average area uptake | 100 uM | NA | NA | Immunohistochemistry | Penetration | GWTLNSAGYLLGKINLKALAALAKKIL |
| 725 | CendRP | NA | Carboxyfluorescein | 25894337 | 0.0 | % Average area uptake | 100 uM | NA | NA | Immunohistochemistry | Penetration | RPARPAR |
| 726 | R6 | HeLa cells | FITC | 25654426 | 24 | Relative Mean Fluorescence intensity (%) | 5 mM | NA | NA | Flow cytometry | Uptake | BRRRRRR |
| 727 | R7 | HeLa cells | FITC | 25654426 | 44 | Relative Mean Fluorescence intensity (%) | 5 mM | NA | NA | Flow cytometry | Uptake | BRRRRRRR |
| 728 | R8 | HeLa cells | FITC | 25654426 | 72 | Relative Mean Fluorescence intensity (%) | 5 mM | NA | NA | Flow cytometry | Uptake | BRRRRRRRR |
| 729 | R9 | HeLa cells | FITC | 25654426 | 100 | Relative Mean Fluorescence intensity (%) | 5 mM | NA | NA | Flow cytometry | Uptake | Ahx-RRRRRRRRR |
| 730 | Cyc-R4 | HeLa cells | FITC | 25654426 | 12 | Relative Mean Fluorescence intensity (%) | 5 mM | NA | NA | Flow cytometry | Uptake | ?A-[KRRRRE] |
| 731 | Cyc-R6 | HeLa cells | FITC | 25654426 | 26 | Relative Mean Fluorescence intensity (%) | 5 mM | NA | NA | Flow cytometry | Uptake | ?A-[KRRRRRRE] |
| 732 | Cyc-R7 | HeLa cells | FITC | 25654426 | 42 | Relative Mean Fluorescence intensity (%) | 5 mM | NA | NA | Flow cytometry | Uptake | ?A-[KRRRRRRRE] |
| 733 | Cyc-R8 | HeLa cells | FITC | 25654426 | 124 | Relative Mean Fluorescence intensity (%) | 5 mM | NA | NA | Flow cytometry | Uptake | ?A-[KRRRRRRRRE] |
| 734 | Cyc-R9 | HeLa cells | FITC | 25654426 | 148 | Relative Mean Fluorescence intensity (%) | 5 mM | NA | NA | Flow cytometry | Uptake | ?A-[KRRRRRRRRRE] |
| 735 | Cyc-r7 | HeLa cells | FITC | 25654426 | 42 | Relative Mean Fluorescence intensity (%) | 5 mM | NA | NA | Flow cytometry | Uptake | ?A-[KrrrrrrrE] |
| 736 | Cyc-r8 | HeLa cells | FITC | 25654426 | 64 | Relative Mean Fluorescence intensity (%) | 5 mM | NA | NA | Flow cytometry | Uptake | ?A-[KrrrrrrrrE] |
| 737 | Cyc-r9 | HeLa cells | FITC | 25654426 | 70 | Relative Mean Fluorescence intensity (%) | 5 mM | NA | NA | Flow cytometry | Uptake | ?A-[KrrrrrrrrE] |
| 738 | Bicyc-0-R6 | HeLa cells | FITC | 25654426 | 17 | Relative Mean Fluorescence intensity (%) | 5 mM | NA | NA | Flow cytometry | Uptake | ?A-[ERRRK]-[KRRRE] |
| 739 | Bicyc-1-R6 | HeLa cells | FITC | 25654426 | 20 | Relative Mean Fluorescence intensity (%) | 5 mM | NA | NA | Flow cytometry | Uptake | ?A-[ERRRK]-?A-[KRRRE] |
| 740 | Bicyc-2-R6 | HeLa cells | FITC | 25654426 | 33 | Relative Mean Fluorescence intensity (%) | 5 mM | NA | NA | Flow cytometry | Uptake | ?A-[ERRRK]-(?A)2-[KRRRE] |
| 741 | Bicyc-3-R6 | HeLa cells | FITC | 25654426 | 30 | Relative Mean Fluorescence intensity (%) | 5 mM | NA | NA | Flow cytometry | Uptake | ?A-[ERRRK]-(?A)3-[KRRRE] |
| 742 | Cyc-R3-R4 | HeLa cells | FITC | 25654426 | 66 | Relative Mean Fluorescence intensity (%) | 5 mM | NA | NA | Flow cytometry | Uptake | ?A-RRRR-[KRRRE] |
| 743 | Cyc-R4-R3 | HeLa cells | FITC | 25654426 | 95 | Relative Mean Fluorescence intensity (%) | 5 mM | NA | NA | Flow cytometry | Uptake | ?A-RRR-[KRRRRE] |
| 744 | Cyc-R5-R2 | HeLa cells | FITC | 25654426 | 75 | Relative Mean Fluorescence intensity (%) | 5 mM | NA | NA | Flow cytometry | Uptake | ?A-RR-[KRRRRRE] |
| 745 | Cyc-R6-R1 | HeLa cells | FITC | 25654426 | 72 | Relative Mean Fluorescence intensity (%) | 5 mM | NA | NA | Flow cytometry | Uptake | ?A-R[KRRRRRRE] |
| 746 | RW9 | CHO-K1 cells | NA | 25445669 | 10.375 | pmol/uM Internalized peptide | 10 uM | 1h | 37ºC | MALDI-TOF | Uptake | GGGGRRWWRRWRR |
| 747 | RFFF9 | CHO-K1 cells | NA | 25445669 | 0.2 | pmol/uM Internalized peptide | 10 uM | 1h | 37ºC | MALDI-TOF | Uptake | GGGGRRFFRRFRR |
| 748 | RFFW9 | CHO-K1 cells | NA | 25445669 | 0.5 | pmol/uM Internalized peptide | 10 uM | 1h | 37ºC | MALDI-TOF | Uptake | GGGGRRFFRRWRR |
| 749 | RWFF9 | CHO-K1 cells | NA | 25445669 | 0.625 | pmol/uM Internalized peptide | 10 uM | 1h | 37ºC | MALDI-TOF | Uptake | GGGGRRWFRRFRR |
| 750 | RFWF9 | CHO-K1 cells | NA | 25445669 | 0.25 | pmol/uM Internalized peptide | 10 uM | 1h | 37ºC | MALDI-TOF | Uptake | GGGGRRFWRRFRR |
| 751 | RFWW9 | CHO-K1 cells | NA | 25445669 | 1 | pmol/uM Internalized peptide | 10 uM | 1h | 37ºC | MALDI-TOF | Uptake | GGGGRRFWRRWRR |
| 752 | RWWF9 | CHO-K1 cells | NA | 25445669 | 0.625 | pmol/uM Internalized peptide | 10 uM | 1h | 37ºC | MALDI-TOF | Uptake | GGGGRRWWRRFRR |
| 753 | RWFW9 | CHO-K1 cells | NA | 25445669 | 0.5 | pmol/uM Internalized peptide | 10 uM | 1h | 37ºC | MALDI-TOF | Uptake | GGGGRRWFRRWRR |
| 754 | NA | MDA-MB-231 cells | RNA-FAM | 34948105 | 65 000 | Fluorescence intensity | NA | 30 min | NA | Flow cytometry | Transduction | FFAARTMIWYpGAWYKRI |
| 755 | TAT | HeLa cells | Carboxyfluorescein | 34504427 | 32.0 | % Positive cells | 10 uM | 2h | NA | Flow cytometry | Internalization | GRKKRRQRRRPPQ |
| 756 | AKIP1 | HeLa cells | Carboxyfluorescein | 34504427 | 38.0 | % Positive cells | 10 uM | 2h | NA | Flow cytometry | Internalization | VLERAKRRAV |
| 757 | CASC3 | HeLa cells | Carboxyfluorescein | 34504427 | 54.0 | % Positive cells | 10 uM | 2h | NA | Flow cytometry | Internalization | PDDIKPRRIRKPRY |
| 758 | CCNL2 | HeLa cells | Carboxyfluorescein | 34504427 | 2.0 | % Positive cells | 10 uM | 2h | NA | Flow cytometry | Internalization | NTKRRLEGAKKA |
| 759 | DAPK1 | HeLa cells | Carboxyfluorescein | 34504427 | 9.0 | % Positive cells | 10 uM | 2h | NA | Flow cytometry | Internalization | AAKFIKKRRTKSS |
| 760 | ING4 | HeLa cells | Carboxyfluorescein | 34504427 | 4.0 | % Positive cells | 10 uM | 2h | NA | Flow cytometry | Internalization | TQKEKKAARARSK |
| 761 | DMAP1 | HeLa cells | Carboxyfluorescein | 34504427 | 10.0 | % Positive cells | 10 uM | 2h | NA | Flow cytometry | Internalization | RKRRESASSSSSVKKAKKP |
| 762 | VP8 | HeLa cells | Carboxyfluorescein | 34504427 | 28.0 | % Positive cells | 10 uM | 2h | NA | Flow cytometry | Internalization | KRKGRLRSKGKK |
| 763 | NOP53 | HeLa cells | Carboxyfluorescein | 34504427 | 8.0 | % Positive cells | 10 uM | 2h | NA | Flow cytometry | Internalization | AEADKPRRLGRLK |
| 764 | AHRR | HeLa cells | Carboxyfluorescein | 34504427 | 38.0 | % Positive cells | 10 uM | 2h | NA | Flow cytometry | Internalization | GECTYAGRKRRRPLQK |
| 765 | CUL4B | HeLa cells | Carboxyfluorescein | 34504427 | 16.0 | % Positive cells | 10 uM | 2h | NA | Flow cytometry | Internalization | TPPTSAKKRKL |
| 766 | FBXO32 | HeLa cells | Carboxyfluorescein | 34504427 | 4.0 | % Positive cells | 10 uM | 2h | NA | Flow cytometry | Internalization | VAAKKRKKDML |
| 767 | TAT | PC3 cells | Carboxyfluorescein | 34504427 | 64.0 | % Positive cells | 10 uM | 2h | NA | Flow cytometry | Internalization | GRKKRRQRRRPPQ |
| 768 | AKIP1 | PC3 cells | Carboxyfluorescein | 34504427 | 60.0 | % Positive cells | 10 uM | 2h | NA | Flow cytometry | Internalization | VLERAKRRAV |
| 769 | CASC3 | PC3 cells | Carboxyfluorescein | 34504427 | 74.0 | % Positive cells | 10 uM | 2h | NA | Flow cytometry | Internalization | PDDIKPRRIRKPRY |
| 770 | CCNL2 | PC3 cells | Carboxyfluorescein | 34504427 | 6.0 | % Positive cells | 10 uM | 2h | NA | Flow cytometry | Internalization | NTKRRLEGAKKA |
| 771 | DAPK1 | PC3 cells | Carboxyfluorescein | 34504427 | 18.0 | % Positive cells | 10 uM | 2h | NA | Flow cytometry | Internalization | AAKFIKKRRTKSS |
| 772 | ING4 | PC3 cells | Carboxyfluorescein | 34504427 | 6.0 | % Positive cells | 10 uM | 2h | NA | Flow cytometry | Internalization | TQKEKKAARARSK |
| 773 | DMAP1 | PC3 cells | Carboxyfluorescein | 34504427 | 22.0 | % Positive cells | 10 uM | 2h | NA | Flow cytometry | Internalization | RKRRESASSSSSVKKAKKP |
| 774 | VP8 | PC3 cells | Carboxyfluorescein | 34504427 | 46.0 | % Positive cells | 10 uM | 2h | NA | Flow cytometry | Internalization | KRKGRLRSKGKK |
| 775 | NOP53 | PC3 cells | Carboxyfluorescein | 34504427 | 18.0 | % Positive cells | 10 uM | 2h | NA | Flow cytometry | Internalization | AEADKPRRLGRLK |
| 776 | AHRR | PC3 cells | Carboxyfluorescein | 34504427 | 54.0 | % Positive cells | 10 uM | 2h | NA | Flow cytometry | Internalization | GECTYAGRKRRRPLQK |
| 777 | CUL4B | PC3 cells | Carboxyfluorescein | 34504427 | 21.0 | % Positive cells | 10 uM | 2h | NA | Flow cytometry | Internalization | TPPTSAKKRKL |
| 778 | FBXO32 | PC3 cells | Carboxyfluorescein | 34504427 | 10.0 | % Positive cells | 10 uM | 2h | NA | Flow cytometry | Internalization | VAAKKRKKDML |
| 779 | TAT | U87 cells | Carboxyfluorescein | 34504427 | 32.0 | % Positive cells | 10 uM | 2h | NA | Flow cytometry | Internalization | GRKKRRQRRRPPQ |
| 780 | AKIP1 | U87 cells | Carboxyfluorescein | 34504427 | 40.0 | % Positive cells | 10 uM | 2h | NA | Flow cytometry | Internalization | VLERAKRRAV |
| 781 | CASC3 | U87 cells | Carboxyfluorescein | 34504427 | 49.0 | % Positive cells | 10 uM | 2h | NA | Flow cytometry | Internalization | PDDIKPRRIRKPRY |
| 782 | CCNL2 | U87 cells | Carboxyfluorescein | 34504427 | 3.0 | % Positive cells | 10 uM | 2h | NA | Flow cytometry | Internalization | NTKRRLEGAKKA |
| 783 | DAPK1 | U87 cells | Carboxyfluorescein | 34504427 | 24.0 | % Positive cells | 10 uM | 2h | NA | Flow cytometry | Internalization | AAKFIKKRRTKSS |
| 784 | ING4 | U87 cells | Carboxyfluorescein | 34504427 | 11.0 | % Positive cells | 10 uM | 2h | NA | Flow cytometry | Internalization | TQKEKKAARARSK |
| 785 | DMAP1 | U87 cells | Carboxyfluorescein | 34504427 | 32.0 | % Positive cells | 10 uM | 2h | NA | Flow cytometry | Internalization | RKRRESASSSSSVKKAKKP |
| 786 | VP8 | U87 cells | Carboxyfluorescein | 34504427 | 28.0 | % Positive cells | 10 uM | 2h | NA | Flow cytometry | Internalization | KRKGRLRSKGKK |
| 787 | NOP53 | U87 cells | Carboxyfluorescein | 34504427 | 10.0 | % Positive cells | 10 uM | 2h | NA | Flow cytometry | Internalization | AEADKPRRLGRLK |
| 788 | AHRR | U87 cells | Carboxyfluorescein | 34504427 | 36.0 | % Positive cells | 10 uM | 2h | NA | Flow cytometry | Internalization | GECTYAGRKRRRPLQK |
| 789 | CUL4B | U87 cells | Carboxyfluorescein | 34504427 | 18.0 | % Positive cells | 10 uM | 2h | NA | Flow cytometry | Internalization | TPPTSAKKRKL |
| 790 | FBXO32 | U87 cells | Carboxyfluorescein | 34504427 | 3.0 | % Positive cells | 10 uM | 2h | NA | Flow cytometry | Internalization | VAAKKRKKDML |
| 791 | RALA | HeLa cells | pCMV-EGFP plasmid DNA | 34443195 | 61.0 | % Positive cells | N/P ratio 6 | 6h | 37ºC | Flow cytometry | Transfection | WEARLARALARALARHLARALARALRACEA |
| 792 | HALA1 | HeLa cells | pCMV-EGFP plasmid DNA | 34443195 | 45.0 | % Positive cells | N/P ratio 6 | 6h | 37ºC | Flow cytometry | Transfection | WEAHLAHALARALARHLARALARALRACEA |
| 793 | HALA2 | HeLa cells | pCMV-EGFP plasmid DNA | 34443195 | 62.0 | % Positive cells | N/P ratio 6 | 6h | 37ºC | Flow cytometry | Transfection | WEARLARALARALARHLARALAHALHACEA |
| 794 | HALA3 | HeLa cells | pCMV-EGFP plasmid DNA | 34443195 | 27.0 | % Positive cells | N/P ratio 6 | 6h | 37ºC | Flow cytometry | Transfection | WEAHLAHALAHALARHLARALARALRACEA |
| 795 | HALA4 | HeLa cells | pCMV-EGFP plasmid DNA | 34443195 | 40.0 | % Positive cells | N/P ratio 6 | 6h | 37ºC | Flow cytometry | Transfection | WEARLARALARALARHLAHALAHALHACEA |
| 796 | RALA | HEK293T cells | pCMV-EGFP plasmid DNA | 34443195 | 41.5 | % Positive cells | N/P ratio 6 | 6h | 37ºC | Flow cytometry | Transfection | WEARLARALARALARHLARALARALRACEA |
| 797 | HALA1 | HEK293T cells | pCMV-EGFP plasmid DNA | 34443195 | 39.0 | % Positive cells | N/P ratio 6 | 6h | 37ºC | Flow cytometry | Transfection | WEAHLAHALARALARHLARALARALRACEA |
| 798 | HALA2 | HEK293T cells | pCMV-EGFP plasmid DNA | 34443195 | 56.5 | % Positive cells | N/P ratio 6 | 6h | 37ºC | Flow cytometry | Transfection | WEARLARALARALARHLARALAHALHACEA |
| 799 | HALA3 | HEK293T cells | pCMV-EGFP plasmid DNA | 34443195 | 21.0 | % Positive cells | N/P ratio 6 | 6h | 37ºC | Flow cytometry | Transfection | WEAHLAHALAHALARHLARALARALRACEA |
| 800 | HALA4 | HEK293T cells | pCMV-EGFP plasmid DNA | 34443195 | 55.0 | % Positive cells | N/P ratio 6 | 6h | 37ºC | Flow cytometry | Transfection | WEARLARALARALARHLAHALAHALHACEA |
| 801 | RALA | A549 cells | pCMV-EGFP plasmid DNA | 34443195 | 13.5 | % Positive cells | N/P ratio 6 | 6h | 37ºC | Flow cytometry | Transfection | WEARLARALARALARHLARALARALRACEA |
| 802 | HALA1 | A549 cells | pCMV-EGFP plasmid DNA | 34443195 | 10.0 | % Positive cells | N/P ratio 6 | 6h | 37ºC | Flow cytometry | Transfection | WEAHLAHALARALARHLARALARALRACEA |
| 803 | HALA2 | A549 cells | pCMV-EGFP plasmid DNA | 34443195 | 25.5 | % Positive cells | N/P ratio 6 | 6h | 37ºC | Flow cytometry | Transfection | WEARLARALARALARHLARALAHALHACEA |
| 804 | HALA3 | A549 cells | pCMV-EGFP plasmid DNA | 34443195 | 4.0 | % Positive cells | N/P ratio 6 | 6h | 37ºC | Flow cytometry | Transfection | WEAHLAHALAHALARHLARALARALRACEA |
| 805 | HALA4 | A549 cells | pCMV-EGFP plasmid DNA | 34443195 | 8.5 | % Positive cells | N/P ratio 6 | 6h | 37ºC | Flow cytometry | Transfection | WEARLARALARALARHLAHALAHALHACEA |
| 806 | PDL | SH-SY5Y cells | EGFP pDNA | 34361142 | 31.10 ± 0.5 | % Transfection | plasmid/PDL ratio 1:4 | 48h | 37ºC | Flow cytometry | Transfection | kkk |
| 807 | PDL | HeLa cells | EGFP pDNA | 34361142 | 1.33 ± 0.18 | % Transfection | plasmid/PDL ratio 1:4 | 48 h | 37ºC | Flow cytometry | Transfection | kkk |
| 808 | PDL | NIH-3T3 cells | EGFP pDNA | 34361142 | 0.16 ± 0.03 | % Transfection | plasmid/PDL ratio 1:4 | 48 h | 37ºC | Flow cytometry | Transfection | kkk |
| 809 | TAT | H1299 | 111In-GFP-G1 | 33789931 | 6.8 | Relative Cellular uptake | 1.5 nM | 1h | 37ºC | Flow cytometry | Uptake | GRKKRRQRRRPPQGYG |
| 810 | Tat(48-57) | HEK293 cells | TAMRA | 33589718 | 68333 | Mean Fluorescence intensity | 5 ug | 16h | NA | Flow cytometry | Penetration efficiencies | GRKKRRQRRR |
| 811 | CTP | HEK293 cells | TAMRA | 33589718 | 43333 | Mean Fluorescence intensity | 5 ug | 16h | NA | Flow cytometry | Penetration efficiencies | GGRRARRRRRR |
| 812 | TatsMTS (TMG) | HEK293 cells | TAMRA | 33589718 | 80000 | Mean Fluorescence intensity | 5 ug | 16h | NA | Flow cytometry | Penetration efficiencies | GRKKRRQRRRMVSAL |
| 813 | Tat(49-57) | HEK293 cells | TAMRA | 33589718 | 48333 | Mean Fluorescence intensity | 5 ug | 16h | NA | Flow cytometry | Penetration efficiencies | RKKRRQRRR |
| 814 | Tat | HEK293 cells | TAMRA | 33589718 | 45833 | Mean Fluorescence intensity | 5 ug | 16h | NA | Flow cytometry | Penetration efficiencies | GRKKRRQRRRPPQRKC |
| 815 | Tat(47-57) | HEK293 cells | TAMRA | 33589718 | 72500 | Mean Fluorescence intensity | 5 ug | 16h | NA | Flow cytometry | Penetration efficiencies | YGRKKRRQRRR |
| 816 | 6-Oct | HEK293 cells | TAMRA | 33589718 | 73333 | Mean Fluorescence intensity | 5 ug | 16h | NA | Flow cytometry | Penetration efficiencies | GRKRKKRT |
| 817 | K9 | HEK293 cells | TAMRA | 33589718 | 72500 | Mean Fluorescence intensity | 5 ug | 16h | NA | Flow cytometry | Penetration efficiencies | KKKKKKKKK |
| 818 | D-R9 | HEK293 cells | TAMRA | 33589718 | 34166 | Mean Fluorescence intensity | 5 ug | 16h | NA | Flow cytometry | Penetration efficiencies | rrrrrrrrr |
| 819 | HIV-1 TAT peptide--Crystallins | HEK293 cells | TAMRA | 33589718 | 48333 | Mean Fluorescence intensity | 5 ug | 16h | NA | Flow cytometry | Penetration efficiencies | GRKKRRQRRRPQ |
| 820 | CRGDK | HEK293 cells | TAMRA | 33589718 | 56666 | Mean Fluorescence intensity | 5 ug | 16h | NA | Flow cytometry | Penetration efficiencies | CRGDK |
| 821 | PAF95 | HEK293 cells | TAMRA | 33589718 | 39166 | Mean Fluorescence intensity | 5 ug | 16h | NA | Flow cytometry | Penetration efficiencies | AAAWFW |
| 822 | iRGD | HEK293 cells | TAMRA | 33589718 | 37500 | Mean Fluorescence intensity | 5 ug | 16h | NA | Flow cytometry | Penetration efficiencies | CRGDKGDPC |
| 823 | Ypep-GFP-Ypep | HEK293 cells | TAMRA | 33589718 | 5000 | Mean Fluorescence intensity | 5 ug | 16h | NA | Flow cytometry | Penetration efficiencies | YTFGLKTSFNVQYTFGLKTSFNVQ |
| 824 | VP1 BC loop (V) peptides | HEK293 cells | TAMRA | 33589718 | 41666 | Mean Fluorescence intensity | 5 ug | 16h | NA | Flow cytometry | Penetration efficiencies | TVDNPASTTNKDKLFAVRK |
| 825 | Peptide 1-NTCS | HEK293 cells | TAMRA | 33589718 | 55000 | Mean Fluorescence intensity | 5 ug | 16h | NA | Flow cytometry | Penetration efficiencies | TWLKYH |
| 826 | Ypep-GFP | HEK293 cells | TAMRA | 33589718 | 10000 | Mean Fluorescence intensity | 5 ug | 16h | NA | Flow cytometry | Penetration efficiencies | YTFGLKTSFNVQ |
| 827 | CPPP-2 | HEK293 cells | TAMRA | 33589718 | 30000 | Mean Fluorescence intensity | 5 ug | 16h | NA | Flow cytometry | Penetration efficiencies | KLPVM |
| 828 | TCTPPTD | HEK293 cells | TAMRA | 33589718 | 40000 | Mean Fluorescence intensity | 5 ug | 16h | NA | Flow cytometry | Penetration efficiencies | MIIYRDLISH |
| 829 | ARF(1-22) | HEK293 cells | TAMRA | 33589718 | 0 | Mean Fluorescence intensity | 5 ug | 16h | NA | Flow cytometry | Penetration efficiencies | MVRRFLVTLRIRRACGPPRVRV |
| 830 | Tat(48-57) | CHO cells | TAMRA | 33589718 | 3500 | Mean Fluorescence intensity | 5 ug | 16h | NA | Flow cytometry | Penetration efficiencies | GRKKRRQRRR |
| 831 | CTP | CHO cells | TAMRA | 33589718 | 2500 | Mean Fluorescence intensity | 5 ug | 16h | NA | Flow cytometry | Penetration efficiencies | GGRRARRRRRR |
| 832 | TatsMTS (TMG) | CHO cells | TAMRA | 33589718 | 7000 | Mean Fluorescence intensity | 5 ug | 16h | NA | Flow cytometry | Penetration efficiencies | GRKKRRQRRRMVSAL |
| 833 | Tat(49-57) | CHO cells | TAMRA | 33589718 | 3000 | Mean Fluorescence intensity | 5 ug | 16h | NA | Flow cytometry | Penetration efficiencies | RKKRRQRRR |
| 834 | Tat | CHO cells | TAMRA | 33589718 | 8000 | Mean Fluorescence intensity | 5 ug | 16h | NA | Flow cytometry | Penetration efficiencies | GRKKRRQRRRPPQRKC |
| 835 | Tat(47-57) | CHO cells | TAMRA | 33589718 | 3000 | Mean Fluorescence intensity | 5 ug | 16h | NA | Flow cytometry | Penetration efficiencies | YGRKKRRQRRR |
| 836 | 6-Oct | CHO cells | TAMRA | 33589718 | 5000 | Mean Fluorescence intensity | 5 ug | 16h | NA | Flow cytometry | Penetration efficiencies | GRKRKKRT |
| 837 | K9 | CHO cells | TAMRA | 33589718 | 9000 | Mean Fluorescence intensity | 5 ug | 16h | NA | Flow cytometry | Penetration efficiencies | KKKKKKKKK |
| 838 | D-R9 | CHO cells | TAMRA | 33589718 | 3500 | Mean Fluorescence intensity | 5 ug | 16h | NA | Flow cytometry | Penetration efficiencies | rrrrrrrrr |
| 839 | HIV-1 TAT peptide--Crystallins | CHO cells | TAMRA | 33589718 | 7000 | Mean Fluorescence intensity | 5 ug | 16h | NA | Flow cytometry | Penetration efficiencies | GRKKRRQRRRPQ |
| 840 | CRGDK | CHO cells | TAMRA | 33589718 | 16500 | Mean Fluorescence intensity | 5 ug | 16h | NA | Flow cytometry | Penetration efficiencies | CRGDK |
| 841 | PAF95 | CHO cells | TAMRA | 33589718 | 20000 | Mean Fluorescence intensity | 5 ug | 16h | NA | Flow cytometry | Penetration efficiencies | AAAWFW |
| 842 | iRGD | CHO cells | TAMRA | 33589718 | 2000 | Mean Fluorescence intensity | 5 ug | 16h | NA | Flow cytometry | Penetration efficiencies | CRGDKGDPC |
| 843 | Ypep-GFP-Ypep | CHO cells | TAMRA | 33589718 | 6000 | Mean Fluorescence intensity | 5 ug | 16h | NA | Flow cytometry | Penetration efficiencies | YTFGLKTSFNVQYTFGLKTSFNVQ |
| 844 | VP1 BC loop (V) peptides | CHO cells | TAMRA | 33589718 | 16000 | Mean Fluorescence intensity | 5 ug | 16h | NA | Flow cytometry | Penetration efficiencies | TVDNPASTTNKDKLFAVRK |
| 845 | Peptide 1-NTCS | CHO cells | TAMRA | 33589718 | 11000 | Mean Fluorescence intensity | 5 ug | 16h | NA | Flow cytometry | Penetration efficiencies | TWLKYH |
| 846 | Ypep-GFP | CHO cells | TAMRA | 33589718 | 5500 | Mean Fluorescence intensity | 5 ug | 16h | NA | Flow cytometry | Penetration efficiencies | YTFGLKTSFNVQ |
| 847 | CPPP-2 | CHO cells | TAMRA | 33589718 | 7500 | Mean Fluorescence intensity | 5 ug | 16h | NA | Flow cytometry | Penetration efficiencies | KLPVM |
| 848 | TCTPPTD | CHO cells | TAMRA | 33589718 | 4500 | Mean Fluorescence intensity | 5 ug | 16h | NA | Flow cytometry | Penetration efficiencies | MIIYRDLISH |
| 849 | ARF(1-22) | CHO cells | TAMRA | 33589718 | 0 | Mean Fluorescence intensity | 5 ug | 16h | NA | Flow cytometry | Penetration efficiencies | MVRRFLVTLRIRRACGPPRVRV |
| 850 | KYKGAIIGNIK | HEK293T cells | pGL3-SV40 | 31861408 | 102500 | RFU/mg | pDNA/peptide ratio 1:2500 | 4h | 37ºC | Fluorescent Microscopy | Transfection | KYKGAIIGNIK |
| 851 | KYRSGAITIGY | HEK293T cells | pGL3-SV40 | 31861408 | 175000 | RFU/mg | pDNA/peptide ratio 1:2500 | 4h | 37ºC | Fluorescent Microscopy | Transfection | KYRSGAITIGY |
| 852 | 4Iphf-HN1 | Cal 27 | IR800 | 31450798 | 0.55 | Fluorescence intensity | 10 uM | 2h | NA | Fluorescent Microscopy | Uptake | TSPLNIHNGQKL |
| 853 | f-HN1 | Cal 27 | IR800 | 31450798 | 1 | Fluorescence intensity | 10 uM | 2h | NA | Fluorescent Microscopy | Uptake | TSPLNIHNGQKL |
| 854 | HNJ | Cal 27 | IR800 | 31450798 | 0.3 | Fluorescence intensity | 10 uM | 2h | NA | Fluorescent Microscopy | Uptake | NQHSKNTLLIGP |
| 855 | 4Iphf-HN17 | Cal 27 | IR800 | 31450798 | 4.5 | Fluorescence intensity | 10 uM | 2h | NA | Fluorescent Microscopy | Uptake | LPNSNHIKQGL |
| 856 | f-HN17 | Cal 27 | IR800 | 31450798 | 1.70 | Fluorescence intensity | 10 uM | 2h | NA | Fluorescent Microscopy | Uptake | TLPNSNHIKQGL |
| 857 | iPTD | HEK293T cells | Fab-F2 | 31375703 | 7750 | Mean Fluorescence intensity | 10 ug/mL | 24h | NA | Flow cytometry | Internalization | MALGPCMLLLLLLLGLRLPGVWAPPRRRRRRRRR |
| 858 | CPP9 | Saos-2 cells | Rho-labeled SNAP-tag | 30410976 | 0.175E-3 | Average Median Fluorescence intensity | 1 uM | 30 min | 37ºC | Flow cytometry | Uptake | FRRRRQ |
| 859 | CPP12 | Saos-2 cells | Rho-labeled SNAP-tag | 30410976 | 0.4E-3 | Average Median Fluorescence intensity | 1 uM | 30 min | 37ºC | Flow cytometry | Uptake | FRRRRQ |
| 860 | aPP5.3 | Saos-2 cells | Rho-labeled SNAP-tag | 30410976 | 0.4E-3 | Average Median Fluorescence intensity | 1 uM | 30 min | 37ºC | Flow cytometry | Uptake | MGPSQPTYPGDDAPVRDLIRFYRDLRRYLNVVTRHRY |
| 861 | R8 | Saos-2 cells | Rho-labeled SNAP-tag | 30410976 | 0.725E-3 | Average Median Fluorescence intensity | 1 uM | 30 min | 37ºC | Flow cytometry | Uptake | MRRRRRRR |
| 862 | ZiF | Saos-2 cells | Rho-labeled SNAP-tag | 30410976 | 0.75E-3 | Average Median Fluorescence intensity | 1 uM | 30 min | 37ºC | Flow cytometry | Uptake | MLEPGEKPYKCPECGKSFSASAALVAHQRTHTGKKTS |
| 863 | Pen | Saos-2 cells | Rho-labeled SNAP-tag | 30410976 | 1.4E-3 | Average Median Fluorescence intensity | 1 uM | 30 min | 37ºC | Flow cytometry | Uptake | MRQIKIWFQNRRMKWKK |
| 864 | ZF5.3 | Saos-2 cells | Rho-labeled SNAP-tag | 30410976 | 2.125E-3 | Average Median Fluorescence intensity | 1 uM | 30 min | 37ºC | Flow cytometry | Uptake | MYSCNVCGKAFVLSRHLNRHLRVHRRAT |
| 865 | TAT | HEK293 cells | EDB_S11 (protein fusions) | 30135446 | 22.0 | % Green viable cells | 40 uM | 1h | 37ºC | Flow cytometry | Uptake (Endosomal escape) | GRKKRRQRRRPPQRKC |
| 866 | 84 | HEK293 cells | EDB_S11 (protein fusions) | 30135446 | 36.0 | % Green viable cells | 40 uM | 1h | 37ºC | Flow cytometry | Uptake (Endosomal escape) | RKQKSLQTKLAENPPVPRKKRQSRPRWKQWLQK |
| 867 | 1746 | HEK293 cells | EDB_S11 (protein fusions) | 30135446 | 72.0 | % Green viable cells | 40 uM | 1h | 37ºC | Flow cytometry | Uptake (Endosomal escape) | PLKPKKPKTQEKKKKQPPKPKKPKTQEKKKKQPPKPKR |
| 868 | PPC1 | eGFP HeLa 654 | PMO | 29721534 | 18400 | Mean Fluorescence intensity | 5 uM | 22h | 37ºC | Flow cytometry | Uptake | KQPRIKRKK |
| 869 | PPC2 | eGFP HeLa 654 | PMO | 29721534 | 17500 | Mean Fluorescence intensity | 5 uM | 22h | 37ºC | Flow cytometry | Uptake | LKKRRKLPKKKPIRNEQ |
| 870 | PPC3 | eGFP HeLa 654 | PMO | 29721534 | 23640 | Mean Fluorescence intensity | 5 uM | 22h | 37ºC | Flow cytometry | Uptake | KKYRGRKRHPR |
| 871 | PPC4 | eGFP HeLa 654 | PMO | 29721534 | 21370 | Mean Fluorescence intensity | 5 uM | 22h | 37ºC | Flow cytometry | Uptake | APKRKKLKKRF |
| 872 | PPC5 | eGFP HeLa 654 | PMO | 29721534 | 18640 | Mean Fluorescence intensity | 5 uM | 22h | 37ºC | Flow cytometry | Uptake | GRKAARAPGRRKQ |
| 873 | NS1 | eGFP HeLa 654 | PMO | 29721534 | 5000 | Mean Fluorescence intensity | 5 uM | 22h | 37ºC | Flow cytometry | Uptake | HDLPKGG |
| 874 | NS2 | eGFP HeLa 654 | PMO | 29721534 | 9320 | Mean Fluorescence intensity | 5 uM | 22h | 37ºC | Flow cytometry | Uptake | AGSHRRL |
| 875 | IMT-P8 | HeLa cells | KLA | 27189051 | 285000 | Mean Fluorescence intensity | 2.5 uM | 30 min | 37ºC | Flow cytometry | Uptake | RRWRRWNRFNRRRCR |
| 876 | IMT-P8 | MDA-MB-231 cells | KLA | 27189051 | 161600 | Mean Fluorescence intensity | 2.5 uM | 30 min | 37ºC | Flow cytometry | Uptake | RRWRRWNRFNRRRCR |
| 877 | IMT-P8 | PC3 cells | KLA | 27189051 | 1037500 | Mean Fluorescence intensity | 2.5 uM | 30 min | 37ºC | Flow cytometry | Uptake | RRWRRWNRFNRRRCR |
| 878 | HR9 | A549 cells | FITC | 26942714 | 94.0 | % Positive cells | 10 uM | 1h | 37ºC | Flow cytometry | Internalization | CHHHHHRRRRRRRRRHHHHHC |
| 879 | Lfcin | A549 cells | FITC | 26942714 | 94.0 | % Positive cells | 10 uM | 1h | 37ºC | Flow cytometry | Internalization | CRRWQWRMKKLGC |
| 880 | L12 | A549 cells | FITC | 26942714 | 97.0 | % Positive cells | 10 uM | 1h | 37ºC | Flow cytometry | Internalization | FKCRRWQWRMKK |
| 881 | L11 | A549 cells | FITC | 26942714 | 93.0 | % Positive cells | 10 uM | 1h | 37ºC | Flow cytometry | Internalization | KCRRWQWRMKK |
| 882 | L9 | A549 cells | FITC | 26942714 | 77.0 | % Positive cells | 10 uM | 1h | 37ºC | Flow cytometry | Internalization | RRWQWRMKK |
| 883 | L6 | A549 cells | FITC | 26942714 | 98.0 | % Positive cells | 10 uM | 1h | 37ºC | Flow cytometry | Internalization | RRWQWR |
| 884 | L5a | A549 cells | FITC | 26942714 | 95.5 | % Positive cells | 10 uM | 1h | 37ºC | Flow cytometry | Internalization | RRWQW |
| 885 | L5b | A549 cells | FITC | 26942714 | 25.0 | % Positive cells | 10 uM | 1h | 37ºC | Flow cytometry | Internalization | RWQWR |
| 886 | L4 | A549 cells | FITC | 26942714 | 9.0 | % Positive cells | 10 uM | 1h | 37ºC | Flow cytometry | Internalization | RWQW |
| 887 | TAT | N2a cells | BoNTA | 35223792 | 158.75 | Relative fluorescence (%) | 100 nM | 2h | 37ºC | Immunofluorescence analysis | Cellular uptake | GRKKRRQRRRPQ |
| 888 | Pep1 | N2a cells | BoNTA | 35223792 | 117.5 | Relative fluorescence (%) | 100 nM | 2h | 37ºC | Immunofluorescence analysis | Cellular uptake | KETWWETWWTEWSQPKKKRKV |
| 889 | ZFP3 (N-Terminal) | N2a cells | BoNTA | 35223792 | 110.0 | Relative fluorescence (%) | 100 nM | 2h | 37ºC | Immunofluorescence analysis | Cellular uptake | EKPYKCPECGKSFSASAALVAHQRTHTGEKPYKCPECGKSFSASAALVAHQRTHTGEKPYKCPECGKSFSASAALVAHQRTHTG |
| 890 | ZFP3 (C-Terminal) | N2a cells | BoNTA | 35223792 | 120.0 | Relative fluorescence (%) | 100 nM | 2h | 37ºC | Immunofluorescence analysis | Cellular uptake | EKPYKCPECGKSFSASAALVAHQRTHTGEKPYKCPECGKSFSASAALVAHQRTHTGEKPYKCPECGKSFSASAALVAHQRTHTG |
| 891 | ZFP3 (N and C-Terminal) | N2a cells | BoNTA | 35223792 | 177.5 | Relative fluorescence (%) | 100 nM | 2h | 37ºC | Immunofluorescence analysis | Cellular uptake | EKPYKCPECGKSFSASAALVAHQRTHTGEKPYKCPECGKSFSASAALVAHQRTHTGEKPYKCPECGKSFSASAALVAHQRTHTG |
| 892 | SynB1 | MCF7 cells | ELP-DOXO | 35216417 | 3.2 | RFU | 2 uM dox equivalent concentration | 24h | NA | Flow cytometry | Cellular uptake | RGGRLSYSRRRFSTSTGR-VPGXGVPGXGVPGXG |
| 893 | SynB1 | MCF7 cells | ELP-GFLG-NCDox | 35216417 | 0.8 | RFU | 2 uM dox equivalent concentration | 24h | NA | Flow cytometry | Cellular uptake | RGGRLSYSRRRFSTSTGR-VPGXGVPGXGVPGXG |
| 894 | SynB1 | NCI/ADR | ELP-DOXO | 35216417 | 1.3 | RFU | 2 uM dox equivalent concentration | 24h | NA | Flow cytometry | Cellular uptake | RGGRLSYSRRRFSTSTGR-VPGXGVPGXGVPGXG |
| 895 | SynB1 | NCI/ADR | ELP-GFLG-NCDox | 35216417 | 1.1 | RFU | 2 uM dox equivalent concentration | 24h | NA | Flow cytometry | Cellular uptake | RGGRLSYSRRRFSTSTGR-VPGXGVPGXGVPGXG |
| 896 | Cys-Penetratin | TR146 cell | Liposomes-salmon calcitonin (sCT) | 35210769 | 3800 | Relative Mean Fluorescence intensity | NA | 2h | 37ºC | Flow cytometry | Relative uptake | CRQIKIWFQNRRMKWKK |
| 897 | G2R2 | HeLa cells | Somatropin-Hyaluronic acid | 35093459 | 0.055 | C/M ratio of somatropin (mL/mg protein) | 50 ug/ml | 2h | 37ºC | ELISA | Uptake | GGRR |
| 898 | G2R4 | HeLa cells | Somatropin-Hyaluronic acid | 35093459 | 0.15 | C/M ratio of somatropin (mL/mg protein) | 50 ug/ml | 2h | 37ºC | ELISA | Uptake | GGRRRR |
| 899 | G4R8 | HeLa cells | Somatropin-Hyaluronic acid | 35093459 | 0.10 | C/M ratio of somatropin (mL/mg protein) | 50 ug/ml | 2h | 37ºC | ELISA | Uptake | GGGGRRRRRRRR |
| 900 | G2R2 | HeLa cells | Exendin-4-Hyaluronic acid | 35093459 | 1.225 | C/M ratio of exendin-4 (uL/mg protein) | 50 ug/ml | 2h | 37ºC | ELISA | Uptake | GGRR |
| 901 | G2R4 | HeLa cells | Exendin-4-Hyaluronic acid | 35093459 | 1.65 | C/M ratio of exendin-4 (uL/mg protein) | 50 ug/ml | 2h | 37ºC | ELISA | Uptake | GGRRRR |
| 902 | G4R8 | HeLa cells | Exendin-4-Hyaluronic acid | 35093459 | 2.125 | C/M ratio of exendin-4 (uL/mg protein) | 50 ug/ml | 2h | 37ºC | ELISA | Uptake | GGGGRRRRRRRR |
| 903 | Crotamine | P. falciparum-infected erythrocytes | Cy3-labeled Crotamine | 35074306 | 46.0 | % Internalization | 5 uM | 30 min | 37ºC | Flow cytometry | Internalization | YKQCHKKGGHCFPKEKICLPPSSDFGKMDCRWRWKCCKKGSG |
| 904 | CKRRMKWKK | HepG2 cells | siRNA | 35024246 | 3600 | Mean Fluorescence intensity | 100 uM | 4h | NA | Flow cytometry | Cellular uptake | CKRRMKWKK-Cys |
| 905 | CKRRMKWKK | HepG2 cells | siRNA-TSL | 35024246 | 1600 | Mean Fluorescence intensity | 100 uM | 4h | NA | Flow cytometry | Cellular uptake | CKRRMKWKK-Cys |
| 906 | CKRRMKWKK | HepG2 cells | siRNA-MTSL | 35024246 | 2100 | Mean Fluorescence intensity | 100 uM | 4h | NA | Flow cytometry | Cellular uptake | CKRRMKWKK-Cys |
| 907 | CKRRMKWKK | HepG2 cells | siRNA-MTSLR | 35024246 | 2550 | Mean Fluorescence intensity | 100 uM | 4h | NA | Flow cytometry | Cellular uptake | CKRRMKWKK-Cys |
| 908 | CKRRMKWKK | HepG2 cells | siRNA-MTSLR-H | 35024246 | 3900 | Mean Fluorescence intensity | 100 uM | 4h | NA | Flow cytometry | Cellular uptake | CKRRMKWKK-Cys |
| 909 | CKRRMKWKK | RAW264.7 cells | siRNA-TSL | 35024246 | 1200 | Mean Fluorescence intensity | 100 uM | 4h | NA | Flow cytometry | Cellular uptake | CKRRMKWKK-Cys |
| 910 | CKRRMKWKK | RAW264.7 cells | siRNA-MTSL | 35024246 | 750 | Mean Fluorescence intensity | 100 uM | 4h | NA | Flow cytometry | Cellular uptake | CKRRMKWKK-Cys |
| 911 | CKRRMKWKK | RAW264.7 cells | siRNA-MTSLR | 35024246 | 875 | Mean Fluorescence intensity | 100 uM | 4h | NA | Flow cytometry | Cellular uptake | CKRRMKWKK-Cys |
| 912 | TmP(Glu)4 | HeLa cells | (alpha-D-glucose)4-TAMRA | 34994362 | 545 | RFU | 10 uM | 30 min | NA | Flow cytometry | Internalization efficency | RKLRRLLRRLKRL |
| 913 | TmP(Glu)6 | HeLa cells | (alpha-D-glucose)6-TAMRA | 34994362 | 660 | RFU | 10 uM | 30 min | NA | Flow cytometry | Internalization efficency | KRKLRRLLRRLKRL |
| 914 | TmP(Man)4 | HeLa cells | (alpha-D-mannose)4-TAMRA | 34994362 | 860 | RFU | 10 uM | 30 min | NA | Flow cytometry | Internalization efficency | RKLRRLLRRLKRL |
| 915 | TmP(Man)6 | HeLa cells | (alpha-D-mannose)6-TAMRA | 34994362 | 720 | RFU | 10 uM | 30 min | NA | Flow cytometry | Internalization efficency | KRKLRRLLRRLKRL |
| 916 | TmP(Gal)4 | HeLa cells | (alpha-D-galactose)4-TAMRA | 34994362 | 845 | RFU | 10 uM | 30 min | NA | Flow cytometry | Internalization efficency | RKLRRLLRRLKRL |
| 917 | TmP(Gal)6 | HeLa cells | (alpha-D-galactose)6-TAMRA | 34994362 | 730 | RFU | 10 uM | 30 min | NA | Flow cytometry | Internalization efficency | KRKLRRLLRRLKRL |
| 918 | Arg | HeLa cells | Carboxyfluorescein | 30718681 | 180 | Mean Fluorescence intensity | 1 uM | 2h | NA | Flow cytometry | Uptake | GRRRRRRRRR |
| 919 | Arg | HeLa cells | Carboxyfluorescein | 30718681 | 180 | Mean Fluorescence intensity | 1 uM | 6h | NA | Flow cytometry | Uptake | GRRRRRRRRR |
| 920 | Arg | HeLa cells | Carboxyfluorescein | 30718681 | 30 | Mean Fluorescence intensity | 1 uM | 24h | NA | Flow cytometry | Uptake | GRRRRRRRRR |
| 921 | Leu | HeLa cells | Carboxyfluorescein | 30718681 | 30 | Mean Fluorescence intensity | 1 uM | 2h | NA | Flow cytometry | Uptake | GRRLRRLRRL |
| 922 | Leu | HeLa cells | Carboxyfluorescein | 30718681 | 35 | Mean Fluorescence intensity | 1 uM | 6h | NA | Flow cytometry | Uptake | GRRLRRLRRL |
| 923 | Leu | HeLa cells | Carboxyfluorescein | 30718681 | 25 | Mean Fluorescence intensity | 1 uM | 24h | NA | Flow cytometry | Uptake | GRRLRRLRRL |
| 924 | (?Me)Leu | HeLa cells | Carboxyfluorescein | 30718681 | 70 | Mean Fluorescence intensity | 1 uM | 2h | NA | Flow cytometry | Uptake | GRRXRRXRRX |
| 925 | (?Me)Leu | HeLa cells | Carboxyfluorescein | 30718681 | 135 | Mean Fluorescence intensity | 1 uM | 6h | NA | Flow cytometry | Uptake | GRRXRRXRRX |
| 926 | (?Me)Leu | HeLa cells | Carboxyfluorescein | 30718681 | 120 | Mean Fluorescence intensity | 1 uM | 24h | NA | Flow cytometry | Uptake | GRRXRRXRRX |
| 927 | Ac5cdOM | HeLa cells | Carboxyfluorescein | 30718681 | 30 | Mean Fluorescence intensity | 1 uM | 2h | NA | Flow cytometry | Uptake | GRRXRRXRRX |
| 928 | Ac5cdOM | HeLa cells | Carboxyfluorescein | 30718681 | 45 | Mean Fluorescence intensity | 1 uM | 6h | NA | Flow cytometry | Uptake | GRRXRRXRRX |
| 929 | Ac5cdOM | HeLa cells | Carboxyfluorescein | 30718681 | 60 | Mean Fluorescence intensity | 1 uM | 24h | NA | Flow cytometry | Uptake | GRRXRRXRRX |
| 930 | Ac5c | HeLa cells | Carboxyfluorescein | 30718681 | 50 | Mean Fluorescence intensity | 1 uM | 2h | NA | Flow cytometry | Uptake | GRRXRRXRRX |
| 931 | Ac5c | HeLa cells | Carboxyfluorescein | 30718681 | 70 | Mean Fluorescence intensity | 1 uM | 6h | NA | Flow cytometry | Uptake | GRRXRRXRRX |
| 932 | Ac5c | HeLa cells | Carboxyfluorescein | 30718681 | 60 | Mean Fluorescence intensity | 1 uM | 24h | NA | Flow cytometry | Uptake | GRRXRRXRRX |
| 933 | Arg | CHO-K1 cells | Carboxyfluorescein | 30718681 | 18 | Mean Fluorescence intensity | 1 uM | 2h | NA | Flow cytometry | Uptake | GRRRRRRRRR |
| 934 | Arg | CHO-K1 cells | Carboxyfluorescein | 30718681 | 12 | Mean Fluorescence intensity | 1 uM | 6h | NA | Flow cytometry | Uptake | GRRRRRRRRR |
| 935 | Arg | CHO-K1 cells | Carboxyfluorescein | 30718681 | 1 | Mean Fluorescence intensity | 1 uM | 24h | NA | Flow cytometry | Uptake | GRRRRRRRRR |
| 936 | Leu | CHO-K1 cells | Carboxyfluorescein | 30718681 | 5 | Mean Fluorescence intensity | 1 uM | 2h | NA | Flow cytometry | Uptake | GRRLRRLRRL |
| 937 | Leu | CHO-K1 cells | Carboxyfluorescein | 30718681 | 5 | Mean Fluorescence intensity | 1 uM | 6h | NA | Flow cytometry | Uptake | GRRLRRLRRL |
| 938 | Leu | CHO-K1 cells | Carboxyfluorescein | 30718681 | 1 | Mean Fluorescence intensity | 1 uM | 24h | NA | Flow cytometry | Uptake | GRRLRRLRRL |
| 939 | (?Me)Leu | CHO-K1 cells | Carboxyfluorescein | 30718681 | 15 | Mean Fluorescence intensity | 1 uM | 2h | NA | Flow cytometry | Uptake | GRRXRRXRRX |
| 940 | (?Me)Leu | CHO-K1 cells | Carboxyfluorescein | 30718681 | 22 | Mean Fluorescence intensity | 1 uM | 6h | NA | Flow cytometry | Uptake | GRRXRRXRRX |
| 941 | (?Me)Leu | CHO-K1 cells | Carboxyfluorescein | 30718681 | 11 | Mean Fluorescence intensity | 1 uM | 24h | NA | Flow cytometry | Uptake | GRRXRRXRRX |
| 942 | Ac5cdOM | CHO-K1 cells | Carboxyfluorescein | 30718681 | 5 | Mean Fluorescence intensity | 1 uM | 2h | NA | Flow cytometry | Uptake | GRRXRRXRRX |
| 943 | Ac5cdOM | CHO-K1 cells | Carboxyfluorescein | 30718681 | 11 | Mean Fluorescence intensity | 1 uM | 6h | NA | Flow cytometry | Uptake | GRRXRRXRRX |
| 944 | Ac5cdOM | CHO-K1 cells | Carboxyfluorescein | 30718681 | 10 | Mean Fluorescence intensity | 1 uM | 24h | NA | Flow cytometry | Uptake | GRRXRRXRRX |
| 945 | Ac5c | CHO-K1 cells | Carboxyfluorescein | 30718681 | 20 | Mean Fluorescence intensity | 1 uM | 2h | NA | Flow cytometry | Uptake | GRRXRRXRRX |
| 946 | Ac5c | CHO-K1 cells | Carboxyfluorescein | 30718681 | 40 | Mean Fluorescence intensity | 1 uM | 6h | NA | Flow cytometry | Uptake | GRRXRRXRRX |
| 947 | Ac5c | CHO-K1 cells | Carboxyfluorescein | 30718681 | 10 | Mean Fluorescence intensity | 1 uM | 24h | NA | Flow cytometry | Uptake | GRRXRRXRRX |
| 948 | KFE8-Tat | BMDC | FITC | 32686113 | 10 | % Positive cells | 0.5uM | 4h | 37ºC | Flow cytometry | Nanofiber uptake | FKFEFKFESGSGSG-RKKRRQRRRPQ |
| 949 | KFE8-Tat | BMDC | FITC | 32686113 | 25 | % Positive cells | 1uM | 4h | 37ºC | Flow cytometry | Nanofiber uptake | FKFEFKFESGSGSG-RKKRRQRRRPQ |
| 950 | KFE8-Tat | BMDC | FITC | 32686113 | 35 | % Positive cells | 2uM | 4h | 37ºC | Flow cytometry | Nanofiber uptake | FKFEFKFESGSGSG-RKKRRQRRRPQ |
| 951 | CyLoP-1 | HeLa cells | FITC | 27836642 | 250 | Mean Fluorescence intensity | 5uM | 2h | 37ºC | Flow cytometry | Cellular uptake | CRWRWKCCKK |
| 952 | CyLoP-1 | HeLa cells | FITC | 27836642 | 260 | Mean Fluorescence intensity | 10uM | 2h | 37ºC | Flow cytometry | Cellular uptake | CRWRWKCCKK |
| 953 | CyLoP-1 | HeLa cells | FITC | 27836642 | 350 | Mean Fluorescence intensity | 15uM | 2h | 37ºC | Flow cytometry | Cellular uptake | CRWRWKCCKK |
| 954 | CyLoP-1 | HeLa cells | FITC | 27836642 | 400 | Mean Fluorescence intensity | 20uM | 2h | 37ºC | Flow cytometry | Cellular uptake | CRWRWKCCKK |
| 955 | CyLoP-1 | HeLa cells | FITC | 27836642 | 450 | Mean Fluorescence intensity | 30uM | 2h | 37ºC | Flow cytometry | Cellular uptake | CRWRWKCCKK |
| 956 | CyLoP-1 | HeLa cells | FITC | 27836642 | 500 | Mean Fluorescence intensity | 40uM | 2h | 37ºC | Flow cytometry | Cellular uptake | CRWRWKCCKK |
| 957 | diTatBim | HeLa cells | AT520 | 29275934 | 50 | Mean Fluorescence intensity | 5uM | 30min | 37ºC | Fluorescent Microscopy | Cellular uptake | RKKRRQRRR-EIWIAQELRRIGDEFNAYYARLL-C-C-LLRAYYANFEDGIRRLEQAIWIE-RRRQRRKKR |
| 958 | mTatBim | HeLa cells | AT521 | 29275934 | 90 | Mean Fluorescence intensity | 10uM | 30min | 37ºC | Fluorescent Microscopy | Cellular uptake | RKKRRQRRR-EIWIAQELRRIGDEFNAYYARLL-C |
| 959 | NP1-EPT | CHO-K1 cells | EPT | 30673275 | 25 | Mean Fluorescence intensity | NA | NA | NA | Flow cytometry | Cellular uptake | stearyl-HHHHHHHHHHHHHHHH-RRRRRRRR-NH2 |
| 960 | NP1-EPT-2X | CHO-K1 cells | EPT | 30673275 | 15 | Mean Fluorescence intensity | NA | NA | NA | Flow cytometry | Cellular uptake | stearyl-HHHHHHHHHHHHHHHH-RRRRRRRR-NH3 |
| 961 | RRCPP | B16 cells | RRCPP/siRNA | 34375118 | 0 | NA | NA | NA | NA | Flow cytometry | Cellular uptake | RGDRRRRRRRRR |
| 962 | Cys-Trp-Trp-Arg8-Cys-Arg8- Cys-Arg8-Cys | Dendritic cells | peptide/OVA-Cy5.5 | 29359945 | 18 000 | Fluorescence intensity | NA | 4h | NA | Flow cytometry | Antigen Uptake | CWWRRRRRRRRCRRRRRRRRCRRRRRRRRC |
| 963 | CLIP6 | Dendritic cells | FITC | 31339694 | 50 | Fluorescence intensity | 10uM | 24h | 37ºC | Flow cytometry | Cellular uptake | KVRVRVRVDPPTRVRERVKC |
| 964 | [(RW)5K](RW) | CCRF-CEM cells | F'-GpYEEI | 34491768 | 120 | Mean Fluorescence intensity | 10uM | 3h | NA | Flow cytometry | Cellular uptake | RWRWRWRWRWKRWRWRWRWRW |
| 965 | [(RW)5K](RW)2 | CCRF-CEM cells | F'-GpYEEI | 34491768 | 100 | Mean Fluorescence intensity | 10uM | 3h | NA | Flow cytometry | Cellular uptake | RWRWRWRWRWKRWRWRWRWRW |
| 966 | [(RW)5K](RW)3 | CCRF-CEM cells | F'-GpYEEI | 34491768 | 200 | Mean Fluorescence intensity | 10uM | 3h | NA | Flow cytometry | Cellular uptake | RWRWRWRWRWKRWRWRWRWRW |
| 967 | [(RW)5K](RW)4 | CCRF-CEM cells | F'-GpYEEI | 34491768 | 300 | Mean Fluorescence intensity | 10uM | 3h | NA | Flow cytometry | Cellular uptake | RWRWRWRWRWKRWRWRWRWRW |
| 968 | [(RW)5K](RW)5 | CCRF-CEM cells | F'-GpYEEI | 34491768 | 500 | Mean Fluorescence intensity | 10uM | 3h | NA | Flow cytometry | Cellular uptake | RWRWRWRWRWKRWRWRWRWRW |
| 969 | [(RW)5K](RW) | SK-OV-3 cells | F'-GpYEEI | 34491768 | 100 | Mean Fluorescence intensity | 10uM | 3h | NA | Flow cytometry | Cellular uptake | RWRWRWRWRWKRWRWRWRWRW |
| 970 | [(RW)5K](RW)2 | SK-OV-3 cells | F'-GpYEEI | 34491768 | 120 | Mean Fluorescence intensity | 10uM | 3h | NA | Flow cytometry | Cellular uptake | RWRWRWRWRWKRWRWRWRWRW |
| 971 | [(RW)5K](RW)3 | SK-OV-3 cells | F'-GpYEEI | 34491768 | 120 | Mean Fluorescence intensity | 10uM | 3h | NA | Flow cytometry | Cellular uptake | RWRWRWRWRWKRWRWRWRWRW |
| 972 | [(RW)5K](RW)4 | SK-OV-3 cells | F'-GpYEEI | 34491768 | 130 | Mean Fluorescence intensity | 10uM | 3h | NA | Flow cytometry | Cellular uptake | RWRWRWRWRWKRWRWRWRWRW |
| 973 | [(RW)5K](RW)5 | SK-OV-3 cells | F'-GpYEEI | 34491768 | 130 | Mean Fluorescence intensity | 10uM | 3h | NA | Flow cytometry | Cellular uptake | RWRWRWRWRWKRWRWRWRWRW |
| 974 | PLL | Caco-2 cells | TPP | 33360901 | 18 | Cellular uptake | NA | 3h | NA | CLSM | Cellular uptake | poly-L-lysine |
| 975 | PLL | Caco-2 cells | PA | 33360901 | 15 | Cellular uptake | NA | 3h | NA | CLSM | Cellular uptake | poly-L-lysine |
| 976 | P1 | HSC-T6 | FITC | 34338123 | 800 | Fluorescence intensity | 5uM | 1h | 37ºC | Fluorescent Microscopy | Cellular uptake | (Acp)-KKKKKRFSFKKSFKLSGFSFKKNKK |
| 977 | P1 | A549 cells | FITC | 34338123 | 750 | Fluorescence intensity | 5uM | 1h | 37ºC | Fluorescent Microscopy | Cellular uptake | (Acp)-KKKKKRFSFKKSFKLSGFSFKKNKK |
| 978 | P1 | BV2 | FITC | 34338123 | 750 | Fluorescence intensity | 5uM | 1h | 37ºC | Fluorescent Microscopy | Cellular uptake | (Acp)-KKKKKRFSFKKSFKLSGFSFKKNKK |
| 979 | P1 | MCF7 cells | FITC | 34338123 | 900 | Fluorescence intensity | 5uM | 1h | 37ºC | Fluorescent Microscopy | Cellular uptake | (Acp)-KKKKKRFSFKKSFKLSGFSFKKNKK |
| 980 | CB1-sC18 | HeLa cells | daunorubicin (Dau) | 34959356 | 0 | Fluorescence intensity | 1uM | 2h | 37ºC | Flow cytometry | Cellular uptake | GLRKRLRKFRNKIKEK |
| 981 | CB2-sC18 | HeLa cells | daunorubicin (Dau) | 34959356 | 1000 | Fluorescence intensity | 1uM | 2h | 37ºC | Flow cytometry | Cellular uptake | GLRKRLRKFRNKIKEK |
| 982 | CB3-sC18 | HeLa cells | daunorubicin (Dau) | 34959356 | 2500 | Fluorescence intensity | 1uM | 2h | 37ºC | Flow cytometry | Cellular uptake | GLRKRLRKFRNKIKEK |
| 983 | CB4-sC18 | HeLa cells | daunorubicin (Dau) | 34959356 | 11000 | Fluorescence intensity | 1uM | 2h | 37ºC | Flow cytometry | Cellular uptake | GLRKRLRKFRNKIKEK |
| 984 | CB5-sC18 | HeLa cells | daunorubicin (Dau) | 34959356 | 2500 | Fluorescence intensity | 1uM | 2h | 37ºC | Flow cytometry | Cellular uptake | GLRKRLRKFRNKIKEK |
| 985 | CB1-sC18 | HeLa cells | daunorubicin (Dau) | 34959356 | 100 | Fluorescence intensity | 1uM | 30 min | 37ºC | Flow cytometry | Cellular uptake | GLRKRLRKFRNKIKEK |
| 986 | CB2-sC18 | HeLa cells | daunorubicin (Dau) | 34959356 | 300 | Fluorescence intensity | 1uM | 30 min | 37ºC | Flow cytometry | Cellular uptake | GLRKRLRKFRNKIKEK |
| 987 | CB3-sC18 | HeLa cells | daunorubicin (Dau) | 34959356 | 350 | Fluorescence intensity | 1uM | 30 min | 37ºC | Flow cytometry | Cellular uptake | GLRKRLRKFRNKIKEK |
| 988 | CB4-sC18 | HeLa cells | daunorubicin (Dau) | 34959356 | 1100 | Fluorescence intensity | 1uM | 30 min | 37ºC | Flow cytometry | Cellular uptake | GLRKRLRKFRNKIKEK |
| 989 | CB5-sC18 | HeLa cells | daunorubicin (Dau) | 34959356 | 200 | Fluorescence intensity | 1uM | 30 min | 37ºC | Flow cytometry | Cellular uptake | GLRKRLRKFRNKIKEK |
| 990 | SARTHI-1 | HeLa cells | Carboxyfluorescein | 30665017 | 500 | Hoechst fluorescence intensity | 10uM | 4h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KRKIFLRCKILV |
| 991 | SARTHI-2 | HeLa cells | Carboxyfluorescein | 30665017 | 600 | Hoechst fluorescence intensity | 10uM | 4h | 37ºC | Fluorescence spectroscopy | Cellular uptake | VLIKCRLFIKRK |
| 992 | SARTHI-3 | HeLa cells | Carboxyfluorescein | 30665017 | 1500 | Hoechst fluorescence intensity | 10uM | 4h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KRKIFLRCKILV |
| 993 | SARTHI-4 | HeLa cells | Carboxyfluorescein | 30665017 | 1000 | Hoechst fluorescence intensity | 10uM | 4h | 37ºC | Fluorescence spectroscopy | Cellular uptake | VLIKCRLFIKRK |
| 994 | SARTHI-1 | HeLa cells | Carboxyfluorescein | 30665017 | 3500 | Hoechst fluorescence intensity | 20uM | 4h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KRKIFLRCKILV |
| 995 | SARTHI-2 | HeLa cells | Carboxyfluorescein | 30665017 | 3500 | Hoechst fluorescence intensity | 20uM | 4h | 37ºC | Fluorescence spectroscopy | Cellular uptake | VLIKCRLFIKRK |
| 996 | SARTHI-3 | HeLa cells | Carboxyfluorescein | 30665017 | 2500 | Hoechst fluorescence intensity | 20uM | 4h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KRKIFLRCKILV |
| 997 | SARTHI-4 | HeLa cells | Carboxyfluorescein | 30665017 | 2000 | Hoechst fluorescence intensity | 20uM | 4h | 37ºC | Fluorescence spectroscopy | Cellular uptake | VLIKCRLFIKRK |
| 998 | SARTHI-1 | HeLa cells | Carboxyfluorescein | 30665017 | 3000 | Hoechst fluorescence intensity | 30uM | 4h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KRKIFLRCKILV |
| 999 | SARTHI-2 | HeLa cells | Carboxyfluorescein | 30665017 | 3200 | Hoechst fluorescence intensity | 30uM | 4h | 37ºC | Fluorescence spectroscopy | Cellular uptake | VLIKCRLFIKRK |
| 1000 | SARTHI-3 | HeLa cells | Carboxyfluorescein | 30665017 | 4000 | Hoechst fluorescence intensity | 30uM | 4h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KRKIFLRCKILV |
| 1001 | SARTHI-4 | HeLa cells | Carboxyfluorescein | 30665017 | 3750 | Hoechst fluorescence intensity | 30uM | 4h | 37ºC | Fluorescence spectroscopy | Cellular uptake | VLIKCRLFIKRK |
| 1002 | SARTHI-1 | HeLa cells | Carboxyfluorescein | 30665017 | 4750 | Hoechst fluorescence intensity | 40uM | 4h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KRKIFLRCKILV |
| 1003 | SARTHI-2 | HeLa cells | Carboxyfluorescein | 30665017 | 5500 | Hoechst fluorescence intensity | 40uM | 4h | 37ºC | Fluorescence spectroscopy | Cellular uptake | VLIKCRLFIKRK |
| 1004 | SARTHI-3 | HeLa cells | Carboxyfluorescein | 30665017 | 3500 | Hoechst fluorescence intensity | 40uM | 4h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KRKIFLRCKILV |
| 1005 | SARTHI-4 | HeLa cells | Carboxyfluorescein | 30665017 | 5400 | Hoechst fluorescence intensity | 40uM | 4h | 37ºC | Fluorescence spectroscopy | Cellular uptake | VLIKCRLFIKRK |
| 1006 | SARTHI-1 | HeLa cells | Carboxyfluorescein | 30665017 | 5800 | Hoechst fluorescence intensity | 50uM | 4h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KRKIFLRCKILV |
| 1007 | SARTHI-2 | HeLa cells | Carboxyfluorescein | 30665017 | 6600 | Hoechst fluorescence intensity | 50uM | 4h | 37ºC | Fluorescence spectroscopy | Cellular uptake | VLIKCRLFIKRK |
| 1008 | SARTHI-3 | HeLa cells | Carboxyfluorescein | 30665017 | 7500 | Hoechst fluorescence intensity | 50uM | 4h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KRKIFLRCKILV |
| 1009 | SARTHI-4 | HeLa cells | Carboxyfluorescein | 30665017 | 7000 | Hoechst fluorescence intensity | 50uM | 4h | 37ºC | Fluorescence spectroscopy | Cellular uptake | VLIKCRLFIKRK |
| 1010 | P2 | HeLa cells | FITC | 34463179 | 1700 | Fluorescence intensity | 5 uM | 1h | NA | Fluorescent Microscopy | Cellular uptake | (Acp)-RKRRQTSMTDFYHSKRRLIFS |
| 1011 | P2 | MCF7 cells | FITC | 34463179 | 1400 | Fluorescence intensity | 5 uM | 1h | NA | Fluorescent Microscopy | Cellular uptake | (Acp)-RKRRQTSMTDFYHSKRRLIFS |
| 1012 | P2 | HepG2 cells | FITC | 34463179 | 1400 | Fluorescence intensity | 5 uM | 1h | NA | Fluorescent Microscopy | Cellular uptake | (Acp)-RKRRQTSMTDFYHSKRRLIFS |
| 1013 | P2 | A549 cells | FITC | 34463179 | 1000 | Fluorescence intensity | 5 uM | 1h | NA | Fluorescent Microscopy | Cellular uptake | (Acp)-RKRRQTSMTDFYHSKRRLIFS |
| 1014 | P2 | HSC-T6 | FITC | 34463179 | 800 | Fluorescence intensity | 5 uM | 1h | NA | Fluorescent Microscopy | Cellular uptake | (Acp)-RKRRQTSMTDFYHSKRRLIFS |
| 1015 | R8 | U87 cells | LP | 30591464 | 7 | Mean Fluorescence intensity | NA | 4h | 37ºC | Flow cytometry | Cellular uptake | RRRRRRRR |
| 1016 | R8 | U87 cells | PLP | 30591464 | 12 | Mean Fluorescence intensity | NA | 4h | 37ºC | Flow cytometry | Cellular uptake | RRRRRRRR |
| 1017 | Tat | CHO cells | icg-labeled lactosomes | 27877876 | 0.38 | Cellular uptake | NA | 2h | 37ºC | Fluorescent Microscopy | Cellular uptake | YGRKKRRQRRR-C |
| 1018 | PTD4 | CHO cells | icg-labeled lactosomes | 27877876 | 0.1 | Cellular uptake | NA | 2h | 37ºC | Fluorescent Microscopy | Cellular uptake | YARAAARQARA-C |
| 1019 | DPV3 | CHO cells | icg-labeled lactosomes | 27877876 | 0.4 | Cellular uptake | NA | 2h | 37ºC | Fluorescent Microscopy | Cellular uptake | RKKRRRESRKKRRRES-C |
| 1020 | MPG?nlS | CHO cells | icg-labeled lactosomes | 27877876 | 0.39 | Cellular uptake | NA | 2h | 37ºC | Fluorescent Microscopy | Cellular uptake | GALFLGFLGAAGSTMGAWSQPKSKRKV-C |
| 1021 | R9MPG | CHO cells | icg-labeled lactosomes | 27877876 | 0.5 | Cellular uptake | NA | 2h | 37ºC | Fluorescent Microscopy | Cellular uptake | RRRRRRRRRGALFLAFLAAALSLMG-C |
| 1022 | Pep1 | CHO cells | icg-labeled lactosomes | 27877876 | 0.6 | Cellular uptake | NA | 2h | 37ºC | Fluorescent Microscopy | Cellular uptake | KETWWETWWTEWSQPKKKRKV-C |
| 1023 | EB1 | CHO cells | icg-labeled lactosomes | 27877876 | 1 | Cellular uptake | NA | 2h | 37ºC | Fluorescent Microscopy | Cellular uptake | LIRLWSHLIHIWFQNRRLKWKKK-C |
| 1024 | PB1-F2 fragment 1 | HEK293T cells | luciferin | 28284862 | 1.9 | Cellular uptake | 1.9 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-GSLKTRVLKR-NH2 |
| 1025 | PB1-F2 fragment 1 | HEK293T cells | luciferin | 28284862 | 2.7 | Cellular uptake | 5.6 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-GSLKTRVLKR-NH2 |
| 1026 | PB1-F2 fragment 1 | HEK293T cells | luciferin | 28284862 | 5.2 | Cellular uptake | 16.7 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-GSLKTRVLKR-NH2 |
| 1027 | PB1-F2 fragment 1 | HEK293T cells | luciferin | 28284862 | 11.2 | Cellular uptake | 50 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-GSLKTRVLKR-NH2 |
| 1028 | PB1-F2 fragment 2 | HEK293T cells | luciferin | 28284862 | 2.3 | Cellular uptake | 1.9 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-SLKTRVLKRW-NH2 |
| 1029 | PB1-F2 fragment 2 | HEK293T cells | luciferin | 28284862 | 3.1 | Cellular uptake | 5.6 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-SLKTRVLKRW-NH2 |
| 1030 | PB1-F2 fragment 2 | HEK293T cells | luciferin | 28284862 | 5.7 | Cellular uptake | 16.7 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-SLKTRVLKRW-NH2 |
| 1031 | PB1-F2 fragment 2 | HEK293T cells | luciferin | 28284862 | 16.7 | Cellular uptake | 50 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-SLKTRVLKRW-NH2 |
| 1032 | PB1-F2 fragment 3 | HEK293T cells | luciferin | 28284862 | 2.1 | Cellular uptake | 1.9 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-LKTRVLKRWK-NH2 |
| 1033 | PB1-F2 fragment 3 | HEK293T cells | luciferin | 28284862 | 3.1 | Cellular uptake | 5.6 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-LKTRVLKRWK-NH2 |
| 1034 | PB1-F2 fragment 3 | HEK293T cells | luciferin | 28284862 | 7.5 | Cellular uptake | 16.7 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-LKTRVLKRWK-NH2 |
| 1035 | PB1-F2 fragment 3 | HEK293T cells | luciferin | 28284862 | 30.1 | Cellular uptake | 50 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-LKTRVLKRWK-NH2 |
| 1036 | PB1-F2 fragment 4 | HEK293T cells | luciferin | 28284862 | 2.4 | Cellular uptake | 1.9 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-KTRVLKRWKL-NH2 |
| 1037 | PB1-F2 fragment 4 | HEK293T cells | luciferin | 28284862 | 3.2 | Cellular uptake | 5.6 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-KTRVLKRWKL-NH2 |
| 1038 | PB1-F2 fragment 4 | HEK293T cells | luciferin | 28284862 | 9.8 | Cellular uptake | 16.7 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-KTRVLKRWKL-NH2 |
| 1039 | PB1-F2 fragment 4 | HEK293T cells | luciferin | 28284862 | 30.7 | Cellular uptake | 50 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-KTRVLKRWKL-NH2 |
| 1040 | PB1-F2 fragment 5 | HEK293T cells | luciferin | 28284862 | 2.3 | Cellular uptake | 1.9 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-TRVLKRWKLF-NH2 |
| 1041 | PB1-F2 fragment 5 | HEK293T cells | luciferin | 28284862 | 3 | Cellular uptake | 5.6 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-TRVLKRWKLF-NH2 |
| 1042 | PB1-F2 fragment 5 | HEK293T cells | luciferin | 28284862 | 18.7 | Cellular uptake | 16.7 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-TRVLKRWKLF-NH2 |
| 1043 | PB1-F2 fragment 5 | HEK293T cells | luciferin | 28284862 | 216.3 | Cellular uptake | 50 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-TRVLKRWKLF-NH2 |
| 1044 | PB1-F2 fragment 6 | HEK293T cells | luciferin | 28284862 | 1.9 | Cellular uptake | 1.9 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-RVLKRWKLFN-NH2 |
| 1045 | PB1-F2 fragment 6 | HEK293T cells | luciferin | 28284862 | 3.4 | Cellular uptake | 5.6 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-RVLKRWKLFN-NH2 |
| 1046 | PB1-F2 fragment 6 | HEK293T cells | luciferin | 28284862 | 12 | Cellular uptake | 16.7 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-RVLKRWKLFN-NH2 |
| 1047 | PB1-F2 fragment 6 | HEK293T cells | luciferin | 28284862 | 198.2 | Cellular uptake | 50 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-RVLKRWKLFN-NH2 |
| 1048 | PB1-F2 fragment 7 | HEK293T cells | luciferin | 28284862 | 1.9 | Cellular uptake | 1.9 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-VLKRWKLFNK-NH2 |
| 1049 | PB1-F2 fragment 7 | HEK293T cells | luciferin | 28284862 | 2.8 | Cellular uptake | 5.6 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-VLKRWKLFNK-NH2 |
| 1050 | PB1-F2 fragment 7 | HEK293T cells | luciferin | 28284862 | 6.2 | Cellular uptake | 16.7 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-VLKRWKLFNK-NH2 |
| 1051 | PB1-F2 fragment 7 | HEK293T cells | luciferin | 28284862 | 30.3 | Cellular uptake | 50 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-VLKRWKLFNK-NH2 |
| 1052 | PB1-F2 fragment 8 | HEK293T cells | luciferin | 28284862 | 2.5 | Cellular uptake | 1.9 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-LKRWKLFNKQ-NH2 |
| 1053 | PB1-F2 fragment 8 | HEK293T cells | luciferin | 28284862 | 3.3 | Cellular uptake | 5.6 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-LKRWKLFNKQ-NH2 |
| 1054 | PB1-F2 fragment 8 | HEK293T cells | luciferin | 28284862 | 8 | Cellular uptake | 16.7 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-LKRWKLFNKQ-NH2 |
| 1055 | PB1-F2 fragment 8 | HEK293T cells | luciferin | 28284862 | 34.5 | Cellular uptake | 50 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-LKRWKLFNKQ-NH2 |
| 1056 | PB1-F2 fragment 9 | HEK293T cells | luciferin | 28284862 | 4 | Cellular uptake | 1.9 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-KRWKLFNKQE-NH2 |
| 1057 | PB1-F2 fragment 9 | HEK293T cells | luciferin | 28284862 | 3 | Cellular uptake | 5.6 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-KRWKLFNKQE-NH2 |
| 1058 | PB1-F2 fragment 9 | HEK293T cells | luciferin | 28284862 | 6.5 | Cellular uptake | 16.7 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-KRWKLFNKQE-NH2 |
| 1059 | PB1-F2 fragment 9 | HEK293T cells | luciferin | 28284862 | 13.6 | Cellular uptake | 50 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-KRWKLFNKQE-NH2 |
| 1060 | PB1-F2 fragment 10 | HEK293T cells | luciferin | 28284862 | 2.7 | Cellular uptake | 1.9 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-RWKLFNKQEW-NH2 |
| 1061 | PB1-F2 fragment 10 | HEK293T cells | luciferin | 28284862 | 3.5 | Cellular uptake | 5.6 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-RWKLFNKQEW-NH2 |
| 1062 | PB1-F2 fragment 10 | HEK293T cells | luciferin | 28284862 | 7.3 | Cellular uptake | 16.7 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-RWKLFNKQEW-NH2 |
| 1063 | PB1-F2 fragment 10 | HEK293T cells | luciferin | 28284862 | 18.2 | Cellular uptake | 50 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-RWKLFNKQEW-NH2 |
| 1064 | PB1-F2 fragment 11 | HEK293T cells | luciferin | 28284862 | 2.4 | Cellular uptake | 1.9 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-WKLFNKQEWT-NH2 |
| 1065 | PB1-F2 fragment 11 | HEK293T cells | luciferin | 28284862 | 3.3 | Cellular uptake | 5.6 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-WKLFNKQEWT-NH2 |
| 1066 | PB1-F2 fragment 11 | HEK293T cells | luciferin | 28284862 | 8 | Cellular uptake | 16.7 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-WKLFNKQEWT-NH2 |
| 1067 | PB1-F2 fragment 11 | HEK293T cells | luciferin | 28284862 | 14.7 | Cellular uptake | 50 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-WKLFNKQEWT-NH2 |
| 1068 | PB1-F2 fragment 12 | HEK293T cells | luciferin | 28284862 | 1.8 | Cellular uptake | 1.9 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-KLFNKQEWTN-NH2 |
| 1069 | PB1-F2 fragment 12 | HEK293T cells | luciferin | 28284862 | 2.4 | Cellular uptake | 5.6 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-KLFNKQEWTN-NH2 |
| 1070 | PB1-F2 fragment 12 | HEK293T cells | luciferin | 28284862 | 4.7 | Cellular uptake | 16.7 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-KLFNKQEWTN-NH2 |
| 1071 | PB1-F2 fragment 12 | HEK293T cells | luciferin | 28284862 | 9.7 | Cellular uptake | 50 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-KLFNKQEWTN-NH2 |
| 1072 | 1-luc | HEK293T cells | luciferin | 28284862 | 5.8 | Cellular uptake | 6.3 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Ac-CVAKYHGYPWCRRR-NH2 |
| 1073 | 1-luc | HEK293T cells | luciferin | 28284862 | 8.7 | Cellular uptake | 12.5 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Ac-CVAKYHGYPWCRRR-NH2 |
| 1074 | 1-luc | HEK293T cells | luciferin | 28284862 | 14.5 | Cellular uptake | 25 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Ac-CVAKYHGYPWCRRR-NH2 |
| 1075 | 1-luc | HEK293T cells | luciferin | 28284862 | 22.8 | Cellular uptake | 50 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Ac-CVAKYHGYPWCRRR-NH2 |
| 1076 | 2-luc | HEK293T cells | luciferin | 28284862 | 6.2 | Cellular uptake | 6.3 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Ac-CVAKYHGYPWCRRR-RRRRR-NH2 |
| 1077 | 2-luc | HEK293T cells | luciferin | 28284862 | 10.6 | Cellular uptake | 12.5 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Ac-CVAKYHGYPWCRRR-RRRRR-NH2 |
| 1078 | 2-luc | HEK293T cells | luciferin | 28284862 | 22.3 | Cellular uptake | 25 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Ac-CVAKYHGYPWCRRR-RRRRR-NH2 |
| 1079 | 2-luc | HEK293T cells | luciferin | 28284862 | 61 | Cellular uptake | 50 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Ac-CVAKYHGYPWCRRR-RRRRR-NH2 |
| 1080 | 5-luc | HEK293T cells | luciferin | 28284862 | 11.6 | Cellular uptake | 6.3 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Ac-CVAKYHGYPWCRRR-TRVLKRWKLF-NH2 |
| 1081 | 5-luc | HEK293T cells | luciferin | 28284862 | 21.3 | Cellular uptake | 12.5 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Ac-CVAKYHGYPWCRRR-TRVLKRWKLF-NH2 |
| 1082 | 5-luc | HEK293T cells | luciferin | 28284862 | 36.1 | Cellular uptake | 25 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Ac-CVAKYHGYPWCRRR-TRVLKRWKLF-NH2 |
| 1083 | 5-luc | HEK293T cells | luciferin | 28284862 | 66.8 | Cellular uptake | 50 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Ac-CVAKYHGYPWCRRR-TRVLKRWKLF-NH2 |
| 1084 | Tf-LPs | U87 cells | Doxorubicin | 31574945 | 40 | Fluorescence intensity | NA | 4h | NA | Flow cytometry | Cellular uptake | RRRRRRRR |
| 1085 | Tf-LPs | GL261 cells | Doxorubicin | 31574945 | 45 | Fluorescence intensity | NA | 4h | NA | Flow cytometry | Cellular uptake | RRRRRRRR |
| 1086 | PAS-pHK | MCF7 cells | miR-126 | 32491855 | 95 | % Internalization | 25 uM | 2h | 37ºC | Flow cytometry | Cellular uptake | GKPILFF |
| 1087 | CAAKA | A375 cells | QDs | 30240193 | 10 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CAAKA |
| 1088 | CAAKA | A375 cells | QDs | 30240193 | 17 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CAAKA |
| 1089 | CAAKA | MSTO cells | QDs | 30240193 | 8 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CAAKA |
| 1090 | CAAKA | MSTO cells | QDs | 30240193 | 25 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CAAKA |
| 1091 | CAAKA | 9L cells | QDs | 30240193 | 3 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CAAKA |
| 1092 | CAAKA | 9L cells | QDs | 30240193 | 3 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CAAKA |
| 1093 | CAAKA | LN18 cells | QDs | 30240193 | 8 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CAAKA |
| 1094 | CAAKA | U87 cells | QDs | 30240193 | 8 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CAAKA |
| 1095 | HSV1-VP22 | A375 cells | QDs | 30240193 | 15 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CDAATATRGRSAASRPTERPRAPARSASRPRRPVD |
| 1096 | HSV1-VP22 | A375 cells | QDs | 30240193 | 40 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CDAATATRGRSAASRPTERPRAPARSASRPRRPVD |
| 1097 | HSV1-VP22 | MSTO cells | QDs | 30240193 | 13 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CDAATATRGRSAASRPTERPRAPARSASRPRRPVD |
| 1098 | HSV1-VP22 | MSTO cells | QDs | 30240193 | 10 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CDAATATRGRSAASRPTERPRAPARSASRPRRPVD |
| 1099 | HSV1-VP22 | 9L cells | QDs | 30240193 | 20 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CDAATATRGRSAASRPTERPRAPARSASRPRRPVD |
| 1100 | HSV1-VP22 | 9L cells | QDs | 30240193 | 20 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CDAATATRGRSAASRPTERPRAPARSASRPRRPVD |
| 1101 | HSV1-VP22 | LN18 cells | QDs | 30240193 | 18 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CDAATATRGRSAASRPTERPRAPARSASRPRRPVD |
| 1102 | HSV1-VP22 | U87 cells | QDs | 30240193 | 36 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CDAATATRGRSAASRPTERPRAPARSASRPRRPVD |
| 1103 | HIV-TAT | A375 cells | QDs | 30240193 | 5 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CYGRKKRRQRRR |
| 1104 | HIV-TAT | A375 cells | QDs | 30240193 | 6 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CYGRKKRRQRRR |
| 1105 | HIV-TAT | MSTO cells | QDs | 30240193 | 4 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CYGRKKRRQRRR |
| 1106 | HIV-TAT | MSTO cells | QDs | 30240193 | 22 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CYGRKKRRQRRR |
| 1107 | HIV-TAT | 9L cells | QDs | 30240193 | 2 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CYGRKKRRQRRR |
| 1108 | HIV-TAT | 9L cells | QDs | 30240193 | 8 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CYGRKKRRQRRR |
| 1109 | HIV-TAT | LN18 cells | QDs | 30240193 | 18 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CYGRKKRRQRRR |
| 1110 | HIV-TAT | U87 cells | QDs | 30240193 | 10 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CYGRKKRRQRRR |
| 1111 | HIV-gp41 | A375 cells | QDs | 30240193 | 15 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CGALFLGWLGAAGSTMGA |
| 1112 | HIV-gp41 | A375 cells | QDs | 30240193 | 20 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CGALFLGWLGAAGSTMGA |
| 1113 | HIV-gp41 | MSTO cells | QDs | 30240193 | 21 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CGALFLGWLGAAGSTMGA |
| 1114 | HIV-gp41 | MSTO cells | QDs | 30240193 | 20 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CGALFLGWLGAAGSTMGA |
| 1115 | HIV-gp41 | 9L cells | QDs | 30240193 | 3 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CGALFLGWLGAAGSTMGA |
| 1116 | HIV-gp41 | 9L cells | QDs | 30240193 | 8 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CGALFLGWLGAAGSTMGA |
| 1117 | HIV-gp41 | LN18 cells | QDs | 30240193 | 15 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CGALFLGWLGAAGSTMGA |
| 1118 | HIV-gp41 | U87 cells | QDs | 30240193 | 10 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CGALFLGWLGAAGSTMGA |
| 1119 | Ku-70 | A375 cells | QDs | 30240193 | 30 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CPMLKE |
| 1120 | Ku-70 | A375 cells | QDs | 30240193 | 75 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CPMLKE |
| 1121 | Ku-70 | MSTO cells | QDs | 30240193 | 50 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CPMLKE |
| 1122 | Ku-70 | MSTO cells | QDs | 30240193 | 18 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CPMLKE |
| 1123 | Ku-70 | 9L cells | QDs | 30240193 | 26 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CPMLKE |
| 1124 | Ku-70 | 9L cells | QDs | 30240193 | 30 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CPMLKE |
| 1125 | Ku-70 | LN18 cells | QDs | 30240193 | 45 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CPMLKE |
| 1126 | Ku-70 | U87 cells | QDs | 30240193 | 50 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CPMLKE |
| 1127 | hCT(9-32) | A375 cells | QDs | 30240193 | 40 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CLGTYTQDFNKFHTFPQTAIGVGAP |
| 1128 | hCT(9-32) | A375 cells | QDs | 30240193 | 90 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CLGTYTQDFNKFHTFPQTAIGVGAP |
| 1129 | hCT(9-32) | MSTO cells | QDs | 30240193 | 40 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CLGTYTQDFNKFHTFPQTAIGVGAP |
| 1130 | hCT(9-32) | MSTO cells | QDs | 30240193 | 18 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CLGTYTQDFNKFHTFPQTAIGVGAP |
| 1131 | hCT(9-32) | 9L cells | QDs | 30240193 | 55 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CLGTYTQDFNKFHTFPQTAIGVGAP |
| 1132 | hCT(9-32) | 9L cells | QDs | 30240193 | 100 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CLGTYTQDFNKFHTFPQTAIGVGAP |
| 1133 | hCT(9-32) | LN18 cells | QDs | 30240193 | 20 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CLGTYTQDFNKFHTFPQTAIGVGAP |
| 1134 | hCT(9-32) | U87 cells | QDs | 30240193 | 40 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CLGTYTQDFNKFHTFPQTAIGVGAP |
| 1135 | integrin ß3 | A375 cells | QDs | 30240193 | 5 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CVTVLALGALAGVGVG |
| 1136 | integrin ß3 | A375 cells | QDs | 30240193 | 6 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CVTVLALGALAGVGVG |
| 1137 | integrin ß3 | MSTO cells | QDs | 30240193 | 10 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CVTVLALGALAGVGVG |
| 1138 | integrin ß3 | MSTO cells | QDs | 30240193 | 18 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CVTVLALGALAGVGVG |
| 1139 | integrin ß3 | 9L cells | QDs | 30240193 | 2 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CVTVLALGALAGVGVG |
| 1140 | integrin ß3 | 9L cells | QDs | 30240193 | 4 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CVTVLALGALAGVGVG |
| 1141 | integrin ß3 | LN18 cells | QDs | 30240193 | 3 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CVTVLALGALAGVGVG |
| 1142 | integrin ß3 | U87 cells | QDs | 30240193 | 18 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CVTVLALGALAGVGVG |
| 1143 | K-FGF | A375 cells | QDs | 30240193 | 6 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CAAVALLPAVLLAHLLAP |
| 1144 | K-FGF | A375 cells | QDs | 30240193 | 10 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CAAVALLPAVLLAHLLAP |
| 1145 | K-FGF | MSTO cells | QDs | 30240193 | 15 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CAAVALLPAVLLAHLLAP |
| 1146 | K-FGF | MSTO cells | QDs | 30240193 | 18 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CAAVALLPAVLLAHLLAP |
| 1147 | K-FGF | 9L cells | QDs | 30240193 | 5 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CAAVALLPAVLLAHLLAP |
| 1148 | K-FGF | 9L cells | QDs | 30240193 | 5 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CAAVALLPAVLLAHLLAP |
| 1149 | K-FGF | LN18 cells | QDs | 30240193 | 5 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CAAVALLPAVLLAHLLAP |
| 1150 | K-FGF | U87 cells | QDs | 30240193 | 23 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CAAVALLPAVLLAHLLAP |
| 1151 | His8 | N. tabacum cells | MBP-RFP | 33791772 | 400 | Fluorescence intensity | 5 uM | 24h | 27ºC | CLSM | Cellular uptake | HHHHHHHH |
| 1152 | His12 | N. tabacum cells | MBP-RFP | 33791772 | 1000 | Fluorescence intensity | 5 uM | 24h | 27ºC | CLSM | Cellular uptake | HHHHHHHHHHHH |
| 1153 | His16 | N. tabacum cells | MBP-RFP | 33791772 | 1500 | Fluorescence intensity | 5 uM | 24h | 27ºC | CLSM | Cellular uptake | HHHHHHHHHHHHHHHH |
| 1154 | His20 | N. tabacum cells | MBP-RFP | 33791772 | 2800 | Fluorescence intensity | 5 uM | 24h | 27ºC | CLSM | Cellular uptake | HHHHHHHHHHHHHHHHHHHH |
| 1155 | His8 | O. Sativa cells | MBP-RFP | 33791772 | 1000 | Fluorescence intensity | 5 uM | 24h | 27ºC | CLSM | Cellular uptake | HHHHHHHH |
| 1156 | His12 | O. Sativa cells | MBP-RFP | 33791772 | 1100 | Fluorescence intensity | 5 uM | 24h | 27ºC | CLSM | Cellular uptake | HHHHHHHHHHHH |
| 1157 | His16 | O. Sativa cells | MBP-RFP | 33791772 | 3000 | Fluorescence intensity | 5 uM | 24h | 27ºC | CLSM | Cellular uptake | HHHHHHHHHHHHHHHH |
| 1158 | His20 | O. Sativa cells | MBP-RFP | 33791772 | 2900 | Fluorescence intensity | 5 uM | 24h | 27ºC | CLSM | Cellular uptake | HHHHHHHHHHHHHHHHHHHH |
| 1159 | His8 | C. japonica cells | MBP-RFP | 33791772 | 800 | Fluorescence intensity | 5 uM | 24h | 27ºC | CLSM | Cellular uptake | HHHHHHHH |
| 1160 | His12 | C. japonica cells | MBP-RFP | 33791772 | 2000 | Fluorescence intensity | 5 uM | 24h | 27ºC | CLSM | Cellular uptake | HHHHHHHHHHHH |
| 1161 | His16 | C. japonica cells | MBP-RFP | 33791772 | 6000 | Fluorescence intensity | 5 uM | 24h | 27ºC | CLSM | Cellular uptake | HHHHHHHHHHHHHHHH |
| 1162 | His20 | C. japonica cells | MBP-RFP | 33791772 | 10100 | Fluorescence intensity | 5 uM | 24h | 27ºC | CLSM | Cellular uptake | HHHHHHHHHHHHHHHHHHHH |
| 1163 | His6 | N. tabacum cells | MBP-RFP-CyaA | 33791772 | 180 | Fluorescence intensity | 2 uM | 6h | 27ºC | CLSM | Cellular uptake | HHHHHH |
| 1164 | His20 | N. tabacum cells | MBP-RFP-CyaA | 33791772 | 350 | Fluorescence intensity | 2 uM | 6h | 27ºC | CLSM | Cellular uptake | HHHHHHHHHHHHHHHHHHHH |
| 1165 | His6 | O. Sativa cells | MBP-RFP-CyaA | 33791772 | 150 | Fluorescence intensity | 2 uM | 1h | 27ºC | CLSM | Cellular uptake | HHHHHH |
| 1166 | His20 | O. Sativa cells | MBP-RFP-CyaA | 33791772 | 380 | Fluorescence intensity | 2 uM | 1h | 27ºC | CLSM | Cellular uptake | HHHHHHHHHHHHHHHHHHHH |
| 1167 | His6 | C. japonica cells | MBP-RFP-CyaA | 33791772 | 100 | Fluorescence intensity | 0.5 uM | 1h | 27ºC | CLSM | Cellular uptake | HHHHHH |
| 1168 | His20 | C. japonica cells | MBP-RFP-CyaA | 33791772 | 160 | Fluorescence intensity | 0.5 uM | 1h | 27ºC | CLSM | Cellular uptake | HHHHHHHHHHHHHHHHHHHH |
| 1169 | Xentry-KALA (XK) | ARPE-19 cells | Cx43AsODN) | 30050146 | 0 | Fluorescence | 1 uM | 4h | 37ºC | Fluorescent Microscopy | Cellular uptake | (biotin)-lclrpvgggweaklakalakalakhlakalakalkacea |
| 1170 | Xentry-Protamine (XP) | ARPE-19 cells | Cx43AsODN) | 30050146 | 0 | Fluorescence | 1 uM | 4h | 37ºC | Fluorescent Microscopy | Cellular uptake | (biotin)-lclrpvggrsqsrsryyrqrqrsrrrrrrs |
| 1171 | WRAP1 | U87 cells | siRNA | 32135145 | 0 | NA | NA | 24h | NA | CLSM | Cellular uptake | LLWRLWRLLW-RLWRLL |
| 1172 | WRAP5 | U87 cells | siRNA | 32135145 | 0 | NA | NA | 24h | NA | CLSM | Cellular uptake | LLRLLRWWWRLLRLL |
| 1173 | pHK-PASA488 | pgsA-745 cells | HKII | 28183803 | 1.63 | Fluorescence intensity | 25uM | 2h | 37ºC | Flow cytometry | Cellular uptake | MIASHLLAYFFTELNGKPILFF |
| 1174 | R16-CD63-GFP | CHO-K1 cells | EVs | 31810935 | 100 | Relative Cellular uptake | NA | 24h | 37ºC | Flow cytometry | Cellular uptake | CGRRRRRRRRRRRRRRRR |
| 1175 | R16-CD63-GFP | CHO-K1 cells | Evs w/ lyophilization | 31810935 | 100 | Relative Cellular uptake | NA | 24h | 37ºC | Flow cytometry | Cellular uptake | CGRRRRRRRRRRRRRRRR |
| 1176 | R16-CD63-GFP | CHO cells | EVs | 31810935 | 55 | Relative Cellular uptake | NA | 24h | 37ºC | Flow cytometry | Cellular uptake | CGRRRRRRRRRRRRRRRR |
| 1177 | R16-CD63-GFP | CHO cells | Evs w/ lyophilization | 31810935 | 49 | Relative Cellular uptake | NA | 24h | 37ºC | Flow cytometry | Cellular uptake | CGRRRRRRRRRRRRRRRR |
| 1178 | AMO/PF6 | A549 cells | 99mTc | 33480702 | 1.6 | Cellular retention (mol/cell x 10-16) | 37 kBq | 1h | 37ºC | CLSM | Cellular uptake | AGYLLGKINLKALAALAKKIL |
| 1179 | AMO/PF6 | A549 cells | 99mTc | 33480702 | 1.8 | Cellular retention (mol/cell x 10-16) | 37 kBq | 2h | 37ºC | CLSM | Cellular uptake | AGYLLGKINLKALAALAKKIL |
| 1180 | AMO/PF6 | A549 cells | 99mTc | 33480702 | 4.5 | Cellular retention (mol/cell x 10-16) | 37 kBq | 4h | 37ºC | CLSM | Cellular uptake | AGYLLGKINLKALAALAKKIL |
| 1181 | AMO/PF6 | A549 cells | 99mTc | 33480702 | 6.8 | Cellular retention (mol/cell x 10-16) | 37 kBq | 6h | 37ºC | CLSM | Cellular uptake | AGYLLGKINLKALAALAKKIL |
| 1182 | AMO/PF6 | A549 cells | 99mTc | 33480702 | 11.24 | Cellular retention (mol/cell x 10-16) | 37 kBq | 12h | 37ºC | CLSM | Cellular uptake | AGYLLGKINLKALAALAKKIL |
| 1183 | AMO/PF6 | A549 cells | 99mTc | 33480702 | 10.42 | Cellular retention (mol/cell x 10-16) | 37 kBq | 24h | 37ºC | CLSM | Cellular uptake | AGYLLGKINLKALAALAKKIL |
| 1184 | misAMO/PF6 | A549 cells | 99mTc | 33480702 | 1.3 | Cellular retention (mol/cell x 10-16) | 37 kBq | 1h | 37ºC | CLSM | Cellular uptake | AGYLLGKINLKALAALAKKIL |
| 1185 | misAMO/PF6 | A549 cells | 99mTc | 33480702 | 1.8 | Cellular retention (mol/cell x 10-16) | 37 kBq | 2h | 37ºC | CLSM | Cellular uptake | AGYLLGKINLKALAALAKKIL |
| 1186 | misAMO/PF6 | A549 cells | 99mTc | 33480702 | 3.3 | Cellular retention (mol/cell x 10-16) | 37 kBq | 4h | 37ºC | CLSM | Cellular uptake | AGYLLGKINLKALAALAKKIL |
| 1187 | misAMO/PF6 | A549 cells | 99mTc | 33480702 | 5.8 | Cellular retention (mol/cell x 10-16) | 37 kBq | 6h | 37ºC | CLSM | Cellular uptake | AGYLLGKINLKALAALAKKIL |
| 1188 | misAMO/PF6 | A549 cells | 99mTc | 33480702 | 10.66 | Cellular retention (mol/cell x 10-16) | 37 kBq | 12h | 37ºC | CLSM | Cellular uptake | AGYLLGKINLKALAALAKKIL |
| 1189 | misAMO/PF6 | A549 cells | 99mTc | 33480702 | 9.2 | Cellular retention (mol/cell x 10-16) | 37 kBq | 24h | 37ºC | CLSM | Cellular uptake | AGYLLGKINLKALAALAKKIL |
| 1190 | LDP-NLS | HeLa cells | FITC | 28159722 | 50100 | FITC Mean Intensity | 20 uM | 1h | 37ºC | Flow cytometry | Cellular uptake | KWRRKLKKLRPKKKRKV |
| 1191 | LDP | HeLa cells | FITC | 28159722 | 8000 | FITC Mean Intensity | 20 uM | 1h | 37ºC | Flow cytometry | Cellular uptake | KWRRKLKKLR |
| 1192 | NLS | HeLa cells | FITC | 28159722 | 0 | FITC Mean Intensity | 20 uM | 1h | 37ºC | Flow cytometry | Cellular uptake | PKKKRKV |
| 1193 | Mut-LDP-NLS | HeLa cells | FITC | 28159722 | 0 | FITC Mean Intensity | 20 uM | 1h | 37ºC | Flow cytometry | Cellular uptake | AWRRKLKALAPAKKAKV |
| 1194 | cR10 | U2OS cells | FITC | 33615660 | 0 | FITC signal | 6 uM | 15 min | NA | CLSM | Cellular uptake | LYRAGLYRAGLYKAGCG |
| 1195 | cR10DABCYL | U2OS cells | FITC | 33615660 | 0 | FITC signal | 6 uM | 15 min | NA | CLSM | Cellular uptake | LYRAGLYRAGLYKAGCG-DABCYL |
| 1196 | Ub-SScR10 | U2OS cells | TAMPA | 33615660 | 18 | TAMPA intensity | 2 uM | 1h | NA | CLSM | Cellular uptake | LYRAGLYRAGLYKAGCGRRRRRRRRRR |
| 1197 | Ub-SScR10D | U2OS cells | TAMPA | 33615660 | 50 | TAMPA intensity | 12 uM | 1h | NA | CLSM | Cellular uptake | LYRAGLYRAGLYKAGCGRRRRRRRRRR |
| 1198 | Tat-PTD | HDF cells | FITC | 32374475 | 264.6±23.21 | Relative fluorescence | 0.2uM | 30min | 37ºC | Flow cytometry | Cellular uptake | GRKKRRQRRK |
| 1199 | Tat-PTD | HDF cells | FITC | 32374475 | 209.00±29.67 | Relative fluorescence | 2uM | 30min | 37ºC | Flow cytometry | Cellular uptake | GRKKRRQRRK |
| 1200 | Ara-27 | HDF cells | FITC | 32374475 | 210.33±17.90 | Relative fluorescence | 0.2uM | 30min | 37ºC | Flow cytometry | Cellular uptake | RNQRKTVRCFRCRQAGHWISDCRLKSK |
| 1201 | Ara-27 | HDF cells | FITC | 32374475 | 1800.33±590.46 | Relative fluorescence | 2uM | 30min | 37ºC | Flow cytometry | Cellular uptake | RNQRKTVRCFRCRQAGHWISDCRLKSK |
| 1202 | Tat-PTD | hDPSC cells | FITC | 32374475 | 174.67±8.45 | Relative fluorescence | 0.2uM | 30min | 37ºC | Flow cytometry | Cellular uptake | GRKKRRQRRK |
| 1203 | Tat-PTD | hDPSC cells | FITC | 32374475 | 231.00±42.12 | Relative fluorescence | 2uM | 30min | 37ºC | Flow cytometry | Cellular uptake | GRKKRRQRRK |
| 1204 | Ara-27 | hDPSC cells | FITC | 32374475 | 240.00±27.75 | Relative fluorescence | 0.2uM | 30min | 37ºC | Flow cytometry | Cellular uptake | RNQRKTVRCFRCRQAGHWISDCRLKSK |
| 1205 | Ara-27 | hDPSC cells | FITC | 32374475 | 4985.67±335.33 | Relative fluorescence | 2uM | 30min | 37ºC | Flow cytometry | Cellular uptake | RNQRKTVRCFRCRQAGHWISDCRLKSK |
| 1206 | MSN@PLA–PEG-CPP | HT29 cells | FITC | 32697099 | 0.65 | Relative Mean Fluorescence intensity | NA | 1h | 37ºC | CLSM | Cellular uptake | VSRRRRRRGGRRRRC |
| 1207 | MSN@PLA–PEG-CPP | HT29 cells | FITC | 32697099 | 1.35 | Relative Mean Fluorescence intensity | NA | 3h | 37ºC | CLSM | Cellular uptake | VSRRRRRRGGRRRRC |
| 1208 | MSN@PLA–PEG-CPP | HT29 cells | FITC | 32697099 | 2.6 | Relative Mean Fluorescence intensity | NA | 6h | 37ºC | CLSM | Cellular uptake | VSRRRRRRGGRRRRC |
| 1209 | CPP-Dot1l | MCF7 cells | FITC | 32024261 | 1100 | Fluorescence intensity | 2.5uM | 1h | NA | Fluorescent Microscopy | Cellular uptake | KARKKKLNKKGRKMAGRKRGRPKK |
| 1210 | CPP-Dot1l | MCF7 cells | FITC | 32024261 | 1400 | Fluorescence intensity | 5uM | 1h | NA | Fluorescent Microscopy | Cellular uptake | KARKKKLNKKGRKMAGRKRGRPKK |
| 1211 | CPP-Dot1l | MCF7 cells | FITC | 32024261 | 1450 | Fluorescence intensity | 7.5uM | 1h | NA | Fluorescent Microscopy | Cellular uptake | KARKKKLNKKGRKMAGRKRGRPKK |
| 1212 | CPP-Dot1l | MCF7 cells | FITC | 32024261 | 1900 | Fluorescence intensity | 10uM | 1h | NA | Fluorescent Microscopy | Cellular uptake | KARKKKLNKKGRKMAGRKRGRPKK |
| 1213 | NCO | MCF7 cells | FITC | 32024261 | 200 | Fluorescence intensity | 2.5uM | 1h | NA | Fluorescent Microscopy | Cellular uptake | KALGISYGRKK |
| 1214 | NCO | MCF7 cells | FITC | 32024261 | 100 | Fluorescence intensity | 5uM | 1h | NA | Fluorescent Microscopy | Cellular uptake | KALGISYGRKK |
| 1215 | NCO | MCF7 cells | FITC | 32024261 | 300 | Fluorescence intensity | 7.5uM | 1h | NA | Fluorescent Microscopy | Cellular uptake | KALGISYGRKK |
| 1216 | NCO | MCF7 cells | FITC | 32024261 | 300 | Fluorescence intensity | 10uM | 1h | NA | Fluorescent Microscopy | Cellular uptake | KALGISYGRKK |
| 1217 | NLS-A | PK15 cells | FITC | 30108178 | 690 | Fluorescence intensity | 6uM | 30 min | 37ºC | Flow cytometry | Cellular uptake | MTYPRRRFRRRRHRPRS |
| 1218 | NLS-A | HeLa cells | FITC | 30108178 | 580 | Fluorescence intensity | 6uM | 30 min | 37ºC | Flow cytometry | Cellular uptake | MTYPRRRFRRRRHRPRS |
| 1219 | NLS-A | NIH-3T3 cells | FITC | 30108178 | 750 | Fluorescence intensity | 6uM | 30 min | 37ºC | Flow cytometry | Cellular uptake | MTYPRRRFRRRRHRPRS |
| 1220 | TAT0 | HeLa cells | HPMA | 31936737 | 8 | Relative Median Fluorescence | 1uM | 1h | 4ºC | Flow cytometry | Cellular uptake | GRKKRRQRRR |
| 1221 | TAT0 | HeLa cells | HPMA | 31936737 | 7 | Relative Median Fluorescence | 10uM | 1h | 4ºC | Flow cytometry | Cellular uptake | GRKKRRQRRR |
| 1222 | TAT0 | HeLa cells | HPMA | 31936737 | 32 | Relative Median Fluorescence | 25uM | 1h | 4ºC | Flow cytometry | Cellular uptake | GRKKRRQRRR |
| 1223 | TAT0 | HeLa cells | HPMA | 31936737 | 28 | Relative Median Fluorescence | 50uM | 1h | 4ºC | Flow cytometry | Cellular uptake | GRKKRRQRRR |
| 1224 | TAT4 | HeLa cells | HPMA | 31936737 | 7 | Relative Median Fluorescence | 1uM | 1h | 4ºC | Flow cytometry | Cellular uptake | GRKKRRQRRR |
| 1225 | TAT4 | HeLa cells | HPMA | 31936737 | 12 | Relative Median Fluorescence | 10uM | 1h | 4ºC | Flow cytometry | Cellular uptake | GRKKRRQRRR |
| 1226 | TAT4 | HeLa cells | HPMA | 31936737 | 50 | Relative Median Fluorescence | 25uM | 1h | 4ºC | Flow cytometry | Cellular uptake | GRKKRRQRRR |
| 1227 | TAT4 | HeLa cells | HPMA | 31936737 | 53 | Relative Median Fluorescence | 50uM | 1h | 4ºC | Flow cytometry | Cellular uptake | GRKKRRQRRR |
| 1228 | TAT12 | HeLa cells | HPMA | 31936737 | 5 | Relative Median Fluorescence | 1uM | 1h | 4ºC | Flow cytometry | Cellular uptake | GRKKRRQRRR |
| 1229 | TAT12 | HeLa cells | HPMA | 31936737 | 22 | Relative Median Fluorescence | 10uM | 1h | 4ºC | Flow cytometry | Cellular uptake | GRKKRRQRRR |
| 1230 | TAT12 | HeLa cells | HPMA | 31936737 | 58 | Relative Median Fluorescence | 25uM | 1h | 4ºC | Flow cytometry | Cellular uptake | GRKKRRQRRR |
| 1231 | TAT12 | HeLa cells | HPMA | 31936737 | 75 | Relative Median Fluorescence | 50uM | 1h | 4ºC | Flow cytometry | Cellular uptake | GRKKRRQRRR |
| 1232 | PEN0 | HeLa cells | HPMA | 31936737 | 11 | Relative Median Fluorescence | 1uM | 1h | 4ºC | Flow cytometry | Cellular uptake | RRMKWKK |
| 1233 | PEN0 | HeLa cells | HPMA | 31936737 | 18 | Relative Median Fluorescence | 10uM | 1h | 4ºC | Flow cytometry | Cellular uptake | RRMKWKK |
| 1234 | PEN0 | HeLa cells | HPMA | 31936737 | 12 | Relative Median Fluorescence | 25uM | 1h | 4ºC | Flow cytometry | Cellular uptake | RRMKWKK |
| 1235 | PEN0 | HeLa cells | HPMA | 31936737 | 12 | Relative Median Fluorescence | 50uM | 1h | 4ºC | Flow cytometry | Cellular uptake | RRMKWKK |
| 1236 | PEN4 | HeLa cells | HPMA | 31936737 | 8 | Relative Median Fluorescence | 1uM | 1h | 4ºC | Flow cytometry | Cellular uptake | RRMKWKK |
| 1237 | PEN4 | HeLa cells | HPMA | 31936737 | 17 | Relative Median Fluorescence | 10uM | 1h | 4ºC | Flow cytometry | Cellular uptake | RRMKWKK |
| 1238 | PEN4 | HeLa cells | HPMA | 31936737 | 13 | Relative Median Fluorescence | 25uM | 1h | 4ºC | Flow cytometry | Cellular uptake | RRMKWKK |
| 1239 | PEN4 | HeLa cells | HPMA | 31936737 | 13 | Relative Median Fluorescence | 50uM | 1h | 4ºC | Flow cytometry | Cellular uptake | RRMKWKK |
| 1240 | PEN12 | HeLa cells | HPMA | 31936737 | 10 | Relative Median Fluorescence | 1uM | 1h | 4ºC | Flow cytometry | Cellular uptake | RRMKWKK |
| 1241 | PEN12 | HeLa cells | HPMA | 31936737 | 27 | Relative Median Fluorescence | 10uM | 1h | 4ºC | Flow cytometry | Cellular uptake | RRMKWKK |
| 1242 | PEN12 | HeLa cells | HPMA | 31936737 | 26 | Relative Median Fluorescence | 25uM | 1h | 4ºC | Flow cytometry | Cellular uptake | RRMKWKK |
| 1243 | PEN12 | HeLa cells | HPMA | 31936737 | 25 | Relative Median Fluorescence | 50uM | 1h | 4ºC | Flow cytometry | Cellular uptake | RRMKWKK |
| 1244 | d-Pen | C2C12 cells | Streptavidin-Alexa555 | 29045142 | 0 | NA | 50uM | 10min | NA | BCARS Imaging | Cellular uptake | GGGGGGRQIKIWFQNRRMKWKKK-biotinyl-NH2 |
| 1245 | rEETI-II | HeLa cells | Alexa488 | 27734922 | 0 | NA | 20uM | 45min | 37ºC | Fluorescence imaging | Cellular uptake | GSGCPRILMRCKQDSDCLAGCVCGPNGFCGGNS |
| 1246 | R8-Alexa488 | A431 cells | Cyt D | 29743505 | 0 | NA | 2uM | 15 min | 37ºC | Flow cytometry | Cellular uptake | RRRRRRR-GC |
| 1247 | R8-Alexa488 | HeLa cells | Cyt D | 29743505 | 0 | NA | 2uM | 15 min | 37ºC | Flow cytometry | Cellular uptake | RRRRRRR-GC |
| 1248 | EGFP-R8 | A431 cells | Lat B | 29743505 | 0 | NA | 2uM | 1h | 37ºC | Flow cytometry | Cellular uptake | RRRRRRR-GC |
| 1249 | EGFP-R8 | A431 cells | JAS | 29743505 | 0 | NA | 2uM | 1h | 37ºC | Flow cytometry | Cellular uptake | RRRRRRR-GC |
| 1250 | RFFR | SH-SY5Y cells | TAMPA | 35019611 | 0 | NA | 100 ug/mL | 30min | 37ºC | CLSM | Cellular uptake | RFFR |
| 1251 | RFFR | NIH-3T3 cells | TAMPA | 35019611 | 0 | NA | 100 ug/mL | 30min | 37ºC | CLSM | Cellular uptake | RFFR |
| 1252 | RFFR | HeLa cells | TAMPA | 35019611 | 0 | NA | 100 ug/mL | 30min | 37ºC | CLSM | Cellular uptake | RFFR |
| 1253 | Tat | HeLa cells | Alexa488 | 34152716 | 1 | Mean Fluorescence intensity | 4uM | 1h | 37ºC | Flow cytometry | Cellular uptake | YGRKKRRQRRRPPQG |
| 1254 | Tat-G | HeLa cells | Alexa488 | 34152716 | 0.2 | Mean Fluorescence intensity | 4uM | 1h | 37ºC | Flow cytometry | Cellular uptake | YGGGKGGQGGGPPQG |
| 1255 | MCNr-2 | HeLa cells | Alexa488 | 34152716 | 0.3 | Mean Fluorescence intensity | 4uM | 1h | 37ºC | Flow cytometry | Cellular uptake | CPKILKKCRRDSDCPGACICRGNGYCGSGSDEETGEGGV |
| 1256 | MCNr-2c | HeLa cells | Alexa488 | 34152716 | 0.4 | Mean Fluorescence intensity | 4uM | 1h | 37ºC | Flow cytometry | Cellular uptake | CPFWRRRRCKRDSDCPGACICRGNGYCGSGCDEETGECGV |
| 1257 | R2W4R2 | MCF7 cells | FITC | 32116040 | 25 | Cell fluorescence (%) | 5uM | 1h | 37ºC | Flow cytometry | Cellular uptake | RRWWWWRR |
| 1258 | R2W4R2 | MCF7 cells | FITC | 32116040 | 72 | Cell fluorescence (%) | 10uM | 1h | 37ºC | Flow cytometry | Cellular uptake | RRWWWWRR |
| 1259 | R2W4R2 | MCF7 cells | FITC | 32116040 | 70 | Cell fluorescence (%) | 15uM | 1h | 37ºC | Flow cytometry | Cellular uptake | RRWWWWRR |
| 1260 | R2W4R2 | MCF7 cells | FITC | 32116040 | 93 | Cell fluorescence (%) | 25uM | 1h | 37ºC | Flow cytometry | Cellular uptake | RRWWWWRR |
| 1261 | W3R4W3 | MCF7 cells | FITC | 32116040 | 2 | Cell fluorescence (%) | 5uM | 1h | 37ºC | Flow cytometry | Cellular uptake | WWWRRRRWWW |
| 1262 | W3R4W3 | MCF7 cells | FITC | 32116040 | 2 | Cell fluorescence (%) | 10uM | 1h | 37ºC | Flow cytometry | Cellular uptake | WWWRRRRWWW |
| 1263 | W3R4W3 | MCF7 cells | FITC | 32116040 | 8 | Cell fluorescence (%) | 15uM | 1h | 37ºC | Flow cytometry | Cellular uptake | WWWRRRRWWW |
| 1264 | W3R4W3 | MCF7 cells | FITC | 32116040 | 12 | Cell fluorescence (%) | 25uM | 1h | 37ºC | Flow cytometry | Cellular uptake | WWWRRRRWWW |
| 1265 | R2W4R2-E12 | MCF7 cells | FITC | 32116040 | 10 | Cell fluorescence (%) | 5uM | 1h | 37ºC | Flow cytometry | Cellular uptake | RRWWWWRR-E12 |
| 1266 | R2W4R2-E12 | MCF7 cells | FITC | 32116040 | 18 | Cell fluorescence (%) | 10uM | 1h | 37ºC | Flow cytometry | Cellular uptake | RRWWWWRR-E12 |
| 1267 | R2W4R2-E12 | MCF7 cells | FITC | 32116040 | 41 | Cell fluorescence (%) | 15uM | 1h | 37ºC | Flow cytometry | Cellular uptake | RRWWWWRR-E12 |
| 1268 | R2W4R2-E12 | MCF7 cells | FITC | 32116040 | 45 | Cell fluorescence (%) | 25uM | 1h | 37ºC | Flow cytometry | Cellular uptake | RRWWWWRR-E12 |
| 1269 | W3R4W3-E12 | MCF7 cells | FITC | 32116040 | 3 | Cell fluorescence (%) | 5uM | 1h | 37ºC | Flow cytometry | Cellular uptake | WWWRRRRWWW-E12 |
| 1270 | W3R4W3-E12 | MCF7 cells | FITC | 32116040 | 2 | Cell fluorescence (%) | 10uM | 1h | 37ºC | Flow cytometry | Cellular uptake | WWWRRRRWWW-E12 |
| 1271 | W3R4W3-E12 | MCF7 cells | FITC | 32116040 | 4 | Cell fluorescence (%) | 15uM | 1h | 37ºC | Flow cytometry | Cellular uptake | WWWRRRRWWW-E12 |
| 1272 | W3R4W3-E12 | MCF7 cells | FITC | 32116040 | 23 | Cell fluorescence (%) | 25uM | 1h | 37ºC | Flow cytometry | Cellular uptake | WWWRRRRWWW-E12 |
| 1273 | TP | CHO cells | AgNPs | 33920021 | 300 | Relative Cellular uptake | 10uM | 1h | 37ºC | Flow cytometry | Cellular uptake | GWTLNSAGYLLGKINLKALAALAKKIL |
| 1274 | TP | CHO cells | AuNPs | 33920021 | 85 | Relative Cellular uptake | 10uM | 1h | 37ºC | Flow cytometry | Cellular uptake | GWTLNSAGYLLGKINLKALAALAKKIL |
| 1275 | TP | CHO cells | IONPs | 33920021 | 38 | Relative Cellular uptake | 10uM | 1h | 37ºC | Flow cytometry | Cellular uptake | GWTLNSAGYLLGKINLKALAALAKKIL |
| 1276 | TP | CHO cells | QDs | 33920021 | 135 | Relative Cellular uptake | 10uM | 1h | 37ºC | Flow cytometry | Cellular uptake | GWTLNSAGYLLGKINLKALAALAKKIL |
| 1277 | TP | CHO cells | BSA | 33920021 | 270 | Relative Cellular uptake | 10uM | 1h | 37ºC | Flow cytometry | Cellular uptake | GWTLNSAGYLLGKINLKALAALAKKIL |
| 1278 | TP | CHO cells | Dextran | 33920021 | 22 | Relative Cellular uptake | 10uM | 1h | 37ºC | Flow cytometry | Cellular uptake | GWTLNSAGYLLGKINLKALAALAKKIL |
| 1279 | TP | H1975 cells | AgNPs | 33920021 | 400 | Relative Cellular uptake | 10uM | 1h | 37ºC | Flow cytometry | Cellular uptake | GWTLNSAGYLLGKINLKALAALAKKIL |
| 1280 | TP | H1975 cells | AuNPs | 33920021 | 40 | Relative Cellular uptake | 10uM | 1h | 37ºC | Flow cytometry | Cellular uptake | GWTLNSAGYLLGKINLKALAALAKKIL |
| 1281 | TP | H1975 cells | IONPs | 33920021 | 29 | Relative Cellular uptake | 10uM | 1h | 37ºC | Flow cytometry | Cellular uptake | GWTLNSAGYLLGKINLKALAALAKKIL |
| 1282 | TP | H1975 cells | QDs | 33920021 | 190 | Relative Cellular uptake | 10uM | 1h | 37ºC | Flow cytometry | Cellular uptake | GWTLNSAGYLLGKINLKALAALAKKIL |
| 1283 | TP | H1975 cells | BSA | 33920021 | 210 | Relative Cellular uptake | 10uM | 1h | 37ºC | Flow cytometry | Cellular uptake | GWTLNSAGYLLGKINLKALAALAKKIL |
| 1284 | TP | H1975 cells | Dextran | 33920021 | 18 | Relative Cellular uptake | 10uM | 1h | 37ºC | Flow cytometry | Cellular uptake | GWTLNSAGYLLGKINLKALAALAKKIL |
| 1285 | TP | HeLa cells | AgNPs | 33920021 | 70 | Relative Cellular uptake | 10uM | 1h | 37ºC | Flow cytometry | Cellular uptake | GWTLNSAGYLLGKINLKALAALAKKIL |
| 1286 | TP | HeLa cells | AuNPs | 33920021 | 15 | Relative Cellular uptake | 10uM | 1h | 37ºC | Flow cytometry | Cellular uptake | GWTLNSAGYLLGKINLKALAALAKKIL |
| 1287 | TP | HeLa cells | IONPs | 33920021 | 10 | Relative Cellular uptake | 10uM | 1h | 37ºC | Flow cytometry | Cellular uptake | GWTLNSAGYLLGKINLKALAALAKKIL |
| 1288 | TP | HeLa cells | QDs | 33920021 | 110 | Relative Cellular uptake | 10uM | 1h | 37ºC | Flow cytometry | Cellular uptake | GWTLNSAGYLLGKINLKALAALAKKIL |
| 1289 | TP | HeLa cells | BSA | 33920021 | 60 | Relative Cellular uptake | 10uM | 1h | 37ºC | Flow cytometry | Cellular uptake | GWTLNSAGYLLGKINLKALAALAKKIL |
| 1290 | TP | HeLa cells | Dextran | 33920021 | 19 | Relative Cellular uptake | 10uM | 1h | 37ºC | Flow cytometry | Cellular uptake | GWTLNSAGYLLGKINLKALAALAKKIL |
| 1291 | sC18 | HEK293 cells | actinomycin D | 27860402 | 70000 | Relative fluorescence | 10uM | 30min | 4ºC | Flow cytometry | Cellular uptake | GLRKRLRKFRNKIKEK |
| 1292 | sC18 | HEK293 cells | actinomycin D | 27860402 | 50000 | Relative fluorescence | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | GLRKRLRKFRNKIKEK |
| 1293 | (sC18)2 | HEK293 cells | actinomycin D | 27860402 | 300000 | Relative fluorescence | 10uM | 30min | 4ºC | Flow cytometry | Cellular uptake | GLRKRLRKFRNKIKEKGLRKRLRKFRNKIKEK |
| 1294 | (sC18)2 | HEK293 cells | actinomycin D | 27860402 | 600000 | Relative fluorescence | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | GLRKRLRKFRNKIKEKGLRKRLRKFRNKIKEK |
| 1295 | sC18 | MCF7 cells | actinomycin D | 27860402 | 100000 | Relative fluorescence | 10uM | 30min | 4ºC | Flow cytometry | Cellular uptake | GLRKRLRKFRNKIKEK |
| 1296 | sC18 | MCF7 cells | actinomycin D | 27860402 | 200000 | Relative fluorescence | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | GLRKRLRKFRNKIKEK |
| 1297 | (sC18)2 | MCF7 cells | actinomycin D | 27860402 | 1800000 | Relative fluorescence | 10uM | 30min | 4ºC | Flow cytometry | Cellular uptake | GLRKRLRKFRNKIKEKGLRKRLRKFRNKIKEK |
| 1298 | (sC18)2 | MCF7 cells | actinomycin D | 27860402 | 1500000 | Relative fluorescence | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | GLRKRLRKFRNKIKEKGLRKRLRKFRNKIKEK |
| 1299 | TAT | HeLa cells | FITC | 34101293 | 70 | Cellular uptake (%) | 10uM | 1h | 4ºC | Flow cytometry | Cellular uptake | YGRKKRRQRRR |
| 1300 | TAT | HeLa cells | FITC | 34101293 | 100 | Cellular uptake (%) | 10uM | 1h | 37ºC | Flow cytometry | Cellular uptake | YGRKKRRQRRR |
| 1301 | HNLS-3 | HeLa cells | FITC | 34101293 | 20 | Cellular uptake (%) | 10uM | 1h | 4ºC | Flow cytometry | Cellular uptake | PFVYLIPKKKRKVHHHHHHGC |
| 1302 | HNLS-3 | HeLa cells | FITC | 34101293 | 100 | Cellular uptake (%) | 10uM | 1h | 37ºC | Flow cytometry | Cellular uptake | PFVYLIPKKKRKVHHHHHHGC |
| 1303 | AF-cGm | HeLa cells | Alexa488 | 32979382 | 0.5 | Relative Cellular uptake | 4uM | 1h | 4ºC | Flow cytometry | Cellular uptake | GCRRLCYKQRCVTYCRGR |
| 1304 | AF-cGm | HeLa cells | Alexa488 | 32979382 | 2.1 | Relative Cellular uptake | 4uM | 1h | 37ºC | Flow cytometry | Cellular uptake | GCRRLCYKQRCVTYCRGR |
| 1305 | Mel-lip | bEnd.3 cells | DiI | 32561686 | 5 | Cellular uptake (%) | 100nM | 0.1h | NA | Fluorescence spectroscopy | Cellular uptake | GIGAVLKVLTTGLPALISWIKRKRQ |
| 1306 | Mel-lip | bEnd.3 cells | DiI | 32561686 | 10 | Cellular uptake (%) | 100nM | 0.25h | NA | Fluorescence spectroscopy | Cellular uptake | GIGAVLKVLTTGLPALISWIKRKRQ |
| 1307 | Mel-lip | bEnd.3 cells | DiI | 32561686 | 20 | Cellular uptake (%) | 100nM | 0.5h | NA | Fluorescence spectroscopy | Cellular uptake | GIGAVLKVLTTGLPALISWIKRKRQ |
| 1308 | Mel-lip | bEnd.3 cells | DiI | 32561686 | 39 | Cellular uptake (%) | 100nM | 1h | NA | Fluorescence spectroscopy | Cellular uptake | GIGAVLKVLTTGLPALISWIKRKRQ |
| 1309 | Mel-lip | bEnd.3 cells | DiI | 32561686 | 70 | Cellular uptake (%) | 100nM | 4h | NA | Fluorescence spectroscopy | Cellular uptake | GIGAVLKVLTTGLPALISWIKRKRQ |
| 1310 | Mel-Tf-lip | bEnd.3 cells | DiI | 32561686 | 5 | Cellular uptake (%) | 100nM | 0.1h | NA | Fluorescence spectroscopy | Cellular uptake | GIGAVLKVLTTGLPALISWIKRKRQ |
| 1311 | Mel-Tf-lip | bEnd.3 cells | DiI | 32561686 | 18 | Cellular uptake (%) | 100nM | 0.25h | NA | Fluorescence spectroscopy | Cellular uptake | GIGAVLKVLTTGLPALISWIKRKRQ |
| 1312 | Mel-Tf-lip | bEnd.3 cells | DiI | 32561686 | 25 | Cellular uptake (%) | 100nM | 0.5h | NA | Fluorescence spectroscopy | Cellular uptake | GIGAVLKVLTTGLPALISWIKRKRQ |
| 1313 | Mel-Tf-lip | bEnd.3 cells | DiI | 32561686 | 37 | Cellular uptake (%) | 100nM | 1h | NA | Fluorescence spectroscopy | Cellular uptake | GIGAVLKVLTTGLPALISWIKRKRQ |
| 1314 | Mel-Tf-lip | bEnd.3 cells | DiI | 32561686 | 70 | Cellular uptake (%) | 100nM | 4h | NA | Fluorescence spectroscopy | Cellular uptake | GIGAVLKVLTTGLPALISWIKRKRQ |
| 1315 | kFGF-lip | bEnd.3 cells | DiI | 32561686 | 10 | Cellular uptake (%) | 100nM | 0.1h | NA | Fluorescence spectroscopy | Cellular uptake | AAVALLPAVLLALLAP |
| 1316 | kFGF-lip | bEnd.3 cells | DiI | 32561686 | 17 | Cellular uptake (%) | 100nM | 0.25h | NA | Fluorescence spectroscopy | Cellular uptake | AAVALLPAVLLALLAP |
| 1317 | kFGF-lip | bEnd.3 cells | DiI | 32561686 | 18 | Cellular uptake (%) | 100nM | 0.5h | NA | Fluorescence spectroscopy | Cellular uptake | AAVALLPAVLLALLAP |
| 1318 | kFGF-lip | bEnd.3 cells | DiI | 32561686 | 39 | Cellular uptake (%) | 100nM | 1h | NA | Fluorescence spectroscopy | Cellular uptake | AAVALLPAVLLALLAP |
| 1319 | kFGF-lip | bEnd.3 cells | DiI | 32561686 | 72 | Cellular uptake (%) | 100nM | 4h | NA | Fluorescence spectroscopy | Cellular uptake | AAVALLPAVLLALLAP |
| 1320 | kFGF-Tf-lip | bEnd.3 cells | DiI | 32561686 | 8 | Cellular uptake (%) | 100nM | 0.1h | NA | Fluorescence spectroscopy | Cellular uptake | AAVALLPAVLLALLAP |
| 1321 | kFGF-Tf-lip | bEnd.3 cells | DiI | 32561686 | 18 | Cellular uptake (%) | 100nM | 0.25h | NA | Fluorescence spectroscopy | Cellular uptake | AAVALLPAVLLALLAP |
| 1322 | kFGF-Tf-lip | bEnd.3 cells | DiI | 32561686 | 22 | Cellular uptake (%) | 100nM | 0.5h | NA | Fluorescence spectroscopy | Cellular uptake | AAVALLPAVLLALLAP |
| 1323 | kFGF-Tf-lip | bEnd.3 cells | DiI | 32561686 | 40 | Cellular uptake (%) | 100nM | 1h | NA | Fluorescence spectroscopy | Cellular uptake | AAVALLPAVLLALLAP |
| 1324 | kFGF-Tf-lip | bEnd.3 cells | DiI | 32561686 | 72 | Cellular uptake (%) | 100nM | 4h | NA | Fluorescence spectroscopy | Cellular uptake | AAVALLPAVLLALLAP |
| 1325 | PasR8-lip | bEnd.3 cells | DiI | 32561686 | 4 | Cellular uptake (%) | 100nM | 0.1h | NA | Fluorescence spectroscopy | Cellular uptake | FFLIPKGRRRRRRRRGC |
| 1326 | PasR8-lip | bEnd.3 cells | DiI | 32561686 | 7 | Cellular uptake (%) | 100nM | 0.25h | NA | Fluorescence spectroscopy | Cellular uptake | FFLIPKGRRRRRRRRGC |
| 1327 | PasR8-lip | bEnd.3 cells | DiI | 32561686 | 30 | Cellular uptake (%) | 100nM | 0.5h | NA | Fluorescence spectroscopy | Cellular uptake | FFLIPKGRRRRRRRRGC |
| 1328 | PasR8-lip | bEnd.3 cells | DiI | 32561686 | 42 | Cellular uptake (%) | 100nM | 1h | NA | Fluorescence spectroscopy | Cellular uptake | FFLIPKGRRRRRRRRGC |
| 1329 | PasR8-lip | bEnd.3 cells | DiI | 32561686 | 67 | Cellular uptake (%) | 100nM | 4h | NA | Fluorescence spectroscopy | Cellular uptake | FFLIPKGRRRRRRRRGC |
| 1330 | PasR8-Tf-lip | bEnd.3 cells | DiI | 32561686 | 4 | Cellular uptake (%) | 100nM | 0.1h | NA | Fluorescence spectroscopy | Cellular uptake | FFLIPKGRRRRRRRRGC |
| 1331 | PasR8-Tf-lip | bEnd.3 cells | DiI | 32561686 | 7 | Cellular uptake (%) | 100nM | 0.25h | NA | Fluorescence spectroscopy | Cellular uptake | FFLIPKGRRRRRRRRGC |
| 1332 | PasR8-Tf-lip | bEnd.3 cells | DiI | 32561686 | 28 | Cellular uptake (%) | 100nM | 0.5h | NA | Fluorescence spectroscopy | Cellular uptake | FFLIPKGRRRRRRRRGC |
| 1333 | PasR8-Tf-lip | bEnd.3 cells | DiI | 32561686 | 40 | Cellular uptake (%) | 100nM | 1h | NA | Fluorescence spectroscopy | Cellular uptake | FFLIPKGRRRRRRRRGC |
| 1334 | PasR8-Tf-lip | bEnd.3 cells | DiI | 32561686 | 73 | Cellular uptake (%) | 100nM | 4h | NA | Fluorescence spectroscopy | Cellular uptake | FFLIPKGRRRRRRRRGC |
| 1335 | Agl-AA 1a | MDA-MB-231 cells | fluorescent tag | 28863239 | 50 | Cellular uptake | 10uM | 3h | 37ºC | FT-IR | Cellular uptake | XRXR |
| 1336 | Agl-AA 1b | MDA-MB-231 cells | fluorescent tag | 28863239 | 30 | Cellular uptake | 10uM | 3h | 37ºC | FT-IR | Cellular uptake | XRXRXRXR |
| 1337 | Agl-AA 1c | MDA-MB-231 cells | fluorescent tag | 28863239 | 60 | Cellular uptake | 10uM | 3h | 37ºC | FT-IR | Cellular uptake | XRXRXRXRXRXR |
| 1338 | Agl-AA 2a | MDA-MB-231 cells | fluorescent tag | 28863239 | 50 | Cellular uptake | 10uM | 3h | 37ºC | FT-IR | Cellular uptake | XWXW |
| 1339 | Agl-AA 2b | MDA-MB-231 cells | fluorescent tag | 28863239 | 150 | Cellular uptake | 10uM | 3h | 37ºC | FT-IR | Cellular uptake | XWXWXWXW |
| 1340 | Agl-AA 2c | MDA-MB-231 cells | fluorescent tag | 28863239 | 650 | Cellular uptake | 10uM | 3h | 37ºC | FT-IR | Cellular uptake | XWXWXWXWXWXW |
| 1341 | Agl-AA 3a | MDA-MB-231 cells | fluorescent tag | 28863239 | 30 | Cellular uptake | 10uM | 3h | 37ºC | FT-IR | Cellular uptake | XFXR |
| 1342 | Agl-AA 3b | MDA-MB-231 cells | fluorescent tag | 28863239 | 30 | Cellular uptake | 10uM | 3h | 37ºC | FT-IR | Cellular uptake | XFXRXFXR |
| 1343 | Agl-AA 3c | MDA-MB-231 cells | fluorescent tag | 28863239 | 40 | Cellular uptake | 10uM | 3h | 37ºC | FT-IR | Cellular uptake | XFXRXFXRXFXR |
| 1344 | Agl-AA 4a | MDA-MB-231 cells | fluorescent tag | 28863239 | 100 | Cellular uptake | 10uM | 3h | 37ºC | FT-IR | Cellular uptake | RQIKIWFQNRRMKWKKGG |
| 1345 | Agl-AA 4b | MDA-MB-231 cells | fluorescent tag | 28863239 | 190 | Cellular uptake | 10uM | 3h | 37ºC | FT-IR | Cellular uptake | RRWWRRWRR |
| 1346 | Agl-AA 5a | MDA-MB-231 cells | fluorescent tag | 28863239 | 40 | Cellular uptake | 10uM | 3h | 37ºC | FT-IR | Cellular uptake | AWARAWARAWAR |
| 1347 | BRC4wt | HeLa cells | TAMRA | 29654063 | 30 | Median TAMRA intensity | 10 umol/L | 1h | NA | Flow cytometry | Cellular uptake | LLGFHTASGKKVKIAK |
| 1348 | R9 | HeLa cells | TAMRA | 29654063 | 5000 | Median TAMRA intensity | 10 umol/L | 1h | NA | Flow cytometry | Cellular uptake | RRRRRRRRR |
| 1349 | R9-BRC4wt | HeLa cells | TAMRA | 29654063 | 4000 | Median TAMRA intensity | 10 umol/L | 1h | NA | Flow cytometry | Cellular uptake | RRRRRRRRR-LLGFHTASGKKVKIAK |
| 1350 | R9-BRC4mut | HeLa cells | TAMRA | 29654063 | 2000 | Median TAMRA intensity | 10 umol/L | 1h | NA | Flow cytometry | Cellular uptake | RRRRRRRRR-LLGATHFSGKKVKIAK |
| 1351 | BRC4wt | U2OS cells | TAMRA | 29654063 | 50 | Median TAMRA intensity | 10 umol/L | 1h | NA | Flow cytometry | Cellular uptake | LLGFHTASGKKVKIAK |
| 1352 | R9 | U2OS cells | TAMRA | 29654063 | 10000 | Median TAMRA intensity | 10 umol/L | 1h | NA | Flow cytometry | Cellular uptake | RRRRRRRRR |
| 1353 | R9-BRC4wt | U2OS cells | TAMRA | 29654063 | 4000 | Median TAMRA intensity | 10 umol/L | 1h | NA | Flow cytometry | Cellular uptake | RRRRRRRRR-LLGFHTASGKKVKIAK |
| 1354 | R9-BRC4mut | U2OS cells | TAMRA | 29654063 | 10000 | Median TAMRA intensity | 10 umol/L | 1h | NA | Flow cytometry | Cellular uptake | RRRRRRRRR-LLGATHFSGKKVKIAK |
| 1355 | GBPECP | A549 cells | FITC | 27936565 | 0 | NA | 5 uM | 1h | 37ºC | Fluorescent Microscopy | Cellular uptake | NYRWRCKNQN |
| 1356 | GBPEDN | A549 cells | FITC | 27936565 | 0 | NA | 5 uM | 1h | 37ºC | Fluorescent Microscopy | Cellular uptake | NYQRRCKNQN |
| 1357 | GBPECP(W4R) | A549 cells | FITC | 27936565 | 0 | NA | 5 uM | 1h | 37ºC | Fluorescent Microscopy | Cellular uptake | NYRRRCKNQN |
| 1358 | IgG-colpep | HeLa cells | FITC | 26725435 | 20 | Fluorescence intensity | 40 ug /mL | 3h | 37ºC | Flow cytometry | Cellular uptake | GPXGPXGPXGPRGPRGPRGPXGPXGPXGP |
| 1359 | IgG-?R8 | HeLa cells | FITC | 26725435 | 14 | Fluorescence intensity | 40 ug /mL | 3h | 37ºC | Flow cytometry | Cellular uptake | XRRRRRRRR |
| 1360 | PepB2 | CHO-K1 cells | PA | 29247010 | 600 | Median Fluorescence intensity | 50 uM | 30min | 37ºC | Flow cytometry | Cellular uptake | NVFKGNTISDKISFNFSDK |
| 1361 | PepB2 | CHO-K1 cells | CROP | 29247010 | 900 | Median Fluorescence intensity | 50 uM | 30min | 37ºC | Flow cytometry | Cellular uptake | NVFKGNTISDKISFNFSDK |
| 1362 | PepB2 | CHO-K1 cells | SLO | 29247010 | 1300 | Median Fluorescence intensity | 50 uM | 30min | 37ºC | Flow cytometry | Cellular uptake | NVFKGNTISDKISFNFSDK |
| 1363 | PepB2 | CHO-K1 cells | CT-B | 29247010 | 600 | Median Fluorescence intensity | 50 uM | 30min | 37ºC | Flow cytometry | Cellular uptake | NVFKGNTISDKISFNFSDK |
| 1364 | PepB2 | CHO-K1 cells | Tf | 29247010 | 1500 | Median Fluorescence intensity | 50 uM | 30min | 37ºC | Flow cytometry | Cellular uptake | NVFKGNTISDKISFNFSDK |
| 1365 | PepB2 | CHO-K1 cells | SA | 29247010 | 1600 | Median Fluorescence intensity | 50 uM | 30min | 37ºC | Flow cytometry | Cellular uptake | NVFKGNTISDKISFNFSDK |
| 1366 | PepB2 | CHO-K1 cells | Dextran | 29247010 | 1500 | Median Fluorescence intensity | 50 uM | 30min | 37ºC | Flow cytometry | Cellular uptake | NVFKGNTISDKISFNFSDK |
| 1367 | PepB2 | CHO-K1 cells | MS | 29247010 | 1000 | Median Fluorescence intensity | 50 uM | 30min | 37ºC | Flow cytometry | Cellular uptake | NVFKGNTISDKISFNFSDK |
| 1368 | IMT-P8 | HeLa cells | KLA | 27189051 | 300000 | Median Fluorescence intensity | 2.5 uM | 30min | 37ºC | Flow cytometry | Cellular uptake | RRWRRWNRFNRRRCR |
| 1369 | IMT-P8 | MDA-MB-231 cells | KLA | 27189051 | 200000 | Median Fluorescence intensity | 2.5 uM | 30min | 37ºC | Flow cytometry | Cellular uptake | RRWRRWNRFNRRRCR |
| 1370 | IMT-P8 | PC3 cells | KLA | 27189051 | 1100000 | Median Fluorescence intensity | 2.5 uM | 30min | 37ºC | Flow cytometry | Cellular uptake | RRWRRWNRFNRRRCR |
| 1371 | IMT-P8 | HeLa cells | GFP | 27189051 | 25000 | Median Fluorescence intensity | 5 uM | 1h | 37ºC | Flow cytometry | Cellular uptake | RRWRRWNRFNRRRCR |
| 1372 | CMR19 | SJSA-1 cells | cR10 | 34977581 | 0 | NA | 5uM | 2h | 37ºC | Fluorescent Microscopy | Cellular uptake | FSDMeSSSVPNBBRNCG |
| 1373 | SI-ULK1 micelle | HepG2 cells | Rho | 29787814 | 0 | Relative fluorescence | 5uM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | FITC-GRKKRRQRRR-NH2 |
| 1374 | Rhodamine micelle | HepG2 cells | Rho | 29787814 | 115 | Relative fluorescence | 5uM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | M-Rho-GRKKRRQRRR-NH2 |
| 1375 | SI-ULK1/Rhodamine micelle | HepG2 cells | Rho | 29787814 | 175 | Relative fluorescence | 5uM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | His6-GRKKRRQRRR-NH2 |
| 1376 | SI-ULK1 micelle | HepG2 cells | FITC | 29787814 | 85 | Relative fluorescence | 5uM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | FITC-GRKKRRQRRR-NH2 |
| 1377 | Rhodamine micelle | HepG2 cells | FITC | 29787814 | 10 | Relative fluorescence | 5uM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | M-Rho-GRKKRRQRRR-NH2 |
| 1378 | SI-ULK1/Rhodamine micelle | HepG2 cells | FITC | 29787814 | 100 | Relative fluorescence | 5uM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | His6-GRKKRRQRRR-NH2 |
| 1379 | Cf | HEK293T cells | FITC | 34277705 | 0 | Fluorescence intensity | 1uM | 24h | 37ºC | Flow cytometry | Cellular uptake | RRPPWLRLDIRR |
| 1380 | Cf | HEK293T cells | FITC | 34277705 | 5 | Fluorescence intensity | 5uM | 24h | 37ºC | Flow cytometry | Cellular uptake | RRPPWLRLDIRR |
| 1381 | Cf | HEK293T cells | FITC | 34277705 | 2 | Fluorescence intensity | 10uM | 24h | 37ºC | Flow cytometry | Cellular uptake | RRPPWLRLDIRR |
| 1382 | Dabcyl | HEK293T cells | FITC | 34277705 | 40 | Fluorescence intensity | 1uM | 24h | 37ºC | Flow cytometry | Cellular uptake | RRRPPWLRLDIRRK |
| 1383 | Dabcyl | HEK293T cells | FITC | 34277705 | 10 | Fluorescence intensity | 5uM | 24h | 37ºC | Flow cytometry | Cellular uptake | RRRPPWLRLDIRRK |
| 1384 | Dabcyl | HEK293T cells | FITC | 34277705 | 120 | Fluorescence intensity | 10uM | 24h | 37ºC | Flow cytometry | Cellular uptake | RRRPPWLRLDIRRK |
| 1385 | E28 | MDA-MB-231 cells | Alexa488 | 31952530 | 0 | NA | NA | 1h | 37ºC | CLSM | Cellular uptake | MSGPGVGVPGVGVPGVGVPGFGVPGVGVPGVGVPGFGVPGVGVPGGGVPGGGVPGVGVPGAGVPGVGVPGGGVPGVGVPGVGVPGVGVPGFGVPGVGVPGVGVPGFGVPGVGVPGGGVPGGGVPGVGVPGAGVPGVGVPGGGVPGWPC |
| 1386 | Tat-E28 | MDA-MB-231 cells | Alexa488 | 31952530 | 0 | NA | NA | 1h | 37ºC | CLSM | Cellular uptake | MSGYGRKKRRQRRRGGGPGVGVPGVGVPGVGVPGFGVPGVGVPGVGVPGFGVPGVGVPGGGVPGGGVPGVGVPGAGVPGVGVPGGGVPVGVPGVGVPGVGVPGFGVPGVGVPGVGVPGFGVPGVGVPGGGVPGGGVPGVGVPGAGVPGVGVPGGGVPGWPC |
| 1387 | Tat-A1E28 | MDA-MB-231 cells | Alexa488 | 31952530 | 0 | NA | NA | 1h | 37ºC | CLSM | Cellular uptake | MSGYGRKKRRQRRRGGGRKRLDRNGGGPGVGVPGVGVPGVGVPGFGVPGVGVPGVGVPGFGVPGVGVPGGGVPGGGVPGVGVPGAGVPGVGVPGGGVPVGVPGVGVPGVGVPGFGVPGVGVPGVGVPGFGVPGVGVPGGGVPGGGVPGVGVPGAGVPGVGVPGGGVPGWPC |
| 1388 | Tat-A4V48 | MDA-MB-231 cells | Alexa488 | 31952530 | 0 | NA | NA | 1h | 37ºC | CLSM | Cellular uptake | MSGYGRKKRRQRRRGGGPGVGRKRLDRNGVGVPGVGVPGVGVPGVGVPGVGVPGVGVPGVGVPGVGVPGVGVPGVGVPGVGVPGVGVPGVGRKRLDRNGVGVPGVGVPGVGVPGVGVPGVGVPGVGVPGVGVPGVGVPGVGVPGVGVPGVGVPGVGVPGVGRKRLDRNGVGVPGVGVPGVGVPGVGVPGVGVPGVGVPGVGVPGVGVPGVGVPGVGVPGVGVPGVGVPGVGRKRLDRNGVGVPGVGVPGVGVPGVGVPGVGVPGVGVPG |
| 1389 | (KW)4 | MCF7 cells | FITC | 28933182 | 85 | Cell fluorescence (%) | 10 uM | 2h | 37ºC | Flow cytometry | Cellular uptake | KWKWKWKW |
| 1390 | (KW)4 | MCF7 cells | FITC | 28933182 | 90 | Cell fluorescence (%) | 25uM | 2h | 37ºC | Flow cytometry | Cellular uptake | KWKWKWKW |
| 1391 | (KW)4 | MCF7 cells | FITC | 28933182 | 70 | Cell fluorescence (%) | 50uM | 2h | 37ºC | Flow cytometry | Cellular uptake | KWKWKWKW |
| 1392 | (KW)5 | MCF7 cells | FITC | 28933182 | 60 | Cell fluorescence (%) | 10 uM | 2h | 37ºC | Flow cytometry | Cellular uptake | KWKWKWKWKW |
| 1393 | (KW)5 | MCF7 cells | FITC | 28933182 | 90 | Cell fluorescence (%) | 25uM | 2h | 37ºC | Flow cytometry | Cellular uptake | KWKWKWKWKW |
| 1394 | (KW)5 | MCF7 cells | FITC | 28933182 | 75 | Cell fluorescence (%) | 50uM | 2h | 37ºC | Flow cytometry | Cellular uptake | KWKWKWKWKW |
| 1395 | K2W4K2 | MCF7 cells | FITC | 28933182 | 80 | Cell fluorescence (%) | 10 uM | 2h | 37ºC | Flow cytometry | Cellular uptake | KKWWWWKK |
| 1396 | K2W4K2 | MCF7 cells | FITC | 28933182 | 90 | Cell fluorescence (%) | 25uM | 2h | 37ºC | Flow cytometry | Cellular uptake | KKWWWWKK |
| 1397 | K2W4K2 | MCF7 cells | FITC | 28933182 | 85 | Cell fluorescence (%) | 50uM | 2h | 37ºC | Flow cytometry | Cellular uptake | KKWWWWKK |
| 1398 | K3W4K3 | MCF7 cells | FITC | 28933182 | 80 | Cell fluorescence (%) | 10 uM | 2h | 37ºC | Flow cytometry | Cellular uptake | KKKWWWWKKK |
| 1399 | K3W4K3 | MCF7 cells | FITC | 28933182 | 90 | Cell fluorescence (%) | 25uM | 2h | 37ºC | Flow cytometry | Cellular uptake | KKKWWWWKKK |
| 1400 | K3W4K3 | MCF7 cells | FITC | 28933182 | 90 | Cell fluorescence (%) | 50uM | 2h | 37ºC | Flow cytometry | Cellular uptake | KKKWWWWKKK |
| 1401 | W2K4W2 | MCF7 cells | FITC | 28933182 | 35 | Cell fluorescence (%) | 10 uM | 2h | 37ºC | Flow cytometry | Cellular uptake | WWKKKKWW |
| 1402 | W2K4W2 | MCF7 cells | FITC | 28933182 | 20 | Cell fluorescence (%) | 25uM | 2h | 37ºC | Flow cytometry | Cellular uptake | WWKKKKWW |
| 1403 | W2K4W2 | MCF7 cells | FITC | 28933182 | 30 | Cell fluorescence (%) | 50uM | 2h | 37ºC | Flow cytometry | Cellular uptake | WWKKKKWW |
| 1404 | W3K4W3 | MCF7 cells | FITC | 28933182 | 80 | Cell fluorescence (%) | 10 uM | 2h | 37ºC | Flow cytometry | Cellular uptake | WWWKKKKWWW |
| 1405 | W3K4W3 | MCF7 cells | FITC | 28933182 | 90 | Cell fluorescence (%) | 25uM | 2h | 37ºC | Flow cytometry | Cellular uptake | WWWKKKKWWW |
| 1406 | W3K4W3 | MCF7 cells | FITC | 28933182 | 85 | Cell fluorescence (%) | 50uM | 2h | 37ºC | Flow cytometry | Cellular uptake | WWWKKKKWWW |
| 1407 | CPP-siRNA | HT1080 cells | siRNA | 27012462 | 120 | Mean Fluorescence intensity | NA | 4h | 37ºC | Flow cytometry | Cellular uptake | CKRRMKWKK |
| 1408 | CPP-siRNA/N-NB | HT1080 cells | siRNA | 27012462 | 30 | Mean Fluorescence intensity | NA | 4h | 37ºC | Flow cytometry | Cellular uptake | CKRRMKWKK |
| 1409 | CPP-siRNA/N-NB(+US) | HT1080 cells | siRNA | 27012462 | 110 | Mean Fluorescence intensity | NA | 4h | 37ºC | Flow cytometry | Cellular uptake | CKRRMKWKK |
| 1410 | CPP-DOX | MCF7 cells | Doxorubicin | 26176270 | 83 | Mean Fluorescence intensity | NA | 24h | 37ºC | Flow cytometry | Cellular uptake | CKRRMKWKK-DOX |
| 1411 | CPP-DOX | HT1080 cells | Doxorubicin | 26176270 | 80 | Mean Fluorescence intensity | NA | 24h | 37ºC | Flow cytometry | Cellular uptake | CKRRMKWKK-DOX |
| 1412 | CPP-DOX/N-NB | MCF7 cells | Doxorubicin | 26176270 | 22 | Mean Fluorescence intensity | NA | 24h | 37ºC | Flow cytometry | Cellular uptake | CKRRMKWKK-DOX |
| 1413 | CPP-DOX/N-NB | HT1080 cells | Doxorubicin | 26176270 | 20 | Mean Fluorescence intensity | NA | 24h | 37ºC | Flow cytometry | Cellular uptake | CKRRMKWKK-DOX |
| 1414 | CPP-DOX/NGR-NB | MCF7 cells | Doxorubicin | 26176270 | 22 | Mean Fluorescence intensity | NA | 24h | 37ºC | Flow cytometry | Cellular uptake | CKRRMKWKK-DOX/CYGGRGNG |
| 1415 | CPP-DOX/NGR-NB | HT1080 cells | Doxorubicin | 26176270 | 40 | Mean Fluorescence intensity | NA | 24h | 37ºC | Flow cytometry | Cellular uptake | CKRRMKWKK-DOX/CYGGRGNG |
| 1416 | CPP-DOX/N-NB (+US) | MCF7 cells | Doxorubicin | 26176270 | 82 | Mean Fluorescence intensity | NA | 24h | 37ºC | Flow cytometry | Cellular uptake | CKRRMKWKK-DOX |
| 1417 | CPP-DOX/N-NB (+US) | HT1080 cells | Doxorubicin | 26176270 | 85 | Mean Fluorescence intensity | NA | 24h | 37ºC | Flow cytometry | Cellular uptake | CKRRMKWKK-DOX |
| 1418 | CPP-DOX/NGR-NB (+US) | MCF7 cells | Doxorubicin | 26176270 | 80 | Mean Fluorescence intensity | NA | 24h | 37ºC | Flow cytometry | Cellular uptake | CKRRMKWKK-DOX/CYGGRGNG |
| 1419 | CPP-DOX/NGR-NB (+US) | HT1080 cells | Doxorubicin | 26176270 | 82 | Mean Fluorescence intensity | NA | 24h | 37ºC | Flow cytometry | Cellular uptake | CKRRMKWKK-DOX/CYGGRGNG |
| 1420 | ENCP | Caco-2 cells | Insulin | 29518466 | 50 | Cellular uptake (%) | NA | 2h | 37ºC | Liquid chromatography | Cellular uptake | RRRRRRRR |
| 1421 | NCP | Caco-2 cells | Insulin | 29518466 | 80 | Cellular uptake (%) | NA | 2h | 37ºC | Liquid chromatography | Cellular uptake | RRRRRRRR |
| 1422 | Insulin+R8 | Caco-2 cells | Insulin | 29518466 | 0 | Cellular uptake (%) | NA | 2h | 37ºC | Liquid chromatography | Cellular uptake | RRRRRRRR |
| 1423 | TAT | Leishmania donovani promastigotes | Doxorubicin | 33053805 | 100 | Internalization | 5uM | 2h | 26ºC | Flow cytometry | Cellular uptake | GRKKRRQRRRPQ |
| 1424 | TAT | Leishmania donovani promastigotes | Doxorubicin | 33053805 | 100 | Internalization | 10uM | 2h | 26ºC | Flow cytometry | Cellular uptake | GRKKRRQRRRPQ |
| 1425 | ?-CC 15 | Leishmania donovani promastigotes | Doxorubicin | 33053805 | 160 | Internalization | 5uM | 2h | 26ºC | Flow cytometry | Cellular uptake | PPPPPPPPPPPPPPP |
| 1426 | ?-CC 15 | Leishmania donovani promastigotes | Doxorubicin | 33053805 | 200 | Internalization | 10uM | 2h | 26ºC | Flow cytometry | Cellular uptake | PPPPPPPPPPPPPPP |
| 1427 | ?-CC 16 | Leishmania donovani promastigotes | Doxorubicin | 33053805 | 170 | Internalization | 5uM | 2h | 26ºC | Flow cytometry | Cellular uptake | PPPPPPPPPPPPPPPP |
| 1428 | ?-CC 16 | Leishmania donovani promastigotes | Doxorubicin | 33053805 | 180 | Internalization | 10uM | 2h | 26ºC | Flow cytometry | Cellular uptake | PPPPPPPPPPPPPPPP |
| 1429 | TAT | Leishmania donovani promastigotes | Doxorubicin | 33053805 | 110 | Internalization | 5uM | 4h | 26ºC | Flow cytometry | Cellular uptake | GRKKRRQRRRPQ |
| 1430 | TAT | Leishmania donovani promastigotes | Doxorubicin | 33053805 | 100 | Internalization | 10uM | 4h | 26ºC | Flow cytometry | Cellular uptake | GRKKRRQRRRPQ |
| 1431 | ?-CC 15 | Leishmania donovani promastigotes | Doxorubicin | 33053805 | 165 | Internalization | 5uM | 4h | 26ºC | Flow cytometry | Cellular uptake | PPPPPPPPPPPPPPP |
| 1432 | ?-CC 15 | Leishmania donovani promastigotes | Doxorubicin | 33053805 | 250 | Internalization | 10uM | 4h | 26ºC | Flow cytometry | Cellular uptake | PPPPPPPPPPPPPPP |
| 1433 | ?-CC 16 | Leishmania donovani promastigotes | Doxorubicin | 33053805 | 160 | Internalization | 5uM | 4h | 26ºC | Flow cytometry | Cellular uptake | PPPPPPPPPPPPPPPP |
| 1434 | ?-CC 16 | Leishmania donovani promastigotes | Doxorubicin | 33053805 | 210 | Internalization | 10uM | 4h | 26ºC | Flow cytometry | Cellular uptake | PPPPPPPPPPPPPPPP |
| 1435 | [RW]3 | A549 cells | FITC | 28694765 | 32 | Cell fluorescence (%) | 10uM | 1.5h | 37ºC | Flow cytometry | Cellular uptake | RWRWRW |
| 1436 | [RW]3 | A549 cells | FITC | 28694765 | 63 | Cell fluorescence (%) | 25uM | 1.5h | 37ºC | Flow cytometry | Cellular uptake | RWRWRW |
| 1437 | [RW]3 | A549 cells | FITC | 28694765 | 90 | Cell fluorescence (%) | 50uM | 1.5h | 37ºC | Flow cytometry | Cellular uptake | RWRWRW |
| 1438 | [RW]4 | A549 cells | FITC | 28694765 | 57 | Cell fluorescence (%) | 10uM | 1.5h | 37ºC | Flow cytometry | Cellular uptake | RWRWRWRW |
| 1439 | [RW]4 | A549 cells | FITC | 28694765 | 79 | Cell fluorescence (%) | 25uM | 1.5h | 37ºC | Flow cytometry | Cellular uptake | RWRWRWRW |
| 1440 | [RW]4 | A549 cells | FITC | 28694765 | 80 | Cell fluorescence (%) | 50uM | 1.5h | 37ºC | Flow cytometry | Cellular uptake | RWRWRWRW |
| 1441 | [RW]5 | A549 cells | FITC | 28694765 | 35 | Cell fluorescence (%) | 10uM | 1.5h | 37ºC | Flow cytometry | Cellular uptake | RWRWRWRWRW |
| 1442 | [RW]5 | A549 cells | FITC | 28694765 | 49 | Cell fluorescence (%) | 25uM | 1.5h | 37ºC | Flow cytometry | Cellular uptake | RWRWRWRWRW |
| 1443 | [RW]5 | A549 cells | FITC | 28694765 | 68 | Cell fluorescence (%) | 50uM | 1.5h | 37ºC | Flow cytometry | Cellular uptake | RWRWRWRWRW |
| 1444 | [RW]6 | A549 cells | FITC | 28694765 | 60 | Cell fluorescence (%) | 10uM | 1.5h | 37ºC | Flow cytometry | Cellular uptake | RWRWRWRWRWRW |
| 1445 | [RW]6 | A549 cells | FITC | 28694765 | 71 | Cell fluorescence (%) | 25uM | 1.5h | 37ºC | Flow cytometry | Cellular uptake | RWRWRWRWRWRW |
| 1446 | [RW]6 | A549 cells | FITC | 28694765 | 79 | Cell fluorescence (%) | 50uM | 1.5h | 37ºC | Flow cytometry | Cellular uptake | RWRWRWRWRWRW |
| 1447 | R5W3R4 | A549 cells | FITC | 28694765 | 47 | Cell fluorescence (%) | 10uM | 1.5h | 37ºC | Flow cytometry | Cellular uptake | RRRRRWWWRRRR |
| 1448 | R5W3R4 | A549 cells | FITC | 28694765 | 59 | Cell fluorescence (%) | 25uM | 1.5h | 37ºC | Flow cytometry | Cellular uptake | RRRRRWWWRRRR |
| 1449 | R5W3R4 | A549 cells | FITC | 28694765 | 88 | Cell fluorescence (%) | 50uM | 1.5h | 37ºC | Flow cytometry | Cellular uptake | RRRRRWWWRRRR |
| 1450 | QD-(Arg9)1 | COS-1 cells | QDs | 28703833 | 0 | Fluorescence intensity | 100 nM | 30min | NA | Fluorescent Microscopy | Cellular uptake | RRRRRRRRRFGWPPPPPPPPPGGHHHHHH |
| 1451 | QD-(Arg9)1 | COS-1 cells | QDs | 28703833 | 0 | Fluorescence intensity | 100 nM | 1h | NA | Fluorescent Microscopy | Cellular uptake | RRRRRRRRRFGWPPPPPPPPPGGHHHHHH |
| 1452 | QD-(Arg9)1 | COS-1 cells | QDs | 28703833 | 0 | Fluorescence intensity | 100 nM | 4h | NA | Fluorescent Microscopy | Cellular uptake | RRRRRRRRRFGWPPPPPPPPPGGHHHHHH |
| 1453 | QD-(Arg9)1 | COS-1 cells | QDs | 28703833 | 0 | Fluorescence intensity | 100 nM | 8h | NA | Fluorescent Microscopy | Cellular uptake | RRRRRRRRRFGWPPPPPPPPPGGHHHHHH |
| 1454 | QD-(Arg9)4 | COS-1 cells | QDs | 28703833 | 0 | Fluorescence intensity | 100 nM | 30min | NA | Fluorescent Microscopy | Cellular uptake | RRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGWPPPPPPPPPGGHHHHHH |
| 1455 | REDV-TAT-NLS-H0 | HUVEC cells | Cy5-oligonucleotide | 29580233 | 23 | Cellular uptake (%) | NA | 4h | NA | Flow cytometry | Cellular uptake | REDVYGRKKRRQRRRPKKKRKVHHHH |
| 1456 | REDV-TAT-NLS-H4 | HUVEC cells | Cy5-oligonucleotide | 29580233 | 30 | Cellular uptake (%) | NA | 4h | NA | Flow cytometry | Cellular uptake | REDVYGRKKRRQRRRPKKKRKVHHHHHHHH |
| 1457 | REDV-TAT-NLS-H8 | HUVEC cells | Cy5-oligonucleotide | 29580233 | 40 | Cellular uptake (%) | NA | 4h | NA | Flow cytometry | Cellular uptake | REDVYGRKKRRQRRRPKKKRKVHHHHHHHHHHHH |
| 1458 | REDV-TAT-NLS-H12 | HUVEC cells | Cy5-oligonucleotide | 29580233 | 88 | Cellular uptake (%) | NA | 4h | NA | Flow cytometry | Cellular uptake | REDV-YGRKKRRQRRR-PKK-KRKV-HHHHHHHHHHHH |
| 1459 | CVP1-N2 | HCT116 cells | FITC | 33141296 | 10 | Relative internalization (%) | 0.1uM | NA | 37ºC | Flow cytometry | Cellular uptake | LKRLRRRYKFRHRRRQRYRRR |
| 1460 | CVP1-N2 | HCT116 cells | FITC | 33141296 | 75 | Relative internalization (%) | 1uM | NA | 37ºC | Flow cytometry | Cellular uptake | LKRLRRRYKFRHRRRQRYRRR |
| 1461 | CVP1-N2 | HCT116 cells | FITC | 33141296 | 100 | Relative internalization (%) | 10uM | NA | 37ºC | Flow cytometry | Cellular uptake | LKRLRRRYKFRHRRRQRYRRR |
| 1462 | CVP1-N2 | HCT116 cells | FITC | 33141296 | 88 | Relative internalization (%) | 10uM | NA | 4ºC | Flow cytometry | Cellular uptake | LKRLRRRYKFRHRRRQRYRRR |
| 1463 | Scp01-b | Caski cells | FITC | 30230543 | 350 | Fluorescence intensity | 2.5uM | 1h | 37ºC | Fluorescent Microscopy | Cellular uptake | VSRRRRRRGGRRRRGGGSYARVRRRGPRRGYARVRRRGPRR |
| 1464 | Scp01-b | Caski cells | FITC | 30230543 | 1100 | Fluorescence intensity | 5uM | 1h | 37ºC | Fluorescent Microscopy | Cellular uptake | VSRRRRRRGGRRRRGGGSYARVRRRGPRRGYARVRRRGPRR |
| 1465 | Scp01-b | Caski cells | FITC | 30230543 | 1350 | Fluorescence intensity | 7.5uM | 1h | 37ºC | Fluorescent Microscopy | Cellular uptake | VSRRRRRRGGRRRRGGGSYARVRRRGPRRGYARVRRRGPRR |
| 1466 | Scp01-b | Caski cells | FITC | 30230543 | 1400 | Fluorescence intensity | 10uM | 1h | 37ºC | Fluorescent Microscopy | Cellular uptake | VSRRRRRRGGRRRRGGGSYARVRRRGPRRGYARVRRRGPRR |
| 1467 | R4-EMCS | CHO-K1 cells | CD63-GFP Evs | 28512335 | 1361 | Relative Cellular uptake | 20uM | 24h | 37ºC | Flow cytometry | Cellular uptake | GRRRR |
| 1468 | R8-EMCS | CHO-K1 cells | CD63-GFP Evs | 28512335 | 2890 | Relative Cellular uptake | 20uM | 24h | 37ºC | Flow cytometry | Cellular uptake | GRRRRRRRR |
| 1469 | R12-EMCS | CHO-K1 cells | CD63-GFP Evs | 28512335 | 2862 | Relative Cellular uptake | 20uM | 24h | 37ºC | Flow cytometry | Cellular uptake | GRRRRRRRRRRRR |
| 1470 | R16-EMCS | CHO-K1 cells | CD63-GFP Evs | 28512335 | 1823 | Relative Cellular uptake | 10uM | 24h | 37ºC | Flow cytometry | Cellular uptake | GRRRRRRRRRRRRRRRR |
| 1471 | cyc-hCT(9-32) | MCF7 cells | Carboxyfluorescein | 27197760 | 15000 | Relative fluorescence | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | CF-Cys-BLGTYTQDFNXFHTFPQTAIGVGAP |
| 1472 | cyc-hCT(9-32) | MCF7 cells | Carboxyfluorescein | 27197760 | 52000 | Relative fluorescence | 50uM | 30min | 37ºC | Flow cytometry | Cellular uptake | CF-Cys-BLGTYTQDFNXFHTFPQTAIGVGAP |
| 1473 | iCREKA | U87 cells | FITC | 29686590 | 14110 | Fluorescence intensity | 10uM | 1h | 37ºC | Flow cytometry | Cellular uptake | CREKAPLGLAGRKKRRQRRRC |
| 1474 | CREKA | U87 cells | FITC | 29686590 | 2569.5 | Fluorescence intensity | 10uM | 1h | 37ºC | Flow cytometry | Cellular uptake | CREKA |
| 1475 | ALD5MTS (2–17) | HeLa cells | TAM | 30367921 | 0.05 | Internalization | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | LSRTRAAAPNSRIFTR |
| 1476 | ALD5MTS (2–17) | HeLa cells | TAM | 30367921 | 0 | Internalization | 1uM | 30min | 37ºC | Flow cytometry | Cellular uptake | LSRTRAAAPNSRIFTR |
| 1477 | ALD5MTS (2–17)-sC18 | HeLa cells | TAM | 30367921 | 0.65 | Internalization | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | LSRTRAAAPNSRIFTRGLRKRLRKFRNKIKEK |
| 1478 | ALD5MTS (2–17)-sC18 | HeLa cells | TAM | 30367921 | 0.1 | Internalization | 1uM | 30min | 37ºC | Flow cytometry | Cellular uptake | LSRTRAAAPNSRIFTRGLRKRLRKFRNKIKEK |
| 1479 | HSP60MTS (2–14) | HeLa cells | TAM | 30367921 | 0.05 | Internalization | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | LRSSVVRSRATLR |
| 1480 | HSP60MTS (2–14) | HeLa cells | TAM | 30367921 | 0 | Internalization | 1uM | 30min | 37ºC | Flow cytometry | Cellular uptake | LRSSVVRSRATLR |
| 1481 | HSP60MTS (2–14)-sC18 | HeLa cells | TAM | 30367921 | 0.8 | Internalization | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | LRSSVVRSRATLRGLRKRLRKFRNKIKEK |
| 1482 | HSP60MTS (2–14)-sC18 | HeLa cells | TAM | 30367921 | 0.1 | Internalization | 1uM | 30min | 37ºC | Flow cytometry | Cellular uptake | LRSSVVRSRATLRGLRKRLRKFRNKIKEK |
| 1483 | BNA3MTS (2–7) | HeLa cells | TAM | 30367921 | 0.05 | Internalization | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | KQRFIR |
| 1484 | BNA3MTS (2–7) | HeLa cells | TAM | 30367921 | 0 | Internalization | 1uM | 30min | 37ºC | Flow cytometry | Cellular uptake | KQRFIR |
| 1485 | BNA3MTS (2–7)-sC18 | HeLa cells | TAM | 30367921 | 0.75 | Internalization | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | KQRFIRGLRKRLRKFRNKIKEK |
| 1486 | BNA3MTS (2–7)-sC18 | HeLa cells | TAM | 30367921 | 0.08 | Internalization | 1uM | 30min | 37ºC | Flow cytometry | Cellular uptake | KQRFIRGLRKRLRKFRNKIKEK |
| 1487 | CalpMTS (2–19)-sC18 | HeLa cells | TAM | 30367921 | 0.4 | Internalization | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | SEEIITPVYCTGVSAQVQKGLRKRLRKFRNKIKEK |
| 1488 | CalpMTS (2–19)-sC18 | HeLa cells | TAM | 30367921 | 0.15 | Internalization | 1uM | 30min | 37ºC | Flow cytometry | Cellular uptake | SEEIITPVYCTGVSAQVQKGLRKRLRKFRNKIKEK |
| 1489 | sC18 | HeLa cells | TAM | 30367921 | 0.2 | Internalization | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | GLRKRLRKFRNKIKEK |
| 1490 | sC18 | HeLa cells | TAM | 30367921 | 0 | Internalization | 1uM | 30min | 37ºC | Flow cytometry | Cellular uptake | GLRKRLRKFRNKIKEK |
| 1491 | ALD5MTS (2–17) | MCF7 cells | TAM | 30367921 | 0.01 | Internalization | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | LSRTRAAAPNSRIFTR |
| 1492 | ALD5MTS (2–17) | MCF7 cells | TAM | 30367921 | 0.01 | Internalization | 1uM | 30min | 37ºC | Flow cytometry | Cellular uptake | LSRTRAAAPNSRIFTR |
| 1493 | ALD5MTS (2–17)-sC18 | MCF7 cells | TAM | 30367921 | 0.35 | Internalization | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | LSRTRAAAPNSRIFTRGLRKRLRKFRNKIKEK |
| 1494 | ALD5MTS (2–17)-sC18 | MCF7 cells | TAM | 30367921 | 0.08 | Internalization | 1uM | 30min | 37ºC | Flow cytometry | Cellular uptake | LSRTRAAAPNSRIFTRGLRKRLRKFRNKIKEK |
| 1495 | HSP60MTS (2–14) | MCF7 cells | TAM | 30367921 | 0.02 | Internalization | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | LRSSVVRSRATLR |
| 1496 | HSP60MTS (2–14) | MCF7 cells | TAM | 30367921 | 0.01 | Internalization | 1uM | 30min | 37ºC | Flow cytometry | Cellular uptake | LRSSVVRSRATLR |
| 1497 | HSP60MTS (2–14)-sC18 | MCF7 cells | TAM | 30367921 | 0.8 | Internalization | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | LRSSVVRSRATLRGLRKRLRKFRNKIKEK |
| 1498 | HSP60MTS (2–14)-sC18 | MCF7 cells | TAM | 30367921 | 0.05 | Internalization | 1uM | 30min | 37ºC | Flow cytometry | Cellular uptake | LRSSVVRSRATLRGLRKRLRKFRNKIKEK |
| 1499 | BNA3MTS (2–7) | MCF7 cells | TAM | 30367921 | 0.04 | Internalization | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | KQRFIR |
| 1500 | BNA3MTS (2–7) | MCF7 cells | TAM | 30367921 | 0 | Internalization | 1uM | 30min | 37ºC | Flow cytometry | Cellular uptake | KQRFIR |
| 1501 | BNA3MTS (2–7)-sC18 | MCF7 cells | TAM | 30367921 | 0.8 | Internalization | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | KQRFIRGLRKRLRKFRNKIKEK |
| 1502 | BNA3MTS (2–7)-sC18 | MCF7 cells | TAM | 30367921 | 0.05 | Internalization | 1uM | 30min | 37ºC | Flow cytometry | Cellular uptake | KQRFIRGLRKRLRKFRNKIKEK |
| 1503 | CalpMTS (2–19)-sC18 | MCF7 cells | TAM | 30367921 | 0.15 | Internalization | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | SEEIITPVYCTGVSAQVQKGLRKRLRKFRNKIKEK |
| 1504 | CalpMTS (2–19)-sC18 | MCF7 cells | TAM | 30367921 | 0.08 | Internalization | 1uM | 30min | 37ºC | Flow cytometry | Cellular uptake | SEEIITPVYCTGVSAQVQKGLRKRLRKFRNKIKEK |
| 1505 | sC18 | MCF7 cells | TAM | 30367921 | 0.1 | Internalization | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | GLRKRLRKFRNKIKEK |
| 1506 | sC18 | MCF7 cells | TAM | 30367921 | 0 | Internalization | 1uM | 30min | 37ºC | Flow cytometry | Cellular uptake | GLRKRLRKFRNKIKEK |
| 1507 | ALD5MTS (2–17) | TDA cells | TAM | 30367921 | 0.01 | Internalization | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | LSRTRAAAPNSRIFTR |
| 1508 | ALD5MTS (2–17) | TDA cells | TAM | 30367921 | 0 | Internalization | 1uM | 30min | 37ºC | Flow cytometry | Cellular uptake | LSRTRAAAPNSRIFTR |
| 1509 | ALD5MTS (2–17)-sC18 | TDA cells | TAM | 30367921 | 0.2 | Internalization | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | LSRTRAAAPNSRIFTRGLRKRLRKFRNKIKEK |
| 1510 | ALD5MTS (2–17)-sC18 | TDA cells | TAM | 30367921 | 0.1 | Internalization | 1uM | 30min | 37ºC | Flow cytometry | Cellular uptake | LSRTRAAAPNSRIFTRGLRKRLRKFRNKIKEK |
| 1511 | HSP60MTS (2–14) | TDA cells | TAM | 30367921 | 0.01 | Internalization | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | LRSSVVRSRATLR |
| 1512 | HSP60MTS (2–14) | TDA cells | TAM | 30367921 | 0 | Internalization | 1uM | 30min | 37ºC | Flow cytometry | Cellular uptake | LRSSVVRSRATLR |
| 1513 | HSP60MTS (2–14)-sC18 | TDA cells | TAM | 30367921 | 0.2 | Internalization | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | LRSSVVRSRATLRGLRKRLRKFRNKIKEK |
| 1514 | HSP60MTS (2–14)-sC18 | TDA cells | TAM | 30367921 | 0.1 | Internalization | 1uM | 30min | 37ºC | Flow cytometry | Cellular uptake | LRSSVVRSRATLRGLRKRLRKFRNKIKEK |
| 1515 | BNA3MTS (2–7) | TDA cells | TAM | 30367921 | 0.01 | Internalization | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | KQRFIR |
| 1516 | BNA3MTS (2–7) | TDA cells | TAM | 30367921 | 0 | Internalization | 1uM | 30min | 37ºC | Flow cytometry | Cellular uptake | KQRFIR |
| 1517 | BNA3MTS (2–7)-sC18 | TDA cells | TAM | 30367921 | 0.3 | Internalization | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | KQRFIRGLRKRLRKFRNKIKEK |
| 1518 | BNA3MTS (2–7)-sC18 | TDA cells | TAM | 30367921 | 0.08 | Internalization | 1uM | 30min | 37ºC | Flow cytometry | Cellular uptake | KQRFIRGLRKRLRKFRNKIKEK |
| 1519 | CalpMTS (2–19)-sC18 | TDA cells | TAM | 30367921 | 0.25 | Internalization | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | SEEIITPVYCTGVSAQVQKGLRKRLRKFRNKIKEK |
| 1520 | CalpMTS (2–19)-sC18 | TDA cells | TAM | 30367921 | 0.2 | Internalization | 1uM | 30min | 37ºC | Flow cytometry | Cellular uptake | SEEIITPVYCTGVSAQVQKGLRKRLRKFRNKIKEK |
| 1521 | sC18 | TDA cells | TAM | 30367921 | 0.15 | Internalization | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | GLRKRLRKFRNKIKEK |
| 1522 | sC18 | TDA cells | TAM | 30367921 | 0.05 | Internalization | 1uM | 30min | 37ºC | Flow cytometry | Cellular uptake | GLRKRLRKFRNKIKEK |
| 1523 | MTX-SCPP-PS | A549 cells | FITC | 29280317 | 0 | NA | NA | 2h | 37ºC | Flow cytometry | Cellular uptake | RLWMRWYSPRTRAYGC |
| 1524 | TI | MDA-MB-435S cells | Alexa488 | 31714739 | 6000 | Fluorescence intensity | 2uM | 1h | 37ºC | Flow cytometry | Cellular uptake | KWCFRVCYRGICYRRCR |
| 1525 | cTI | MDA-MB-435S cells | Alexa488 | 31714739 | 1000 | Fluorescence intensity | 2uM | 1h | 37ºC | Flow cytometry | Cellular uptake | KWCFRVCYRGICYRRCRG |
| 1526 | [Y8SI11S]cTI | MDA-MB-435S cells | Alexa488 | 31714739 | 5000 | Fluorescence intensity | 2uM | 1h | 37ºC | Flow cytometry | Cellular uptake | KWCFRVCSRGSCYRRCRG |
| 1527 | [F4S-Y13S]cTI | MDA-MB-435S cells | Alexa488 | 31714739 | 500 | Fluorescence intensity | 2uM | 1h | 37ºC | Flow cytometry | Cellular uptake | KWCSRVCYRGICSRRCRG |
| 1528 | TI | MM96L cells | Alexa488 | 31714739 | 5500 | Fluorescence intensity | 2uM | 1h | 37ºC | Flow cytometry | Cellular uptake | KWCFRVCYRGICYRRCR |
| 1529 | cTI | MM96L cells | Alexa488 | 31714739 | 2500 | Fluorescence intensity | 2uM | 1h | 37ºC | Flow cytometry | Cellular uptake | KWCFRVCYRGICYRRCRG |
| 1530 | [Y8SI11S]cTI | MM96L cells | Alexa488 | 31714739 | 4500 | Fluorescence intensity | 2uM | 1h | 37ºC | Flow cytometry | Cellular uptake | KWCFRVCSRGSCYRRCRG |
| 1531 | [F4S-Y13S]cTI | MM96L cells | Alexa488 | 31714739 | 2000 | Fluorescence intensity | 2uM | 1h | 37ºC | Flow cytometry | Cellular uptake | KWCSRVCYRGICSRRCRG |
| 1532 | TI | HeLa cells | Alexa488 | 31714739 | 3000 | Fluorescence intensity | 2uM | 1h | 37ºC | Flow cytometry | Cellular uptake | KWCFRVCYRGICYRRCR |
| 1533 | cTI | HeLa cells | Alexa488 | 31714739 | 1000 | Fluorescence intensity | 2uM | 1h | 37ºC | Flow cytometry | Cellular uptake | KWCFRVCYRGICYRRCRG |
| 1534 | [Y8SI11S]cTI | HeLa cells | Alexa488 | 31714739 | 2000 | Fluorescence intensity | 2uM | 1h | 37ºC | Flow cytometry | Cellular uptake | KWCFRVCSRGSCYRRCRG |
| 1535 | [F4S-Y13S]cTI | HeLa cells | Alexa488 | 31714739 | 500 | Fluorescence intensity | 2uM | 1h | 37ºC | Flow cytometry | Cellular uptake | KWCSRVCYRGICSRRCRG |
| 1536 | TI | HaCaT cells | Alexa488 | 31714739 | 2500 | Fluorescence intensity | 2uM | 1h | 37ºC | Flow cytometry | Cellular uptake | KWCFRVCYRGICYRRCR |
| 1537 | cTI | HaCaT cells | Alexa488 | 31714739 | 1500 | Fluorescence intensity | 2uM | 1h | 37ºC | Flow cytometry | Cellular uptake | KWCFRVCYRGICYRRCRG |
| 1538 | [Y8SI11S]cTI | HaCaT cells | Alexa488 | 31714739 | 2000 | Fluorescence intensity | 2uM | 1h | 37ºC | Flow cytometry | Cellular uptake | KWCFRVCSRGSCYRRCRG |
| 1539 | [F4S-Y13S]cTI | HaCaT cells | Alexa488 | 31714739 | 1000 | Fluorescence intensity | 2uM | 1h | 37ºC | Flow cytometry | Cellular uptake | KWCSRVCYRGICSRRCRG |
| 1540 | SynB1–ELP1–dnMAML | D54 cells | Fluorescein | 28140690 | 9 | Relative fluorescence | 30 uM | 1h | 37ºC | Flow cytometry | Cellular uptake | RGGRLSYSRRRFSTSTGRVPGVVVVVGGGAAGLPRHSAVMERLRRRIELCRRHHSTCEARYEAVSPERLELERQHTFALHQRCIQAKAKRAGKH |
| 1541 | SynB1–ELP1–dnMAML | D54 cells | Fluorescein | 28140690 | 37 | Relative fluorescence | 30 uM | 1h | 42ºC | Flow cytometry | Cellular uptake | RGGRLSYSRRRFSTSTGRVPGVVVVVGGGAAGLPRHSAVMERLRRRIELCRRHHSTCEARYEAVSPERLELERQHTFALHQRCIQAKAKRAGKH |
| 1542 | SynB1–ELP2–dnMAML | D54 cells | Fluorescein | 28140690 | 5 | Relative fluorescence | 30 uM | 1h | 37ºC | Flow cytometry | Cellular uptake | RGGRLSYSRRRFSTSTGRVPGVGGGGGGGAAAAAAAAGLPRHSAVMERLRRRIELCRRHHSTCEARYEAVSPERLELERQHTFALHQRCIQAKAKRAGKH |
| 1543 | SynB1–ELP2–dnMAML | D54 cells | Fluorescein | 28140690 | 8 | Relative fluorescence | 30 uM | 1h | 42ºC | Flow cytometry | Cellular uptake | RGGRLSYSRRRFSTSTGRVPGVGGGGGGGAAAAAAAAGLPRHSAVMERLRRRIELCRRHHSTCEARYEAVSPERLELERQHTFALHQRCIQAKAKRAGKH |
| 1544 | SynB1–ELP1–dnMAML | U251 cells | Fluorescein | 28140690 | 8 | Relative fluorescence | 30 uM | 1h | 37ºC | Flow cytometry | Cellular uptake | RGGRLSYSRRRFSTSTGRVPGVVVVVGGGAAGLPRHSAVMERLRRRIELCRRHHSTCEARYEAVSPERLELERQHTFALHQRCIQAKAKRAGKH |
| 1545 | SynB1–ELP1–dnMAML | U251 cells | Fluorescein | 28140690 | 24 | Relative fluorescence | 30 uM | 1h | 42ºC | Flow cytometry | Cellular uptake | RGGRLSYSRRRFSTSTGRVPGVVVVVGGGAAGLPRHSAVMERLRRRIELCRRHHSTCEARYEAVSPERLELERQHTFALHQRCIQAKAKRAGKH |
| 1546 | SynB1–ELP2–dnMAML | U251 cells | Fluorescein | 28140690 | 7 | Relative fluorescence | 30 uM | 1h | 37ºC | Flow cytometry | Cellular uptake | RGGRLSYSRRRFSTSTGRVPGVGGGGGGGAAAAAAAAGLPRHSAVMERLRRRIELCRRHHSTCEARYEAVSPERLELERQHTFALHQRCIQAKAKRAGKH |
| 1547 | SynB1–ELP2–dnMAML | U251 cells | Fluorescein | 28140690 | 10 | Relative fluorescence | 30 uM | 1h | 42ºC | Flow cytometry | Cellular uptake | RGGRLSYSRRRFSTSTGRVPGVGGGGGGGAAAAAAAAGLPRHSAVMERLRRRIELCRRHHSTCEARYEAVSPERLELERQHTFALHQRCIQAKAKRAGKH |
| 1548 | KT2 | HCT116 cells | FITC | 31073999 | 100 | Mean Fluorescence intensity | 1.25uM | 4h | 37ºC | Flow cytometry | Cellular uptake | NGVQPKYKWWKWWKKWW-NH2 |
| 1549 | KT2 | HCT116 cells | FITC | 31073999 | 200 | Mean Fluorescence intensity | 2.5uM | 4h | 37ºC | Flow cytometry | Cellular uptake | NGVQPKYKWWKWWKKWW-NH2 |
| 1550 | KT2 | HCT116 cells | FITC | 31073999 | 500 | Mean Fluorescence intensity | 5uM | 4h | 37ºC | Flow cytometry | Cellular uptake | NGVQPKYKWWKWWKKWW-NH2 |
| 1551 | KT2 | HCT116 cells | FITC | 31073999 | 800 | Mean Fluorescence intensity | 10uM | 4h | 37ºC | Flow cytometry | Cellular uptake | NGVQPKYKWWKWWKKWW-NH2 |
| 1552 | palmitoyl-cyclic-(D-Arg)12 | HeLa cells | FITC | 29530390 | 100 | Mean Fluorescence intensity | 9.0 uM | 30min | 37ºC | Flow cytometry | Cellular uptake | C37H66N7O17P3S-rrrrrrrrrrrr |
| 1553 | palmitoyl-cyclic-(D-Arg)12 | HeLa cells | FITC | 29530390 | 300 | Mean Fluorescence intensity | 9.0 uM | 1h | 37ºC | Flow cytometry | Cellular uptake | C37H66N7O17P3S-rrrrrrrrrrrr |
| 1554 | palmitoyl-cyclic-(D-Arg)12 | HeLa cells | FITC | 29530390 | 1000 | Mean Fluorescence intensity | 9.0 uM | 2h | 37ºC | Flow cytometry | Cellular uptake | C37H66N7O17P3S-rrrrrrrrrrrr |
| 1555 | palmitoyl-cyclic-(D-Arg)12 | HeLa cells | FITC | 29530390 | 50 | Mean Fluorescence intensity | 9.0 uM | 30min | 4ºC | Flow cytometry | Cellular uptake | C37H66N7O17P3S-rrrrrrrrrrrr |
| 1556 | palmitoyl-cyclic-(D-Arg)12 | HeLa cells | FITC | 29530390 | 50 | Mean Fluorescence intensity | 9.0 uM | 1h | 4ºC | Flow cytometry | Cellular uptake | C37H66N7O17P3S-rrrrrrrrrrrr |
| 1557 | palmitoyl-cyclic-(D-Arg)12 | HeLa cells | FITC | 29530390 | 200 | Mean Fluorescence intensity | 9.0 uM | 2h | 4ºC | Flow cytometry | Cellular uptake | C37H66N7O17P3S-rrrrrrrrrrrr |
| 1558 | P-(dNP2)-DOX | HeLa cells | Doxorubicin | 30205127 | 2.5 | Fluorescence intensity | 10 ug/ml | 2h | 37ºC | Flow cytometry | Cellular uptake | CKIKKVKKKGRKKIKKVKKKGRK |
| 1559 | P-(dNP2)-DOX | HeLa cells | Doxorubicin | 30205127 | 3.5 | Fluorescence intensity | 10 ug/ml | 4h | 37ºC | Flow cytometry | Cellular uptake | CKIKKVKKKGRKKIKKVKKKGRK |
| 1560 | KD3 | MCF7 cells | Alexa488 | 33533253 | 5 | Relative Cellular uptake | 2 uM | 1h | 37ºC | Flow cytometry | Cellular uptake | LTFKEYWDQLTSAA |
| 1561 | cTAT | MCF7 cells | Alexa488 | 33533253 | 10 | Relative Cellular uptake | 2 uM | 1h | 37ºC | Flow cytometry | Cellular uptake | KrRrGgKkRrD |
| 1562 | cR10 | MCF7 cells | Alexa488 | 33533253 | 15 | Relative Cellular uptake | 2 uM | 1h | 37ºC | Flow cytometry | Cellular uptake | KrRrRrRrRrRE |
| 1563 | cTAT-KD3 | MCF7 cells | Alexa488 | 33533253 | 25 | Relative Cellular uptake | 2 uM | 1h | 37ºC | Flow cytometry | Cellular uptake | KrRrGgKkRrDLTFKEYWDQLTSAA |
| 1564 | cR10-KD3 | MCF7 cells | Alexa488 | 33533253 | 45 | Relative Cellular uptake | 2 uM | 1h | 37ºC | Flow cytometry | Cellular uptake | KrRrRrRrRrRELTFKEYWDQLTSAA |
| 1565 | KD3 | HeLa cells | Alexa488 | 33533253 | 3 | Relative Cellular uptake | 2 uM | 1h | 37ºC | Flow cytometry | Cellular uptake | LTFKEYWDQLTSAA |
| 1566 | cTAT | HeLa cells | Alexa488 | 33533253 | 15 | Relative Cellular uptake | 2 uM | 1h | 37ºC | Flow cytometry | Cellular uptake | KrRrGgKkRrD |
| 1567 | cR10 | HeLa cells | Alexa488 | 33533253 | 18 | Relative Cellular uptake | 2 uM | 1h | 37ºC | Flow cytometry | Cellular uptake | KrRrRrRrRrRE |
| 1568 | cTAT-KD3 | HeLa cells | Alexa488 | 33533253 | 18 | Relative Cellular uptake | 2 uM | 1h | 37ºC | Flow cytometry | Cellular uptake | KrRrGgKkRrDLTFKEYWDQLTSAA |
| 1569 | cR10-KD3 | HeLa cells | Alexa488 | 33533253 | 20 | Relative Cellular uptake | 2 uM | 1h | 37ºC | Flow cytometry | Cellular uptake | KrRrRrRrRrRELTFKEYWDQLTSAA |
| 1570 | KD3 | MCF7 cells | Alexa488 | 33533253 | 0 | Relative Cellular uptake | 2 uM | 2h | 4ºC | Flow cytometry | Cellular uptake | LTFKEYWDQLTSAA |
| 1571 | cTAT | MCF7 cells | Alexa488 | 33533253 | 1 | Relative Cellular uptake | 2 uM | 2h | 4ºC | Flow cytometry | Cellular uptake | KrRrGgKkRrD |
| 1572 | cR10 | MCF7 cells | Alexa488 | 33533253 | 15 | Relative Cellular uptake | 2 uM | 2h | 4ºC | Flow cytometry | Cellular uptake | KrRrRrRrRrRE |
| 1573 | cTAT-KD3 | MCF7 cells | Alexa488 | 33533253 | 0 | Relative Cellular uptake | 2 uM | 2h | 4ºC | Flow cytometry | Cellular uptake | KrRrGgKkRrDLTFKEYWDQLTSAA |
| 1574 | cR10-KD3 | MCF7 cells | Alexa488 | 33533253 | 1 | Relative Cellular uptake | 2 uM | 2h | 4ºC | Flow cytometry | Cellular uptake | KrRrRrRrRrRELTFKEYWDQLTSAA |
| 1575 | KD3 | HeLa cells | Alexa488 | 33533253 | 0.2 | Relative Cellular uptake | 2 uM | 2h | 4ºC | Flow cytometry | Cellular uptake | LTFKEYWDQLTSAA |
| 1576 | cTAT | HeLa cells | Alexa488 | 33533253 | 1.3 | Relative Cellular uptake | 2 uM | 2h | 4ºC | Flow cytometry | Cellular uptake | KrRrGgKkRrD |
| 1577 | cR10 | HeLa cells | Alexa488 | 33533253 | 3 | Relative Cellular uptake | 2 uM | 2h | 4ºC | Flow cytometry | Cellular uptake | KrRrRrRrRrRE |
| 1578 | cTAT-KD3 | HeLa cells | Alexa488 | 33533253 | 0.8 | Relative Cellular uptake | 2 uM | 2h | 4ºC | Flow cytometry | Cellular uptake | KrRrGgKkRrD-LTFKEYWDQLTSAA |
| 1579 | cR10-KD3 | HeLa cells | Alexa488 | 33533253 | 2.1 | Relative Cellular uptake | 2 uM | 2h | 4ºC | Flow cytometry | Cellular uptake | KrRrRrRrRrRE-LTFKEYWDQLTSAA |
| 1580 | N50-sC18* | HeLa cells | Carboxyfluorescein | 29977402 | 15000 | Fluorescence intensity | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | VQRKRQKLMPGLRKRLRKFRNK |
| 1581 | N50-sC18* | HeLa cells | Carboxyfluorescein | 29977402 | 7000 | Fluorescence intensity | 10uM | 120min | 37ºC | Flow cytometry | Cellular uptake | VQRKRQKLMPGLRKRLRKFRNK |
| 1582 | N50-sC18* | HeLa cells | Carboxyfluorescein | 29977402 | 1000 | Fluorescence intensity | 10uM | 30min | 4ºC | Flow cytometry | Cellular uptake | VQRKRQKLMPGLRKRLRKFRNK |
| 1583 | NrTP-sC18* | HeLa cells | Carboxyfluorescein | 29977402 | 13000 | Fluorescence intensity | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | YKQCHKKGGKKGSGGLRKRLRKFRNK |
| 1584 | NrTP-sC18* | HeLa cells | Carboxyfluorescein | 29977402 | 10000 | Fluorescence intensity | 10uM | 120min | 37ºC | Flow cytometry | Cellular uptake | YKQCHKKGGKKGSGGLRKRLRKFRNK |
| 1585 | NrTP-sC18* | HeLa cells | Carboxyfluorescein | 29977402 | 2900 | Fluorescence intensity | 10uM | 30min | 4ºC | Flow cytometry | Cellular uptake | YKQCHKKGGKKGSGGLRKRLRKFRNK |
| 1586 | N50-sC18* | MCF7 cells | Carboxyfluorescein | 29977402 | 17000 | Fluorescence intensity | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | VQRKRQKLMPGLRKRLRKFRNK |
| 1587 | N50-sC18* | MCF7 cells | Carboxyfluorescein | 29977402 | 13000 | Fluorescence intensity | 10uM | 120min | 37ºC | Flow cytometry | Cellular uptake | VQRKRQKLMPGLRKRLRKFRNK |
| 1588 | N50-sC18* | MCF7 cells | Carboxyfluorescein | 29977402 | 16000 | Fluorescence intensity | 10uM | 30min | 4ºC | Flow cytometry | Cellular uptake | VQRKRQKLMPGLRKRLRKFRNK |
| 1589 | NrTP-sC18* | MCF7 cells | Carboxyfluorescein | 29977402 | 21000 | Fluorescence intensity | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | YKQCHKKGGKKGSGGLRKRLRKFRNK |
| 1590 | NrTP-sC18* | MCF7 cells | Carboxyfluorescein | 29977402 | 7000 | Fluorescence intensity | 10uM | 120min | 37ºC | Flow cytometry | Cellular uptake | YKQCHKKGGKKGSGGLRKRLRKFRNK |
| 1591 | NrTP-sC18* | MCF7 cells | Carboxyfluorescein | 29977402 | 7500 | Fluorescence intensity | 10uM | 30min | 4ºC | Flow cytometry | Cellular uptake | YKQCHKKGGKKGSGGLRKRLRKFRNK |
| 1592 | Conjugate 1a | U87 cells | Carboxyfluorescein | 31243977 | 0.4 | Fluorescence intensity | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | c[DKP-RGD]-PEG4-GLRKRLRK(CF)FRNKIKEK-CONH2 |
| 1593 | Conjugate 1a | HT29 cells | Carboxyfluorescein | 31243977 | 0.38 | Fluorescence intensity | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | c[DKP-RGD]-PEG4-GLRKRLRK(CF)FRNKIKEK-CONH2 |
| 1594 | Conjugate 1a | MCF7 cells | Carboxyfluorescein | 31243977 | 0.3 | Fluorescence intensity | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | c[DKP-RGD]-PEG4-GLRKRLRK(CF)FRNKIKEK-CONH2 |
| 1595 | Conjugate 2a | U87 cells | Carboxyfluorescein | 31243977 | 1 | Fluorescence intensity | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | GLRKRLRK(CF)FRNKIKEK-CONH2 |
| 1596 | Conjugate 2a | HT29 cells | Carboxyfluorescein | 31243977 | 0.37 | Fluorescence intensity | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | GLRKRLRK(CF)FRNKIKEK-CONH2 |
| 1597 | Conjugate 2a | MCF7 cells | Carboxyfluorescein | 31243977 | 0.35 | Fluorescence intensity | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | GLRKRLRK(CF)FRNKIKEK-CONH2 |
| 1598 | Conjugate 1a | U87 cells | Carboxyfluorescein | 31243977 | 0.8 | Fluorescence intensity | 10uM | 1h | 37ºC | Flow cytometry | Cellular uptake | c[DKP-RGD]-PEG4-GLRKRLRK(CF)FRNKIKEK-CONH2 |
| 1599 | Conjugate 1a | HT29 cells | Carboxyfluorescein | 31243977 | 0.75 | Fluorescence intensity | 10uM | 1h | 37ºC | Flow cytometry | Cellular uptake | c[DKP-RGD]-PEG4-GLRKRLRK(CF)FRNKIKEK-CONH2 |
| 1600 | Conjugate 1a | MCF7 cells | Carboxyfluorescein | 31243977 | 0.4 | Fluorescence intensity | 10uM | 1h | 37ºC | Flow cytometry | Cellular uptake | c[DKP-RGD]-PEG4-GLRKRLRK(CF)FRNKIKEK-CONH2 |
| 1601 | Conjugate 2a | U87 cells | Carboxyfluorescein | 31243977 | 1.2 | Fluorescence intensity | 10uM | 1h | 37ºC | Flow cytometry | Cellular uptake | GLRKRLRK(CF)FRNKIKEK-CONH2 |
| 1602 | Conjugate 2a | HT29 cells | Carboxyfluorescein | 31243977 | 0.43 | Fluorescence intensity | 10uM | 1h | 37ºC | Flow cytometry | Cellular uptake | GLRKRLRK(CF)FRNKIKEK-CONH2 |
| 1603 | Conjugate 2a | MCF7 cells | Carboxyfluorescein | 31243977 | 0.6 | Fluorescence intensity | 10uM | 1h | 37ºC | Flow cytometry | Cellular uptake | GLRKRLRK(CF)FRNKIKEK-CONH2 |
| 1604 | R8-Lip | C6 cells | CFPE | 26877777 | 40 | Fluorescence intensity | NA | 4h | 37ºC | Flow cytometry | Cellular uptake | RRRRRRRR-Lip |
| 1605 | R8-RGD-Lip | C6 cells | CFPE | 26877777 | 60 | Fluorescence intensity | NA | 4h | 37ºC | Flow cytometry | Cellular uptake | Cys-RRRRRRRR-RGD-Lip |
| 1606 | R8-EGR-Lip | C6 cells | CFPE | 26877777 | 80 | Fluorescence intensity | NA | 4h | 37ºC | Flow cytometry | Cellular uptake | Cys-RRRRRRRR-EGR-Lip |
| 1607 | R8-dGR-Lip | C6 cells | CFPE | 26877777 | 90 | Fluorescence intensity | NA | 4h | 37ºC | Flow cytometry | Cellular uptake | Cys-RRRRRRRR-dGR-Lip |
| 1608 | R8-Lip | bEnd.3 cells | CFPE | 26877777 | 10 | Fluorescence intensity | NA | 4h | 37ºC | Flow cytometry | Cellular uptake | RRRRRRRR-Lip |
| 1609 | R8-RGD-Lip | bEnd.3 cells | CFPE | 26877777 | 20 | Fluorescence intensity | NA | 4h | 37ºC | Flow cytometry | Cellular uptake | Cys-RRRRRRRR-RGD-Lip |
| 1610 | R8-EGR-Lip | bEnd.3 cells | CFPE | 26877777 | 18 | Fluorescence intensity | NA | 4h | 37ºC | Flow cytometry | Cellular uptake | Cys-RRRRRRRR-EGR-Lip |
| 1611 | R8-dGR-Lip | bEnd.3 cells | CFPE | 26877777 | 25 | Fluorescence intensity | NA | 4h | 37ºC | Flow cytometry | Cellular uptake | Cys-RRRRRRRR-dGR-Lip |
| 1612 | R8-Lip | HeLa cells | CFPE | 26877777 | 6 | Fluorescence intensity | NA | 4h | 37ºC | Flow cytometry | Cellular uptake | RRRRRRRR-Lip |
| 1613 | R8-RGD-Lip | HeLa cells | CFPE | 26877777 | 7 | Fluorescence intensity | NA | 4h | 37ºC | Flow cytometry | Cellular uptake | Cys-RRRRRRRR-RGD-Lip |
| 1614 | R8-EGR-Lip | HeLa cells | CFPE | 26877777 | 8 | Fluorescence intensity | NA | 4h | 37ºC | Flow cytometry | Cellular uptake | Cys-RRRRRRRR-EGR-Lip |
| 1615 | R8-dGR-Lip | HeLa cells | CFPE | 26877777 | 9 | Fluorescence intensity | NA | 4h | 37ºC | Flow cytometry | Cellular uptake | Cys-RRRRRRRR-dGR-Lip |
| 1616 | HL6 | A549 cells | FITC | 31253836 | 0 | NA | NA | 1h | 37ºC | Fluorescent Microscopy | Cellular uptake | CHHHHHRRWQWRHHHHHC |
| 1617 | hPep1 | HeLa cells | AF568-SSO | 34440250 | 100 | Relative fluorescence | 25nM | 4h | NA | Fluorescence spectroscopy | Cellular uptake | H-LAKLAKA(R8)AKLLKA(S5)AKAL-NH2 |
| 1618 | hPep2 | HeLa cells | AF568-SSO | 34440250 | 100 | Relative fluorescence | 25nM | 4h | NA | Fluorescence spectroscopy | Cellular uptake | H-LAKLAKA(R8)AKLLKA(S8)AKAL-NH2 |
| 1619 | hPep3 | HeLa cells | AF568-SSO | 34440250 | 300 | Relative fluorescence | 25nM | 4h | NA | Fluorescence spectroscopy | Cellular uptake | H-L(R8)KLAKA(R8)AKLLKA(R8)AKAL-NH2 |
| 1620 | hPep1 | HeLa cells | AF568-SSO | 34440250 | 100 | Relative fluorescence | 50nM | 4h | NA | Fluorescence spectroscopy | Cellular uptake | H-LAKLAKA(R8)AKLLKA(S5)AKAL-NH2 |
| 1621 | hPep2 | HeLa cells | AF568-SSO | 34440250 | 300 | Relative fluorescence | 50nM | 4h | NA | Fluorescence spectroscopy | Cellular uptake | H-LAKLAKA(R8)AKLLKA(S8)AKAL-NH2 |
| 1622 | hPep3 | HeLa cells | AF568-SSO | 34440250 | 1000 | Relative fluorescence | 50nM | 4h | NA | Fluorescence spectroscopy | Cellular uptake | H-L(R8)KLAKA(R8)AKLLKA(R8)AKAL-NH2 |
| 1623 | hPep1 | HeLa cells | AF568-SSO | 34440250 | 1000 | Relative fluorescence | 100nM | 4h | NA | Fluorescence spectroscopy | Cellular uptake | H-LAKLAKA(R8)AKLLKA(S5)AKAL-NH2 |
| 1624 | hPep2 | HeLa cells | AF568-SSO | 34440250 | 1500 | Relative fluorescence | 100nM | 4h | NA | Fluorescence spectroscopy | Cellular uptake | H-LAKLAKA(R8)AKLLKA(S8)AKAL-NH2 |
| 1625 | hPep3 | HeLa cells | AF568-SSO | 34440250 | 2500 | Relative fluorescence | 100nM | 4h | NA | Fluorescence spectroscopy | Cellular uptake | H-L(R8)KLAKA(R8)AKLLKA(R8)AKAL-NH2 |
| 1626 | hPep1 | HeLa cells | AF568-SSO | 34440250 | 5500 | Relative fluorescence | 200nM | 4h | NA | Fluorescence spectroscopy | Cellular uptake | H-LAKLAKA(R8)AKLLKA(S5)AKAL-NH2 |
| 1627 | hPep2 | HeLa cells | AF568-SSO | 34440250 | 6000 | Relative fluorescence | 200nM | 4h | NA | Fluorescence spectroscopy | Cellular uptake | H-LAKLAKA(R8)AKLLKA(S8)AKAL-NH2 |
| 1628 | hPep3 | HeLa cells | AF568-SSO | 34440250 | 7000 | Relative fluorescence | 200nM | 4h | NA | Fluorescence spectroscopy | Cellular uptake | H-L(R8)KLAKA(R8)AKLLKA(R8)AKAL-NH2 |
| 1629 | VaspinN | HEK293 cells | TAMRA | 33866927 | 150 | Relative fluorescence | 10uM | 30min | 37ºC | Fluorescent Microscopy | Cellular uptake | LKPSFSPRNY |
| 1630 | VaspinHA1 | HEK293 cells | TAMRA | 33866927 | 80 | Relative fluorescence | 10uM | 30min | 37ºC | Fluorescent Microscopy | Cellular uptake | KALSEVQGWKQRMAAKELAR |
| 1631 | VaspinHA2 | HEK293 cells | TAMRA | 33866927 | 150 | Relative fluorescence | 10uM | 30min | 37ºC | Fluorescent Microscopy | Cellular uptake | KQRMAAKELAR |
| 1632 | VaspinN | NIH-3T3 cells | TAMRA | 33866927 | 2500 | Relative fluorescence | 10uM | 30min | 37ºC | Fluorescent Microscopy | Cellular uptake | LKPSFSPRNY |
| 1633 | VaspinHA1 | NIH-3T3 cells | TAMRA | 33866927 | 2000 | Relative fluorescence | 10uM | 30min | 37ºC | Fluorescent Microscopy | Cellular uptake | KALSEVQGWKQRMAAKELAR |
| 1634 | VaspinHA2 | NIH-3T3 cells | TAMRA | 33866927 | 2000 | Relative fluorescence | 10uM | 30min | 37ºC | Fluorescent Microscopy | Cellular uptake | KQRMAAKELAR |
| 1635 | NLC-RGE | MDA-MB-231 cells | Cou-6 | 29528244 | 70 | Fluorescence intensity | 0.002ug/mL | 30min | 37ºC | Flow cytometry | Cellular uptake | RGERPPR |
| 1636 | NLC-cRGD | MDA-MB-231 cells | Cou-6 | 29528244 | 50 | Fluorescence intensity | 0.002ug/mL | 30min | 37ºC | Flow cytometry | Cellular uptake | CRGDRGPDC |
| 1637 | NLC-RGE/cRG | MDA-MB-231 cells | Cou-6 | 29528244 | 60 | Fluorescence intensity | 0.002ug/mL | 30min | 37ºC | Flow cytometry | Cellular uptake | RGERPPRCRGDRGPDC |
| 1638 | NLC-RGE | MDA-MB-231 cells | Cou-6 | 29528244 | 210 | Fluorescence intensity | 0.002ug/mL | 2h | 37ºC | Flow cytometry | Cellular uptake | RGERPPR |
| 1639 | NLC-cRGD | MDA-MB-231 cells | Cou-6 | 29528244 | 160 | Fluorescence intensity | 0.002ug/mL | 2h | 37ºC | Flow cytometry | Cellular uptake | CRGDRGPDC |
| 1640 | NLC-RGE/cRG | MDA-MB-231 cells | Cou-6 | 29528244 | 120 | Fluorescence intensity | 0.002ug/mL | 2h | 37ºC | Flow cytometry | Cellular uptake | RGERPPRCRGDRGPDC |
| 1641 | NLC-RGE | MDA-MB-231 cells | Cou-6 | 29528244 | 250 | Fluorescence intensity | 0.002ug/mL | 4h | 37ºC | Flow cytometry | Cellular uptake | RGERPPR |
| 1642 | NLC-cRGD | MDA-MB-231 cells | Cou-6 | 29528244 | 230 | Fluorescence intensity | 0.002ug/mL | 4h | 37ºC | Flow cytometry | Cellular uptake | CRGDRGPDC |
| 1643 | NLC-RGE/cRG | MDA-MB-231 cells | Cou-6 | 29528244 | 200 | Fluorescence intensity | 0.002ug/mL | 4h | 37ºC | Flow cytometry | Cellular uptake | RGERPPRCRGDRGPDC |
| 1644 | NLC-RGE | MDA-MB-231 cells | Cou-6 | 29528244 | 342.34 | Fluorescence intensity | 0.002ug/mL | 12h | 37ºC | Flow cytometry | Cellular uptake | RGERPPR |
| 1645 | NLC-cRGD | MDA-MB-231 cells | Cou-6 | 29528244 | 254.4 | Fluorescence intensity | 0.002ug/mL | 12h | 37ºC | Flow cytometry | Cellular uptake | CRGDRGPDC |
| 1646 | NLC-RGE/cRG | MDA-MB-231 cells | Cou-6 | 29528244 | 245.8 | Fluorescence intensity | 0.002ug/mL | 12h | 37ºC | Flow cytometry | Cellular uptake | RGERPPRCRGDRGPDC |
| 1647 | CPP–siRNA/N-NB | MCF7 cells | siRNA | 26492155 | 30 | Mean Fluorescence intensity | NA | 4h | 37ºC | Flow cytometry | Cellular uptake | CKRRMKWKK |
| 1648 | CPP–siRNA/YSA-NB | MCF7 cells | siRNA | 26492155 | 40 | Mean Fluorescence intensity | NA | 4h | 37ºC | Flow cytometry | Cellular uptake | CKRRMKWKK-YSAYPDSVPMMS |
| 1649 | CPP-siRNA/N-NB (+US) | MCF7 cells | siRNA | 26492155 | 110 | Mean Fluorescence intensity | NA | 4h | 37ºC | Flow cytometry | Cellular uptake | CKRRMKWKK |
| 1650 | CPP–siRNA/YSA-NB (+US) | MCF7 cells | siRNA | 26492155 | 130 | Mean Fluorescence intensity | NA | 4h | 37ºC | Flow cytometry | Cellular uptake | CKRRMKWKK-YSAYPDSVPMMS |
| 1651 | I-LCP | HCT116 cells | Radiolabelled Iodine (125I) | 31445852 | 10 | Cellular uptake (%) | NA | 2h | 37ºC | Flow cytometry | Cellular uptake | Ac-eeeeeeeeeXPAANVGrrrrrrrrrXk([125I]IB)-NH2 |
| 1652 | I-NCP | HCT116 cells | Radiolabelled Iodine (125I) | 31445852 | 2 | Cellular uptake (%) | NA | 2h | 37ºC | Flow cytometry | Cellular uptake | Ac-eeeeeeeeeXPAACtVGrrrrrrrrrXk([125I]IB)-NH2 |
| 1653 | LPC | HCT116 cells | FL | 31445852 | 5 | Cellular uptake (%) | NA | 2h | 37ºC | Flow cytometry | Cellular uptake | Ac-eeeeeeeeeXPAANVGrrrrrrrrrXk(FL)-NH2 |
| 1654 | NCP | HCT116 cells | FL | 31445852 | 7 | Cellular uptake (%) | NA | 2h | 37ºC | Flow cytometry | Cellular uptake | Ac-eeeeeeeeeXPAACtVGrrrrrrrrrXk(FL)-NH2 |
| 1655 | LCP-r | HCT116 cells | FL | 31445852 | 31 | Cellular uptake (%) | NA | 2h | 37ºC | Flow cytometry | Cellular uptake | Ac-XPAANVGrrrrrrrrrXk(FL)-NH2 |
| 1656 | NCP-r | HCT116 cells | FL | 31445852 | 33 | Cellular uptake (%) | NA | 2h | 37ºC | Flow cytometry | Cellular uptake | Ac-XPAACtVGrrrrrrrrrXk(FL)-NH2 |
| 1657 | R9 | A549 cells | FITC | 27074859 | 65 | Relative fraction of positive cells (%) | 10uM | 1.5h | 37ºC | Flow cytometry | Cellular uptake | RRRRRRRRR |
| 1658 | R5W3R4 | A549 cells | FITC | 27074859 | 70 | Relative fraction of positive cells (%) | 10uM | 1.5h | 37ºC | Flow cytometry | Cellular uptake | RRRRRWWWRRRR |
| 1659 | [RW]6 | A549 cells | FITC | 27074859 | 72 | Relative fraction of positive cells (%) | 10uM | 1.5h | 37ºC | Flow cytometry | Cellular uptake | RWRWRWRWRWRW |
| 1660 | R9 | A549 cells | FITC | 27074859 | 73 | Relative fraction of positive cells (%) | 25uM | 1.5h | 37ºC | Flow cytometry | Cellular uptake | RRRRRRRRR |
| 1661 | R5W3R4 | A549 cells | FITC | 27074859 | 80 | Relative fraction of positive cells (%) | 25uM | 1.5h | 37ºC | Flow cytometry | Cellular uptake | RRRRRWWWRRRR |
| 1662 | [RW]6 | A549 cells | FITC | 27074859 | 79 | Relative fraction of positive cells (%) | 25uM | 1.5h | 37ºC | Flow cytometry | Cellular uptake | RWRWRWRWRWRW |
| 1663 | R9 | A549 cells | FITC | 27074859 | 88 | Relative fraction of positive cells (%) | 50uM | 1.5h | 37ºC | Flow cytometry | Cellular uptake | RRRRRRRRR |
| 1664 | R5W3R4 | A549 cells | FITC | 27074859 | 95 | Relative fraction of positive cells (%) | 50uM | 1.5h | 37ºC | Flow cytometry | Cellular uptake | RRRRRWWWRRRR |
| 1665 | [RW]6 | A549 cells | FITC | 27074859 | 85 | Relative fraction of positive cells (%) | 50uM | 1.5h | 37ºC | Flow cytometry | Cellular uptake | RWRWRWRWRWRW |
| 1666 | R9/E9 | A549 cells | FITC | 27074859 | 52 | Relative fraction of positive cells (%) | 10uM | 1.5h | 37ºC | Flow cytometry | Cellular uptake | RRRRRRRRR-EEEEEEEEE |
| 1667 | R5W3R4/E9 | A549 cells | FITC | 27074859 | 55 | Relative fraction of positive cells (%) | 10uM | 1.5h | 37ºC | Flow cytometry | Cellular uptake | RRRRRWWWRRRR-EEEEEEEEE |
| 1668 | [RW]6/E9 | A549 cells | FITC | 27074859 | 56 | Relative fraction of positive cells (%) | 10uM | 1.5h | 37ºC | Flow cytometry | Cellular uptake | RWRWRWRWRWRW-EEEEEEEEE |
| 1669 | R9/E9 | A549 cells | FITC | 27074859 | 72 | Relative fraction of positive cells (%) | 25uM | 1.5h | 37ºC | Flow cytometry | Cellular uptake | RRRRRRRRR-EEEEEEEEE |
| 1670 | R5W3R4/E9 | A549 cells | FITC | 27074859 | 75 | Relative fraction of positive cells (%) | 25uM | 1.5h | 37ºC | Flow cytometry | Cellular uptake | RRRRRWWWRRRR-EEEEEEEEE |
| 1671 | [RW]6/E9 | A549 cells | FITC | 27074859 | 78 | Relative fraction of positive cells (%) | 25uM | 1.5h | 37ºC | Flow cytometry | Cellular uptake | RWRWRWRWRWRW-EEEEEEEEE |
| 1672 | R9/E9 | A549 cells | FITC | 27074859 | 82 | Relative fraction of positive cells (%) | 50uM | 1.5h | 37ºC | Flow cytometry | Cellular uptake | RRRRRRRRR-EEEEEEEEE |
| 1673 | R5W3R4/E9 | A549 cells | FITC | 27074859 | 85 | Relative fraction of positive cells (%) | 50uM | 1.5h | 37ºC | Flow cytometry | Cellular uptake | RRRRRWWWRRRR-EEEEEEEEE |
| 1674 | [RW]6/E9 | A549 cells | FITC | 27074859 | 86 | Relative fraction of positive cells (%) | 50uM | 1.5h | 37ºC | Flow cytometry | Cellular uptake | RWRWRWRWRWRW-EEEEEEEEE |
| 1675 | Dabcyl–Arg6–Lys(Rh)–NH2 | HeLa cells | Carboxyfluorescein | 34032919 | 200000 | Fluorescence intensity | 2.5uM | 30min | 37ºC | Flow cytometry | Cellular uptake | Dabcyl-RRRRRRK-Rho-NH2 |
| 1676 | Dabcyl–Arg6–Lys(Rh)–NH2 | HeLa cells | Carboxyfluorescein | 34032919 | 800000 | Fluorescence intensity | 5uM | 30min | 37ºC | Flow cytometry | Cellular uptake | Dabcyl-RRRRRRK-Rho-NH2 |
| 1677 | Dabcyl–Arg6–Lys(Rh)–NH2 | HeLa cells | Carboxyfluorescein | 34032919 | 1050000 | Fluorescence intensity | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | Dabcyl-RRRRRRK-Rho-NH2 |
| 1678 | H–Arg6–Lys(Rh)–NH2 | HeLa cells | Carboxyfluorescein | 34032919 | 0 | Fluorescence intensity | 2.5uM | 30min | 37ºC | Flow cytometry | Cellular uptake | H-RRRRRRK-Rho-NH2 |
| 1679 | H–Arg6–Lys(Rh)–NH2 | HeLa cells | Carboxyfluorescein | 34032919 | 5000 | Fluorescence intensity | 5uM | 30min | 37ºC | Flow cytometry | Cellular uptake | H-RRRRRRK-Rho-NH2 |
| 1680 | H–Arg6–Lys(Rh)–NH2 | HeLa cells | Carboxyfluorescein | 34032919 | 5000 | Fluorescence intensity | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | H-RRRRRRK-Rho-NH2 |
| 1681 | biotinyl-GM3BP | HeLa cells | GFP | 28051846 | 8 | Fluorescence intensity | 5uM | 1h | 37ºC | Flow cytometry | Cellular uptake | GWWYKGRARPVSAVAK |
| 1682 | biotinyl-GM3BP | HeLa cells | GFP | 28051846 | 1 | Fluorescence intensity | 5uM | 1h | 4ºC | Flow cytometry | Cellular uptake | GWWYKGRARPVSAVAK |
| 1683 | biotinyl-TAT | HeLa cells | GFP | 28051846 | 0 | NA | NA | NA | NA | Flow cytometry | Cellular uptake | YGRKKRRQRRRK |
| 1684 | biotinyl-CP8 | HeLa cells | GFP | 28051846 | 0 | NA | NA | NA | NA | Flow cytometry | Cellular uptake | AETVESCLAKPHTENK |
| 1685 | GGL27 | A375 cells | TAMRA | 31672541 | 25 | Corrected total cell fluorescence | 5uM | 2h | 37ºC | Flow cytometry | Cellular uptake | GGLIKTKRKRKKQRVKIAYEEIFVKNM |
| 1686 | GGL27 | A375 cells | TAMRA | 31672541 | 8 | Corrected total cell fluorescence | 5uM | 2h | 4ºC | Flow cytometry | Cellular uptake | GGLIKTKRKRKKQRVKIAYEEIFVKNM |
| 1687 | GGL27 | HeLa cells | TAMRA | 31672541 | 35 | Corrected total cell fluorescence | 5uM | 2h | 37ºC | Flow cytometry | Cellular uptake | GGLIKTKRKRKKQRVKIAYEEIFVKNM |
| 1688 | GGL27 | HeLa cells | TAMRA | 31672541 | 18 | Corrected total cell fluorescence | 5uM | 2h | 4ºC | Flow cytometry | Cellular uptake | GGLIKTKRKRKKQRVKIAYEEIFVKNM |
| 1689 | GA-TAT | EJ cells | NA | 29670331 | 1 | Cellular uptake | 0.25uM | 2h | NA | Flow cytometry | Cellular uptake | GA-YGRKKRRQRRR |
| 1690 | GA-TAT | EJ cells | NA | 29670331 | 2 | Cellular uptake | 1uM | 2h | NA | Flow cytometry | Cellular uptake | GA-YGRKKRRQRRR |
| 1691 | GA-TAT | EJ cells | NA | 29670331 | 5 | Cellular uptake | 2.5uM | 2h | NA | Flow cytometry | Cellular uptake | GA-YGRKKRRQRRR |
| 1692 | GA-TAT | EJ cells | NA | 29670331 | 6 | Cellular uptake | 5uM | 2h | NA | Flow cytometry | Cellular uptake | GA-YGRKKRRQRRR |
| 1693 | GA-TAT | SV-HUC-1 cells | NA | 29670331 | 1 | Cellular uptake | 0.25uM | 2h | NA | Flow cytometry | Cellular uptake | GA-YGRKKRRQRRR |
| 1694 | GA-TAT | SV-HUC-1 cells | NA | 29670331 | 2 | Cellular uptake | 1uM | 2h | NA | Flow cytometry | Cellular uptake | GA-YGRKKRRQRRR |
| 1695 | GA-TAT | SV-HUC-1 cells | NA | 29670331 | 5 | Cellular uptake | 2.5uM | 2h | NA | Flow cytometry | Cellular uptake | GA-YGRKKRRQRRR |
| 1696 | GA-TAT | SV-HUC-1 cells | NA | 29670331 | 7 | Cellular uptake | 5uM | 2h | NA | Flow cytometry | Cellular uptake | GA-YGRKKRRQRRR |
| 1697 | SNEDDS F-1 | Caco-2 cells | sodium fluorescein | 27458781 | 1.5 | Cellular uptake (%) | NA | 2h | 37ºC | Fluorescent Microscopy | Cellular uptake | RKKRRQRRR-pDNA |
| 1698 | SNEDDS F-1 | Caco-2 cells | sodium fluorescein | 27458781 | 2 | Cellular uptake (%) | NA | 4h | 37ºC | Fluorescent Microscopy | Cellular uptake | RKKRRQRRR-pDNA |
| 1699 | SNEDDS F-2 | Caco-2 cells | sodium fluorescein | 27458781 | 3 | Cellular uptake (%) | NA | 2h | 37ºC | Fluorescent Microscopy | Cellular uptake | RKKRRQRRR-OL-Pdna |
| 1700 | SNEDDS F-2 | Caco-2 cells | sodium fluorescein | 27458781 | 5 | Cellular uptake (%) | NA | 4h | 37ºC | Fluorescent Microscopy | Cellular uptake | RKKRRQRRR-OL-Pdna |
| 1701 | L1 | HeLa cells | Carboxyfluorescein | 27966361 | 14 | Normalized Mean Fluorescence intensity | 5uM | 30 min | NA | Flow cytometry | Cellular uptake | MIILIIGSTSRDHMVLHEYVNAAGIT |
| 1702 | L2 | HeLa cells | Carboxyfluorescein | 27966361 | 4 | Normalized Mean Fluorescence intensity | 5uM | 30 min | NA | Flow cytometry | Cellular uptake | FLLIRRVLGSTSRDHMVLHEYVNAAGIT |
| 1703 | L3 | HeLa cells | Carboxyfluorescein | 27966361 | 3 | Normalized Mean Fluorescence intensity | 5uM | 30 min | NA | Flow cytometry | Cellular uptake | PWPRVPWRWGSTSRDHMVLHEYVNAAGIT |
| 1704 | L4 | HeLa cells | Carboxyfluorescein | 27966361 | 3 | Normalized Mean Fluorescence intensity | 5uM | 30 min | NA | Flow cytometry | Cellular uptake | LKRAIWLIKGSTSRDHMVLHEYVNAAGIT |
| 1705 | C1 | HeLa cells | Carboxyfluorescein | 27966361 | 7 | Normalized Mean Fluorescence intensity | 5uM | 30 min | NA | Flow cytometry | Cellular uptake | FIDLKRKIWLIK |
| 1706 | C2 | HeLa cells | Carboxyfluorescein | 27966361 | 5 | Normalized Mean Fluorescence intensity | 5uM | 30 min | NA | Flow cytometry | Cellular uptake | YLKFIPLKDAIWKIK |
| 1707 | L1 | HeLa cells | Carboxyfluorescein | 27966361 | 1 | Normalized Mean Fluorescence intensity | 2uM | 30 min | NA | Flow cytometry | Cellular uptake | MIILIIGSTSRDHMVLHEYVNAAGIT |
| 1708 | L2 | HeLa cells | Carboxyfluorescein | 27966361 | 1 | Normalized Mean Fluorescence intensity | 2uM | 30 min | NA | Flow cytometry | Cellular uptake | FLLIRRVLGSTSRDHMVLHEYVNAAGIT |
| 1709 | L3 | HeLa cells | Carboxyfluorescein | 27966361 | 1 | Normalized Mean Fluorescence intensity | 2uM | 30 min | NA | Flow cytometry | Cellular uptake | PWPRVPWRWGSTSRDHMVLHEYVNAAGIT |
| 1710 | L4 | HeLa cells | Carboxyfluorescein | 27966361 | 1 | Normalized Mean Fluorescence intensity | 2uM | 30 min | NA | Flow cytometry | Cellular uptake | LKRAIWLIKGSTSRDHMVLHEYVNAAGIT |
| 1711 | C1 | HeLa cells | Carboxyfluorescein | 27966361 | 6 | Normalized Mean Fluorescence intensity | 2uM | 30 min | NA | Flow cytometry | Cellular uptake | FIDLKRKIWLIK |
| 1712 | C2 | HeLa cells | Carboxyfluorescein | 27966361 | 7 | Normalized Mean Fluorescence intensity | 2uM | 30 min | NA | Flow cytometry | Cellular uptake | YLKFIPLKDAIWKIK |
| 1713 | L1 | HeLa cells | Carboxyfluorescein | 27966361 | 13 | Normalized Mean Fluorescence intensity | 2uM | 2h | NA | Flow cytometry | Cellular uptake | MIILIIGSTSRDHMVLHEYVNAAGIT |
| 1714 | L2 | HeLa cells | Carboxyfluorescein | 27966361 | 4 | Normalized Mean Fluorescence intensity | 2uM | 2h | NA | Flow cytometry | Cellular uptake | FLLIRRVLGSTSRDHMVLHEYVNAAGIT |
| 1715 | L3 | HeLa cells | Carboxyfluorescein | 27966361 | 7 | Normalized Mean Fluorescence intensity | 2uM | 2h | NA | Flow cytometry | Cellular uptake | PWPRVPWRWGSTSRDHMVLHEYVNAAGIT |
| 1716 | L4 | HeLa cells | Carboxyfluorescein | 27966361 | 4 | Normalized Mean Fluorescence intensity | 2uM | 2h | NA | Flow cytometry | Cellular uptake | LKRAIWLIKGSTSRDHMVLHEYVNAAGIT |
| 1717 | C1 | HeLa cells | Carboxyfluorescein | 27966361 | 1 | Normalized Mean Fluorescence intensity | 2uM | 2h | NA | Flow cytometry | Cellular uptake | FIDLKRKIWLIK |
| 1718 | C2 | HeLa cells | Carboxyfluorescein | 27966361 | 1 | Normalized Mean Fluorescence intensity | 2uM | 2h | NA | Flow cytometry | Cellular uptake | YLKFIPLKDAIWKIK |
| 1719 | L1-1 | HeLa cells | Carboxyfluorescein | 27966361 | 3 | Median Fluorescence intensity | 2uM | 2h | NA | Flow cytometry | Cellular uptake | KIIIIDGSTSRDHVLHEYVNAAGIT |
| 1720 | L1-2 | HeLa cells | Carboxyfluorescein | 27966361 | 4 | Median Fluorescence intensity | 2uM | 2h | NA | Flow cytometry | Cellular uptake | KIILIIDGSTSRDHVLHEYVNAAGIT |
| 1721 | L1-3 | HeLa cells | Carboxyfluorescein | 27966361 | 16 | Median Fluorescence intensity | 2uM | 2h | NA | Flow cytometry | Cellular uptake | IILIIGSTSRDHVLHEYVNAAGIT |
| 1722 | L1-4 | HeLa cells | Carboxyfluorescein | 27966361 | 5 | Median Fluorescence intensity | 2uM | 2h | NA | Flow cytometry | Cellular uptake | MLILIIGSTSRDHVLHEYVNAAGIT |
| 1723 | L1-5 | HeLa cells | Carboxyfluorescein | 27966361 | 9 | Median Fluorescence intensity | 2uM | 2h | NA | Flow cytometry | Cellular uptake | MIILIIMGVADLIKKFESISKEE |
| 1724 | L1-6 | HeLa cells | Carboxyfluorescein | 27966361 | 15 | Median Fluorescence intensity | 2uM | 2h | NA | Flow cytometry | Cellular uptake | PLILLRLLRGSTSRDHVLHEYVNAAGIT |
| 1725 | L1-7 | HeLa cells | Carboxyfluorescein | 27966361 | 35 | Median Fluorescence intensity | 2uM | 2h | NA | Flow cytometry | Cellular uptake | FIDIIIKILLIGSTSRDHVLHEYVNAAGIT |
| 1726 | R8HNPs | R1 ESC cells | NA | 33464088 | 59 | Relative fluorescence | 25 ug/mL | 30 min | NA | CLSM | Cellular uptake | RRRRRRRR-H-NPs-siScr |
| 1727 | R8HNPs | R1 ESC cells | NA | 33464088 | 43 | Relative fluorescence | 25 ug/mL | 1h | NA | CLSM | Cellular uptake | RRRRRRRR-H-NPs-siScr |
| 1728 | R8HNPs | R1 ESC cells | NA | 33464088 | 38 | Relative fluorescence | 25 ug/mL | 3h | NA | CLSM | Cellular uptake | RRRRRRRR-H-NPs-siScr |
| 1729 | R8HNPs | R1 ESC cells | NA | 33464088 | 27 | Relative fluorescence | 25 ug/mL | 6h | NA | CLSM | Cellular uptake | RRRRRRRR-H-NPs-siScr |
| 1730 | R8HNPs | R1 ESC cells | NA | 33464088 | 20 | Relative fluorescence | 25 ug/mL | 12h | NA | CLSM | Cellular uptake | RRRRRRRR-H-NPs-siScr |
| 1731 | R8HNPs | R1 ESC cells | NA | 33464088 | 19 | Relative fluorescence | 25 ug/mL | 24h | NA | CLSM | Cellular uptake | RRRRRRRR-H-NPs-siScr |
| 1732 | R8HNPs | R1 ESC cells | NA | 33464088 | -20 | Relative fluorescence | 25 ug/mL | 48h | NA | CLSM | Cellular uptake | RRRRRRRR-H-NPs-siScr |
| 1733 | SR11 | HeLa cells | FITC | 26752214 | 20 | Mean Fluorescence intensity | 20 ug/ml | 30min | NA | Flow cytometry | Cellular uptake | SGASDDEEIAR |
| 1734 | SR11 | HeLa cells | FITC | 26752214 | 110 | Mean Fluorescence intensity | 20 ug/ml | 1h | NA | Flow cytometry | Cellular uptake | SGASDDEEIAR |
| 1735 | SR11 | HeLa cells | FITC | 26752214 | 130 | Mean Fluorescence intensity | 20 ug/ml | 1.5h | NA | Flow cytometry | Cellular uptake | SGASDDEEIAR |
| 1736 | SR11 | HeLa cells | FITC | 26752214 | 140 | Mean Fluorescence intensity | 20 ug/ml | 2h | NA | Flow cytometry | Cellular uptake | SGASDDEEIAR |
| 1737 | IR15 | HeLa cells | FITC | 26752214 | 90 | Mean Fluorescence intensity | 20 ug/ml | 30min | NA | Flow cytometry | Cellular uptake | ICSSHYEPTVRIGGR |
| 1738 | IR15 | HeLa cells | FITC | 26752214 | 135 | Mean Fluorescence intensity | 20 ug/ml | 1h | NA | Flow cytometry | Cellular uptake | ICSSHYEPTVRIGGR |
| 1739 | IR15 | HeLa cells | FITC | 26752214 | 150 | Mean Fluorescence intensity | 20 ug/ml | 1.5h | NA | Flow cytometry | Cellular uptake | ICSSHYEPTVRIGGR |
| 1740 | IR15 | HeLa cells | FITC | 26752214 | 170 | Mean Fluorescence intensity | 20 ug/ml | 2h | NA | Flow cytometry | Cellular uptake | ICSSHYEPTVRIGGR |
| 1741 | PAK | A375 cells | FITC | 30904618 | 0 | NA | 20uM | 48h | 37ºC | Fluorescent Microscopy | Cellular uptake | GGEEEEEEEEPLGLAGRRRRRRRRGG |
| 1742 | ?1H | HeLa cells | FITC | 28096156 | 18 | Fluorescence intensity | 1uM | 2h | 37ºC | Flow cytometry | Cellular uptake | KSKTEYYNAWAVWERNAP |
| 1743 | ?1H | HeLa cells | FITC | 28096156 | 18 | Fluorescence intensity | 1uM | 4h | 37ºC | Flow cytometry | Cellular uptake | KSKTEYYNAWAVWERNAP |
| 1744 | ?1H | HeLa cells | FITC | 28096156 | 19 | Fluorescence intensity | 1uM | 6h | 37ºC | Flow cytometry | Cellular uptake | KSKTEYYNAWAVWERNAP |
| 1745 | ?1H | HeLa cells | FITC | 28096156 | 12 | Fluorescence intensity | 1uM | 24h | 37ºC | Flow cytometry | Cellular uptake | KSKTEYYNAWAVWERNAP |
| 1746 | ?2H | HeLa cells | FITC | 28096156 | 13 | Fluorescence intensity | 1uM | 2h | 37ºC | Flow cytometry | Cellular uptake | GNGEQREMAVSRLRDCLDRQA |
| 1747 | ?2H | HeLa cells | FITC | 28096156 | 14 | Fluorescence intensity | 1uM | 4h | 37ºC | Flow cytometry | Cellular uptake | GNGEQREMAVSRLRDCLDRQA |
| 1748 | ?2H | HeLa cells | FITC | 28096156 | 12 | Fluorescence intensity | 1uM | 6h | 37ºC | Flow cytometry | Cellular uptake | GNGEQREMAVSRLRDCLDRQA |
| 1749 | ?2H | HeLa cells | FITC | 28096156 | 8 | Fluorescence intensity | 1uM | 24h | 37ºC | Flow cytometry | Cellular uptake | GNGEQREMAVSRLRDCLDRQA |
| 1750 | ?1H | HBMEC cells | FITC | 28096156 | 25 | Fluorescence intensity | 1uM | 2h | 37ºC | Flow cytometry | Cellular uptake | KSKTEYYNAWAVWERNAP |
| 1751 | ?1H | HBMEC cells | FITC | 28096156 | 30 | Fluorescence intensity | 1uM | 4h | 37ºC | Flow cytometry | Cellular uptake | KSKTEYYNAWAVWERNAP |
| 1752 | ?1H | HBMEC cells | FITC | 28096156 | 23 | Fluorescence intensity | 1uM | 6h | 37ºC | Flow cytometry | Cellular uptake | KSKTEYYNAWAVWERNAP |
| 1753 | ?1H | HBMEC cells | FITC | 28096156 | 30 | Fluorescence intensity | 1uM | 24h | 37ºC | Flow cytometry | Cellular uptake | KSKTEYYNAWAVWERNAP |
| 1754 | ?2H | HBMEC cells | FITC | 28096156 | 40 | Fluorescence intensity | 1uM | 2h | 37ºC | Flow cytometry | Cellular uptake | GNGEQREMAVSRLRDCLDRQA |
| 1755 | ?2H | HBMEC cells | FITC | 28096156 | 45 | Fluorescence intensity | 1uM | 4h | 37ºC | Flow cytometry | Cellular uptake | GNGEQREMAVSRLRDCLDRQA |
| 1756 | ?2H | HBMEC cells | FITC | 28096156 | 35 | Fluorescence intensity | 1uM | 6h | 37ºC | Flow cytometry | Cellular uptake | GNGEQREMAVSRLRDCLDRQA |
| 1757 | ?2H | HBMEC cells | FITC | 28096156 | 40 | Fluorescence intensity | 1uM | 24h | 37ºC | Flow cytometry | Cellular uptake | GNGEQREMAVSRLRDCLDRQA |
| 1758 | R8-CM?CD | MCF7 cells | FITC | 32589088 | 12 | Mean fluorescence intensity (%) | NA | 2h | NA | CLSM | Cellular uptake | RRRRRRRR-CM?CD |
| 1759 | R8-CM?CD | MCF7 cells | FITC | 32589088 | 15 | Mean fluorescence intensity (%) | NA | 6h | NA | CLSM | Cellular uptake | RRRRRRRR-CM?CD |
| 1760 | R8-CM?CD | MCF7 cells | FITC | 32589088 | 35 | Mean fluorescence intensity (%) | NA | 12h | NA | CLSM | Cellular uptake | RRRRRRRR-CM?CD |
| 1761 | Cf-OT20 | MonoMac6 cells | FITC | 30099595 | 5000 | FITC Mean Intensity | 10uM | 2h | 37ºC | Flow cytometry | Cellular uptake | CF-TKPKGTKPKGTKPKGTKPKG |
| 1762 | Cf-Penetratin | MonoMac6 cells | FITC | 30099595 | 140000 | FITC Mean Intensity | 10uM | 2h | 37ºC | Flow cytometry | Cellular uptake | CF-RQIKIWFQNRRMKWKK |
| 1763 | Cf-Dhvar4 | MonoMac6 cells | FITC | 30099595 | 200000 | FITC Mean Intensity | 10uM | 2h | 37ºC | Flow cytometry | Cellular uptake | CF-KRLFKKLLFSLRKY |
| 1764 | Cf-Transportan | MonoMac6 cells | FITC | 30099595 | 40000 | FITC Mean Intensity | 10uM | 2h | 37ºC | Flow cytometry | Cellular uptake | CF-AGYLLGKINLKALAALAKKIL |
| 1765 | Cf-Magainin | MonoMac6 cells | FITC | 30099595 | 10000 | FITC Mean Intensity | 10uM | 2h | 37ºC | Flow cytometry | Cellular uptake | CF-GIGKFLHSAKKFGKAFVGEIMNS |
| 1766 | Cf-Melittin | MonoMac6 cells | FITC | 30099595 | 175000 | FITC Mean Intensity | 10uM | 2h | 37ºC | Flow cytometry | Cellular uptake | CF-GIGAVLKVLTTGLPALISWIKRKRQQ |
| 1767 | A1 | HeLa cells | FITC | 33355559 | 100 | Relative Mean Fluorescence intensity (%) | 2uM | 2h | NA | Flow cytometry | Cellular uptake | YGRKKRRQRRR |
| 1768 | A2 | HeLa cells | FITC | 33355559 | 210 | Relative Mean Fluorescence intensity (%) | 2uM | 2h | NA | Flow cytometry | Cellular uptake | S5GRKS5RRQRRR |
| 1769 | A3 | HeLa cells | FITC | 33355559 | 220 | Relative Mean Fluorescence intensity (%) | 2uM | 2h | NA | Flow cytometry | Cellular uptake | R8GRKKRRS5RRR |
| 1770 | A4 | HeLa cells | FITC | 33355559 | 410 | Relative Mean Fluorescence intensity (%) | 2uM | 2h | NA | Flow cytometry | Cellular uptake | YGRKS5RRQS5RR |
| 1771 | A5 | HeLa cells | FITC | 33355559 | 80 | Relative Mean Fluorescence intensity (%) | 2uM | 2h | NA | Flow cytometry | Cellular uptake | YGRKERRQKRR |
| 1772 | A6 | HeLa cells | FITC | 33355559 | 370 | Relative Mean Fluorescence intensity (%) | 2uM | 2h | NA | Flow cytometry | Cellular uptake | YGRAS5RRQS5RA |
| 1773 | A7 | HeLa cells | FITC | 33355559 | 120 | Relative Mean Fluorescence intensity (%) | 2uM | 2h | NA | Flow cytometry | Cellular uptake | YGRAS5RRQS5RA |
| 1774 | A8 | HeLa cells | FITC | 33355559 | 25 | Relative Mean Fluorescence intensity (%) | 2uM | 2h | NA | Flow cytometry | Cellular uptake | YGRAS5ARQS5RA |
| 1775 | A9 | HeLa cells | FITC | 33355559 | 200 | Relative Mean Fluorescence intensity (%) | 2uM | 2h | NA | Flow cytometry | Cellular uptake | YGRKR8RRQS5RR |
| 1776 | A10 | HeLa cells | FITC | 33355559 | 100 | Relative Mean Fluorescence intensity (%) | 2uM | 2h | NA | Flow cytometry | Cellular uptake | YGRKR8RRQXRR |
| 1777 | A11 | HeLa cells | FITC | 33355559 | 90 | Relative Mean Fluorescence intensity (%) | 2uM | 2h | NA | Flow cytometry | Cellular uptake | YGRKS5RRQXRR |
| 1778 | A3u | HeLa cells | FITC | 33355559 | 80 | Relative Mean Fluorescence intensity (%) | 2uM | 2h | NA | Flow cytometry | Cellular uptake | R8GRRKKRRS5RRR |
| 1779 | A4u | HeLa cells | FITC | 33355559 | 100 | Relative Mean Fluorescence intensity (%) | 2uM | 2h | NA | Flow cytometry | Cellular uptake | YGRKS5RRQS5RR |
| 1780 | A6u | HeLa cells | FITC | 33355559 | 90 | Relative Mean Fluorescence intensity (%) | 2uM | 2h | NA | Flow cytometry | Cellular uptake | YGRAS5RRQS5RR |
| 1781 | C6M3 | CHO-K1 cells | siRNA-Cy3 labeled | 28349343 | 90 | Fluorescent cells (%) | NA | NA | NA | Flow cytometry | Cellular uptake | RLWHLLWRLWRRLHRLLR |
| 1782 | AntpOVA | Dendritic cells | FITC | 27138940 | 50 | Cellular uptake (%) | 100ug/ml | 30min | 37ºC | Flow cytometry | Cellular uptake | RQIKIWFQNRRMKWKK-SIINFEKL |
| 1783 | AntpOVA | Dendritic cells | FITC | 27138940 | 45 | Cellular uptake (%) | 100ug/ml | 1h | 37ºC | Flow cytometry | Cellular uptake | RQIKIWFQNRRMKWKK-SIINFEKL |
| 1784 | AntpOVA | Dendritic cells | FITC | 27138940 | 45 | Cellular uptake (%) | 100ug/ml | 2h | 37ºC | Flow cytometry | Cellular uptake | RQIKIWFQNRRMKWKK-SIINFEKL |
| 1785 | Tylotoin-sC18* | HaCaT cells | Carboxyfluorescein | 30389988 | 1400 | Relative fluorescence | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | KCVRQNNKRVCKGLRKRLRKFRNK-NH2 |
| 1786 | TDCS-Tat NPs | Caco-2 cells | Cou-6 | 30672923 | 13 | Cellular uptake | NA | 1h | 37ºC | Fluorescent Microscopy | Cellular uptake | GRKKRRQRRRPQ |
| 1787 | TDCS-Pen NPs | Caco-2 cells | Cou-6 | 30672923 | 10 | Cellular uptake | NA | 1h | 37ºC | Fluorescent Microscopy | Cellular uptake | RQIKIWFQNRRMKWKKGG |
| 1788 | TDCS-R8 NPs | Caco-2 cells | Cou-6 | 30672923 | 9 | Cellular uptake | NA | 1h | 37ºC | Fluorescent Microscopy | Cellular uptake | RRRRRRRR |
| 1789 | TDCS-Tat NPs | Caco-2 cells | Cou-6 | 30672923 | 15 | Cellular uptake | NA | 2h | 37ºC | Fluorescent Microscopy | Cellular uptake | GRKKRRQRRRPQ |
| 1790 | TDCS-Pen NPs | Caco-2 cells | Cou-6 | 30672923 | 13 | Cellular uptake | NA | 2h | 37ºC | Fluorescent Microscopy | Cellular uptake | RQIKIWFQNRRMKWKKGG |
| 1791 | TDCS-R8 NPs | Caco-2 cells | Cou-6 | 30672923 | 12 | Cellular uptake | NA | 2h | 37ºC | Fluorescent Microscopy | Cellular uptake | RRRRRRRR |
| 1792 | TDCS-Tat NPs | Caco-2 cells | Cou-6 | 30672923 | 26 | Cellular uptake | NA | 4h | 37ºC | Fluorescent Microscopy | Cellular uptake | GRKKRRQRRRPQ |
| 1793 | TDCS-Pen NPs | Caco-2 cells | Cou-6 | 30672923 | 23 | Cellular uptake | NA | 4h | 37ºC | Fluorescent Microscopy | Cellular uptake | RQIKIWFQNRRMKWKKGG |
| 1794 | TDCS-R8 NPs | Caco-2 cells | Cou-6 | 30672923 | 21 | Cellular uptake | NA | 4h | 37ºC | Fluorescent Microscopy | Cellular uptake | RRRRRRRR |
| 1795 | DsC18 | MCF7 cells | Carboxyfluorescein | 28332260 | 39 | Relative fluorescence | 25uM | 30min | 37ºC | Fluorescent Microscopy | Cellular uptake | CF-glrkrlrkfrnkikek |
| 1796 | DsC18(NIA)2 | MCF7 cells | Carboxyfluorescein | 28332260 | 40 | Relative fluorescence | 25uM | 30min | 37ºC | Fluorescent Microscopy | Cellular uptake | CF-?A-glrk-?A?A-NIA-rlrkfrnk-?A?A-NIA-ikek |
| 1797 | DsC18 | MCF7 cells | Carboxyfluorescein | 28332260 | 130 | Relative fluorescence | 50uM | 30min | 37ºC | Fluorescent Microscopy | Cellular uptake | CF-glrkrlrkfrnkikek |
| 1798 | DsC18(NIA)2 | MCF7 cells | Carboxyfluorescein | 28332260 | 150 | Relative fluorescence | 50uM | 30min | 37ºC | Fluorescent Microscopy | Cellular uptake | CF-?A-glrk-?A?A-NIA-rlrkfrnk-?A?A-NIA-ikek |
| 1799 | BR2-Lp | HepG2 cells | Cou-6 | 28644728 | 125 | Mean Fluorescence intensity | 0.1ug/ml | 3h | 37ºC | Flow cytometry | Cellular uptake | RAGLQFPVGRLLRRL |
| 1800 | BR2-Lp | Miha cells | Cou-6 | 28644728 | 100 | Mean Fluorescence intensity | 0.1ug/ml | 3h | 37ºC | Flow cytometry | Cellular uptake | RAGLQFPVGRLLRRL |
| 1801 | CCMV | HeLa cells | Cy5 | 31257379 | 4000 | Mean Fluorescence intensity | NA | 6h | 37ºC | Flow cytometry | Cellular uptake | IWLTALKFLGKHAAKHEAKQQLSKL |
| 1802 | SPIONs-PEG-gH625 | MDA-MB-231 cells | Cy5.5 | 28388503 | 384.8 | Fluorescence intensity | 100 mg/L | 15min | NA | Fluorescent Microscopy | Cellular uptake | AcHGLASTLTRWAHYNALIRAFC-CONH2 |
| 1803 | SPIONs-PEG-gH625 | MDA-MB-231 cells | Cy5.5 | 28388503 | 656.2 | Fluorescence intensity | 100 mg/L | 30min | NA | Fluorescent Microscopy | Cellular uptake | AcHGLASTLTRWAHYNALIRAFC-CONH2 |
| 1804 | 9R | HEK293 cells | dsRED | 30293549 | 0 | NA | NA | NA | NA | Fluorescent Microscopy | Penetration | RRRRRRRRR |
| 1805 | 9K | HEK293 cells | dsRED | 30293549 | 0.7 | Mean Intensity | 20ug | 30min | NA | Fluorescent Microscopy | Penetration | KKKKKKKKK |
| 1806 | 9K | HEK293 cells | dsRED | 30293549 | 1.3 | Mean Intensity | 20ug | 1h | NA | Fluorescent Microscopy | Penetration | KKKKKKKKK |
| 1807 | 9K | HEK293 cells | dsRED | 30293549 | 1.4 | Mean Intensity | 20ug | 4h | NA | Fluorescent Microscopy | Penetration | KKKKKKKKK |
| 1808 | 9K | HEK293 cells | dsRED | 30293549 | 1.8 | Mean Intensity | 20ug | 12h | NA | Fluorescent Microscopy | Penetration | KKKKKKKKK |
| 1809 | 9K | HEK293 cells | dsRED | 30293549 | 1.6 | Mean Intensity | 20ug | 24h | NA | Fluorescent Microscopy | Penetration | KKKKKKKKK |
| 1810 | F6G6(rR)3R2 | HeLa cells | 4CzIPN | 30525541 | 97.2 | Fluorescence intensity (%) | 2ug/mL | 5min | 37ºC | Flow cytometry | Cellular internalization of NPs | FFFFFFGGGGGGrrrRR |
| 1811 | F6G6(rR)3R2 | HeLa cells | NAI-DPAC | 30525541 | 44.1 | Fluorescence intensity (%) | 2ug/mL | 5min | 37ºC | Flow cytometry | Cellular internalization of NPs | FFFFFFGGGGGGrrrRR |
| 1812 | F6G6(rR)3R2 | HeLa cells | BTZ-DMAC | 30525541 | 59.7 | Fluorescence intensity (%) | 2ug/mL | 5min | 37ºC | Flow cytometry | Cellular internalization of NPs | FFFFFFGGGGGGrrrRR |
| 1813 | F6G6(rR)3R2 | NIH-3T3 cells | 4CzIPN | 30525541 | 57 | Fluorescence intensity (%) | 2ug/mL | 5min | 37ºC | Flow cytometry | Cellular internalization of NPs | FFFFFFGGGGGGrrrRR |
| 1814 | F6G6(rR)3R2 | NIH-3T3 cells | NAI-DPAC | 30525541 | 10.3 | Fluorescence intensity (%) | 2ug/mL | 5min | 37ºC | Flow cytometry | Cellular internalization of NPs | FFFFFFGGGGGGrrrRR |
| 1815 | F6G6(rR)3R2 | NIH-3T3 cells | BTZ-DMAC | 30525541 | 18 | Fluorescence intensity (%) | 2ug/mL | 5min | 37ºC | Flow cytometry | Cellular internalization of NPs | FFFFFFGGGGGGrrrRR |
| 1816 | RLA | C6 cells | DB | 31617510 | 42.6 | Cellular uptake | 25uM | 30min | 37ºC | ELISA | Cellular uptake | B12H11S(CH2)2COOH-rlarlarrlarlar |
| 1817 | r8 | C6 cells | DB | 31617510 | 4.6 | Cellular uptake | 25uM | 30min | 37ºC | ELISA | Cellular uptake | B12H11S(CH2)2COOH-rrrrrrrr |
| 1818 | PEP-1 | HEK293T cells | GFP | 27516189 | 57.58 | GFP-positive population (%) | 20uM | 4h | NA | Flow cytometry | Transfection | Ac-KETWWETWWTEWSQPKKKRKV-Cya |
| 1819 | CADY-2 | HEK293T cells | GFP | 27516189 | 58.7 | GFP-positive population (%) | 20uM | 4h | NA | Flow cytometry | Transfection | Ac-GLWWRLWWRLRSWFRLWFRA-Cya |
| 1820 | R9 | Endothelial cells | CmLN | 26748549 | 18 | Mean Fluorescence intensity | 10uM | 4h | 37ºC | Flow cytometry | Cellular uptake | RRRRRRRRR |
| 1821 | R9 | Endothelial cells | CmLN | 26748549 | 35 | Mean Fluorescence intensity | 25uM | 4h | 37ºC | Flow cytometry | Cellular uptake | RRRRRRRRR |
| 1822 | R9 | Endothelial cells | CmLN | 26748549 | 50 | Mean Fluorescence intensity | 50uM | 4h | 37ºC | Flow cytometry | Cellular uptake | RRRRRRRRR |
| 1823 | pHLIP | MCF7 cells | SS-DOX | 25853477 | 20 | Mean Fluorescence intensity | 7uM | 3h | 37ºC | Flow cytometry | Cellular uptake | AEQNPIYWARYADWLFTTPLLLLDLALLVDADEGTCG |
| 1824 | pHLIP | MCF7 cells | SS-DOX | 25853477 | 40 | Mean Fluorescence intensity | 7uM | 3h | 37ºC | Flow cytometry | Cellular uptake | AEQNPIYWARYADWLFTTPLLLLDLALLVDADEGTCG |
| 1825 | pHLIP | MCF7 cells | SS-DOX | 25853477 | 24 | Mean Fluorescence intensity | 7uM | 3h | 37ºC | Flow cytometry | Cellular uptake | AEQNPIYWARYADWLFTTPLLLLDLALLVDADEGTCG |
| 1826 | pHLIP | MCF7 cells | SS-DOX | 25853477 | 35 | Mean Fluorescence intensity | 7uM | 3h | 37ºC | Flow cytometry | Cellular uptake | AEQNPIYWARYADWLFTTPLLLLDLALLVDADEGTCG |
| 1827 | HSF | HTB-55 cells | FP | 30465781 | 0.15 | Drug transport | 1uM | 3h | NA | Fluorescent Microscopy | Drug transport | KCFQWQRNMRKVRGPPVSCIKR |
| 1828 | HSF | HTB-55 cells | SX/FP | 30465781 | 0.14 | Drug transport | 1uM | 3h | NA | Fluorescent Microscopy | Drug transport | KCFQWQRNMRKVRGPPVSCIKR |
| 1829 | Tpl | T98G cell | FITC | 31726199 | 40 | Percentage of FITC | 3uM | 1h | 37ºC | Flow cytometry | CPP activity | KWCFRVCYRGICYRRCR |
| 1830 | Tpl | T98G cell | FITC | 31726199 | 55 | Percentage of FITC | 5uM | 1h | 37ºC | Flow cytometry | CPP activity | KWCFRVCYRGICYRRCR |
| 1831 | Tpl | T98G cell | FITC | 31726199 | 70 | Percentage of FITC | 7uM | 1h | 37ºC | Flow cytometry | CPP activity | KWCFRVCYRGICYRRCR |
| 1832 | Tpl | L929 cells | FITC | 31726199 | 3 | Percentage of FITC | 3uM | 1h | 37ºC | Flow cytometry | CPP activity | KWCFRVCYRGICYRRCR |
| 1833 | Tpl | L929 cells | FITC | 31726199 | 5 | Percentage of FITC | 5uM | 1h | 37ºC | Flow cytometry | CPP activity | KWCFRVCYRGICYRRCR |
| 1834 | Tpl | L929 cells | FITC | 31726199 | 2 | Percentage of FITC | 7uM | 1h | 37ºC | Flow cytometry | CPP activity | KWCFRVCYRGICYRRCR |
| 1835 | Hpp3 | ECV304 cells | FITC | 27070736 | 3000 | Fluorescence intensity | 2.5uM | 1h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KPKRKRRKKKGHGWSR |
| 1836 | Hpp3 | ECV304 cells | FITC | 27070736 | 5000 | Fluorescence intensity | 5uM | 1h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KPKRKRRKKKGHGWSR |
| 1837 | Hpp3 | ECV304 cells | FITC | 27070736 | 5200 | Fluorescence intensity | 7.5uM | 1h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KPKRKRRKKKGHGWSR |
| 1838 | Hpp3 | ECV304 cells | FITC | 27070736 | 5800 | Fluorescence intensity | 10uM | 1h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KPKRKRRKKKGHGWSR |
| 1839 | Kkd-5 | HeLa cells | FITC | 28349160 | 30 | Relative Mean Fluorescence intensity (%) | 5uM | 4h | 37ºC | Flow cytometry | Cellular uptake | |
| 1840 | Kkd-5 | HeLa cells | FITC | 28349160 | 70 | Relative Mean Fluorescence intensity (%) | 10uM | 4h | 37ºC | Flow cytometry | Cellular uptake | |
| 1841 | Kkd-5 | HeLa cells | FITC | 28349160 | 97 | Relative Mean Fluorescence intensity (%) | 25uM | 4h | 37ºC | Flow cytometry | Cellular uptake | |
| 1842 | Fol-Pep1 | HeLa cells | FITC | 26544061 | 17 | Mean Fluorescence intensity | NA | 2h | 37ºC | Flow cytometry | Cellular uptake | KETWWETWWTEWSQPKKKRKVC |
| 1843 | Fol-Pep2 | HaCaT cells | FITC | 26544061 | 8 | Mean Fluorescence intensity | NA | 2h | 37ºC | Flow cytometry | Cellular uptake | KETWWETWWTEWSQPKKKRKVC |
| 1844 | R8-modified MITO-Porter | HeLa cells | NBD | 27056631 | 28 | Cellular uptake | 2.5 | NA | 37ºC | Flow cytometry | Cellular uptake | RRRRRRRR |
| 1845 | RP/R8-modified MITO-Porter | HeLa cells | NBD | 27056631 | 58 | Cellular uptake | 2.5 | NA | 37ºC | Flow cytometry | Cellular uptake | RRRRRRRR |
| 1846 | MRP/R8-modified MITO-Porter | HeLa cells | NBD | 27056631 | 35 | Cellular uptake | 2.5 | NA | 37ºC | Flow cytometry | Cellular uptake | RRRRRRRR |
| 1847 | D-arm/R8-modified MITO-Porter | HeLa cells | NBD | 27056631 | 40 | Cellular uptake | 2.5 | NA | 37ºC | Flow cytometry | Cellular uptake | RRRRRRRR |
| 1848 | CPP 2 | RAW264.7 cells | FITC | 30095906 | 71.9 | Intracellular FITC-labeled peptides (%) | 5uM | 2h | 37ºC | Flow cytometry | Cellular uptake | GFAWNVCVYRNGVRVCHRRAN |
| 1849 | CPP 6 | RAW264.7 cells | FITC | 30095906 | 95.8 | Intracellular FITC-labeled peptides (%) | 5uM | 2h | 37ºC | Flow cytometry | Cellular uptake | YGRKKRRQRRR-C-MC-VC-PABC-GFAWNVCVYRNGVRVCHRRAN |
| 1850 | CPP 7 | RAW264.7 cells | FITC | 30095906 | 75.2 | Intracellular FITC-labeled peptides (%) | 5uM | 2h | 37ºC | Flow cytometry | Cellular uptake | GFAWNVCVYRNGVRVCHRRAN-NH2 |
| 1851 | gH625 | HeLa cells | PtNPs | 28758654 | 0 | NA | NA | NA | NA | STEM | Cellular uptake | HGLASTLTRWAHYNALIRAFKGGGC |
| 1852 | SAP(E) | NA | NA | 27237727 | 0 | NA | NA | NA | NA | NA | NA | CGGWVELPPPVELPPPVELPPP |
| 1853 | CGA-N9 | C. tropicaliscells | Propidium iodide (PI) | 30610128 | 2.25 | Fluorescence intensity | 3.9mg/ml | 2h | 28ºC | Flow cytometry | Cellular uptake | RILSILRHQ |
| 1854 | MeG10 | HeLa cells | FITC | 27039278 | 2200 | Mean Fluorescence intensity | 5uM | NA | 37ºC | CLSM | Cellular uptake | RRRRRRRR |
| 1855 | dG5 | HeLa cells | FITC | 27039278 | 200 | Mean Fluorescence intensity | 5uM | NA | 37ºC | CLSM | Cellular uptake | RRRRRRRR |
| 1856 | dG10 | HeLa cells | FITC | 27039278 | 1500 | Mean Fluorescence intensity | 5uM | NA | 37ºC | CLSM | Cellular uptake | RRRRRRRR |
| 1857 | PGON20 | HeLa cells | FITC | 27039278 | 2200 | Mean Fluorescence intensity | 5uM | NA | 37ºC | CLSM | Cellular uptake | RRRRRRRR |
| 1858 | MePh10-b-dG5 | HeLa cells | FITC | 27039278 | 500 | Mean Fluorescence intensity | 5uM | NA | 37ºC | CLSM | Cellular uptake | RRRRRRRR |
| 1859 | RG301 | HeLa cells | Carboxyfluorescein | 34333729 | 100 | Cellular uptake (%) | 10uM | 4h | 37ºC | Flow cytometry | Cellular uptake | RaDPAYQaRFLGKrKfIcL |
| 1860 | RG302 | HeLa cells | Carboxyfluorescein | 34333729 | 100 | Cellular uptake (%) | 10uM | 4h | 37ºC | Flow cytometry | Cellular uptake | KrKfIcLGRaDPAYQaRFL |
| 1861 | CTX-M1 | HeLa cells | Alexa488 | 28459137 | 40 | Relative fluorescence (%) | 6uM | 1h | 37ºC | Flow cytometry | Internalization of fluorescently labeled peptides | MCMPCFTTDHQMARRCDDCCGGRGRGKCYGPQCLCR |
| 1862 | CTX-M2 | HeLa cells | Alexa488 | 28459137 | 38 | Relative fluorescence (%) | 6uM | 1h | 37ºC | Flow cytometry | Internalization of fluorescently labeled peptides | MCMPCFTTDHQMARRCDDCCGGRGRGKCWGPQCLCR |
| 1863 | CTX-M1 | HeLa cells | Cy5.5 | 28459137 | 49 | Relative fluorescence (%) | 6uM | 1h | 37ºC | Flow cytometry | Internalization of fluorescently labeled peptides | MCMPCFTTDHQMARRCDDCCGGRGRGKCYGPQCLCR |
| 1864 | CTX-M2 | HeLa cells | Cy5.5 | 28459137 | 75 | Relative fluorescence (%) | 6uM | 1h | 37ºC | Flow cytometry | Internalization of fluorescently labeled peptides | MCMPCFTTDHQMARRCDDCCGGRGRGKCWGPQCLCR |
| 1865 | HBHAc | HepG2 cells | eGFP | 31524004 | 55 | Mean Fluorescence intensity | 3uM | 1h | 37ºC | Flow cytometry | Cellular uptake | KKAAPAKKAAAKKAPAKKAAAKK |
| 1866 | HBHAc | HepG2 cells | eGFP | 31524004 | 30 | Mean Fluorescence intensity | 3uM | 1h | 37ºC | Flow cytometry | Cellular uptake | KKAAPAKKAAAKKAPAKKAAAKK |
| 1867 | HBHAc | HepG2 cells | eGFP | 31524004 | 20 | Mean Fluorescence intensity | 3uM | 1h | 37ºC | Flow cytometry | Cellular uptake | KKAAPAKKAAAKKAPAKKAAAKK |
| 1868 | [WR]5 | CCRF-CEM cells | F'-GpYEEI | 32498339 | 1000 | Mean Fluorescence intensity | 25uM | 3h | 37ºC | Flow cytometry | Cellular uptake | WRWRWRWRWR |
| 1869 | c[C(WR)4C] | CCRF-CEM cells | F'-GpYEEI | 32498339 | 200 | Mean Fluorescence intensity | 25uM | 3h | 37ºC | Flow cytometry | Cellular uptake | CWRWRWRWRC |
| 1870 | l(C(WR)4C) | CCRF-CEM cells | F'-GpYEEI | 32498339 | 700 | Mean Fluorescence intensity | 25uM | 3h | 37ºC | Flow cytometry | Cellular uptake | CWRWRWRWRC |
| 1871 | c[C(WR)5C] | CCRF-CEM cells | F'-GpYEEI | 32498339 | 1050 | Mean Fluorescence intensity | 25uM | 3h | 37ºC | Flow cytometry | Cellular uptake | CWRWRWRWRWRC |
| 1872 | l(C(WR)5C) | CCRF-CEM cells | F'-GpYEEI | 32498339 | 1100 | Mean Fluorescence intensity | 25uM | 3h | 37ºC | Flow cytometry | Cellular uptake | CWRWRWRWRWRC |
| 1873 | CPP 12 | HeLa cells | Carboxyfluorescein | 33838611 | 550 | Mean Fluorescence intensity | 2uM | 2h | NA | Flow cytometry | Intracellular levels of peptides | CF-GRR-Ac6cNH2-RR-Ac6cNH2-RR-Ac6cNH2-NH2 |
| 1874 | CPP 13 | HeLa cells | Carboxyfluorescein | 33838611 | 400 | Mean Fluorescence intensity | 2uM | 2h | NA | Flow cytometry | Intracellular levels of peptides | CF-GRR-Ac5cNH2-RR-Ac5cNH2-RR-Ac5cNH2-NH2 |
| 1875 | CPP 14 | HeLa cells | Carboxyfluorescein | 33838611 | 2600 | Mean Fluorescence intensity | 2uM | 2h | NA | Flow cytometry | Intracellular levels of peptides | CF-GRRRRRRRRR-NH2 |
| 1876 | CPP 12 | HEK293 cells | Carboxyfluorescein | 33838611 | 110 | Mean Fluorescence intensity | 2uM | 2h | NA | Flow cytometry | Intracellular levels of peptides | CF-GRR-Ac6cNH2-RR-Ac6cNH2-RR-Ac6cNH2-NH2 |
| 1877 | CPP 13 | HEK293 cells | Carboxyfluorescein | 33838611 | 1200 | Mean Fluorescence intensity | 2uM | 2h | NA | Flow cytometry | Intracellular levels of peptides | CF-GRR-Ac5cNH2-RR-Ac5cNH2-RR-Ac5cNH2-NH2 |
| 1878 | CPP 14 | HEK293 cells | Carboxyfluorescein | 33838611 | 2800 | Mean Fluorescence intensity | 2uM | 2h | NA | Flow cytometry | Intracellular levels of peptides | CF-GRRRRRRRRR-NH2 |
| 1879 | SAHM1 | HeLa cells | FITC | 28757184 | 16 | Mean Fluorescence intensity | 5uM | 90min | NA | Flow cytometry | Cellular uptake | ?A1a-ERLRRRI-S5-LCR-S5-HHST |
| 1880 | StAx | HeLa cells | FITC | 28757184 | 3 | Mean Fluorescence intensity | 5uM | 90min | NA | Flow cytometry | Cellular uptake | RRWPRXILDXHVRRVWR |
| 1881 | PI | A549 cells | siRNA | 27480031 | 90 | Mean Fluorescence intensity/mg protein | 2.5uM | 8h | 37ºC | Fluorometer | Cellular uptake | KLXLKLXLKXLKAXLKLXGC |
| 1882 | PI-acetamide | A549 cells | siRNA | 27480031 | 50 | Mean Fluorescence intensity/mg protein | 2.5uM | 8h | 37ºC | Fluorometer | Cellular uptake | KLXLKLXLKXLKAXLKLXGC |
| 1883 | PII | A549 cells | siRNA | 27480031 | 20 | Mean Fluorescence intensity/mg protein | 2.5uM | 8h | 37ºC | Fluorometer | Cellular uptake | KLXLKLXLKXLKACLKLXG |
| 1884 | PIII | A549 cells | siRNA | 27480031 | 92 | Mean Fluorescence intensity/mg protein | 2.5uM | 8h | 37ºC | Fluorometer | Cellular uptake | KCXLKLXLKXLKACLKLXG |
| 1885 | PIV | A549 cells | siRNA | 27480031 | 5 | Mean Fluorescence intensity/mg protein | 2.5uM | 8h | 37ºC | Fluorometer | Cellular uptake | KLXLKLXCKXLKACLKLXG |
| 1886 | PV | A549 cells | siRNA | 27480031 | 15 | Mean Fluorescence intensity/mg protein | 2.5uM | 8h | 37ºC | Fluorometer | Cellular uptake | KCXLKLXCKXLKACLKLXG |
| 1887 | Lys-peptide 1 | HeLa cells | NA | 26814673 | 90 | RFU/mg | 1uM | 2h | 4ºC | Fluorescence spectroscopy | Cellular uptake | TMR-GKKKKKKKKK-NH2 |
| 1888 | Arg-peptide 2 | HeLa cells | NA | 26814673 | 500 | RFU/mg | 1uM | 2h | 4ºC | Fluorescence spectroscopy | Cellular uptake | TMR-GRRRRRRRRR-NH2 |
| 1889 | Lys(AEt)-peptide 3 | HeLa cells | NA | 26814673 | 10 | RFU/mg | 1uM | 2h | 4ºC | Fluorescence spectroscopy | Cellular uptake | TMR-G(AEt)(AEt)(AEt)(AEt)(AEt)(AEt)(AEt)(AEt)(AEt)-NH2 |
| 1890 | Lys(GEt)-peptide 4 | HeLa cells | NA | 26814673 | 200 | RFU/mg | 1uM | 2h | 4ºC | Fluorescence spectroscopy | Cellular uptake | TMR-G(GEt)(GEt)(GEt)(GEt)(GEt)(GEt)(GEt)(GEt)(GEt)-NH2 |
| 1891 | KIW7 | HeLa cells | pDNA | 32329496 | 0 | NA | NA | NA | NA | CLSM | NA | KIWFQNR |
| 1892 | mPrPA488 | N2a cells | Alexa488 | 27818203 | 1 | Cellular uptake | 1uM | 24h | 4ºC | CLSM | Cellular uptake | ALFVKLMGTPLDNAKWTLCPVLRGMWKY |
| 1893 | bPrPA488 | N2a cells | Alexa488 | 27818203 | 1 | Cellular uptake | 1uM | 24h | 4ºC | CLSM | Cellular uptake | KPACVIKMVS-WKIGPVSDLKLVKSFGLMRW |
| 1894 | mPrPA488 | HeLa cells | Alexa488 | 27818203 | 1 | Cellular uptake | 1uM | 24h | 4ºC | CLSM | Cellular uptake | ALFVKLMGTPLDNAKWTLCPVLRGMWKY |
| 1895 | bPrPA488 | HeLa cells | Alexa488 | 27818203 | 1 | Cellular uptake | 1uM | 24h | 4ºC | CLSM | Cellular uptake | KPACVIKMVS-WKIGPVSDLKLVKSFGLMRW |
| 1896 | stearyl-r8 | HeLa cells | CD63-GFP Evs | 27748399 | 3340 | Relative Cellular uptake | 16uM | 24h | 37ºC | CLSM | Cellular uptake | CH3(CH2)16-CO-NH-rrrrrrrr-NH2 |
| 1897 | stearyl-sC18 | MCF7 cells | CD63-GFP Evs | 34365796 | 692 | Relative Cellular uptake | 10uM | 24h | 37ºC | Flow cytometry | Cellular uptake | CH3(CH2)16-CONH-GGGGLRKRLRKFRNKIKEK-NH2 |
| 1898 | stearyl-(sC18)2 | MCF7 cells | CD63-GFP Evs | 34365796 | 777 | Relative Cellular uptake | 2uM | 24h | 37ºC | Flow cytometry | Cellular uptake | NH2-GLRK(KEKIKNRFKRLRKRLGGGG-NH2CO-CH3(CH2)16)RLRKFRNKIKEK-NH2 |
| 1899 | sC18 | MCF7 cells | CD63-GFP Evs | 34365796 | 128 | Relative Cellular uptake | 10uM | 24h | 37ºC | Flow cytometry | Cellular uptake | NH2-GLRKRLRKFRNKIKEK-amide |
| 1900 | (sC18)2 | MCF7 cells | CD63-GFP Evs | 34365796 | 78 | Relative Cellular uptake | 2uM | 24h | 37ºC | Flow cytometry | Cellular uptake | NH2-GLRK(RLRKFRKEKIKNRFKRLRKRLG-NH2)NKIKEK-amide |
| 1901 | T-hNP | B16 cells | Rh-PE | 28954191 | 9 | Mean Fluorescence intensity | NA | 15 min | 37ºC | Flow cytometry | Cellular uptake | GRKKRRQRRRPQ |
| 1902 | peptide 1 | HeLa cells | DUB | 32831622 | 0 | NA | NA | NA | NA | NA | NA | Ac-RWVRVPGRWIRQLRGG-AFC |
| 1903 | peptide 2 | HeLa cells | DUB | 32831622 | 0 | NA | NA | NA | NA | NA | NA | Ac-RWVRVPGRWIRQLVLRLRGG-AFC |
| 1904 | peptide 3 | HeLa cells | DUB | 32831622 | 0 | NA | NA | NA | NA | NA | NA | Z-LRGG-AMC |
| 1905 | peptide 4 | HeLa cells | DUB | 32831622 | 0 | NA | 30uM | 1h | 37ºC | Flow cytometry | Cellular uptake | Ac-RWVRVPGX(-CF)WIRQLRGG-NH2 |
| 1906 | COSS 4 | HeLa cells | TAMRA | 27774725 | 150 | Mean Fluorescence intensity | NA | 1h | 37ºC | Flow cytometry | Cellular uptake | NA |
| 1907 | POSS-(PEG-NLS-G-TAT)8 | Endothelial cells | Cy5-oligonucleotide | 32254599 | 2000 | Mean Fluorescence intensity | NA | 4h | 37ºC | Flow cytometry | Cellular uptake | CPKKKRKVEDPGGRKKRRQRRRPQ |
| 1908 | POSS-(PEG-NLS-G-TAT-G-REDV)8 | Endothelial cells | Cy5-oligonucleotide | 32254599 | 2100 | Mean Fluorescence intensity | NA | 4h | 37ºC | Flow cytometry | Cellular uptake | CPKKKRKVEDPGGRKKRRQRRRPQGREDV |
| 1909 | TP-H12 | Endothelial cells | Cy5-oligonucleotide | 32254599 | 7000 | Mean Fluorescence intensity | NA | 4h | 37ºC | Flow cytometry | Cellular uptake | REDVGRKKRRQRRRPQCPKKKRKVEDPHHHHHHHHHHHH |
| 1910 | L6 | A549 cells | FITC | 30360131 | 0 | NA | NA | NA | NA | Fluorescent Microscopy | Cellular internalization of CPP-FITC | RRWQWR |
| 1911 | H6 | BY-2 plant cells | TAMRA | 27885926 | 9000 | Cellular uptake | 1uM | 12h | 27ºC | CLSM | Cellular uptake | HHHHHH-NH2 |
| 1912 | H8 | BY-2 plant cells | TAMRA | 27885926 | 15000 | Cellular uptake | 1uM | 12h | 27ºC | CLSM | Cellular uptake | HHHHHHHH-NH2 |
| 1913 | H10 | BY-2 plant cells | TAMRA | 27885926 | 12000 | Cellular uptake | 1uM | 12h | 27ºC | CLSM | Cellular uptake | HHHHHHHHHH-NH2 |
| 1914 | H12 | BY-2 plant cells | TAMRA | 27885926 | 5000 | Cellular uptake | 1uM | 12h | 27ºC | CLSM | Cellular uptake | HHHHHHHHHHHH-NH2 |
| 1915 | H14 | BY-2 plant cells | TAMRA | 27885926 | 6000 | Cellular uptake | 1uM | 12h | 27ºC | CLSM | Cellular uptake | HHHHHHHHHHHHHH-NH2 |
| 1916 | H16 | BY-2 plant cells | TAMRA | 27885926 | 6000 | Cellular uptake | 1uM | 12h | 27ºC | CLSM | Cellular uptake | HHHHHHHHHHHHHHHH-NH2 |
| 1917 | H18 | BY-2 plant cells | TAMRA | 27885926 | 3000 | Cellular uptake | 1uM | 12h | 27ºC | CLSM | Cellular uptake | HHHHHHHHHHHHHHHHHH-NH2 |
| 1918 | H20 | BY-2 plant cells | TAMRA | 27885926 | 3000 | Cellular uptake | 1uM | 12h | 27ºC | CLSM | Cellular uptake | HHHHHHHHHHHHHHHHHHHH-NH2 |
| 1919 | H22 | BY-2 plant cells | TAMRA | 27885926 | 1000 | Cellular uptake | 1uM | 12h | 27ºC | CLSM | Cellular uptake | HHHHHHHHHHHHHHHHHHHHHH-NH2 |
| 1920 | H24 | BY-2 plant cells | TAMRA | 27885926 | 2000 | Cellular uptake | 1uM | 12h | 27ºC | CLSM | Cellular uptake | HHHHHHHHHHHHHHHHHHHHHHHH-NH2 |
| 1921 | Lip-Cou6 | MCF7 cells | Cou-6 | 35539172 | 40 | Mean Fluorescence intensity | NA | 1h | 37ºC | Flow cytometry | Cellular uptake | PFVYL-Cou6 |
| 1922 | PFV-Lip-Cou6 | MCF7 cells | Cou-6 | 35539172 | 90 | Mean Fluorescence intensity | NA | 1h | 37ºC | Flow cytometry | Cellular uptake | PFVYL-Lip-Cou6 |
| 1923 | His16-Lyso | HT1080 cells | lysosomes | 31426598 | 100 | Relative cellular uptake (%) | NA | NA | 37ºC | Flow cytometry | Cellular uptake | stearly-His6-HHHHHHHHHHHHHHHH–NH2 |
| 1924 | R9 | A549 cells | chitosan/siRNA | 26568525 | 70 | Cellular uptake (%) | NA | NA | NA | Flow cytometry | Cellular uptake | RRRRRRRRR |
| 1925 | R9G4 | A549 cells | chitosan/siRNA | 26568525 | 80 | Cellular uptake (%) | NA | NA | NA | Flow cytometry | Cellular uptake | RRRRRRRRRGGGG |
| 1926 | R9G10 | A549 cells | chitosan/siRNA | 26568525 | 90 | Cellular uptake (%) | NA | NA | NA | Flow cytometry | Cellular uptake | RRRRRRRRRGGGGGGGGGG |
| 1927 | RhB-NLC-R11 | HaCaT cells | RhB | 31447556 | 350 | Mean Fluorescence intensity | 6ug/mL | 1h | 37ºC | Flow cytometry | Cellular uptake | HHHHHH-RRRRRRRRRRR |
| 1928 | RhB-NLC-R11 | HaCaT cells | RhB | 31447556 | 800 | Mean Fluorescence intensity | 12ug/mL | 2h | 37ºC | Flow cytometry | Cellular uptake | HHHHHH-RRRRRRRRRRR |
| 1929 | RhB-NLC-R11 | HaCaT cells | RhB | 31447556 | 1050 | Mean Fluorescence intensity | 25ug/mL | 4h | 37ºC | Flow cytometry | Cellular uptake | HHHHHH-RRRRRRRRRRR |
| 1930 | ppTG21 | HepG2 cells | GFP | 30994954 | 0.3 | Fluorescence intensity | 30uM | 90min | NA | CLSM | Cellular uptake | GLFHALLHLLHSLWHLLLHA |
| 1931 | Cys-penetratin | TR146 cell | Alexa 647-sCT | 35210769 | 3800 | Relative Mean Fluorescence intensity | NA | 24h | 37ºC | Flow cytometry | Cellular uptake | CRQIKIWFQNRRMKWKK |
| 1932 | PFV | U87 cells | Doxorubicin | 30261346 | 52 | Cellular uptake (%) | NA | 2h | 37ºC | Flow cytometry | Cellular uptake | PFVYLI |
| 1933 | PFV | bEnd.3 cells | Doxorubicin | 30261346 | 50 | Cellular uptake (%) | NA | 2h | 37ºC | Flow cytometry | Cellular uptake | PFVYLI |
| 1934 | PFV | Glial cells | Doxorubicin | 30261346 | 50 | Cellular uptake (%) | NA | 2h | 37ºC | Flow cytometry | Cellular uptake | PFVYLI |
| 1935 | Tf-PFV | U87 cells | Doxorubicin | 30261346 | 65 | Cellular uptake (%) | NA | 2h | 37ºC | Flow cytometry | Cellular uptake | Tf-PFVYLI |
| 1936 | Tf-PFV | bEnd.3 cells | Doxorubicin | 30261346 | 5 | Cellular uptake (%) | NA | 2h | 37ºC | Flow cytometry | Cellular uptake | Tf-PFVYLI |
| 1937 | Tf-PFV | Glial cells | Doxorubicin | 30261346 | 62 | Cellular uptake (%) | NA | 2h | 37ºC | Flow cytometry | Cellular uptake | Tf-PFVYLI |
| 1938 | PFV | U87 cells | Erlo | 30261346 | 45 | Cellular uptake (%) | NA | 2h | 37ºC | Flow cytometry | Cellular uptake | PFVYLI |
| 1939 | PFV | bEnd.3 cells | Erlo | 30261346 | 47 | Cellular uptake (%) | NA | 2h | 37ºC | Flow cytometry | Cellular uptake | PFVYLI |
| 1940 | PFV | Glial cells | Erlo | 30261346 | 43 | Cellular uptake (%) | NA | 2h | 37ºC | Flow cytometry | Cellular uptake | PFVYLI |
| 1941 | Tf-PFV | U87 cells | Erlo | 30261346 | 70 | Cellular uptake (%) | NA | 2h | 37ºC | Flow cytometry | Cellular uptake | Tf-PFVYLI |
| 1942 | Tf-PFV | bEnd.3 cells | Erlo | 30261346 | 69 | Cellular uptake (%) | NA | 2h | 37ºC | Flow cytometry | Cellular uptake | Tf-PFVYLI |
| 1943 | Tf-PFV | Glial cells | Erlo | 30261346 | 65 | Cellular uptake (%) | NA | 2h | 37ºC | Flow cytometry | Cellular uptake | Tf-PFVYLI |
| 1944 | PPP | MCF7 cells | NPs | 27043442 | 90 | Mean Fluorescence intensity | NA | 30min | NA | Flow cytometry | Cellular uptake | CGRRMKWKKXXXXGGGGEEEERRRR |
| 1945 | PPP | MCF7 cells | NPs | 27043442 | 110 | Mean Fluorescence intensity | NA | 30min | NA | Flow cytometry | Cellular uptake | CGRRMKWKKXXXXGGGGEEEERRRR |
| 1946 | RU006 | HeLa cells | Doxorubicin | 29113134 | 0.4 | Fluorescence intensity | 10uM | 6h | 25ºC | CLSM | Dox encapsulation | AIAKAXKIA |
| 1947 | RU006 | HeLa cells | Doxorubicin | 29113134 | 0.6 | Fluorescence intensity | 20uM | 6h | 25ºC | CLSM | Dox encapsulation | AIAKAXKIA |
| 1948 | RU006 | HeLa cells | Doxorubicin | 29113134 | 0.8 | Fluorescence intensity | 50uM | 6h | 25ºC | CLSM | Dox encapsulation | AIAKAXKIA |
| 1949 | BP9 | HepG2 cells | Doxorubicin | 31452330 | 0 | NA | NA | 3h | 37ºC | CLSM | Cellular uptake | AHLHNRS |
| 1950 | TH | HeLa cells | FITC | 28603674 | 1600 | Fluorescence intensity | 5uM | 1h | 37ºC | Flow cytometry | Cellular uptake | AGYLLGHINLHHLAHL(Aib)HHIL-NH2 |
| 1951 | TH | HeLa cells | FITC | 28603674 | 1700 | Fluorescence intensity | 5uM | 1h | 37ºC | Flow cytometry | Cellular uptake | AGYLLGHINLHHLAHL(Aib)HHIL-NH2 |
| 1952 | TH | HeLa cells | FITC | 28603674 | 2750 | Fluorescence intensity | 5uM | 1h | 37ºC | Flow cytometry | Cellular uptake | AGYLLGHINLHHLAHL(Aib)HHIL-NH2 |
| 1953 | Methly-TH | HeLa cells | FITC | 28603674 | 1550 | Fluorescence intensity | 5uM | 1h | 37ºC | Flow cytometry | Cellular uptake | AGYLLGHMINLHMHMLAHML(Aib)HMHMIL-NH2 |
| 1954 | Methly-TH | HeLa cells | FITC | 28603674 | 1600 | Fluorescence intensity | 5uM | 1h | 37ºC | Flow cytometry | Cellular uptake | AGYLLGHMINLHMHMLAHML(Aib)HMHMIL-NH2 |
| 1955 | Methly-TH | HeLa cells | FITC | 28603674 | 1900 | Fluorescence intensity | 5uM | 1h | 37ºC | Flow cytometry | Cellular uptake | AGYLLGHMINLHMHMLAHML(Aib)HMHMIL-NH2 |
| 1956 | Ethyl-TH | HeLa cells | FITC | 28603674 | 1200 | Fluorescence intensity | 5uM | 1h | 37ºC | Flow cytometry | Cellular uptake | AGYLLGHEINLHEHELAHEL(Aib)HEHEIL-NH2 |
| 1957 | Ethyl-TH | HeLa cells | FITC | 28603674 | 1100 | Fluorescence intensity | 5uM | 1h | 37ºC | Flow cytometry | Cellular uptake | AGYLLGHEINLHEHELAHEL(Aib)HEHEIL-NH2 |
| 1958 | Ethyl-TH | HeLa cells | FITC | 28603674 | 2250 | Fluorescence intensity | 5uM | 1h | 37ºC | Flow cytometry | Cellular uptake | AGYLLGHEINLHEHELAHEL(Aib)HEHEIL-NH2 |
| 1959 | Isopropyl-TH | HeLa cells | FITC | 28603674 | 1750 | Fluorescence intensity | 5uM | 1h | 37ºC | Flow cytometry | Cellular uptake | AGYLLGHIINLHIHILAHIL(Aib)HIHIIL-NH2 |
| 1960 | Isopropyl-TH | HeLa cells | FITC | 28603674 | 1500 | Fluorescence intensity | 5uM | 1h | 37ºC | Flow cytometry | Cellular uptake | AGYLLGHIINLHIHILAHIL(Aib)HIHIIL-NH2 |
| 1961 | Isopropyl-TH | HeLa cells | FITC | 28603674 | 2250 | Fluorescence intensity | 5uM | 1h | 37ºC | Flow cytometry | Cellular uptake | AGYLLGHIINLHIHILAHIL(Aib)HIHIIL-NH2 |
| 1962 | Butyl-TH | HeLa cells | FITC | 28603674 | 2200 | Fluorescence intensity | 5uM | 1h | 37ºC | Flow cytometry | Cellular uptake | AGYLLGHBINLHBHBLAHBL(Aib)HBHBIL-NH2 |
| 1963 | Butyl-TH | HeLa cells | FITC | 28603674 | 2800 | Fluorescence intensity | 5uM | 1h | 37ºC | Flow cytometry | Cellular uptake | AGYLLGHBINLHBHBLAHBL(Aib)HBHBIL-NH2 |
| 1964 | Butyl-TH | HeLa cells | FITC | 28603674 | 2500 | Fluorescence intensity | 5uM | 1h | 37ºC | Flow cytometry | Cellular uptake | AGYLLGHBINLHBHBLAHBL(Aib)HBHBIL-NH2 |
| 1965 | NC-2 | hPSC cells | FAM-labeled AMO | 28524768 | 155 | Mean Fluorescence intensity | NA | 6h | 37ºC | Flow cytometry | Cellular uptake | RRRRGGRRRRRRSVCSSCVSRRRRRRGGRRRR |
| 1966 | NC-2 | BJ-fibroblasts | FAM-labeled AMO | 28524768 | 15 | Mean Fluorescence intensity | NA | 6h | 37ºC | Flow cytometry | Cellular uptake | RRRRGGRRRRRRSVCSSCVSRRRRRRGGRRRR |
| 1967 | NC-2 | Panc-1 | FAM-labeled AMO | 28524768 | 10 | Mean Fluorescence intensity | NA | 6h | 37ºC | Flow cytometry | Cellular uptake | RRRRGGRRRRRRSVCSSCVSRRRRRRGGRRRR |
| 1968 | NC-2 | AsPc-1 | FAM-labeled AMO | 28524768 | 3 | Mean Fluorescence intensity | NA | 6h | 37ºC | Flow cytometry | Cellular uptake | RRRRGGRRRRRRSVCSSCVSRRRRRRGGRRRR |
| 1969 | NC-2 | MiaPaCa-2 | FAM-labeled AMO | 28524768 | 3 | Mean Fluorescence intensity | NA | 6h | 37ºC | Flow cytometry | Cellular uptake | RRRRGGRRRRRRSVCSSCVSRRRRRRGGRRRR |
| 1970 | dNP2 | HeLa cells | FITC | 32254889 | 100 | Fluorescence intensity | NA | 4h | NA | Flow cytometry | Cellular uptake | CKIKKVKKKGRKKIKKVKKKGRK |
| 1971 | dNP2 | HeLa cells | FITC | 32254889 | 350 | Fluorescence intensity | NA | 18h | NA | Flow cytometry | Cellular uptake | CKIKKVKKKGRKKIKKVKKKGRK |
| 1972 | SAH-P53-8 | HeLa cells | Rho | 29150077 | 700 | Cellular uptake | NA | 30min | 37ºC | Flow cytometry | Cellular uptake | QSQQTFNLWKLLQN |
| 1973 | SAH-p53-4 | HeLa cells | Rho | 29150077 | 500 | Cellular uptake | NA | 30min | 37ºC | Flow cytometry | Cellular uptake | LSQETFDLWKLLEN |
| 1974 | BP1.2 | HeLa cells | Rho | 29150077 | 1200 | Cellular uptake | NA | 30min | 37ºC | Flow cytometry | Cellular uptake | RSQRRFRLWRLLEN |
| 1975 | BP1.3 | HeLa cells | Rho | 29150077 | 1700 | Cellular uptake | NA | 30min | 37ºC | Flow cytometry | Cellular uptake | RRRRRFDLWKLLEN |
| 1976 | BP1.4 | HeLa cells | Rho | 29150077 | 3500 | Cellular uptake | NA | 30min | 37ºC | Flow cytometry | Cellular uptake | RSQERFDLWKLLEN |
| 1977 | BP1.5 | HeLa cells | Rho | 29150077 | 1500 | Cellular uptake | NA | 30min | 37ºC | Flow cytometry | Cellular uptake | LRRETFDRWKRLRR |
| 1978 | BP1.6 | HeLa cells | Rho | 29150077 | 2500 | Cellular uptake | NA | 30min | 37ºC | Flow cytometry | Cellular uptake | LSQETFRLWRRLRR |
| 1979 | BP1.7 | HeLa cells | Rho | 29150077 | 1600 | Cellular uptake | NA | 30min | 37ºC | Flow cytometry | Cellular uptake | LRRETFDLWKRLRR |
| 1980 | NR2B9c | BCECs cells | TAMRA | 32674358 | 0.02 | Cell peptide accumulation (mol*cm^-2) | 100uM | 3h | 37ºC | Fluorescent Microscopy | Live cell peptide uptake | KLSSIESDV |
| 1981 | Tat-NR2B9c | BCECs cells | TAMRA | 32674358 | 0.09 | Cell peptide accumulation (mol*cm^-2) | 100uM | 3h | 37ºC | Fluorescent Microscopy | Live cell peptide uptake | YGRKKRRQRRRKLSSIESDV |
| 1982 | Tat-N-dimer | BCECs cells | TAMRA | 32674358 | 0.05 | Cell peptide accumulation (mol*cm^-2) | 100uM | 3h | 37ºC | Fluorescent Microscopy | Live cell peptide uptake | YGRKKRRQRRRN |
| 1983 | CB5005-Cy | U87 cells | Carboxyfluorescein | 30243823 | 1500 | Mean value of cellular uptake | 1uM | 4h | 37ºC | Flow cytometry | Cellular uptake | KLKLALALALAVQRKRQKLMPC |
| 1984 | CB5005-Cy | U87 cells | Carboxyfluorescein | 30243823 | 500 | Mean value of cellular uptake | 0.1uM | 4h | 37ºC | Flow cytometry | Cellular uptake | KLKLALALALAVQRKRQKLMPC |
| 1985 | CB5005-Cy | U87 cells | Carboxyfluorescein | 30243823 | 70 | Mean value of cellular uptake | 0.01uM | 4h | 37ºC | Flow cytometry | Cellular uptake | KLKLALALALAVQRKRQKLMPC |
| 1986 | Dox-SS[C(WR)4K] | HT1080 cells | Doxorubicin | 30396106 | 8000 | Mean Fluorescence intensity | 50uM | 3h | 37ºC | Flow cytometry | Cellular uptake | CWRWRWRWRK |
| 1987 | Dox-SS[C(WR)4K] | HEK293 cells | Doxorubicin | 30396106 | 6000 | Mean Fluorescence intensity | 50uM | 3h | 37ºC | Flow cytometry | Cellular uptake | CWRWRWRWRK |
| 1988 | Dox-SS[C(WR)4K] | SK-OV-3 cells | Doxorubicin | 30396106 | 13000 | Mean Fluorescence intensity | 50uM | 3h | 37ºC | Flow cytometry | Cellular uptake | CWRWRWRWRK |
| 1989 | Dox-SS[C(WR)4K] | CCRF-CEM cells | Doxorubicin | 30396106 | 5000 | Mean Fluorescence intensity | 50uM | 3h | 37ºC | Flow cytometry | Cellular uptake | CWRWRWRWRK |
| 1990 | KL4 | A549 cells | siRNA | 32352853 | 75 | Cellular uptake (%) | 3000 pmol | 4h | 37ºC | Flow cytometry | Cellular uptake | KLLLLKLLLLKLLLLKLLLLK |
| 1991 | KA2 | A549 cells | siRNA | 32352853 | 0 | Cellular uptake (%) | 3000 pmol | 4h | 37ºC | Flow cytometry | Cellular uptake | KAALLKAALLKAALLKAALLK |
| 1992 | KV4 | A549 cells | siRNA | 32352853 | 90 | Cellular uptake (%) | 3000 pmol | 4h | 37ºC | Flow cytometry | Cellular uptake | KVVVVKVVVVKVVVVKVVVVK |
| 1993 | DNP | Caco-2 cells | Carboxyfluorescein | 28757359 | 2 | Uptake amount (x10^3 pfu/ug protein) | 10uM | 10min | 37ºC | CLSM | Cellular uptake | ACDNPGNETCGGGS |
| 1994 | DRIM | HEK293 cells | NA | 28921993 | 8 | Normalized fluorescence intensities | 2uM | 4h | 37ºC | Flow cytometry | Cellular uptake | QQRKRKIWSILAPLGTTLVKLVAGIG |
| 1995 | WWSP | HEK293 cells | NA | 28921993 | 10 | Normalized fluorescence intensities | 2uM | 4h | 37ºC | Flow cytometry | Cellular uptake | PLILLRLLRGQF |
| 1996 | KFGF | HEK293 cells | NA | 28921993 | 1 | Normalized fluorescence intensities | 2uM | 4h | 37ºC | Flow cytometry | Cellular uptake | AAVLLPVLLAAP |
| 1997 | MAP-1 | HEK293 cells | NA | 28921993 | 20 | Normalized fluorescence intensities | 2uM | 4h | 37ºC | Flow cytometry | Cellular uptake | KLALKALKALKAALKLA |
| 1998 | sDRIM | HEK293 cells | NA | 28921993 | 5 | Normalized fluorescence intensities | 2uM | 4h | 37ºC | Flow cytometry | Cellular uptake | QQRKRKIWSKLAPDGTTLVKLVAGIG |
| 1999 | sWWSP | HEK293 cells | NA | 28921993 | 2 | Normalized fluorescence intensities | 2uM | 4h | 37ºC | Flow cytometry | Cellular uptake | PLIKLRLDRGQF |
| 2000 | sKFGF | HEK293 cells | NA | 28921993 | 1 | Normalized fluorescence intensities | 2uM | 4h | 37ºC | Flow cytometry | Cellular uptake | AAKLLPDLLAAP |
| 2001 | sMAP-1 | HEK293 cells | NA | 28921993 | 18 | Normalized fluorescence intensities | 2uM | 4h | 37ºC | Flow cytometry | Cellular uptake | KLALKALKKLKADLKLA |
| 2002 | DRIM | HeLa cells | NA | 28921993 | 20 | Normalized fluorescence intensities | 2uM | 4h | 37ºC | Flow cytometry | Cellular uptake | QQRKRKIWSILAPLGTTLVKLVAGIG |
| 2003 | WWSP | HeLa cells | NA | 28921993 | 10 | Normalized fluorescence intensities | 2uM | 4h | 37ºC | Flow cytometry | Cellular uptake | PLILLRLLRGQF |
| 2004 | KFGF | HeLa cells | NA | 28921993 | 1 | Normalized fluorescence intensities | 2uM | 4h | 37ºC | Flow cytometry | Cellular uptake | AAVLLPVLLAAP |
| 2005 | MAP-1 | HeLa cells | NA | 28921993 | 25 | Normalized fluorescence intensities | 2uM | 4h | 37ºC | Flow cytometry | Cellular uptake | KLALKALKALKAALKLA |
| 2006 | sDRIM | HeLa cells | NA | 28921993 | 3 | Normalized fluorescence intensities | 2uM | 4h | 37ºC | Flow cytometry | Cellular uptake | QQRKRKIWSKLAPDGTTLVKLVAGIG |
| 2007 | sWWSP | HeLa cells | NA | 28921993 | 2 | Normalized fluorescence intensities | 2uM | 4h | 37ºC | Flow cytometry | Cellular uptake | PLIKLRLDRGQF |
| 2008 | sKFGF | HeLa cells | NA | 28921993 | 1 | Normalized fluorescence intensities | 2uM | 4h | 37ºC | Flow cytometry | Cellular uptake | AAKLLPDLLAAP |
| 2009 | sMAP-1 | HeLa cells | NA | 28921993 | 15 | Normalized fluorescence intensities | 2uM | 4h | 37ºC | Flow cytometry | Cellular uptake | KLALKALKKLKADLKLA |
| 2010 | Cur | MCF7 cells | NPs | 31691601 | 5500 | Fluorescence intensity | 25ug/ml | 4h | 37ºC | Flow cytometry | Cellular uptake | GPLGIAGQrrrrrrrrr |
| 2011 | Cur | MCF7 cells | P-NPs | 31691601 | 9000 | Fluorescence intensity | 25ug/ml | 4h | 37ºC | Flow cytometry | Cellular uptake | GPLGIAGQrrrrrrrrr |
| 2012 | PEG2k-ppTAT-PEG1k-PE | A549 cells | MMP2 | 28870072 | 280 | PTX | 2mg/ml | 4h | 37ºC | Flow cytometry | Cellular uptake | GPLGIAGQYGRKKRRQRRRC |
| 2013 | PEG2k-ppTAT-PEG1k-PE | MCF7 cells | MMP2 | 28870072 | 200 | PTX | 2mg/ml | 4h | 37ºC | Flow cytometry | Cellular uptake | GPLGIAGQYGRKKRRQRRRC |
| 2014 | StA-R8 | HepG2 cells | Cy3-siRNA | 27354583 | 40 | Mean Fluorescence intensity | NA | 4h | 37ºC | Flow cytometry | Cellular uptake | CH3(CH2)16-CONH-RRRRRRRR |
| 2015 | StA-R8 | A549 cells | Cy3-siRNA | 27354583 | 48 | Mean Fluorescence intensity | NA | 4h | 37ºC | Flow cytometry | Cellular uptake | CH3(CH2)16-CONH-RRRRRRRR |
| 2016 | StA-R8 liposome | HepG2 cells | Cy3-siRNA | 27354583 | 45 | Mean Fluorescence intensity | NA | 4h | 37ºC | Flow cytometry | Cellular uptake | CH3(CH2)16-CONH-RRRRRRRRRR |
| 2017 | StA-R8 liposome | A549 cells | Cy3-siRNA | 27354583 | 50 | Mean Fluorescence intensity | NA | 4h | 37ºC | Flow cytometry | Cellular uptake | CH3(CH2)16-CONH-RRRRRRRRRR |
| 2018 | vaults 1a | RAW264.7 cells | FITC | 28029784 | 10000 | Mean Fluorescence intensity | 10ug | 16h | 37ºC | Flow cytometry | Cellular uptake | MAGCGCPCGCGA |
| 2019 | Vault-r8Cleavable 8 | RAW264.7 cells | FITC | 28029784 | 20000 | Mean Fluorescence intensity | 10ug | 16h | 37ºC | Flow cytometry | Cellular uptake | MAGCGCPCGCGA |
| 2020 | Vault-r8Noncleavable 12 | RAW264.7 cells | FITC | 28029784 | 80000 | Mean Fluorescence intensity | 10ug | 16h | 37ºC | Flow cytometry | Cellular uptake | MAGCGCPCGCGA |
| 2021 | vaults 1a | HeLa cells | FITC | 28029784 | 3500 | Mean Fluorescence intensity | 10ug | 16h | 37ºC | Flow cytometry | Cellular uptake | MAGCGCPCGCGA |
| 2022 | Vault-r8Cleavable 8 | HeLa cells | FITC | 28029784 | 4500 | Mean Fluorescence intensity | 10ug | 16h | 37ºC | Flow cytometry | Cellular uptake | MAGCGCPCGCGA |
| 2023 | Vault-r8Noncleavable 12 | HeLa cells | FITC | 28029784 | 6000 | Mean Fluorescence intensity | 10ug | 16h | 37ºC | Flow cytometry | Cellular uptake | MAGCGCPCGCGA |
| 2024 | vaults 1a | CHO-K1 cells | FITC | 28029784 | 1800 | Mean Fluorescence intensity | 10ug | 16h | 37ºC | Flow cytometry | Cellular uptake | MAGCGCPCGCGA |
| 2025 | Vault-r8Cleavable 8 | CHO-K1 cells | FITC | 28029784 | 2300 | Mean Fluorescence intensity | 10ug | 16h | 37ºC | Flow cytometry | Cellular uptake | MAGCGCPCGCGA |
| 2026 | Vault-r8Noncleavable 12 | CHO-K1 cells | FITC | 28029784 | 2600 | Mean Fluorescence intensity | 10ug | 16h | 37ºC | Flow cytometry | Cellular uptake | MAGCGCPCGCGA |
| 2027 | C6M1 | CHO-K1 cells | Cy3-siRNA | 26682443 | 100 | Relative fluorescence (%) | NA | 4h | 37ºC | Flow cytometry | Cellular uptake | Acetyl-RLWRLLWRLWRRLWRLLR-NH2 |
| 2028 | DM1 | CHO-K1 cells | Cy3-siRNA | 26682443 | 95 | Relative fluorescence (%) | NA | 4h | 37ºC | Flow cytometry | Cellular uptake | DEG-RLWRLLWRLWRRLWRLLR-NH2 |
| 2029 | R1PECL | HeLa cells | NA | 27532744 | 1000 | Fluorescence intensity | NA | 24h | NA | Flow cytometry | Cellular uptake | RC-PEG-b-PCL |
| 2030 | R4PECL | HeLa cells | NA | 27532744 | 2500 | Fluorescence intensity | NA | 24h | NA | Flow cytometry | Cellular uptake | RRRRC-PEG-b-PCL |
| 2031 | R8PECL | HeLa cells | NA | 27532744 | 8000 | Fluorescence intensity | NA | 24h | NA | Flow cytometry | Cellular uptake | RRRRRRRRC-PEG-b-PCL |
| 2032 | R7E7 | MDA-MB-231 cells | FITC | 30774914 | 40 | Intensity | 10uM | 10min | NA | Flow cytometry | Cellular uptake | RRRRRRREEEEEEE |
| 2033 | R7E7 | MDA-MB-231 cells | FITC | 30774914 | 160 | Intensity | 50uM | 10min | NA | Flow cytometry | Cellular uptake | RRRRRRREEEEEEE |
| 2034 | R7E7 | MDA-MB-231 cells | FITC | 30774914 | 200 | Intensity | 100uM | 10min | NA | Flow cytometry | Cellular uptake | RRRRRRREEEEEEE |
| 2035 | PLGA/R6LRVG | Caco-2 cells | FITC | 34239301 | 1500 | Mean Fluorescence intensity | 600 ug/ml | 3h | NA | Flow cytometry | Cellular uptake | RRRRRRLRVG |
| 2036 | HPRP-A1 | A549 cells | FITC | 29396568 | 25 | Fluorescence intensity | 16uM | 100s | 37ºC | Flow cytometry | Cellular uptake | FKKLKKLFSKLWNWK |
| 2037 | HPRP-A1-iRGD | A549 cells | FITC | 29396568 | 35 | Fluorescence intensity | 16uM | 100s | 37ºC | Flow cytometry | Cellular uptake | FKKLKKLFSKLWNWKCRGDKGPDC |
| 2038 | RCCNPs | HepG2 cells | NA | 34893294 | 8000 | Mean Fluorescence intensity | NA | 3h | 37ºC | Flow cytometry | Cellular uptake | RRRRRRHHHH |
| 2039 | RCCNPs | HepG2 cells | NA | 34893294 | 11000 | Mean Fluorescence intensity | NA | 3h | 37ºC | Flow cytometry | Cellular uptake | RRRRRRHHHH |
| 2040 | NFL-TBS.40-63 | J3T cells | LNC-(DiD) | 34144141 | 17 | Fluorescent cells (%) | 1 mg/ml | 12h | 37ºC | Flow cytometry | Cellular uptake of LNC-(DiD) | YSSYSAPVSSSLSVRRSYSSSSGS |
| 2041 | R-NLC | A549 cells | Cou-6 | 32104313 | 3500 | Cou 6/protein /ug/mg) | 2ug/ml | 2h | NA | Flow cytometry | Cellular uptake | RRRRRRRRNLC |
| 2042 | dNP2 | MDA-MB-231 cells | Cou-6-NLC | 33921919 | 2300 | Mean Fluorescence intensity | NA | 4h | 37ºC | Flow cytometry | Cellular uptake | CKIKKVKKKGRKKIKKVKKKGRK |
| 2043 | dNP2 | MDA-MB-231 cells | Cou-6-NLC | 33921919 | 2200 | Mean Fluorescence intensity | NA | 8h | 37ºC | Flow cytometry | Cellular uptake | CKIKKVKKKGRKKIKKVKKKGRK |
| 2044 | dNP2 | 4T1 cells | Cou-6-NLC | 33921919 | 2000 | Mean Fluorescence intensity | NA | 4h | 37ºC | Flow cytometry | Cellular uptake | CKIKKVKKKGRKKIKKVKKKGRK |
| 2045 | dNP2 | 4T1 cells | Cou-6-NLC | 33921919 | 2200 | Mean Fluorescence intensity | NA | 8h | 37ºC | Flow cytometry | Cellular uptake | CKIKKVKKKGRKKIKKVKKKGRK |
| 2046 | dNP2 | MCF7 cells | Cou-6-NLC | 33921919 | 3000 | Mean Fluorescence intensity | NA | 4h | 37ºC | Flow cytometry | Cellular uptake | CKIKKVKKKGRKKIKKVKKKGRK |
| 2047 | dNP2 | MCF7 cells | Cou-6-NLC | 33921919 | 3400 | Mean Fluorescence intensity | NA | 8h | 37ºC | Flow cytometry | Cellular uptake | CKIKKVKKKGRKKIKKVKKKGRK |
| 2048 | tLyP-1-HFtn | MDA-MB-231 cells | FITC | 33568906 | 120 | Mean Fluorescence intensity | NA | 4h | 37ºC | Flow cytometry | Cellular uptake | CGNKRTR |
| 2049 | M-tLyP-1-HFtn | MDA-MB-231 cells | FITC | 33568906 | 20 | Mean Fluorescence intensity | NA | 4h | 37ºC | Flow cytometry | Cellular uptake | CGNARTA |
| 2050 | P7 | A549 cells | Carboxyfluorescein | 33995950 | 100 | Cell Fluorescence | 25uM | 90min | 37ºC | Flow cytometry | Cellular uptake | COOH-RRRRRRRRRR-NH2 |
| 2051 | P8 | A549 cells | Carboxyfluorescein | 33995950 | 75 | Cell Fluorescence | 25uM | 90min | 37ºC | Flow cytometry | Cellular uptake | COOH-KKKKKKKKKK-NH2 |
| 2052 | TAT-ASA-MNP-CDDP | HNE-1 cells | FITC | 30826059 | 1800 | Fluorescence intensity | 5ug/ml | 2h | NA | Flow cytometry | Intracellular uptake | YGRKKRRQRRR |
| 2053 | TAT-ASA-MNP-CDDP | CNE-2 cells | FITC | 30826059 | 800 | Fluorescence intensity | 5ug/ml | 2h | NA | Flow cytometry | Intracellular uptake | YGRKKRRQRRR |
| 2054 | IF-7 | A549 cells | CMNC | 31686810 | 5000 | Mean Fluorescence intensity | 100ug | 30min | 37ºC | Flow cytometry | Cellular uptake | IFLLWQ |
| 2055 | IF-7 | A549 cells | CMNC | 31686810 | 10000 | Mean Fluorescence intensity | 100ug | 1h | 37ºC | Flow cytometry | Cellular uptake | IFLLWQ |
| 2056 | IF-7 | A549 cells | CMNC | 31686810 | 16000 | Mean Fluorescence intensity | 100ug | 2h | 37ºC | Flow cytometry | Cellular uptake | IFLLWQ |
| 2057 | IF-7 | A549 cells | CMNC | 31686810 | 17000 | Mean Fluorescence intensity | 100ug | 4h | 37ºC | Flow cytometry | Cellular uptake | IFLLWQ |
| 2058 | PP1 | HUVEC cells | Cy5 | 30855618 | 1000 | Mean Fluorescence intensity | NA | 4h | 37ºC | Flow cytometry | Cellular uptake | CGPKKKRKVGYGRKKRRQRRR |
| 2059 | PP1 | HUVEC cells | BCPs | 30855618 | 5000 | Mean Fluorescence intensity | NA | 4h | 37ºC | Flow cytometry | Cellular uptake | CGPKKKRKVGYGRKKRRQRRR |
| 2060 | PP1 | HUVEC cells | TCPs-1 | 30855618 | 3800 | Mean Fluorescence intensity | NA | 4h | 37ºC | Flow cytometry | Cellular uptake | CGPKKKRKVGYGRKKRRQRRR |
| 2061 | PP1 | HUVEC cells | TCPs-2 | 30855618 | 3500 | Mean Fluorescence intensity | NA | 4h | 37ºC | Flow cytometry | Cellular uptake | CGPKKKRKVGYGRKKRRQRRR |
| 2062 | PP1 | HUVEC cells | TCPs-3 | 30855618 | 3000 | Mean Fluorescence intensity | NA | 4h | 37ºC | Flow cytometry | Cellular uptake | CGPKKKRKVGYGRKKRRQRRR |
| 2063 | DP7-C | GL261 cells | siRNA | 34973309 | 130000 | Mean Fluorescence intensity | NA | 4h | NA | Flow cytometry | Cellular uptake | VQWRIRVAVIRK |
| 2064 | GBP(L) | A549 cells | L-DOX | 32241176 | 1.1 | Cellular uptake | NA | 24h | 37ºC | Flow cytometry | Cellular uptake | NYRWRCKN |
| 2065 | GBP(M) | A549 cells | L-DOX | 32241176 | 2.6 | Cellular uptake | NA | 24h | 37ºC | Flow cytometry | Cellular uptake | NYRWRCKN |
| 2066 | GBP(H) | A549 cells | L-DOX | 32241176 | 5.7 | Cellular uptake | NA | 24h | 37ºC | Flow cytometry | Cellular uptake | NYRWRCKN |
| 2067 | R8NLS | A2780 cells | P-GFLG-FITC | 26784985 | 42 | Mean Fluorescence intensity | 5uM | 1h | 37ºC | Flow cytometry | Cellular uptake | CRRRRRRRRVKRKKKP |
| 2068 | R8NLS | A2780 cells | P-GFLG-FITC | 26784985 | 78 | Mean Fluorescence intensity | 10uM | 1h | 37ºC | Flow cytometry | Cellular uptake | CRRRRRRRRVKRKKKP |
| 2069 | R8NLS | A2780 cells | P-GFLG-FITC | 26784985 | 100 | Mean Fluorescence intensity | 15uM | 1h | 37ºC | Flow cytometry | Cellular uptake | CRRRRRRRRVKRKKKP |
| 2070 | R8NLS | A2780 cells | P-GFLG-FITC | 26784985 | 115 | Mean Fluorescence intensity | 20uM | 1h | 37ºC | Flow cytometry | Cellular uptake | CRRRRRRRRVKRKKKP |
| 2071 | R8NLS | A2780 cells | P-GFLG-FITC | 26784985 | 120 | Mean Fluorescence intensity | 25uM | 1h | 37ºC | Flow cytometry | Cellular uptake | CRRRRRRRRVKRKKKP |
| 2072 | R8NLS | A2780 cells | P-GFLG-FITC | 26784985 | 130 | Mean Fluorescence intensity | 30uM | 1h | 37ºC | Flow cytometry | Cellular uptake | CRRRRRRRRVKRKKKP |
| 2073 | NT4 | HT29 cells | QDs | 29501065 | 14000 | Mean Fluorescence intensity | 20uM | 30min | 37ºC | Flow cytometry | QD internalization | ELYENKPRRPYIL |
| 2074 | NT4 | HT29 cells | QDs | 29501065 | 9000 | Mean Fluorescence intensity | 10uM | 30min | 37ºC | Flow cytometry | QD internalization | ELYENKPRRPYIL |
| 2075 | NT4 | HT29 cells | QDs | 29501065 | 5000 | Mean Fluorescence intensity | 5uM | 30min | 37ºC | Flow cytometry | QD internalization | ELYENKPRRPYIL |
| 2076 | NT4 | HT29 cells | QDs | 29501065 | 1000 | Mean Fluorescence intensity | 1uM | 30min | 37ºC | Flow cytometry | QD internalization | ELYENKPRRPYIL |
| 2077 | P2 | HeLa cells | FITC-siRNA | 35575337 | 5000 | Relative fluorescence | NA | 6h | NA | Flow cytometry | Cellular uptake | P(LAEMA37)-b-P(FPMA2-st-DMA2)-KRRKRRRRRK |
| 2078 | P3 | HeLa cells | FITC-siRNA | 35575337 | 4800 | Relative fluorescence | NA | 6h | NA | Flow cytometry | Cellular uptake | P(LAEMA23-st-FPMA3)-KRRKRRRRRK |
| 2079 | P4 | HeLa cells | FITC-siRNA | 35575337 | 5500 | Relative fluorescence | NA | 6h | NA | Flow cytometry | Cellular uptake | P(LAEMA25-st-FPMA2-st-DMA2)-KRRKRRRRRK |
| 2080 | L17E | HeLa cells | FITC | 35395514 | 100 | Relative Cellular uptake | 6uM | 1h | 37ºC | Flow cytometry | Cellular uptake | IWLTALKFLGKHAAKHEAKQQLSKL-GK(FITC)-NH2 |
| 2081 | L17ER2 | HeLa cells | FITC | 35395514 | 200 | Relative Cellular uptake | 6uM | 1h | 37ºC | Flow cytometry | Cellular uptake | IWLTALKFLGKHAAKHEAKQQLSKL-GRRGK(FITC)-NH2 |
| 2082 | L17ER4 | HeLa cells | FITC | 35395514 | 900 | Relative Cellular uptake | 6uM | 1h | 37ºC | Flow cytometry | Cellular uptake | IWLTALKFLGKHAAKHEAKQQLSKL-GRRRRGK(FITC)-NH2 |
| 2083 | R2L17E | HeLa cells | FITC | 35395514 | 220 | Relative Cellular uptake | 6uM | 1h | 37ºC | Flow cytometry | Cellular uptake | RRG-IWLTALKFLGKHAAKHEAKQQLSKL-GK(FITC)-NH2 |
| 2084 | R4L17E | HeLa cells | FITC | 35395514 | 800 | Relative Cellular uptake | 6uM | 1h | 37ºC | Flow cytometry | Cellular uptake | RRRRG-IWLTALKFLGKHAAKHEAKQQLSKL-GK(FITC)-NH2 |
| 2085 | JTS-1 | TF cells | FITC | 35601335 | 0 | NA | 1uM | 1h | NA | CLSM | Peptide uptake | GLFEALLELLESLWELLLEA |
| 2086 | STRAP-1 | MDA-MB-231 cells | Carboxyfluorescein | 35839086 | 500 | Mean Fluorescence intensity | 10uM | 4h | NA | Flow cytometry | Cellular uptake | KrKiFcL |
| 2087 | STRAP-2 | MDA-MB-231 cells | Carboxyfluorescein | 35839086 | 400 | Mean Fluorescence intensity | 10uM | 4h | NA | Flow cytometry | Cellular uptake | kRkIfCl |
| 2088 | STRAP-3 | MDA-MB-231 cells | Carboxyfluorescein | 35839086 | 800 | Mean Fluorescence intensity | 10uM | 4h | NA | Flow cytometry | Cellular uptake | KrKfIcL |
| 2089 | STRAP-4 | MDA-MB-231 cells | Carboxyfluorescein | 35839086 | 2000 | Mean Fluorescence intensity | 10uM | 4h | NA | Flow cytometry | Cellular uptake | kRkFiCl |
| 2090 | Oleyl-(HR)4 | MDA-MB-231 cells | siRNA-A488 | 35456715 | 10 | Mean Fluorescence intensity | 50nM | 24h | 37ºC | Flow cytometry | Cellular internalization of oleyl | HRHRHRHR |
| 2091 | Oleyl-R1-(HR)4 | MDA-MB-231 cells | siRNA-A489 | 35456715 | 50 | Mean Fluorescence intensity | 50nM | 24h | 37ºC | Flow cytometry | Cellular internalization of oleyl | RHRHRHRHR |
| 2092 | Oleyl-R2-(HR)4 | MDA-MB-231 cells | siRNA-A490 | 35456715 | 100 | Mean Fluorescence intensity | 50nM | 24h | 37ºC | Flow cytometry | Cellular internalization of oleyl | RRHRHRHRHR |
| 2093 | Oleyl-R3-(HR)4 | MDA-MB-231 cells | siRNA-A491 | 35456715 | 250 | Mean Fluorescence intensity | 50nM | 24h | 37ºC | Flow cytometry | Cellular internalization of oleyl | RRRHRHRHRHR |
| 2094 | Oleyl-R4-(HR)4 | MDA-MB-231 cells | siRNA-A492 | 35456715 | 400 | Mean Fluorescence intensity | 50nM | 24h | 37ºC | Flow cytometry | Cellular internalization of oleyl | RRRRHRHRHRHR |
| 2095 | Oleyl-R5-(HR)4 | MDA-MB-231 cells | siRNA-A493 | 35456715 | 500 | Mean Fluorescence intensity | 50nM | 24h | 37ºC | Flow cytometry | Cellular internalization of oleyl | RRRRRHRHRHRHR |
| 2096 | CyLoP-1 | NIH-3T3 cells | Carboxyfluorescein | 35752142 | 7000 | corr. Fluorescence | 2.5uM | 18h | 37ºC | Flow cytometry | Cellular internalization of oleyl | CRWRWKCCKK |